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List of works by William J. Kerr

A Practical and General Amidation Method from Isocyanates Enabled by Flow Technology

scientific article published on 17 August 2018

A tetrahydropentaleno[1,6a-a]naphthalen-4(2H)-one of defined relative stereochemistry for use towards Agariblazeispirol C

article

Anion effects to deliver enhanced iridium catalysts for hydrogen isotope exchange processes

scientific article

Application of neutral iridium(I) N-heterocyclic carbene complexes in ortho-directed hydrogen isotope exchange

scientific article published on 19 July 2013

Bismesitylmagnesium: a thermally stable and non-nucleophilic carbon-centred base reagent for the efficient preparation of silyl enol ethers

scientific article published on 27 September 2007

Boron phenylalanine and related impurities: HPLC analysis, stability profile and degradation pathways

scientific article published on 01 July 2011

C-H Functionalisation for Hydrogen Isotope Exchange

scientific article

Characterization of route specific impurities found in methamphetamine synthesized by the Leuckart and reductive amination methods

scientific article

Clarification of route specific impurities found in methylamphetamine synthesised using the Birch method

scientific article published on 03 November 2012

Cobalt close-up

scientific article published on 01 June 2011

Design, synthesis and antibacterial properties of pyrimido[4,5-b]indol-8-amine inhibitors of DNA gyrase

scientific article published on 26 May 2018

Deuterium- and Tritium-Labelled Compounds: Applications in the Life Sciences.

scientific article published on 16 August 2017

Discovery of Novel Irreversible Inhibitors of Interleukin (IL)-2-inducible Tyrosine Kinase (Itk) by Targeting Cysteine 442 in the ATP Pocket

scientific article

E- and Z-stereoselectivity in the preparation of enamides from glycidyl sulfonamides and carbamates

scientific article published on 29 November 2011

Efficient methods for enol phosphate synthesis using carbon-centred magnesium bases

scientific article published on 28 September 2015

Elemental profiling using ICPMS of methylamphetamine hydrochloride prepared from proprietary medication using the Moscow and hypophosphorous synthesis

scientific article published on 12 December 2012

Emerging use of isotope ratio mass spectrometry as a tool for discrimination of 3,4-methylenedioxymethamphetamine by synthetic route

scientific article published on 21 March 2008

Flexible access to conformationally-locked bicyclic morpholines.

scientific article

Formal total synthesis of (+/-)-alpha- and beta-cedrene by preparation of cedrone. Construction of the tricyclic carbon skeleton by the use of a highly efficient intramolecular Khand annulation.

scientific article

Highly active iridium(I) complexes for catalytic hydrogen isotope exchange.

scientific article published on 3 January 2008

Highly active iridium(I) complexes for the selective hydrogenation of carbon-carbon multiple bonds

scientific article published on 29 September 2011

Highly efficient methods for the one-pot synthesis of beta-substituted enones

scientific article published on 25 November 2005

Hydrogen isotope exchange with highly active iridium(I) NHC/phosphine complexes: a comparative counterion study.

scientific article published on 27 July 2016

In situ generation of Mes2Mg as a non-nucleophilic carbon-centred base reagent for the efficient one-pot conversion of ketones to silyl enol ethers.

scientific article

Influence of precursor solvent extraction on stable isotope signatures of methylamphetamine prepared from over-the-counter medicines using the Moscow and Hypophosphorous routes

scientific article published on 15 December 2012

Investigation of the reaction impurities associated with methylamphetamine synthesized using the Nagai method

scientific article

Iridium(I) N-Heterocyclic Carbene (NHC)/Phosphine Catalysts for Mild and Chemoselective Hydrogenation Processes

scientific article published on 8 February 2016

Iridium(I)-catalyzed regioselective C-H activation and hydrogen-isotope exchange of non-aromatic unsaturated functionality

scientific article published on 05 October 2014

Iridium-Catalysed ortho-Directed Deuterium Labelling of Aromatic Esters—An Experimental and Theoretical Study on Directing Group Chemoselectivity

article

Iridium-Catalyzed Formyl-Selective Deuteration of Aldehydes

scientific article published on 16 May 2017

Iridium-catalysed ortho-H/D and -H/T exchange under basic conditions: C-H activation of unprotected tetrazoles.

scientific article

Modified Shapiro reactions with bismesitylmagnesium as an efficient base reagent

scientific article published on 17 April 2012

On-site determination of formaldehyde: a low cost measurement device for museum environments.

scientific article

Oxygenated Cyclopentenones via the Pauson–Khand Reaction of Silyl Enol Ether Substrates

scientific article published in 2022

PROTAC-Mediated Degradation of Bruton's Tyrosine Kinase Is Inhibited by Covalent Binding

scientific article published on 27 February 2019

Practically convenient and industrially-aligned methods for iridium-catalysed hydrogen isotope exchange processes

scientific article published on 22 April 2014

Preparation of [(3) H]fluoroethyl tosylate and its use in the labelling of the dopamine transporter radioligand [(3) H]FE-PE2I.

scientific article

Profile of a Highly Selective Quaternized Pyrrolidine Betaine αvβ6 Integrin Inhibitor-(3S)-3-(3-(3,5-Dimethyl-1H-pyrazol-1-yl)phenyl)-4-((1S and 1R,3R)-1-methyl-3-(2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl)pyrrolidin-1-ium-1-yl)butanoate Syn

scientific article published on 05 August 2019

Recent advances in iridium(I) catalysis towards directed hydrogen isotope exchange

scientific article published on 12 November 2019

Stereocontrolled access to optically-enriched oxabispidines

scientific article published on 12 April 2012

Structure-Based Design of a Bromodomain and Extraterminal Domain (BET) Inhibitor Selective for the N-Terminal Bromodomains That Retains an Anti-inflammatory and Antiproliferative Phenotype

scientific article published on 03 August 2020

Synthesis of [3 H] and [14 C]genipin

scientific article published on 04 February 2020

The microwave-assisted Dötz benzannulation process

scientific article published on 01 October 2002

Towards energetically viable asymmetric deprotonations: selectivity at more elevated temperatures with C2-symmetric magnesium bisamides

scientific article published on 18 January 2011