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List of works by Saverio Cellamare

1,3-Dialkyl-8-(hetero)aryl-9-OH-9-deazaxanthines as potent A2B adenosine receptor antagonists: design, synthesis, structure-affinity and structure-selectivity relationships

scientific article

Alpidem analogues containing a GABA or glycine moiety as new anticonvulsant agents

scientific article published in March 2003

Application of a new chiral stationary phase containing the glycopeptide antibiotic A-40,926 in the direct chromatographic resolution of β-amino acids

article by Ilaria D’Acquarica et al published June 2000 in Tetrahedron: Asymmetry

Carbamate prodrug concept for hydroxamate HDAC inhibitors

scientific article

Design, Synthesis, and Biological Evaluation of 2-Aminobenzanilide Derivatives as Potent and Selective HDAC Inhibitors

scientific article published on 24 May 2012

Design, synthesis and biological evaluation of 5-hydroxy, 5-substituted-pyrimidine-2,4,6-triones as potent inhibitors of gelatinases MMP-2 and MMP-9

article by Orazio Nicolotti et al published December 2012 in European Journal of Medicinal Chemistry

Design, synthesis and biological evaluation of coumarin alkylamines as potent and selective dual binding site inhibitors of acetylcholinesterase

scientific article

Design, synthesis and biological evaluation of indane-2-arylhydrazinylmethylene-1,3-diones and indol-2-aryldiazenylmethylene-3-ones as beta-amyloid aggregation inhibitors

scientific article published on 23 December 2009

Design, synthesis, and biological evaluation of coumarin derivatives tethered to an edrophonium-like fragment as highly potent and selective dual binding site acetylcholinesterase inhibitors

scientific article published on September 2010

Design, synthesis, and biological evaluation of glycine-based molecular tongs as inhibitors of Abeta1-40 aggregation in vitro

scientific article published on 25 March 2008

Development and analytical characterization of vitamin(s)-loaded chitosan nanoparticles for potential food packaging applications

Direct chromatographic resolution of carnitine and O-acylcarnitine enantiomers on a teicoplanin-bonded chiral stationary phase

scientific article published on 01 October 1999

Discovery of Potent Dual Binding Site Acetylcholinesterase Inhibitors via Homo- and Heterodimerization of Coumarin-Based Moieties

scientific article published in June 2017

Discovery of new 7-substituted-4-imidazolylmethyl coumarins and 4′-substituted-2-imidazolyl acetophenones open analogues as potent and selective inhibitors of steroid-11β-hydroxylase

scholarly article by Angela Stefanachi et al published January 2015 in European Journal of Medicinal Chemistry

Discovery, biological evaluation, and structure-activity and -selectivity relationships of 6'-substituted (E)-2-(benzofuran-3(2H)-ylidene)-N-methylacetamides, a novel class of potent and selective monoamine oxidase inhibitors.

scientific article published on 13 March 2013

Docking-based classification models for exploratory toxicology studies on high-quality estrogenic experimental data

scientific article

Effect of Thapsia Essential Oils on Bile Composition in Rats

article

Effects of isoquinoline derivatives structurally related to 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine (MPTP) on mitochondrial respiration.

scientific article published in June 1996

Enantiomeric resolution of sulfoxides on a DACH-DNB chiral stationary phase: A quantitative structure-enantioselective retention relationship (QSERR) study

article by Cosimo Altomare et al published 1993 in Chirality

Extended form of a retro-inverso peptide stabilized by beta-sheet unidirectional H-bonds: Crystallographic and NMR evidence

scientific article published in January 2001

Galloyl benzamide-based compounds modulating tumour necrosis factor α-stimulated c-Jun N-terminal kinase and p38 mitogen-activated protein kinase signalling pathways

scientific article published on 16 June 2015

Hydroxy-Propil-β-Cyclodextrin Inclusion Complexes of two Biphenylnicotinamide Derivatives: Formulation and Anti-Proliferative Activity Evaluation in Pancreatic Cancer Cell Models

