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List of works by Etsuo Yonemochi

A new solvate of epalerstat, a drug for diabetic neuropathy.

scientific article

Applicability of DPI formulations for novel neurokinin receptor antagonist

scientific article

Application and mechanism of inhalation profile improvement of DPI formulations by mechanofusion with magnesium stearate

scientific article published in May 2008

Application of Eudragit RS to thermo-sensitive drug delivery systems: II. Effect of temperature on drug permeability through membrane consisting of Eudragit RS/PEG 400 blend polymers

scientific article published in January 2005

Application of eudragit RS to thermo-sensitive drug delivery systems. I. Thermo-sensitive drug release from acetaminophen matrix tablets consisting of eudragit RS/PEG 400 blend polymers

scientific article published in March 2002

Applying terahertz technology for nondestructive detection of crack initiation in a film-coated layer on a swelling tablet

scientific article published on 13 April 2012

Changes in surface properties by granulation and physicochemical stability of granulated amorphous cefditoren pivoxil with additives

scientific article

Characterization and Quality Control of Pharmaceutical Cocrystals

scientific article published on 18 June 2016

Characterization of complexes between phenethylamine enantiomers and β-cyclodextrin derivatives by capillary electrophoresis-Determination of binding constants and complex mobilities.

scientific article published on 28 January 2017

Characterization of polymorphs of a novel quinolinone derivative, TA-270 (4-hydroxy-1-methyl-3-octyloxy-7-sinapinoylamino-2(1H)-quinolinone)

scientific article published on 01 October 2001

Clarifying the mechanism of aggregation of particles in high-shear granulation based on their surface properties by using micro-spectroscopy.

scientific article published on 22 December 2013

Cocrystallization and amorphization induced by drug-excipient interaction improves the physical properties of acyclovir.

scientific article published on 3 November 2011

Comparison of molecular mobility in the glassy state between amorphous indomethacin and salicin based on spin-lattice relaxation times

scientific article published on 17 May 2005

Competition of thermodynamic and dynamic factors during formation of multicomponent particles via spray drying

scientific article

Component crystallization and physical collapse during freeze-drying of L-arginine-citric acid mixtures

scientific article published on 01 January 2012

Correlation between glass-forming ability and fragility of pharmaceutical compounds.

scientific article

Crystal Structure Determination of Dimenhydrinate after More than 60 Years: Solving Salt–Cocrystal Ambiguity via Solid-State Characterizations and Solubility Study

Determination for dry layer resistance of sucrose under various primary drying conditions using a novel simulation program for designing pharmaceutical lyophilization cycle

scientific article published on 15 May 2013

Development of a method for the determination of caffeine anhydrate in various designed intact tablets [correction of tables] by near-infrared spectroscopy: a comparison between reflectance and transmittance technique

scientific article published on 10 April 2008

Development of a rapid process monitoring method for dry-coated tableting process by using near-infrared spectroscopy.

scientific article

Development of fast disintegrating compressed tablets using amino acid as disintegration accelerator: evaluation of wetting and disintegration of tablet on the basis of surface free energy

scientific article published in December 2005

Development of microparticles coated with poly-γ-glutamic acid to improve oral absorption of a poorly water-soluble drug

scientific article published on 18 June 2019

Differences in crystallization behavior between quenched and ground amorphous ursodeoxycholic acid

scientific article published on 01 June 1999

Do amorphous troglitazones prepared from two diastereomer-pairs have the same molecular mobility and crystallization rate at the surface?

scientific article published on 01 January 2011

Effect of Polymers and Storage Relative Humidity on Amorphous Rebamipide and Its Solid Dispersion Transformation: Multiple Spectra Chemometrics of Powder X-Ray Diffraction and Near-Infrared Spectroscopy

scientific article published on 10 July 2020

Effect of physical properties of troglitazone crystal on the molecular interaction with PVP during heating

scientific article published on 26 November 2006

Effect of sulfobutyl ether-β-cyclodextrin and propylene glycol alginate on the solubility of clozapine

scientific article published on 11 September 2018

Effect of the type of lubricant on the characteristics of orally disintegrating tablets manufactured using the phase transition of sugar alcohol

scientific article published on 23 February 2008

Effect of water-soluble carriers on dissolution characteristics of nifedipine solid dispersions

