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List of works by Giuseppe Caliendo

5-Amino-2-hydroxybenzoic Acid 4-(5-Thioxo-5H-[1,2]dithiol-3yl)-phenyl Ester (ATB-429), a Hydrogen Sulfide-Releasing Derivative of Mesalamine, Exerts Antinociceptive Effects in a Model of Postinflammatory Hypersensitivity

scientific article published on 19 July 2006

5-HT(1A) receptor: an old target as a new attractive tool in drug discovery from central nervous system to cancer

scientific article published on 10 December 2013

A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold

A convenient synthesis by microwave heating and pharmacological evaluation of novel benzoyltriazole and saccharine derivatives as 5-HT(1A) receptor ligands.

scientific article

A convenient synthesis of N-Fmoc-N,N′-bis-Boc-7-guanyl-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (Fmoc-N,N′-bis-Boc-7-guanyl-Tic-OH, GTIC)

A nitro-arginine derivative of trimebutine (NO2-Arg-Trim) attenuates pain induced by colorectal distension in conscious rats.

scientific article published on 29 January 2009

A suitable 1,2,4-oxadiazoles synthesis by microwave irradiation

scientific article published on 01 September 2004

Bromazepam determination in human plasma by high-performance liquid chromatography coupled to tandem mass spectrometry: a highly sensitive and specific tool for bioequivalence studies.

scientific article published in February 2004

Conformation-activity relationship of peptide T and new pseudocyclic hexapeptide analogs

scientific article published on 01 June 2007

Conformational analysis of three NK1 tripeptide antagonists: a proton nuclear magnetic resonance study

scientific article published in February 1997

Derivatives as 5HT1A receptor ligands--past and present.

scientific article

Design of Inhibitors for Human Tissue Kallikrein Using Non-Natural Aromatic and Basic Amino Acids

scientific article published on 01 May 2002

Development of 1,2,3-Triazole-Based Sphingosine Kinase Inhibitors and Their Evaluation as Antiproliferative Agents.

scientific article published on 5 November 2017

Efficient microwave combinatorial parallel and nonparallel synthesis of N-alkylated glycine methyl esters as peptide building blocks.

scientific article published in July 2005

Efficient microwave combinatorial synthesis of novel indolic arylpiperazine derivatives as serotoninergic ligands.

scientific article

Enhanced activity of a hydrogen sulphide-releasing derivative of mesalamine (ATB-429) in a mouse model of colitis

scientific article

Evidence for a protective role played by the Na+/Ca2+ exchanger in cerebral ischemia induced by middle cerebral artery occlusion in male rats

scientific article published in March 2004

Gastrointestinal Safety and Anti-Inflammatory Effects of a Hydrogen Sulfide–Releasing Diclofenac Derivative in the Rat

scientific article published on 29 November 2006

Identification of a pepducin acting as S1P3 receptor antagonist.

scientific article published on 20 September 2013

In vitro mutagenicity of anti-inflammatory parsalmide analogues PA7, PA10, and PA31 triggered by biotransformation into hydroxy derivatives

scientific article published on 18 January 2006

Kallikrein protease activated receptor (PAR) axis: an attractive target for drug development

scientific article

Markedly reduced toxicity of a hydrogen sulphide-releasing derivative of naproxen (ATB-346).

scientific article

Minimal structural requirements for agonist activity of PAR-2 activating peptides.

scientific article published in January 2002

Neurounina-1, a novel compound that increases Na+/Ca2+ exchanger activity, effectively protects against stroke damage

scientific article

Nevirapine quantification in human plasma by high-performance liquid chromatography coupled to electrospray tandem mass spectrometry. Application to bioequivalence study.

scientific article

New 5-HT(1A) receptor ligands containing a N'-cyanoisonicotinamidine nucleus: synthesis and in vitro pharmacological evaluation

scientific article published on 3 March 2010

New 5-hydroxytryptamine(1A) receptor ligands containing a norbornene nucleus: synthesis and in vitro pharmacological evaluation.

scientific article published in August 2005

New potent 5-HT2A receptor ligands containing an N′-cyanopicolinamidine nucleus: Synthesis and in vitro pharmacological evaluation

scientific article published on 20 November 2011

Nitric Oxide Related Therapeutic Phenomenon: A Challenging Task

scientific article published on 01 January 2002

PAR1 antagonism protects against experimental liver fibrosis. Role of proteinase receptors in stellate cell activation

scientific article published on February 2004

Peptide T revisited: conformational mimicry of epitopes of anti-HIV proteins

scientific article published in April 2001

Perfusion of rat colon with sennosides, rhein and rheinanthrone. Concentration-related histamine release

scientific article published on 01 November 1990

Pharmacokinetics of dihydroergocristine and its major metabolite 8'-hydroxy-dihydroergocristine in human plasma

scientific article published in December 2005

Probing the shape of a hydrophobic pocket in the active site of delta-opioid antagonists.

