Search filters

List of works by Anthony P Davenport

(18)F-Endothelin-1, a positron emission tomography (PET) radioligand for the endothelin receptor system: radiosynthesis and in vivo imaging using microPET

article

18F-Fluoride and 18F-Fluorodeoxyglucose Positron Emission Tomography After Transient Ischemic Attack or Minor Ischemic Stroke: Case-Control Study

scientific article

A sensitive radioimmunoassay measuring endothelin-like immunoreactivity in human plasma: comparison of levels in patients with essential hypertension and normotensive control subjects

article by Anthony P Davenport et al published March 1990 in Clinical Science

Advances in therapeutic peptides targeting G protein-coupled receptors

scientific article published on 19 March 2020

Alternative pathway to endothelin-converting enzyme for the synthesis of endothelin in human blood vessels

scientific article

Alternatively spliced mRNAs for human endothelin-2 and their tissue distribution

scientific article

Analysis of endogenous human endothelin peptides by high-performance liquid chromatography and mass spectrometry

scientific article published on 01 January 1995

Analysis of endothelins by enzyme-linked immunosorbent assay and radioimmunoassay

scientific article published on 01 January 2002

Anatomical localization and pharmacological activity of mature endothelins and their precursors in human vascular tissue

scholarly article by P G Howard et al published November 1992 in Journal of Hypertension

Apelin, Elabela/Toddler, and biased agonists as novel therapeutic agents in the cardiovascular system

scientific article published in September 2015

Apoptosis of vascular smooth muscle cells induces features of plaque vulnerability in atherosclerosis.

scientific article

Arteriojugular endothelin-1 gradients in aneurysmal subarachnoid haemorrhage

scientific article published in August 2002

Automated synthesis of the generic peptide labelling agent N-succinimidyl 4-[(18)F]fluorobenzoate and application to (18)F-label the vasoactive transmitter urotensin-II as a ligand for positron emission tomography

scientific article

Autoradiographic study of endothelin receptors in human cerebral arteries

scientific article published on 01 January 1995

Autoradiographical localization of binding sites for porcine [125I]endothelin-1 in humans, pigs, and rats: functional relevance in humans

scientific article published on 01 January 1989

Binding sites for 125I ET-1, ET-2, ET-3 and vasoactive intestinal contractor are present in adult rat brain and neurone-enriched primary cultures of embryonic brain cells

scientific article published in July 1991

Binding sites for 125I-labelled endothelin-1 in the kidneys: differential distribution in rat, pig and man demonstrated by using quantitative autoradiography

article published in 1989

Binding sites for iodinated endothelin-1, endothelin-2 and endothelin-3 demonstrated on human uterine glandular epithelial cells by quantitative high-resolution autoradiography

scientific article

Biogenic amines in the brain of the honeybee, Apis mellifera

scientific article published in January 1983

CRF2 receptors are highly expressed in the human cardiovascular system and their cognate ligands urocortins 2 and 3 are potent vasodilators

scientific article

Cardiac action of the first G protein biased small molecule apelin agonist

scientific article published on 27 July 2016

Cellular Expression of Isoforms of Endothelin-Converting Enzyme-1 (ECE-1c, ECE-1b and ECE-1a) and Endothelin-Converting Enzyme-2

scientific article published on 01 November 2000

Cellular distribution of immunoreactive urotensin-II in human tissues with evidence of increased expression in atherosclerosis and a greater constrictor response of small compared to large coronary arteries

article

Cellular localization of receptors using antibodies visualized by light and dual labeling confocal microscopy

scientific article

Cerebellar neurons and glia respond differentially to endothelins and sarafotoxin S6b.

scientific article published in May 1992

Changes in ETA-, AT1- and AT2-Receptors in the Phenotypically Transformed Intimal Smooth Muscle Layer of Human Atherosclerotic Coronary Arteries

scientific article published on 01 November 2000

Changes in biomechanical properties of the coronary artery wall contribute to maintained contractile responses to endothelin-1 in atherosclerosis

scientific article published on 8 April 2014

Changes in haemolymph octopamine levels associated with food deprivation in the locust, Schistocerca gregaria