Effects of formulation and process factors on the crystal structure of freeze-dried Myo-inositol

scientific article published on 10 June 2014

Effects of solute miscibility on the micro- and macroscopic structural integrity of freeze-dried solids

scientific article published on 01 November 2010

Effects of sugar ester and hydroxypropyl methylcellulose on the physicochemical stability of amorphous cefditoren pivoxil in aqueous suspension

scientific article published on 8 January 2005

Effects of water content in physical mixture and heating temperature on crystallinity of troglitazone-PVP K30 solid dispersions prepared by closed melting method

scientific article published in September 2005

Enhanced dissolution and skin permeation profiles of epalrestat with β-cyclodextrin derivatives using a cogrinding method

scientific article published on 22 May 2017

Epalrestat tetra-hydro-furan monosolvate: crystal structure and phase transition

scientific article published on 2 June 2017

Estimation of initial dissolution rate of drug substance by thermal analysis: application for carbamazepine hydrate

scientific article published in January 2002

Evaluation of amorphous ursodeoxycholic acid by thermal methods

scientific article published on 01 June 1997

Evaluation of antitumor effect of zoledronic acid entrapped in folate-linked liposome for targeting to tumor-associated macrophages

scientific article published on 9 September 2014

Evaluation of rapidly disintegrating tablets containing glycine and carboxymethylcellulose

scientific article published on 23 January 2006

Evaluation of solid dispersions on a molecular level by the Raman mapping technique

scientific article published on 16 May 2008

Evaluation of the crystalline and amorphous states of drug products by nanothermal analysis and Raman imaging

scientific article published on 23 November 2012

Evaluation of the physical properties of dry surface-modified ibuprofen using a powder rheometer (FT4) and analysis of the influence of pharmaceutical additives on improvement of the powder flowability

scientific article published on 18 February 2020

Factors affecting the apparent solubility of ursodeoxycholic acid in the grinding process

scientific article published in April 2003

Fluorometric Studies of Pyrene Adsorption on Porous Crystalline Cellulose

scientific article published on 01 September 1998

Fluorometric study of the molecular states of 2,5-diphenyloxazole in ground mixtures with gamma-cyclodextrin

scientific article published on 01 February 1994

Formulation design of a novel fast-disintegrating tablet

scientific article published on 27 October 2005

Freeze-drying of proteins in glass solids formed by basic amino acids and dicarboxylic acids

scientific article published in January 2009

Freeze-drying of proteins with glass-forming oligosaccharide-derived sugar alcohols

scientific article published on 25 January 2010

Glass-state amorphous salt solids formed by freeze-drying of amines and hydroxy carboxylic acids: effect of hydrogen-bonding and electrostatic interactions

scientific article published in June 2008

Importance of excipient wettability on tablet characteristics prepared by moisture activated dry granulation (MADG).

scientific article

In vivo siRNA delivery system for targeting to the liver by poly-l-glutamic acid-coated lipoplex

scientific article

Interaction of microcrystalline cellulose and water in granules prepared by a high-shear mixer

scientific article published on 01 April 2001

Investigation of the dynamic process during spray-drying to improve aerodynamic performance of inhalation particles.

scientific article published on 17 February 2010

Low-density microparticles with petaloid surface structure for pulmonary drug delivery

scientific article published on 12 February 2014

Mechanisms for Improved Hygroscopicity of L-Arginine Valproate Revealed by X-Ray Single Crystal Structure Analysis

scientific article published on 13 December 2016

Microscopic molecular mobility of amorphous AG-041R measured by solid-state 13C NMR.

scientific article published in May 2004

Molecular Dynamics of Amorphous Sulfamethazine With Structurally Related Sulfonamide Impurities Evaluated Using Thermal Analysis

scientific article published on 19 December 2016

Molecular properties of propranolol hydrochloride prepared as drug-resin complexes

scientific article published in April 2001

Molecular states of p-dimethylaminobenzonitrile coground with β-cyclodextrin investigated using solid-state fluorescence spectroscopy

scientific article published on 01 January 2011

Near IR spectroscopy to quantify the silica content and difference between silicified microcrystalline cellulose and physical mixtures of microcrystalline cellulose and silica

scientific article published on 01 March 2000

New approach to optimizing risk management of the sticking problem using scale-independent critical material attributes and the quantitative process parameter

scientific article published on 15 January 2020

Novel approach to DPI carrier lactose with mechanofusion process with additives and evaluation by IGC.

