List of works - Walter Cabri

4,5,6,7-Tetrahydro-isoxazolo-[4,5-c]-pyridines as a new class of cytotoxic Hsp90 inhibitors

scientific article

A new group of oxime carbamates as reversible inhibitors of fatty acid amide hydrolase.

scientific article published on 15 June 2010

A translation of the twelve principles of green chemistry to guide the development of cross-coupling reactions

scientific article published in 2022

Application of Af4-Multidetection to Liraglutide in Its Formulation: Preserving and Representing Native Aggregation

scientific article published in 2022

Azetidinones as zinc-binding groups to design selective HDAC8 inhibitors

scientific article published in December 2009

Benefits of a Mixed-Mode Stationary Phase to Address the Challenging Purification of an Industrially Relevant Peptide: A Proof-of-Concept Study

scientific article published in 2022

Biotechnological lycopene production by mated fermentation of Blakeslea trispora

scientific article published on 10 July 2004

Biotransformation of colchicinoids into their corresponding 3-O-glucosyl derivatives by selected strains of Bacillus megaterium

scientific article published in July 2014

Camptothecins in tumor homing via an RGD sequence mimetic.

scientific article published on 26 July 2012

Cefdinir: A comparative study of anhydrous vs. monohydrate form. Microstructure and tabletting behaviour

scientific article published on 26 May 2006

Combination of HPLC "inverted chirality columns approach" and MS/MS detection for extreme enantiomeric excess determination even in absence of reference samples. Application to camptothecin derivatives

scientific article published on 29 June 2007

Derivatives of R-aminocarnitine without ammonium moiety as liver carnitine palmitoyltransferase I (L-CPT I) inhibitors

scientific article published on 10 August 2011

Direct B-alkyl Suzuki-Miyaura cross-coupling of 2-halopurines. Practical synthesis of ST1535, a potent adenosine A2A receptor antagonist.

scientific article published in August 2010

Discovery of potent inhibitors of human and mouse fatty acid amide hydrolases

scientific article published on 26 July 2012

Divergent synthesis of novel 9-deazaxanthine derivatives via late-stage cross-coupling reactions.

scientific article

Effect of SAMITAL® in the treatment of chemotherapy-induced mucositis in adult oncohematological patients

scientific article

Efficient organic monoliths prepared by γ-radiation induced polymerization in the evaluation of histone deacetylase inhibitors by capillary(nano)-high performance liquid chromatography and ion trap mass spectrometry

scientific article published on 27 April 2011

Enol carbamates as inhibitors of fatty acid amide hydrolase (FAAH) endowed with high selectivity for FAAH over the other targets of the endocannabinoid system

scientific article published in March 2010

Evolution of an acylase active on cephalosporin C

scientific article published on 31 October 2005

Extending the use of "Inverted Chirality Columns Approach" for enantiomeric excess determination in absence of reference samples: Application to a water-soluble camptothecin derivative.

scientific article published on 17 October 2009

Fast Heck-Cassar-Sonogashira (HCS) Reactions in Green Solvents

scientific article published on 28 April 2020

Ganoderma lucidum Ethanol Extracts Enhance Re-Epithelialization and Prevent Keratinocytes from Free-Radical Injury

scientific article published on 29 August 2020

Histone deacetylase inhibitors in the treatment of cancer: overview and perspectives.

scientific article published on July 2012

Identification of a novel arylpiperazine scaffold for fatty acid amide hydrolase inhibition with improved drug disposition properties

scientific article published on 22 November 2012

Identification of impurities in artemisinin, their behavior in high performance liquid chromatography and implications for the quality of derived anti-malarial drugs

scientific article published on 30 July 2011

Innovative chemical synthesis and conformational hints on the lipopeptide liraglutide.

scientific article published on 30 May 2016

Investigating the Neuroprotective Effects of Turmeric Extract: Structural Interactions of β-Amyloid Peptide with Single Curcuminoids.

scientific article published on 22 December 2016

Isoxazolo(aza)naphthoquinones: a new class of cytotoxic Hsp90 inhibitors

scientific article published on 28 March 2012

Lactam based 7-amino suberoylamide hydroxamic acids as potent HDAC inhibitors

scientific article published on 4 December 2013

Modeling the nonlinear behavior of a bioactive peptide in reversed-phase gradient elution chromatography

scientific article published on 19 December 2019

N-Hydroxy-(4-oxime)-cinnamide: a versatile scaffold for the synthesis of novel histone deacetylase [correction of deacetilase] (HDAC) inhibitors

scientific article

Natural Occurring and Engineered Enzymes for Peptide Ligation and Cyclization

scientific article published on 29 November 2019

New retinoid derivatives as back-ups of Adarotene

scientific article

Non-natural macrocyclic inhibitors of histone deacetylases: design, synthesis, and activity.