Characterization and localization of endothelin receptor subtypes in the human atrioventricular conducting system and myocardium

scientific article published on March 1, 1993

Characterization of Site-Directed Antisera Against Endothelin-Converting Enzymes

article

Characterization of [125I]-PD164333, an ETA selective non-peptide radiolabelled antagonist, in normal and diseased human tissues

scientific article

Characterization of [¹²⁵I]GLP-1(9-36), a novel radiolabeled analog of the major metabolite of glucagon-like peptide 1 to a receptor distinct from GLP1-R and function of the peptide in murine aorta

scientific article published on 15 March 2014

Characterization of endothelin isoforms in human heart: endothelin-2 demonstrated

scientific article published on 01 January 1993

Characterization of endothelin receptors in human brain cortex, gliomas, and meningiomas

article

Characterization of endothelin receptors in the human pulmonary vasculature using bosentan, SB209670, and 97-139

scientific article published on 01 January 1995

Characterization of peptide and nonpeptide antagonists in human kidney

scientific article published on 01 January 1995

Characterization of the binding of endothelin ETB selective ligands in human and rat heart

scientific article

Characterization of the endothelin receptor selective agonist, BQ3020 and antagonists BQ123, FR139317, BQ788, 50235, Ro462005 and bosentan in the heart.

scientific article published on February 1996

Characterization of the snake venom ligand [125I]-DNP binding to natriuretic peptide receptor-A in human artery and potent DNP mediated vasodilatation.

scientific article published on 16 October 2006

Characterization of two new ETB selective radioligands, [125I]-BQ3020 and [125I]-[Ala1,3,11,15]ET-1 in human heart

scientific article published on November 1, 1992

Chemerin Elicits Potent Constrictor Actions via Chemokine-Like Receptor 1 (CMKLR1), not G-Protein-Coupled Receptor 1 (GPR1), in Human and Rat Vasculature

scientific article

Chemokine receptor CCR5: from AIDS to atherosclerosis

scientific article

Chronic Apoptosis of Vascular Smooth Muscle Cells Accelerates Atherosclerosis and Promotes Calcification and Medial Degeneration

scientific article published on 22 May 2008

Class A Orphans (version 2019.5) in the IUPHAR/BPS Guide to Pharmacology Database

Class A Orphans (version 2020.5) in the IUPHAR/BPS Guide to Pharmacology Database

Class A Orphans in GtoPdb v.2021.3

Comparative quantification of endothelin receptor mRNA in human kidney: new tools for direct investigation of human tissue

article

Comparison between brain paste and polymer [125I]standards for quantitative receptor autoradiography

scientific article published on 01 August 1988

Comparison of Endothelin-A and Endothelin-B Receptor Distribution Visualized by Radioligand Binding versus Immunocytochemical Localization using Subtype Selective Antisera

scientific article published on 01 November 2004

Comparison of endothelin receptors in normal versus cirrhotic human liver and in the liver from endothelial cell-specific ETB knockout mice

scientific article published on 18 February 2012

Comparison of human ETA and ETB receptor signalling via G-protein and β-arrestin pathways

scientific article published on 27 March 2012

Comparison of the effects of atherosclerosis and nitrate therapy on responses to nitric oxide and endothelin-1 in human arteries in vitro

scientific article published in August 2002

Comparison of vasodilators in human internal mammary artery: ghrelin is a potent physiological antagonist of endothelin-1.

scientific article

Davenport and Maguire reply

Defining the affinity and receptor sub-type selectivity of four classes of endothelin antagonists in clinically relevant human cardiovascular tissues

scientific article published on 23 May 2012

Deletion of Endothelial Cell Endothelin B Receptors Does Not Affect Blood Pressure or Sensitivity to Salt

Delineation of endothelin receptors in human left ventricular smooth-muscle cells

scientific article published on 01 January 1995

Depressor and regionally-selective vasodilator effects of human and rat urotensin II in conscious rats

scientific article published in April 2001

Design, characterization, and first-in-human study of the vascular actions of a novel biased apelin receptor agonist

scientific article

Detection of Atherosclerotic Inflammation by 68Ga-DOTATATE PET Compared to [18F]FDG PET Imaging

scientific article published on April 2017

Detection of Endothelin Receptors in Human Coronary Artery Vascular Smooth Muscle Cells But Not Endothelial Cells by Using Electron Microscope Autoradiography

scientific article published on June 1, 1997

Development and validation of an LC-MS/MS method for detection and quantification of in vivo derived metabolites of [Pyr1]apelin-13 in humans

scientific article published on 27 December 2019

Differential distribution of endothelin peptides and receptors in human adrenal gland

scientific article published on 01 November 1996

Differential distribution of endothelin receptor subtypes in placentae from normal and growth-restricted pregnancies

scientific article published on 01 March 1997

Discovery of a competitive apelin receptor (APJ) antagonist.

