List of works - Kensuke Okuda

10'-Chloro-3',4'-dihydro-2'H-spiro-[cyclo-propane-1,7'(6'H)-pyrimido[2,1-a]isoquinolin]-6'-one.

scientific article published on 31 October 2012

2-Nitroimidazole-tricarbocyanine conjugate as a near-infrared fluorescent probe for in vivo imaging of tumor hypoxia

scientific article

3-(2-Oxo-2,3,4,5-tetra-hydro-furan-3-yl)-1-benzofuran-2-carbonitrile.

scientific article published on 31 August 2012

7-Chloro-1,2-dihydro-furo[2,3-c]isoquinolin-5-amine.

scientific article published on 30 October 2010

A fluorogenic probe using a catalytic reaction for the detection of trace intracellular zinc

scientific article published on 16 October 2020

A highly sensitive assay of IRE1 activity using the small luciferase NanoLuc: Evaluation of ALS-related genetic and pathological factors.

scientific article published on 06 June 2015

A new class of high-contrast Fe(II) selective fluorescent probes based on spirocyclized scaffolds for visualization of intracellular labile iron delivered by transferrin

scientific article published in September 2014

A universal fluorogenic switch for Fe(ii) ion based on N-oxide chemistry permits the visualization of intracellular redox equilibrium shift towards labile iron in hypoxic tumor cells

scientific article published on 24 April 2017

An uncharged amine in the transition state of the ribosomal peptidyl transfer reaction

scientific article published on May 2008

Bismuth-rhodamine: a new red light-excitable photosensitizer

scientific article published on 6 October 2017

Development of a hypoxia-selective near-infrared fluorescent probe for non-invasive tumor imaging.

scientific article

Effect of hexasulfobutylated C(60) on the isolated aortic ring of guinea pig.

scientific article published in February 2002

Elucidating the rapid action of 2-(2-chlorophenyl)ethylbiguanide on HT-29 cells under a serum- and glucose-deprived condition

scientific article

Elucidation of a novel phenformin derivative on glucose-deprived stress responses in HT-29 cells.

scientific article published on 8 July 2016

FRET-based imaging of transbilayer movement of pepducin in living cells by novel intracellular bioreductively activatable fluorescent probes

scientific article published in May 2013

Facile one-pot synthesis of [1, 2, 3]triazolo[1, 5-a]pyridines from 2-acylpyridines by copper(II)-catalyzed oxidative N-N bond formation.

scientific article published on 25 February 2014

In vivo retinal and choroidal hypoxia imaging using a novel activatable hypoxia-selective near-infrared fluorescent probe

scientific article published on 29 August 2016

Inhibition of E. coli growth by fullerene derivatives and inhibition mechanism

scientific article published on 01 October 1999

Isolation, identification, and biological evaluation of HIF-1-modulating compounds from Brazilian green propolis

scientific article published on 4 August 2011

Kinetic isotope effect analysis of the ribosomal peptidyl transferase reaction

scientific article

Optimization of biguanide derivatives as selective antitumor agents blocking adaptive stress responses in the tumor microenvironment.

scientific article published on 6 June 2014

Polycyclic N-heterocyclic compounds. Part 62: Reaction of N-(quinazolin-4-yl)amidine derivatives with hydroxylamine hydrochloride and anti-platelet aggregation activity of the products.

scientific article published in March 2010

Polycyclic N-heterocyclic compounds. part 59: rearrangement reactions of fused tricyclic 3-(2-bromoethyl)pyrimidin-4(3h)-ones with primary amines via a dimroth-type rearrangement

scientific article published on 01 July 2009

Respiratory chain inhibition by fullerene derivatives: hydrogen peroxide production caused by fullerene derivatives and a respiratory chain system

scientific article published in April 2003

Solution-phase synthesis and biological evaluation of triostin A and its analogues

scientific article published on 18 January 2016

Synthesis and evaluation of cyclic RGD-boron cluster conjugates to develop tumor-selective boron carriers for boron neutron capture therapy.

