List of works - Erki Enkvist

A Selective Biligand Inhibitor of CK2 Increases Caspase-3 Activity in Cancer Cells and Inhibits Platelet Aggregation

scientific article published on 24 August 2017

A subnanomolar fluorescent probe for protein kinase CK2 interaction studies

scientific article

Acetoxymethyl Ester of Tetrabromobenzimidazole-Peptoid Conjugate for Inhibition of Protein Kinase CK2 in Living Cells

scientific article published on 12 November 2015

Adenosine analogue-oligo-arginine conjugates (ARCs) serve as high-affinity inhibitors and fluorescence probes of type I cGMP-dependent protein kinase (PKGIalpha)

scientific article

Adenosine-derived non-phosphate antagonists for P2Y(1) purinoceptors.

scientific article published in June 2000

Benzoselenadiazole-based responsive long-lifetime photoluminescent probes for protein kinases.

scientific article published in April 2014

Bifunctional Ligands for Inhibition of Tight-Binding Protein-Protein Interactions

scientific article

Bisubstrate inhibitors of protein kinases: from principle to practical applications

scientific article published on January 2010

Carbocyclic 3'-deoxyadenosine-based highly potent bisubstrate-analog inhibitor of basophilic protein kinases

scientific article published on 15 August 2007

Combining chemical and genetic approaches for development of responsive FRET-based sensor systems for protein kinases.

scientific article published on 25 January 2016

Conjugates of 5-isoquinolinesulfonylamides and oligo-d-arginine possess high affinity and selectivity towards Rho kinase (ROCK) ⬇️

scientific article published on April 4, 2012

Conjugation of adenosine and hexa-(D-arginine) leads to a nanomolar bisubstrate-analog inhibitor of basophilic protein kinases

scientific article published on 01 November 2006

Correction to "Deoxygenation Increases Photoluminescence Lifetime of Protein-Responsive Organic Probes with Triplet-Singlet Resonant Energy Transfer".

scientific article published on 23 September 2016

Deoxygenation Increases Photoluminescence Lifetime of Protein-Responsive Organic Probes with Triplet-Singlet Resonant Energy Transfer.

scientific article

Diversity of bisubstrate binding modes of adenosine analogue-oligoarginine conjugates in protein kinase a and implications for protein substrate interactions

scientific article

Efficient photocaging of a tight-binding bisubstrate inhibitor of cAMP-dependent protein kinase

scientific article published on 29 August 2019

FRET-based screening assay using small-molecule photoluminescent probes in lysate of cells overexpressing RFP-fused protein kinases.

scientific article published on 10 April 2015

High-affinity bisubstrate probe for fluorescence anisotropy binding/displacement assays with protein kinases PKA and ROCK.

scientific article published on 31 October 2008

Inhibition of CREB phosphorylation by conjugates of adenosine analogues and arginine-rich peptides, inhibitors of PKA catalytic subunit

scientific article published on 8 December 2014

Long residence times revealed by Aurora A kinase-targeting fluorescent probes derived from inhibitors MLN8237 and VX-689.

scientific article

Oligo-aspartic acid conjugates with benzo[c][2,6]naphthyridine-8-carboxylic acid scaffold as picomolar inhibitors of CK2.

scientific article published on 28 February 2017

Protein-induced long lifetime luminescence of nonmetal probes.

scientific article

Selective bisubstrate inhibitors with sub-nanomolar affinity for protein kinase Pim-1.

scientific article published on 24 April 2013

Slowly on, Slowly off: Bisubstrate-Analogue Conjugates of 5-Iodotubercidin and Histone H3 Peptide Targeting Protein Kinase Haspin.