scientific article published on 10 May 2011

Discovery of recently adopted orphan receptors for apelin, urotensin II, and ghrelin identified using novel radioligands and functional role in the human cardiovascular system.

scientific article

Distribution of endothelin receptors in atherosclerotic human coronary arteries

scientific article published on 01 January 1995

Down-regulation of ETA receptors in ETB receptor-deficient mice

scientific article published in November 2004

Dynamic In Vivo Imaging of Receptors in Small Animals Using Positron Emission Tomography

scientific article published on 01 January 2012

Dynamic in vivo imaging of receptors in small animals using positron emission tomography

scientific article published in January 2005

ETA and ETB endothelin receptors in human myometrium characterized by the subtype selective ligands BQ123, BQ3020, FR139317 and PD151242.

scientific article published on January 1995

ETA receptor antagonists inhibit intimal smooth muscle cell proliferation in human vessels

scientific article published in August 2002

ETA receptors predominate in the human vasculature and mediate constriction

scientific article published on 01 January 1995

ETA receptor‐mediated constrictor responses to endothelin peptides in human blood vessels in vitro

scientific article published on May 1, 1995

Effect of in vivo fetal infusion of dexamethasone at 0.75 GA on fetal ovine resistance artery responses to ET-1.

scientific article published in July 2001

Effect of the formamidine insecticide chordimeform on feeding and reproduction in the noctuid moth, Spodoptera littoralis (Boisduval)

scholarly article by Anthony P Davenport & Denis J. Wright published February 1987 in Crop Protection

Effects of an ET1-receptor antagonist, FR139317, on regional haemodynamic responses to endothelin-1 and [Ala11,15]Ac-endothelin-1 (6-21) in conscious rats.

scientific article published on June 1994

Elabela/Toddler Is an Endogenous Agonist of the Apelin APJ Receptor in the Adult Cardiovascular System, and Exogenous Administration of the Peptide Compensates for the Downregulation of Its Expression in Pulmonary Arterial Hypertension

scientific article published on 30 January 2017

Elevated systemic levels of endothelin-1 and blood pressure correlate with blunted constrictor responses and downregulation of endothelin(A), but not endothelin(B), receptors in an animal model of hypertension.

scientific article published in August 2002

Emerging pharmacology and physiology of neuromedin U and the structurally related peptide neuromedin S

scientific article

Emerging roles for orphan G-protein-coupled receptors in the cardiovascular system

scientific article

Emerging roles of apelin in biology and medicine

scientific article

Endothelial cell-specific ETB receptor knockout: autoradiographic and histological characterisation and crucial role in the clearance of endothelin-1.

scientific article

Endothelin

scientific article

Endothelin

scholarly article

Endothelin ETA receptors predominate in chronic thromboembolic pulmonary hypertension

scientific article published on 10 February 2016

Endothelin Peptide and Converting Enzymes in Human Endothelium

scientific article published on 01 January 1998

Endothelin Peptide and Receptors in Human Atherosclerotic Coronary Artery and Aorta

scientific article published on 01 October 1996

Endothelin and the human kidney: a potential target for new drugs

scientific article published on 01 January 1994

Endothelin receptor antagonism in patients with chronic heart failure

scientific article published on 01 July 2000

Endothelin receptor pharmacology and function in the mouse: comparison with rat and man.

scientific article published in November 2004

Endothelin receptor subtypes and their functional relevance in human small coronary arteries

scientific article

Endothelin receptors and their antagonists

scientific article

Endothelin-1 mRNA is widely expressed in porcine and human tissues

scientific article published on May 1, 1990

Endothelin-1 stimulates prostaglandin F2 alpha release from human endometrium

scientific article published in March 1991

Endothelin-2, the forgotten isoform: emerging role in the cardiovascular system, ovarian development, immunology and cancer.