scientific article published on 18 January 2011

Synthesis of a fluorine-substituted puromycin derivative for Brønsted studies of ribosomal-catalyzed peptide bond formation

scientific article published in March 2009

Synthesis of water-soluble C60-porphyrin hybrid compounds.

scientific article

Uncovering the enzymatic pKa of the ribosomal peptidyl transferase reaction utilizing a fluorinated puromycin derivative

scientific article published in May 2005

List of works by Kensuke Okuda

10'-Chloro-3',4'-dihydro-2'H-spiro-[cyclo-propane-1,7'(6'H)-pyrimido[2,1-a]isoquinolin]-6'-one.

2-Nitroimidazole-tricarbocyanine conjugate as a near-infrared fluorescent probe for in vivo imaging of tumor hypoxia

3-(2-Oxo-2,3,4,5-tetra-hydro-furan-3-yl)-1-benzofuran-2-carbonitrile.

7-Chloro-1,2-dihydro-furo[2,3-c]isoquinolin-5-amine.

A fluorogenic probe using a catalytic reaction for the detection of trace intracellular zinc

A highly sensitive assay of IRE1 activity using the small luciferase NanoLuc: Evaluation of ALS-related genetic and pathological factors.

A new class of high-contrast Fe(II) selective fluorescent probes based on spirocyclized scaffolds for visualization of intracellular labile iron delivered by transferrin

A universal fluorogenic switch for Fe(ii) ion based on N-oxide chemistry permits the visualization of intracellular redox equilibrium shift towards labile iron in hypoxic tumor cells

An uncharged amine in the transition state of the ribosomal peptidyl transfer reaction

Bismuth-rhodamine: a new red light-excitable photosensitizer

Development of a hypoxia-selective near-infrared fluorescent probe for non-invasive tumor imaging.

Effect of hexasulfobutylated C(60) on the isolated aortic ring of guinea pig.

Elucidating the rapid action of 2-(2-chlorophenyl)ethylbiguanide on HT-29 cells under a serum- and glucose-deprived condition

Elucidation of a novel phenformin derivative on glucose-deprived stress responses in HT-29 cells.

FRET-based imaging of transbilayer movement of pepducin in living cells by novel intracellular bioreductively activatable fluorescent probes

Facile one-pot synthesis of [1, 2, 3]triazolo[1, 5-a]pyridines from 2-acylpyridines by copper(II)-catalyzed oxidative N-N bond formation.

In vivo retinal and choroidal hypoxia imaging using a novel activatable hypoxia-selective near-infrared fluorescent probe

Inhibition of E. coli growth by fullerene derivatives and inhibition mechanism

Isolation, identification, and biological evaluation of HIF-1-modulating compounds from Brazilian green propolis

Kinetic isotope effect analysis of the ribosomal peptidyl transferase reaction

Optimization of biguanide derivatives as selective antitumor agents blocking adaptive stress responses in the tumor microenvironment.

Polycyclic N-heterocyclic compounds. Part 62: Reaction of N-(quinazolin-4-yl)amidine derivatives with hydroxylamine hydrochloride and anti-platelet aggregation activity of the products.

Polycyclic N-heterocyclic compounds. part 59: rearrangement reactions of fused tricyclic 3-(2-bromoethyl)pyrimidin-4(3h)-ones with primary amines via a dimroth-type rearrangement

Respiratory chain inhibition by fullerene derivatives: hydrogen peroxide production caused by fullerene derivatives and a respiratory chain system

Solution-phase synthesis and biological evaluation of triostin A and its analogues

Synthesis and evaluation of cyclic RGD-boron cluster conjugates to develop tumor-selective boron carriers for boron neutron capture therapy.

Synthesis of a fluorine-substituted puromycin derivative for Brønsted studies of ribosomal-catalyzed peptide bond formation

Synthesis of water-soluble C60-porphyrin hybrid compounds.

Uncovering the enzymatic pKa of the ribosomal peptidyl transferase reaction utilizing a fluorinated puromycin derivative