List of works - Noriki Kutsumura

A formal total synthesis of (−)-brevisamide ⬇️

scientific article published on April 27, 2011

Antitrichomonal activity of δ opioid receptor antagonists, 7-benzylidenenaltrexone derivatives

scientific article published on 15 June 2017

Design and Synthesis of Non-Peptide, Selective Orexin Receptor 2 Agonists.

scientific article published on 12 August 2015

Design and Synthesis of Potent and Highly Selective Orexin 1 Receptor Antagonists with a Morphinan Skeleton and Their Pharmacologies

scientific article published on 4 January 2017

Dibenzopyrrolo[1,2-a][1,8]naphthyridines: Synthesis and Structural Modification of Fluorescent L-Shaped Heteroarenes.

scientific article published on 12 December 2017

Essential structure of orexin 1 receptor antagonist YNT-707, Part I: Role of the 4,5-epoxy ring for binding with orexin 1 receptor

scientific article published on 4 July 2017

Essential structure of orexin 1 receptor antagonist YNT-707, Part II: Drastic effect of the 14-hydroxy group on the orexin 1 receptor antagonistic activity.

scientific article published on 30 December 2017

Essential structure of orexin 1 receptor antagonist YNT-707, Part IV: The role of D-ring in 4,5-epoxymorphinan on the orexin 1 receptor antagonistic activity

scientific article published on 24 July 2019

Essential structure of orexin 1 receptor antagonist YNT-707, part III: Role of the 14-hydroxy and the 3-methoxy groups in antagonistic activity toward the orexin 1 receptor in YNT-707 derivatives lacking the 4,5-epoxy ring

scientific article published on 05 March 2019

Favorskii-Type Rearrangement of the 4,5-Epoxymorphinan Skeleton.

scientific article published on 7 March 2018

Intramolecular [2+2+2] cycloaddition of bis(propargylphenyl)carbodiimides: synthesis of L-shaped π-extended compounds with pyrrolo[1,2-a][1,8]naphthyridine corner units.

scientific article published in July 2013

Investigation of 7-benzylidenenaltrexone derivatives as a novel structural antitrichomonal lead compound

scientific article published on 10 June 2015

Novel one-pot method for chemoselective bromination and sequential Sonogashira coupling.

scientific article published in August 2010

Palladium-catalyzed highly regio- and stereoselective synthesis of 4-alkylidene-4H-3,1-benzoxazines from N-acyl-o-alkynylanilines

scientific article published on 03 February 2011

Structure-Activity Relationship between Thiol Group-Trapping Ability of Morphinan Compounds with a Michael Acceptor and Anti-Plasmodium falciparum Activities

scientific article published on 02 March 2020

Synthesis of novel triplets with a 1,3,5-trioxazatriquinane skeleton and their pharmacologies for opioid receptors.

scientific article published on 12 May 2015

Total Syntheses of 3- epi-Litsenolide D2 and Lincomolide A

scientific article published on 23 August 2018

Total Synthesis of 3-epi-Juruenolide C

scientific article published on 01 January 2019

Triflic acid-promoted cycloisomerization of 2-alkynylphenyl isothiocyanates and isocyanates: a novel synthetic method for a variety of indole derivatives

scientific article published on 01 November 2014

ZnCl2-Promoted Intramolecular Hetero-Diels-Alder Reaction of o-Alkynylphenylcarbodiimides for Synthesis of Dihydrodibenzo[b,g][1,8]naphthyridines

scientific article

List of works by Noriki Kutsumura