scientific article published on January 2013

Endothelin-A-Receptors in Human Aorta and Pulmonary Arteries are Downregulated in Patients With Cardiovascular Disease

scientific article published on 01 November 2000

Endothelin-converting enzyme in the human vasculature: evidence for differential conversion of big endothelin-3 by endothelial and smooth-muscle cells.

scientific article published on January 1998

Endothelin-like immunoreactivity in human endometrium

scientific article published on 01 July 1992

Endothelin-mediated vasoconstriction in early atherosclerosis is markedly increased in ApoE-/- mouse but prevented by atorvastatin

scientific article published on 01 June 2006

Endothelin: progress in pharmacology and physiology

article

Endothelin@25 - new agonists, antagonists, inhibitors and emerging research frontiers: IUPHAR Review 12

scientific article (publication date: December 2014)

Epidermal growth factor in human endometrium: proliferative effects in culture and immunocytochemical localization in normal and endometriotic tissues

scientific article

Evidence for a novel vasospastic transmitter system, neuromedin U, in the equine digital circulation

scientific article

Evidence using immunoelectron microscopy for regulated and constitutive pathways in the transport and release of endothelin.

scientific article

Evolving pharmacology of orphan GPCRs: IUPHAR Commentary

scientific article published on October 2013

Experimental hemiparkinsonism in the rat following chronic unilateral infusion of MPP+ into the nigrostriatal dopamine pathway—II. Differential localization of dopamine and cholecystokinin receptors

scientific article published on 01 October 1988

Expression and Characterization of the Human Endothelin-A-Receptor in Pichia pastoris

scientific article published on 01 November 2000

Expression and vasoconstrictor function of anorexigenic peptides neuromedin U-25 and S in the human cardiovascular system

scientific article

Expression of endothelin(A) receptors in human gliomas and meningiomas, with high affinity for the selective antagonist PD156707.

scientific article published in October 1998

FDG-PET can distinguish inflamed from non-inflamed plaque in an animal model of atherosclerosis.

scientific article published on 22 September 2009

Failure of BQ123, a more potent antagonist of sarafotoxin 6b than of endothelin-1, to distinguish between these agonists in binding experiments

scientific article published in May 1996

Functional and immunocytochemical evidence for a role of ghrelin and des-octanoyl ghrelin in the regulation of vascular tone in man.

scientific article

G-protein-coupled receptors in human atherosclerosis: comparison of vasoconstrictors (endothelin and thromboxane) with recently de-orphanized (urotensin-II, apelin and ghrelin) receptors.

scientific article published in August 2002

GuideToPharmacology.org--an update

scientific article

Haemodynamic and renal effects of endothelin receptor antagonism in patients with chronic kidney disease

article

Human embryonic stem cell-derived cardiomyocyte platform screens inhibitors of SARS-CoV-2 infection

scientific article published on 29 July 2021

Human endothelin receptors characterized using reverse transcriptase-polymerase chain reaction, in situ hybridization, and subtype-selective ligands BQ123 and BQ3020: evidence for expression of ETB receptors in human vascular smooth muscle.

scientific article

Human kidney: endothelin isoforms detected by HPLC with radioimmunoassay and receptor subtypes detected using ligands BQ123 and BQ3020

scientific article published on 01 January 1993

IUPHAR-DB: the IUPHAR database of G protein-coupled receptors and ion channels

scientific article

IUPHAR-DB: updated database content and new features

scientific article

Identification and cellular localisation of NPW1 (GPR7) receptors for the novel neuropeptide W-23 by [125I]-NPW radioligand binding and immunocytochemistry

scientific article

Identification of endothelin-1, endothelin-2 and endothelin-3 in human endometrium

scientific article published on 01 May 1993

Identifying active vascular microcalcification by (18)F-sodium fluoride positron emission tomography.

scientific article

Imaging and characterization of radioligands for positron emission tomography using quantitative phosphor imaging autoradiography

scientific article published in January 2005

Imaging atherosclerotic plaque inflammation with [18F]-fluorodeoxyglucose positron emission tomography.

scientific article

Imaging endothelin ET(B) receptors using [18F]-BQ3020: in vitro characterization and positron emission tomography (microPET).

