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List of works by Zdzisław Chilmonczyk

13C cross-polarization magic angle spinning NMR and gauge-independent atomic orbital, coupled Hartree-Fock calculations of buspirone analogues. Part 2. Hydrochlorides and perchlorates of 1-arylpiperazine-4-alkylimides

scientific article published on 01 June 1999

1H, 13C, 15N NMR analysis of sildenafil base and citrate (Viagra) in solution, solid state and pharmaceutical dosage forms

scientific article published on 2 April 2005

3D QSAR study of hypolipidemic asarones by comparative molecular surface analysis.

scientific article published on 3 November 2005

A linear combination of pharmacophore hypotheses as a new tool in search of new active compounds--an application for 5-HT1A receptor ligands

scientific article (publication date: 2013)

Assessment of the genotoxic activity of alpha-asarone and its derivatives in the comet assay

scientific article published in March 2013

Autophagic cell death and premature senescence: New mechanism of 5-fluorouracil and sulforaphane synergistic anticancer effect in MDA-MB-231 triple negative breast cancer cell line.

scientific article published on 2 November 2017

Buspirone Analogs as Ligands of the 5-HT1A Receptor. 1. The Molecular Structure of Buspirone and Its Two Analogs

scientific article published on 01 May 1995

Conformational flexibility of serotonin1A receptor ligands from crystallographic data. Updated model of the receptor pharmacophore.

scientific article published on May 1997

Corrigendum to 'Autophagic cell death and premature senescence: New mechanism of 5-fluorouracil and sulforaphane synergistic anticancer effect in MDA-MB-231 triple negative breast cancer cell line' Food Chem Toxicol. 111 (2018) 1-8

scientific article published on 04 May 2018

Deoxynucleosides with benzimidazoles as aglycone moiety are potent anticancer agents.

scientific article

Does molecular docking reveal alternative chemopreventive mechanism of activation of oxidoreductase by sulforaphane isothiocyanates?

scientific article published on 22 December 2009

Enantioselective separation of 1,4-disubstituted piperazine derivatives on two cellulose chiralcel OD and OJ and one amylose chiralpak AD chiral selectors

scientific article published on 01 January 1999

Fluoroaryl analogs of sulforaphane - A group of compounds of anticancer and antimicrobial activity

scientific article published on 20 November 2019

From Homology Models to a Set of Predictive Binding Pockets-a 5-HT1A Receptor Case Study

scientific article published on 05 January 2017

Fullerene Derivatives of Nucleoside HIV Reverse Transcriptase Inhibitors-In Silico Activity Prediction

article

Functional Selectivity and Antidepressant Activity of Serotonin 1A Receptor Ligands

scientific article (publication date: 2015)

Genotoxicity of alpha-asarone analogues.

scientific article

Hypolipidaemic and antiplatelet agents

scientific article published in August 2001

Identification of novel serotonin transporter compounds by virtual screening

scientific article published on 26 February 2014

In Vitro Evaluation of Sulforaphane and a Natural Analog as Potent Inducers of 5-Fluorouracil Anticancer Activity

article published in 2018

In the triple-negative breast cancer MDA-MB-231 cell line, sulforaphane enhances the intracellular accumulation and anticancer action of doxorubicin encapsulated in liposomes

scientific article published on 12 January 2019

In-vivo effects of the 1,2,4-piperazine derivatives MM5 and MC1, putative 5-HT agonists, on dopamine and serotonin release in rat prefrontal cortex

scientific article

Interaction of 1,2,4-substituted piperazines, new serotonin receptor ligands, with 5-HT1A and 5-HT2A receptors

scientific article

Intrinsic activity and comparative molecular dynamics of buspirone analogues at the 5-HT(1A) receptors.

scientific article

Ligand-5-HT1A receptor interaction

scientific article published on 01 March 2000

Ligand-directed trafficking of receptor stimulus

scientific article

Mass-spectrometric studies of new 6-nitroquipazines-serotonin transporter inhibitors

scientific article published on October 2011

Models of 5-hydroxytryptamine receptors. A review.