scientific article published in November 2006

Novel approach to evaluating granulation and segregation level considering the contribution of hydroxypropyl cellulose to the surface property change of granules

scientific article published on 24 March 2020

Novel, lean and environment-friendly granulation method: Green fluidized bed granulation (GFBG)

scientific article published on 17 December 2018

Optimization of primary drying condition for pharmaceutical lyophilization using a novel simulation program with a predictive model for dry layer resistance

scientific article published on 01 January 2014

Physicochemical Properties of Ursodeoxycholic Acid Dispersed in Controlled Pore Glass

scientific article published on 01 August 1999

Physicochemical and crystal structure analysis of pranlukast pseudo-polymorphs I: anhydrates and hydrate.

scientific article published on 13 December 2014

Physicochemical and crystal structure analysis of pranlukast pseudo-polymorphs II: Solvate and cocrystal

scientific article published on 17 March 2015

Physicochemical properties of amorphous clarithromycin obtained by grinding and spray drying

scientific article published on 01 March 1999

Potential of synchrotron X-ray powder diffractometry for detection and quantification of small amounts of crystalline drug substances in pharmaceutical tablets

scientific article published on 06 June 2011

Practical approach for measuring heat capacity of pharmaceutical crystals/glasses by modulated-temperature differential scanning calorimetry

scientific article published on 01 January 2013

Quantitative correlation between initial dissolution rate and heat of fusion of drug substance

scientific article published on 01 August 2000

Quantitative correlation between initial dissolution rate and heat of solution of drug.

scientific article published in August 2000

Quantitative determination of amorphous nicardipine hydrochloride in long acting formula (NIC-LA) using light anhydrous silicic acid

scientific article published in December 2004

Quantitative relationship between solubility, initial dissolution rate and heat of solution of chiral drugs.

scientific article published in January 2000

Reevaluation of solubility of tolbutamide and polymorphic transformation from Form I to unknown crystal form.

scientific article published on 5 November 2008

Relationship between crystallization tendencies during cooling from melt and isothermal storage: toward a general understanding of physical stability of pharmaceutical glasses

scientific article published on 25 April 2014

Sequential intravenous injection of anionic polymer and cationic lipoplex of siRNA could effectively deliver siRNA to the liver

scientific article published in December 2014

Solid states fluorescence study of p-dimethylaminobenzonitrile by co-grinding with cyclodextrins

scientific article published in February 2009

Solid-state 13C NMR study of indomethacin polymorphism

scientific article published on 01 April 2006

Solid-state fluorescence study of naphthalene adsorption on porous material.

scientific article

Solubility Improvement of Benexate through Salt Formation Using Artificial Sweetener.

scientific article

Stabilization of protein structure in freeze-dried amorphous organic acid buffer salts.

scientific article

Study of the pseudo-crystalline transformation from form i to form II of thiamine hydrochloride (vitamin B(1))

scientific article published on 01 January 2011

Studying the morphology of lyophilized protein solids using X-ray micro-CT: effect of post-freeze annealing and controlled nucleation

scientific article

Swelling kinetics of spray-dried chitosan acetate assessed by magnetic resonance imaging and their relation to drug release kinetics of chitosan matrix tablets

scientific article published on 30 November 2010

Synthesis and Characterization of Cholesteryl Conjugated Lysozyme (CHLysozyme)

scientific article published on 14 August 2020

The effect of structurally related impurities on crystallinity reduction of sulfamethazine by grinding.

scientific article

The importance of binder moisture content in Metformin HCL high-dose formulations prepared by moist aqueous granulation (MAG).

scientific article published on 3 October 2015

Therapeutic effect for liver-metastasized tumor by sequential intravenous injection of anionic polymer and cationic lipoplex of siRNA.

scientific article

Triboelectrification of active pharmaceutical ingredients: week acids and their salts

scientific article published on 04 August 2015

Tumor delivery of liposomal doxorubicin prepared with poly-L-glutamic acid as a drug-trapping agent.

scientific article published on 16 March 2016

Uniformity and physical states of troglitazone in solid dispersions determined by electron probe microanalysis and microthermal analysis

scientific article

Water sorption and near IR spectroscopy to study the differences between microcrystalline cellulose and silicified microcrystalline cellulose before and after wet granulation

scientific article published on 01 April 1999

Zoledronic acid enhances antitumor efficacy of liposomal doxorubicin

scientific article published on 7 May 2015

siRNA delivery to lung-metastasized tumor by systemic injection with cationic liposomes

scientific article published on 4 September 2015

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