scientific article published in June 2006

Immunocytochemical Localization of Receptors Using Light and Confocal Microscopy With Application to the Phenotypic Characterization of Knock-Out Mice

scientific article published on 01 January 2005

Immunocytochemical localisation of the apelin receptor, APJ, to human cardiomyocytes, vascular smooth muscle and endothelial cells

scientific article

Immunocytochemical localization of the endogenous vasoactive peptide apelin to human vascular and endocardial endothelial cells

scientific article published in May 2004

Immunocytochemical localization of the urotensin-II receptor, UT, to rat and human tissues: Relevance to function

scientific article published on 26 August 2007

In Vivo Mapping of Vascular Inflammation Using the Translocator Protein Tracer 18F-FEDAA1106.

scientific article

In vitro enzymatic processing of radiolabelled big ET-1 in human kidney

scientific article published on 01 March 1998

In vivo imaging of cardiovascular endothelin receptors using the novel radiolabelled antagonist [18F]-SB209670 and positron emission tomography (microPET).

scientific article published in November 2004

Increased response to big endothelin-1 in atherosclerotic human coronary artery: functional evidence for up-regulation of endothelin-converting enzyme activity in disease.

scientific article

Inotropic action of the puberty hormone kisspeptin in rat, mouse and human: cardiovascular distribution and characteristics of the kisspeptin receptor

scientific article

International Union of Basic and Clinical Pharmacology CIII: Chemerin Receptors CMKLR1 (Chemerin1) and GPR1 (Chemerin2) Nomenclature, Pharmacology, and Function

scientific article published on 26 December 2017

International Union of Basic and Clinical Pharmacology. LXXIV. Apelin receptor nomenclature, distribution, pharmacology, and function

scientific article published on 06 July 2010

International Union of Basic and Clinical Pharmacology. LXXVII. Kisspeptin receptor nomenclature, distribution, and function

scientific article

International Union of Basic and Clinical Pharmacology. LXXXVIII. G protein-coupled receptor list: recommendations for new pairings with cognate ligands

scientific article

International Union of Pharmacology. LVI. Ghrelin receptor nomenclature, distribution, and function

scientific article

International Union of Pharmacology. LXXII. Recommendations for trace amine receptor nomenclature

scientific article

International Union of Pharmacology. XLVI. G protein-coupled receptor list.

scientific article

International Union of Pharmacology. XXIX. Update on endothelin receptor nomenclature

scientific article (publication date: June 2002)

Introduction

Is urotensin-II the new endothelin?

scientific article

Kisspeptins are novel potent vasoconstrictors in humans, with a discrete localization of their receptor, G protein-coupled receptor 54, to atherosclerosis-prone vessels

scientific article published on 5 October 2006

LGR5 Activates Noncanonical Wnt Signaling and Inhibits Aldosterone Production in the Human Adrenal

scientific article published on 27 April 2015

Life before birth: effects of cortisol on future cardiovascular and metabolic function.

scientific article published on July 2003

Localization of endothelin peptides in human kidney

scientific article published on 01 February 1996

Localization of endothelin receptors in human uterus throughout the menstrual cycle.

scientific article published on June 1996

Localization of endothelin-1 (ET-1), ET-2, and ET-3, mouse VIC, and sarafotoxin S6b binding sites in mammalian heart and kidney

scientific article published in January 1991

Localization of immunoreactive endothelin and proendothelin in the human lung

scientific article

Maternal dexamethasone increases endothelin-1 sensitivity and endothelin a receptor expression in ovine foetal placental arteries

scientific article published in April 2003

Measurement of C-terminal fragment of big endothelin-1: a novel method for assessing the generation of endothelin-1 in humans

scientific article published on 01 January 1995

Modulation of endothelin receptors in the failing right ventricle of the heart and vasculature of the lung in human pulmonary arterial hypertension

scientific article

Modulation of the apelin/APJ system in heart failure and atherosclerosis in man

scientific article

Molecular aspects of atrial natriuretic factor physiology.