scientific article published on October 1995

Molecular dynamics of 5-HT1A and 5-HT2A serotonin receptors with methylated buspirone analogues.

scientific article published in November 2001

Molecular mechanism of serotonin transporter inhibition elucidated by a new flexible docking protocol

scientific article

Molecular structure of some 3-amino-2-oxazolidinone derivatives.

scientific article

New benzimidazole-derived isothioureas as potential antileukemic agents--studies in vitro

scientific article

New enantiomeric fluorine-containing derivatives of sulforaphane: synthesis, absolute configurations and biological activity.

scientific article published on 14 February 2014

New validated HPLC methodology for the determination of (-)-trans-paroxetine and its enantiomer in pharmaceutical formulations with use of ovomucoid chiral stationary phase

scientific article

Oncotoxic Properties of Serotonin Transporter Inhibitors and 5-HT Receptor Ligands

scientific article published on 20 October 2018

Organofluorine Isoselenocyanate Analogues of Sulforaphane: Synthesis and Anticancer Activity.

scientific article published on 7 October 2016

Pharmacological properties and SAR of new 1,4-disubstituted piperazine derivatives with hypnotic-sedative activity

scientific article

Proapoptotic activity of heterocyclic compounds containing succinimide moiety in the promyelocytic leukemia cell line HL-60.

scientific article published on May 2013

Proapoptotic effects of new pentabromobenzylisothiouronium salts in a human prostate adenocarcinoma cell line.

scientific article

Proapoptotic effects of novel pentabromobenzylisothioureas in human leukemia cell lines

scientific article

Rigid analogues of buspirone and gepirone, 5-HT1A receptors partial agonists

scientific article

Serotonin transporter and receptor ligands with antidepressant activity as neuroprotective and proapoptotic agents

scientific article published on 22 January 2017

Some analogues of 1,4-disubstituted piperazines as hypnotic and sedative agents

scientific article published on 01 February 1995

Structure-retention relationship in a series of chiral 1,4-disubstituted piperazine derivatives on carbohydrate chiral stationary phases.

scientific article published on 14 April 2005

Sulforaphane Regulates NFE2L2/Nrf2-Dependent Xenobiotic Metabolism Phase II and Phase III Enzymes Differently in Human Colorectal Cancer and Untransformed Epithelial Colon Cells.

scientific article published on 16 September 2016

Synergistic anti-leukemic effects of CK2 inhibitors and pentabromobenzylisothioureas in vitro

scientific article published on November 2013

Synthesis and hypolipidemic and antiplatelet activities of alpha-asarone isomers in humans (in vitro), mice (in vivo), and rats (in vivo)

scientific article published on 01 October 2000

Synthesis and proapoptotic properties of new casein kinase II inhibitors

scientific article published on November 1, 2010

Synthesis, antidepressant evaluation and docking studies of long-chain alkylnitroquipazines as serotonin transporter inhibitors

scientific article published on 11 April 2013

Synthesis, in vitro binding studies and docking of long-chain arylpiperazine nitroquipazine analogues, as potential serotonin transporter inhibitors

scientific article

The Comparison of MTT and CVS Assays for the Assessment of Anticancer Agent Interactions

scientific article

The development and validation of a novel virtual screening cascade protocol to identify potential serotonin 5-HT(7)R antagonists

scientific article published on 6 March 2010

The ligand-binding site of buspirone analogues at the 5-HT1A receptor.

scientific article

The molecular interactions of buspirone analogues with the serotonin transporter

scientific article published on 5 September 2008

The new HPLC methodology for the chiral separation of tamsulosin enantiomers on amylose tris(3,5-dimethylphenylcarbamate) stationary phase

scientific article published on 09 June 2012

Up-regulation of glutathione-related genes, enzyme activities and transport proteins in human cervical cancer cells treated with doxorubicin

scientific article published on 14 July 2016

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