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List of works by Jerome Wielens

A three-dimensional model of the human immunodeficiency virus type 1 integration complex

scientific article

Characterization of two distinct modes of drug binding to human intestinal fatty acid binding protein

scientific article

Corrigendum: Fragment-Based Design of Ligands Targeting a Novel Site on the Integrase Enzyme of Human Immunodeficiency Virus 1

scholarly article published in ChemMedChem

Crystal structure of the HIV-1 integrase core domain in complex with sucrose reveals details of an allosteric inhibitory binding site

scientific article

Cyclic Hexapeptide Mimics of the LEDGF Integrase Recognition Loop in Complex with HIV-1 Integrase

article

Diuretic drug binding to human glutathione transferase P1-1: potential role of Cys-101 revealed in the double mutant C47S/Y108V

scientific article

Fragment-based design of ligands targeting a novel site on the integrase enzyme of human immunodeficiency virus 1

scientific article

Oncogenic protein interfaces: small molecules, big challenges.

scientific article published on 13 March 2014

Parallel screening of low molecular weight fragment libraries: do differences in methodology affect hit identification?

scientific article

Phosphorylation of syndapin I F-BAR domain at two helix-capping motifs regulates membrane tubulation

scientific journal article

Potent hepatitis C inhibitors bind directly to NS5A and reduce its affinity for RNA.

scientific article

Preparation, crystallization and preliminary X-ray diffraction analysis of two intestinal fatty-acid binding proteins in the presence of 11-(dansylamino)undecanoic acid

scientific article

Probing the fibrate binding specificity of rat liver fatty acid binding protein.

scientific article published in September 2009

Propargyloxyproline Regio- and Stereoisomers for Click-Conjugation of Peptides: Synthesis and Application in Linear and Cyclic Peptides

article

Structural and biochemical characterization of the oxidoreductase NmDsbA3 from Neisseria meningitidis

scientific article

The Binding of Syndapin SH3 Domain to Dynamin Proline-rich Domain Involves Short and Long Distance Elements

scientific article published on 18 February 2016

The Structure of the Bacterial Oxidoreductase Enzyme DsbA in Complex with a Peptide Reveals a Basis for Substrate Specificity in the Catalytic Cycle of DsbA Enzymes

scientific article

The interaction of lipophilic drugs with intestinal fatty acid-binding protein.

scientific article