scientific article published on 9 February 2017

Structural analysis of ARC-type inhibitor (ARC-1034) binding to protein kinase A catalytic subunit and rational design of bisubstrate analogue inhibitors of basophilic protein kinases

scientific article

Synthesis of potential purinoceptor antagonists: application of P1-tBU phosphazene base for alkylation of adenine in solution and on solid phase

scientific article published on 01 January 2006

Targeting Plasmodium falciparum protein kinases with adenosine analogue-oligoarginine conjugates

scientific article published on 15 February 2014

Time-gated luminescence microscopy with responsive nonmetal probes for mapping activity of protein kinases in living cells

scientific article

List of works by Erki Enkvist

A Selective Biligand Inhibitor of CK2 Increases Caspase-3 Activity in Cancer Cells and Inhibits Platelet Aggregation

A subnanomolar fluorescent probe for protein kinase CK2 interaction studies

Acetoxymethyl Ester of Tetrabromobenzimidazole-Peptoid Conjugate for Inhibition of Protein Kinase CK2 in Living Cells

Adenosine analogue-oligo-arginine conjugates (ARCs) serve as high-affinity inhibitors and fluorescence probes of type I cGMP-dependent protein kinase (PKGIalpha)

Adenosine-derived non-phosphate antagonists for P2Y(1) purinoceptors.

Benzoselenadiazole-based responsive long-lifetime photoluminescent probes for protein kinases.

Bifunctional Ligands for Inhibition of Tight-Binding Protein-Protein Interactions

Bisubstrate inhibitors of protein kinases: from principle to practical applications

Carbocyclic 3'-deoxyadenosine-based highly potent bisubstrate-analog inhibitor of basophilic protein kinases

Combining chemical and genetic approaches for development of responsive FRET-based sensor systems for protein kinases.

Conjugates of 5-isoquinolinesulfonylamides and oligo-d-arginine possess high affinity and selectivity towards Rho kinase (ROCK) ⬇️

Conjugation of adenosine and hexa-(D-arginine) leads to a nanomolar bisubstrate-analog inhibitor of basophilic protein kinases

Correction to "Deoxygenation Increases Photoluminescence Lifetime of Protein-Responsive Organic Probes with Triplet-Singlet Resonant Energy Transfer".

Deoxygenation Increases Photoluminescence Lifetime of Protein-Responsive Organic Probes with Triplet-Singlet Resonant Energy Transfer.

Diversity of bisubstrate binding modes of adenosine analogue-oligoarginine conjugates in protein kinase a and implications for protein substrate interactions

Efficient photocaging of a tight-binding bisubstrate inhibitor of cAMP-dependent protein kinase

FRET-based screening assay using small-molecule photoluminescent probes in lysate of cells overexpressing RFP-fused protein kinases.

High-affinity bisubstrate probe for fluorescence anisotropy binding/displacement assays with protein kinases PKA and ROCK.

Inhibition of CREB phosphorylation by conjugates of adenosine analogues and arginine-rich peptides, inhibitors of PKA catalytic subunit

Long residence times revealed by Aurora A kinase-targeting fluorescent probes derived from inhibitors MLN8237 and VX-689.

Oligo-aspartic acid conjugates with benzo[c][2,6]naphthyridine-8-carboxylic acid scaffold as picomolar inhibitors of CK2.

Protein-induced long lifetime luminescence of nonmetal probes.

Selective bisubstrate inhibitors with sub-nanomolar affinity for protein kinase Pim-1.

Slowly on, Slowly off: Bisubstrate-Analogue Conjugates of 5-Iodotubercidin and Histone H3 Peptide Targeting Protein Kinase Haspin.

Structural analysis of ARC-type inhibitor (ARC-1034) binding to protein kinase A catalytic subunit and rational design of bisubstrate analogue inhibitors of basophilic protein kinases

Synthesis of potential purinoceptor antagonists: application of P1-tBU phosphazene base for alkylation of adenine in solution and on solid phase

Targeting Plasmodium falciparum protein kinases with adenosine analogue-oligoarginine conjugates

Time-gated luminescence microscopy with responsive nonmetal probes for mapping activity of protein kinases in living cells