scientific article published on 12 November 2010

Novel 3,4-Isoxazolediamides as Potent Inhibitors of Chaperone Heat Shock Protein 90 ⬇️

scientific article published on November 23, 2011

Novel insights into the chemistry of an old medicine: A general degradative pathway for penicillins from a piperacillin/tazobactam stability study

scientific article published on 14 June 2019

Novel substituted aminoalkylguanidines as potential antihyperglycemic and food intake-reducing agents

scientific article published on 9 May 2008

Omega-alkoxy analogues of SAHA (vorinostat) as inhibitors of HDAC: a study of chain-length and stereochemical dependence.

scientific article

On-column epimerization of dihydroartemisinin: an effective analytical approach to overcome the shortcomings of the International Pharmacopoeia monograph.

scientific article published in November 2008

Oxime amides as a novel zinc binding group in histone deacetylase inhibitors: synthesis, biological activity, and computational evaluation.

scientific article

Polymorphisms and Patent, Market, and Legal Battles: Cefdinir Case Study

scientific article (publication date: 2007)

Potent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2A Receptor Ligands

scientific article published on 07 May 2015

Production of peptides as generic drugs: a patent landscape of octreotide

scientific article published on 29 February 2016

Protective effect of Panax ginseng in cisplatin-induced cachexia in rats.

scientific article published on May 2014

Reducing effect of the Chinese medicinal herb, Salvia miltiorrhiza, on alcohol self-administration in Sardinian alcohol-preferring rats

scientific article

SAMITAL®: a new botanical drug for the treatment of mucositis induced by oncological therapies.

scientific article

ST7612AA1, a thioacetate-ω(γ-lactam carboxamide) derivative selected from a novel generation of oral HDAC inhibitors

scientific article

Stereodynamic investigation of labile stereogenic centres in dihydroartemisinin.

scientific article published on 05 March 2010

Stereolability of dihydroartemisinin, an antimalarial drug: a comprehensive kinetic investigation. Part 2.

scientific article published on 16 May 2011

Stereolability of dihydroartemisinin, an antimalarial drug: a comprehensive thermodynamic investigation. Part 1.

scientific article published on 22 February 2011

Synthesis and biological activity of fluorinated combretastatin analogues

scientific article

Synthesis and biological evaluation of metabolites of 2-n-butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine (ST1535), a potent antagonist of the A2A adenosine receptor for the treatment of Parkinson's disease.

scientific article published on 24 June 2013

Synthesis and evaluation of new Hsp90 inhibitors based on a 1,4,5-trisubstituted 1,2,3-triazole scaffold.

scientific article

Synthesis of (E)-8-(3-chlorostyryl)caffeine analogues leading to 9-deazaxanthine derivatives as dual A(2A) antagonists/MAO-B inhibitors.

scientific article published on 16 January 2013

Towards the development of 5-HT7 ligands combining serotonin-like and arylpiperazine moieties

scientific article published on 13 April 2014

Vorinostat-like molecules as structural, stereochemical, and pharmacological tools

scientific article

List of works by Walter Cabri

4,5,6,7-Tetrahydro-isoxazolo-[4,5-c]-pyridines as a new class of cytotoxic Hsp90 inhibitors

A new group of oxime carbamates as reversible inhibitors of fatty acid amide hydrolase.

A translation of the twelve principles of green chemistry to guide the development of cross-coupling reactions

Application of Af4-Multidetection to Liraglutide in Its Formulation: Preserving and Representing Native Aggregation

Azetidinones as zinc-binding groups to design selective HDAC8 inhibitors

Benefits of a Mixed-Mode Stationary Phase to Address the Challenging Purification of an Industrially Relevant Peptide: A Proof-of-Concept Study

Biotechnological lycopene production by mated fermentation of Blakeslea trispora

Biotransformation of colchicinoids into their corresponding 3-O-glucosyl derivatives by selected strains of Bacillus megaterium

Camptothecins in tumor homing via an RGD sequence mimetic.

Cefdinir: A comparative study of anhydrous vs. monohydrate form. Microstructure and tabletting behaviour

Combination of HPLC "inverted chirality columns approach" and MS/MS detection for extreme enantiomeric excess determination even in absence of reference samples. Application to camptothecin derivatives

Derivatives of R-aminocarnitine without ammonium moiety as liver carnitine palmitoyltransferase I (L-CPT I) inhibitors

Direct B-alkyl Suzuki-Miyaura cross-coupling of 2-halopurines. Practical synthesis of ST1535, a potent adenosine A2A receptor antagonist.

