List of works - György Dormán

A New Paclitaxel Photoaffinity Analog with a 3-(4-Benzoylphenyl)propanoyl Probe for Characterization of Drug-Binding Sites on Tubulin and P-Glycoprotein

scientific article published on 01 September 1995

Benzophenone photophores in biochemistry.

scientific article published on May 1994

Combination of 2D/3D ligand-based similarity search in rapid virtual screening from multimillion compound repositories. Selection and biological evaluation of potential PDE4 and PDE5 inhibitors.

scientific article

Combination of Pharmacophore Matching, 2D Similarity Search, and In Vitro Biological Assays in the Selection of Potential 5-HT6 Antagonists from Large Commercial Repositories

scientific article published on 30 March 2015

Combining 2D and 3D in silico methods for rapid selection of potential PDE5 inhibitors from multimillion compounds' repositories: biological evaluation

scientific article

Design, selection, and evaluation of a general kinase-focused library

scientific article published in August 2009

Enhanced hit-to-lead process using bioanalogous lead evolution and chemogenomics: application in designing selective matrix metalloprotease inhibitors

scientific article published on 01 May 2007

Explicit Diversity Index (EDI): a novel measure for assessing the diversity of compound databases

scientific article published in September 2006

Identification of potential glutaminyl cyclase inhibitors from lead-like libraries by in silico and in vitro fragment-based screening

scientific article

MMP inhibitors in cardiac diseases: an update

scientific article published on 01 November 2007

Meldrum's Acid in Multicomponent Reactions: Applications to Combinatorial and Diversity-Oriented Synthesis

N-Acylhydrazones as inhibitors of PDE10A

scientific article published on 02 June 2011

Phosphoinositide binding specificity among phospholipase C isozymes as determined by photo-cross-linking to novel substrate and product analogs

scientific article published on 01 June 1997

Procedure for the parallel preparation of 3-imidazo[1,2-a]pyridin-3-yl-propionic acid derivatives involving Meldrum's acid

scientific article published in July 2005

Purified inositol hexakisphosphate kinase is an ATP synthase: diphosphoinositol pentakisphosphate as a high-energy phosphate donor

scientific article published on April 1996

Special issue in flow chemistry

scientific article published on 13 July 2011

Stepwise aromatic nucleophilic substitution in continuous flow. Synthesis of an unsymmetrically substituted 3,5-diamino-benzonitrile library.

scientific article

Substrate specificity of Escherichia coli MutY protein.

scientific article

Synthesis of enzymatically noncleavable carbocyclic nucleosides for DNA-N-glycosylase studies

scientific article published on 01 March 1998

Tethered benzophenone reagents for the synthesis of photoactivatable ligands

scientific article published on 01 July 1995

The Life of Pi Star: Exploring the Exciting and Forbidden Worlds of the Benzophenone Photophore

scientific article published on 16 December 2016

Using photolabile ligands in drug discovery and development.

scientific article

List of works by György Dormán

A New Paclitaxel Photoaffinity Analog with a 3-(4-Benzoylphenyl)propanoyl Probe for Characterization of Drug-Binding Sites on Tubulin and P-Glycoprotein

Benzophenone photophores in biochemistry.

Combination of 2D/3D ligand-based similarity search in rapid virtual screening from multimillion compound repositories. Selection and biological evaluation of potential PDE4 and PDE5 inhibitors.

Combination of Pharmacophore Matching, 2D Similarity Search, and In Vitro Biological Assays in the Selection of Potential 5-HT6 Antagonists from Large Commercial Repositories

Combining 2D and 3D in silico methods for rapid selection of potential PDE5 inhibitors from multimillion compounds' repositories: biological evaluation

Design, selection, and evaluation of a general kinase-focused library

Enhanced hit-to-lead process using bioanalogous lead evolution and chemogenomics: application in designing selective matrix metalloprotease inhibitors

Explicit Diversity Index (EDI): a novel measure for assessing the diversity of compound databases

Identification of potential glutaminyl cyclase inhibitors from lead-like libraries by in silico and in vitro fragment-based screening

MMP inhibitors in cardiac diseases: an update

Meldrum's Acid in Multicomponent Reactions: Applications to Combinatorial and Diversity-Oriented Synthesis

N-Acylhydrazones as inhibitors of PDE10A

Phosphoinositide binding specificity among phospholipase C isozymes as determined by photo-cross-linking to novel substrate and product analogs

Procedure for the parallel preparation of 3-imidazo[1,2-a]pyridin-3-yl-propionic acid derivatives involving Meldrum's acid

Purified inositol hexakisphosphate kinase is an ATP synthase: diphosphoinositol pentakisphosphate as a high-energy phosphate donor

Special issue in flow chemistry

Stepwise aromatic nucleophilic substitution in continuous flow. Synthesis of an unsymmetrically substituted 3,5-diamino-benzonitrile library.

Substrate specificity of Escherichia coli MutY protein.

Synthesis of enzymatically noncleavable carbocyclic nucleosides for DNA-N-glycosylase studies

Tethered benzophenone reagents for the synthesis of photoactivatable ligands

The Life of Pi Star: Exploring the Exciting and Forbidden Worlds of the Benzophenone Photophore

Using photolabile ligands in drug discovery and development.