scientific article published in July 2001

Pyrrolobenzoxazepinone derivatives as non-nucleoside HIV-1 RT inhibitors: further structure-activity relationship studies and identification of more potent broad-spectrum HIV-1 RT inhibitors with antiviral activity

scientific article

S1 subsite specificity of a recombinant cysteine proteinase, CPB, of Leishmania mexicana compared with cruzain, human cathepsin L and papain using substrates containing non-natural basic amino acids

scientific article

Specificity studies on Kallikrein-related peptidase 7 (KLK7) and effects of osmolytes and glycosaminoglycans on its peptidase activity.

scientific article published on 30 October 2014

Structure—affinity relationship studies on benzotriazole derivatives binding to 5-HT receptor subtypes

Synthesis and Pharmacological Screening of Pyridopyrimidines as Effective Anti-Diarrheal Agents through the Suppression of Cyclic Nucleotide Accumulation

scientific article published on 08 April 2019

Synthesis and antiinflammatory—analgesic profile of 1-methyl-2-(4-X-benzoyl) imidazole-5-carboxylic acids

article published in 1995

Synthesis and antimicrobial activities of 5-amidobenzotriazole derivatives

Synthesis and antinociceptive activity of peptides related to interleukin-1 beta 193-195 Lys-Pro-Thr

scientific article published on 01 January 1996

Synthesis and biological activity of benzotriazole derivatives structurally related to trazodone

Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids.

scientific article

Synthesis and biological activity of tripeptide FR113680 analogues containing unconventional amino acids.

scientific article

Synthesis and biological effects of hydrogen sulfide (H2S): development of H2S-releasing drugs as pharmaceuticals

scientific article published on September 2010

Synthesis and hydrolysis by cathepsin B of fluorogenic substrates with the general structure benzoyl-X-ARG-MCA containing non-natural basic amino acids at position X.

scientific article

Synthesis and in vitro pharmacological evaluation of novel 2-hydroxypropyl-4-arylpiperazine derivatives as serotoninergic ligands

scientific article published on 11 August 2014

Synthesis and in-vitro pharmacological evaluation of new 5-HT1A receptor ligands containing a benzotriazinone nucleus.

scientific article published in January 2008

Synthesis and pharmacological activity of deltorphin and dermorphin-related glycopeptides.

scientific article published in August 1997

Synthesis and pharmacological evaluation of a set of N-[2-(alkylamino)ethyl]benzotriazol-X-yl isobutyramides acting as local anesthetics

scholarly article by Giuseppe Caliendo et al published January 1996 in European Journal of Medicinal Chemistry

Synthesis and pharmacological evaluation of peptide-mimetic protease-activated receptor-1 antagonists containing novel heterocyclic scaffolds.

scientific article published on 26 April 2008

Synthesis and pharmacological evaluations of sildenafil analogues for treatment of erectile dysfunction.

scientific article

Synthesis and structure-activity relationships of antiinflammatory 1-methyl-2-(4-X-benzoyl)imidazole-5-acetic acids

Synthesis and vasorelaxant activity of new 1,4-benzoxazine derivatives potassium channel openers

scientific article

Synthesis by microwave irradiation and antidiarrhoeal activity of benzotriazinone and saccharine derivatives

scientific article

Synthesis by microwave irradiation and binding properties of novel 5-HT(1A) receptor ligands

scientific article published in November 2001

Synthesis of 1-naphtylpiperazine derivatives as serotoninergic ligands and their evaluation as antiproliferative agents

scientific article published on 08 March 2011

Synthesis of 2-Methyl-3-indolylacetic Derivatives as Anti-Inflammatory Agents That Inhibit Preferentially Cyclooxygenase 1 without Gastric Damage

scientific article published on 01 December 2006

Synthesis of benzamide derivatives and their evaluation as antiprion agents

scientific article

Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands

scientific article published on 01 March 2000

Synthesis of novel anti-inflammatory peptides derived from the amino-acid sequence of the bioactive protein SV-IV.

scientific article published in June 2001

Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage

scientific article published in June 2001

Synthesis ofN α-FmocN,N′-bis-Boc-5-, 6- and 8-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic Acid (5-GTIC, 6-GTIC and 8-GTIC)

article

Synthesis, antimicrobial data and correlation analysis in a set of 2-alkyl-5-amidobenzotriazoles

Synthesis, biological evaluation, and docking studies of PAR2-AP-derived pseudopeptides as inhibitors of kallikrein 5 and 6

scientific article published on 01 January 2015

Synthesis, local anesthetic activity and QSAR studies for a set of N-[2-(alkylamino)ethyl]benzotriazol-x-yl acetamides

Synthesis, pharmacological evaluation, and molecular modeling studies of novel peptidic CAAX analogues as farnesyl-protein-transferase inhibitors

scientific article published on March 2006

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