Discovery of potent inhibitors of human and mouse fatty acid amide hydrolases

Divergent synthesis of novel 9-deazaxanthine derivatives via late-stage cross-coupling reactions.

Effect of SAMITAL® in the treatment of chemotherapy-induced mucositis in adult oncohematological patients

Efficient organic monoliths prepared by γ-radiation induced polymerization in the evaluation of histone deacetylase inhibitors by capillary(nano)-high performance liquid chromatography and ion trap mass spectrometry

Enol carbamates as inhibitors of fatty acid amide hydrolase (FAAH) endowed with high selectivity for FAAH over the other targets of the endocannabinoid system

Evolution of an acylase active on cephalosporin C

Extending the use of "Inverted Chirality Columns Approach" for enantiomeric excess determination in absence of reference samples: Application to a water-soluble camptothecin derivative.

Fast Heck-Cassar-Sonogashira (HCS) Reactions in Green Solvents

Ganoderma lucidum Ethanol Extracts Enhance Re-Epithelialization and Prevent Keratinocytes from Free-Radical Injury

Histone deacetylase inhibitors in the treatment of cancer: overview and perspectives.

Identification of a novel arylpiperazine scaffold for fatty acid amide hydrolase inhibition with improved drug disposition properties

Identification of impurities in artemisinin, their behavior in high performance liquid chromatography and implications for the quality of derived anti-malarial drugs

Innovative chemical synthesis and conformational hints on the lipopeptide liraglutide.

Investigating the Neuroprotective Effects of Turmeric Extract: Structural Interactions of β-Amyloid Peptide with Single Curcuminoids.

Isoxazolo(aza)naphthoquinones: a new class of cytotoxic Hsp90 inhibitors

Lactam based 7-amino suberoylamide hydroxamic acids as potent HDAC inhibitors

Modeling the nonlinear behavior of a bioactive peptide in reversed-phase gradient elution chromatography

N-Hydroxy-(4-oxime)-cinnamide: a versatile scaffold for the synthesis of novel histone deacetylase [correction of deacetilase] (HDAC) inhibitors

Natural Occurring and Engineered Enzymes for Peptide Ligation and Cyclization

New retinoid derivatives as back-ups of Adarotene

Non-natural macrocyclic inhibitors of histone deacetylases: design, synthesis, and activity.

Novel 3,4-Isoxazolediamides as Potent Inhibitors of Chaperone Heat Shock Protein 90 ⬇️

Novel insights into the chemistry of an old medicine: A general degradative pathway for penicillins from a piperacillin/tazobactam stability study

Novel substituted aminoalkylguanidines as potential antihyperglycemic and food intake-reducing agents

Omega-alkoxy analogues of SAHA (vorinostat) as inhibitors of HDAC: a study of chain-length and stereochemical dependence.

On-column epimerization of dihydroartemisinin: an effective analytical approach to overcome the shortcomings of the International Pharmacopoeia monograph.

Oxime amides as a novel zinc binding group in histone deacetylase inhibitors: synthesis, biological activity, and computational evaluation.

Polymorphisms and Patent, Market, and Legal Battles: Cefdinir Case Study

Potent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2A Receptor Ligands

Production of peptides as generic drugs: a patent landscape of octreotide

Protective effect of Panax ginseng in cisplatin-induced cachexia in rats.

Reducing effect of the Chinese medicinal herb, Salvia miltiorrhiza, on alcohol self-administration in Sardinian alcohol-preferring rats

SAMITAL®: a new botanical drug for the treatment of mucositis induced by oncological therapies.

ST7612AA1, a thioacetate-ω(γ-lactam carboxamide) derivative selected from a novel generation of oral HDAC inhibitors

Stereodynamic investigation of labile stereogenic centres in dihydroartemisinin.

Stereolability of dihydroartemisinin, an antimalarial drug: a comprehensive kinetic investigation. Part 2.

Stereolability of dihydroartemisinin, an antimalarial drug: a comprehensive thermodynamic investigation. Part 1.

Synthesis and biological activity of fluorinated combretastatin analogues

Synthesis and biological evaluation of metabolites of 2-n-butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine (ST1535), a potent antagonist of the A2A adenosine receptor for the treatment of Parkinson's disease.

Synthesis and evaluation of new Hsp90 inhibitors based on a 1,4,5-trisubstituted 1,2,3-triazole scaffold.

Synthesis of (E)-8-(3-chlorostyryl)caffeine analogues leading to 9-deazaxanthine derivatives as dual A(2A) antagonists/MAO-B inhibitors.

Towards the development of 5-HT7 ligands combining serotonin-like and arylpiperazine moieties

Vorinostat-like molecules as structural, stereochemical, and pharmacological tools