scientific article published on January 1991

Myricerone caffeoyl ester (50-235) is a non-peptide antagonist selective for human ETA receptors

scientific article published on 01 June 1994

Neuropeptide B and W: neurotransmitters in an emerging G-protein-coupled receptor system

scientific article

No Alteration in Vasoconstrictor Endothelin-B-Receptor Density or Function in Human Coronary Artery Disease

scientific article published on 01 November 2000

No evidence for a local renin-angiotensin system in liver mitochondria

scientific journal article

Novel Nitric Oxide Donors Reverse Endothelin-1-Mediated Constriction in Human Blood Vessels

article

Novel ligands BQ123 and BQ3020 characterize endothelin receptor subtypes ETA and ETB in human kidney

scientific article published on 01 July 1993

Novel snake venom ligand dendroaspis natriuretic peptide is selective for natriuretic peptide receptor-A in human heart: downregulation of natriuretic peptide receptor-A in heart failure

scientific article published on 15 June 2006

Octopamine distribution in the larvae and adults of two species of moth, Spodoptera littoralis and Manduca sexta

article by Anthony P Davenport & Denis J. Wright published January 1986 in Journal of Insect Physiology

Of mice and men: advances in endothelin research and first antagonist gains FDA approval

scientific article

PD156707: A Potent Antagonist of Endothelin-1 in Human Diseased Coronary Arteries and Vein Grafts

article

Peptide and trace amine orphan receptors: prospects for new therapeutic targets

scientific article

Pharmacological targeting of apelin impairs glioblastoma growth.

scientific article

Pharmacology of renal endothelin receptors

scientific article published on August 30, 2011

Phosphoramidon inhibition of the in vivo conversion of big endothelin-1 to endothelin-1 in the human forearm.

scientific article published on September 1995

Positron emission tomography of [18F]-big endothelin-1 reveals renal excretion but tissue-specific conversion to [18F]-endothelin-1 in lung and liver

scientific article

Positron emission tomography using 18F-labelled endothelin-1 reveals prevention of binding to cardiac receptors owing to tissue-specific clearance by ET B receptors in vivo

scientific article published in January 2005

Potency of PD155080, an orally active ETA receptor antagonist, determined for human endothelin receptors

scientific article published on 01 January 1995

Quantification of endothelin receptor subtypes in peripheral tissues reveals downregulation of ET(A) receptors in ET(B)-deficient mice.

scientific article

Quantitative Phosphor Imaging Autoradiography of Radioligands for Positron Emission Tomography

scientific article published on 01 January 2012

Quantitative autoradiography reveals higher densities of specific calcitonin-gene-related peptide receptors in small intramyocardial compared with large epicardial coronary arteries

article

Radioligand Binding Assays and Their Analysis

article

Radioligand binding assays and quantitative autoradiography of endothelin receptors

article

Radioligand binding reveals chymase as the predominant enzyme for mediating tissue conversion of angiotensin I in the normal human heart

scientific article published in January 2002

Radioligand-binding and molecular-imaging techniques for the quantitative analysis of established and emerging orphan receptor systems

scientific article published in January 2005

Regional hemodynamic actions of selective corticotropin-releasing factor type 2 receptor ligands in conscious rats

scientific article

Regional heterogeneity in the haemodynamic responses to urotensin II infusion in relation to UT receptor localisation

scientific article published on March 2006

Regulation of endothelin receptor expression in vascular smooth-muscle cells

scientific article published on 01 January 1995

Regulation of vascular reactivity by established and emerging GPCRs

scientific article published in September 2005

Relative contribution of endothelin A and endothelin B receptors to vasoconstriction in small arteries from human heart and brain

scientific article published in January 1998

Screening β-arrestin recruitment for the identification of natural ligands for orphan G-protein-coupled receptors

scientific article

Secretion of endothelin-1 and endothelin-3 by human cultured vascular smooth muscle cells

scientific article

Secretory pathways in endothelin synthesis.

scientific article

Selectivity of [125I]-PD151242 for human, rat and porcine endothelin ETA receptors in the heart.

scientific article published on January 1995

Sex-related differences in the concentration of Met-enkephalin-like immunoreactivity in the nervous system of an insect, Schistocerca gregaria, revealed by radioimmunoassay

scientific article

Smooth Muscle Endothelin B Receptors Regulate Blood Pressure but Not Vascular Function or Neointimal Remodeling

scientific article published on 27 December 2016

Somatic mutations in ATP1A1 and CACNA1D underlie a common subtype of adrenal hypertension.

scientific article

Strategy for improved [(11)C]DAA1106 radiosynthesis and in vivo peripheral benzodiazepine receptor imaging using microPET, evaluation of [(11)C]DAA1106.

scientific article

Stress-induced changes in the octopamine levels of insect haemolymph

scholarly article by Anthony P Davenport & Peter D. Evans published January 1984 in Insect biochemistry