scientific article published on 07 September 2020

Inhibition of [3H]dopamine uptake into striatal synaptosomes by isoquinoline derivatives structurally related to 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine

scientific article published in July 1996

Inhibition of complex I by isoquinoline derivatives structurally related to 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine(MPTP)

scientific article published on 01 November 1995

Inhibition of monoamine oxidase-B by condensed pyridazines and pyrimidines: effects of lipophilicity and structure-activity relationships

scientific article published in September 1998

Insights into structure-activity relationships from lipophilicity profiles of pyridin-2(1H)-one analogs of the cardiotonic agent milrinone

scientific article published in September 2005

Investigating Structural Requirements for the Antiproliferative Activity of Biphenyl Nicotinamides.

scientific article published on 30 June 2017

Investigation of platelet aggregation inhibitory activity by phenyl amides and esters of piperidinecarboxylic acids

scientific article (publication date: 3 April 2003)

Ionization behaviour and tautomerism-dependent lipophilicity of pyridine-2(1 H )-one cardiotonic agents

scientific article published on 01 May 2000

LFER and CoMFA studies on optical resolution of alpha-alkyl alpha-aryloxy acetic acid methyl esters on DACH-DNB chiral stationary phase.

scientific article published in April 1995

Linear Solvation Energy Relationships in Reversed-Phase Liquid Chromatography. Examination of Deltabond C8as Stationary Phase for Measuring Lipophilicity Parameters

article by Cosimo Altomare et al published 1993 in QSAR and Combinatorial Science

Lipophilicity measurements of benzenesulfonamide inhibitors of carbonic anhydrase by reversed-phase HPLC

scholarly article by C. Altomare et al published December 1989 in International Journal of Pharmaceutics

Lipophilicity of teicoplanin antibiotics as assessed by reversed phase high-performance liquid chromatography: quantitative structure-property and structure-activity relationships.

scientific article published in December 1994

Lipophilicity-related inhibition of blood platelet aggregation by nipecotic acid anilides

scientific article

New organic nitrate-containing benzyloxy isonipecotanilide derivatives with vasodilatory and anti-platelet activity

scientific article published on 10 March 2015

Nigral cell loss produced by infusion of isoquinoline derivatives structurally related to 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine

scientific article published in September 1996

Novel Antiproliferative Biphenyl Nicotinamide: NMR Metabolomic Study of its Effect on the MCF-7 Cell in Comparison with Cisplatin and Vinblastine

scientific article published on 31 July 2020

Pharmacophore Modeling and 3D-QSAR Study of Indole and Isatin Derivatives as Antiamyloidogenic Agents Targeting Alzheimer's Disease

scientific article published on 07 December 2020

Potent galloyl-based selective modulators targeting multidrug resistance associated protein 1 and P-glycoprotein

scientific article

Pyrrolo[3,2- c ]pyridine derivatives as inhibitors of platelet aggregation

scientific article published on 01 March 2000

Solid-phase synthesis and insights into structure-activity relationships of safinamide analogues as potent and selective inhibitors of type B monoamine oxidase

scientific article (publication date: 4 October 2007)

Substituent effects on the enantioselective retention of anti-HIV 5-aryl-delta 2-1,2,4-oxadiazolines on R,R-DACH-DNB chiral stationary phase.

scientific article published in January 1996

Teicoplanin-Based Enantiomeric Separations in CZE Using a Partial Filling Technique

article by Angelo Carotti et al published 1 June 1999 in Journal of Separation Science

Toward a fragment-based approach to MMPs inhibitors: an expedite and efficient synthesis of N-hydroxylactams

Toxicity to PC12 cells of isoquinoline derivatives structurally related to 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine

scientific article published on 01 March 1996

Trimethoxybenzanilide-based P-glycoprotein modulators: an interesting case of lipophilicity tuning by intramolecular hydrogen bonding

scientific article

X-ray crystal structure, partitioning behavior, and molecular modeling study of piracetam-type nootropics: insights into the pharmacophore

scientific article published on January 1995