Syntheses of the First Endothelin-A- and -B-Selective Radioligands for Positron Emission Tomography

scientific article published on 01 November 2000

THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: G protein-coupled receptors

scientific article published on December 2017

THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: Overview

scientific article published on December 2017

THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: G protein-coupled receptors

scientific article published on 01 December 2019

THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: Introduction and Other Protein Targets

scientific article published on 01 December 2019

THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: G protein‐coupled receptors

journal article from 'British Journal of Pharmacology' published in 2021

The CCR5 chemokine receptor mediates vasoconstriction and stimulates intimal hyperplasia in human vessels in vitro.

scientific article published on 09 December 2013

The Concise Guide to PHARMACOLOGY 2013/14: overview

scientific article

The Concise Guide to PHARMACOLOGY 2015/16: G protein-coupled receptors

scientific article (publication date: December 2015)

The Concise Guide to PHARMACOLOGY 2015/16: Overview

scientific article

The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands

scientific article

The IUPHAR/BPS Guide to PHARMACOLOGY in 2018: updates and expansion to encompass the new guide to IMMUNOPHARMACOLOGY.

scientific article published on 15 November 2017

The IUPHAR/BPS Guide to PHARMACOLOGY: an expert-driven knowledgebase of drug targets and their ligands

scientific article (publication date: 2014)

The IUPHAR/BPS guide to PHARMACOLOGY in 2022: curating pharmacology for COVID-19, malaria and antibacterials

scientific article published on 01 January 2022

The Prodomain-bound Form of Bone Morphogenetic Protein 10 Is Biologically Active on Endothelial Cells

scientific article

The Twelfth International Conference on Endothelin (ET-12), Cambridge 2011

scientific article published on July 26, 2012

The action of formamidines on octopamine receptors in the locust

scientific article published in 1985

The dual endothelin converting enzyme/neutral endopeptidase inhibitor SLV-306 (daglutril), inhibits systemic conversion of big endothelin-1 in humans

scientific article published on 28 March 2012

The endothelin peptides ET-1, ET-2, ET-3 and sarafotoxin S6b are co-mitogenic with platelet-derived growth factor for vascular smooth muscle cells

article

The endothelin system in pulmonary and renal vasculopathy: les liaisons dangereuses.

scientific article published on December 2009

The haemodynamic effects of iodinated water soluble radiographic contrast media: a review

article

The therapeutic potential of PD156707 and related butenolide endothelin antagonists.

scientific article published in January 1999

The use of quantitative immunocytochemistry (QICC) to measure calbindin D28k-like immunoreactivity in the rat brain

scientific article published on 01 January 1990

Themed section: Imaging in pharmacology

scientific article

Themed section: endothelin

scientific article published in January 2013

Thromboxane receptor density is increased in human cardiovascular disease with evidence for inhibition at therapeutic concentrations by the AT(1) receptor antagonist losartan

scientific article

Tissue-Specific Modulation of Endothelin Receptors in a Rat Model of Hypertension

Toxicity of chlordimeform and amitraz to the egyptian cotton leafworm (Spodoptera littoralis) and the tobacco budworm (Heliothis virescens)

article

Translating the human genome: renaissance of cardiovascular receptor pharmacology

scientific article published on 01 April 2003

Triptan-induced contractile (5-HT1B receptor) responses in human cerebral and coronary arteries: relationship to clinical effect

scientific article published in September 2005

Vascular Imaging With 18F-Fluorodeoxyglucose Positron Emission Tomography Is Influenced by Hypoxia

scientific article published on April 2017

Vasoconstrictor activity of novel endothelin peptide, ET-1(1 - 31), in human mammary and coronary arteries in vitro

scientific article

[125I]-PD151242: a selective ligand for endothelin ETA receptors in human kidney which localizes to renal vasculature.

scientific article published on December 1994

[125I]-PD151242: a selective radioligand for human ETA receptors

scientific article

[Pyr1]Apelin-13(1-12) Is a Biologically Active ACE2 Metabolite of the Endogenous Cardiovascular Peptide [Pyr1]Apelin-13.

scientific article published on 28 February 2017

[Pyr1]apelin-13 identified as the predominant apelin isoform in the human heart: vasoactive mechanisms and inotropic action in disease.

scientific article published on 13 July 2009