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List of works by Benoit Crousse

(19)F NMR monitoring of the eukaryotic 20S proteasome chymotrypsin-like activity: an investigative tool for studying allosteric regulation

scientific article published on 01 July 2014

A one-pot synthesis of 3-trifluoromethyl-2-isoxazolines from trifluoromethyl aldoxime.

scientific article published on 7 November 2013

Access to novel amino trifluoromethyl cyclopropane carboxylic acid derivatives

Access to novel functionalized trifluoromethyl β-lactams by ring expansion of aziridines

Aminocyclopropanes as precursors of endoperoxides with antimalarial activity ⬇️

scientific article published on October 11, 2010

Analogues of key precursors of aspartyl protease inhibitors: synthesis of trifluoromethyl amino epoxides

scientific article published in January 2005

Benefits of a Dual Chemical and Physical Activation: Direct aza-Michael Addition of Anilines Promoted by Solvent Effect under High Pressure

article

Bisulfate Salt-Catalyzed Friedel-Crafts Benzylation of Arenes with Benzylic Alcohols

scientific article published on 07 November 2018

Carbonylhydrazide-based molecular tongs inhibit wild-type and mutated HIV-1 protease dimerization

scientific article published on 31 July 2012

Designed Glycopeptidomimetics Disrupt Protein-Protein Interactions Mediating Amyloid β-Peptide Aggregation and Restore Neuroblastoma Cell Viability.

scientific article published on 20 January 2016

Electrophilic amination of fluoroalkyl groups on azodicarboxylate derivatives.

scientific article published on 16 January 2015

Facile ring opening of oxiranes with aromatic amines in fluoro alcohols

scientific article published on 01 October 2000

First synthesis of 10 alpha-(trifluoromethyl)deoxoartemisinin

scientific article published on 01 March 2002

Fluorinated Alcohols: A New Medium for Selective and Clean Reaction

Fluoro artemisinins: difluoromethylene ketones

scientific article published in November 2001

Fluoroartemisinin: trifluoromethyl analogues of artemether and artesunate.

scientific article published in May 2004

Fluorous 4-N,N-dimethylaminopyridine (DMAP) salts as simple recyclable acylation catalysts

scientific article published in February 2010

Fluorous tagging of DABCO through halogen bonding: recyclable catalyst for the Morita-Baylis-Hillman reaction

scientific article published on 15 April 2011

In vitro antileishmanial activity of fluoro-artemisinin derivatives against Leishmania donovani

scientific article

Influence of the structure of polyfluorinated alcohols on Brønsted acidity/hydrogen-bond donor ability and consequences on the promoter effect

scientific article published on 18 January 2011

Intramolecular Pd-catalyzed carbocyclization, Heck reactions, and aryl-radical cyclizations with planar chiral arene tricarbonyl chromium complexes

scientific article

N-Difluoromethyl-triazole as a constrained scaffold in peptidomimetics

scientific article published on 01 May 2017

Non Lewis acid catalysed epoxide ring opening with amino acid esters.

scientific article published on 26 March 2009

Nonmetal catalyzed insertion reactions of diazocarbonyls to acid derivatives in fluorinated alcohols

scientific article published on 19 January 2011

Novel [1,2]- and [2,3]-Wittig rearrangements of alpha-benzyloxy beta-CF(3)-beta-lactam enolates

scientific article published on 01 August 2001

Orally active antimalarials: hydrolytically stable derivatives of 10-trifluoromethyl anhydrodihydroartemisinin

scientific article published in March 2004

Preparation of 10-trifluoromethyl artemether and artesunate. Influence of hexafluoropropan-2-ol on substitution reaction

scientific article

Reactivity of carbon dioxide in hydrofluoroethers: a facile access to cyclic carbonates

scientific article published in July 2015

Regioselective Halogenation of Arenes and Heterocycles in Hexafluoroisopropanol

scientific article

S(N)/S(N)' competition: selective access to new 10-fluoro artemisinins.

scientific article

Solubility switch of gold nanoparticles through hydrogen bond association

scientific article

Solvent-promoted and -controlled aza-Michael reaction with aromatic amines.

scientific article published in August 2009

Stereoselective Barbier-type allylation reaction of trifluoromethyl aldimines

scientific article published in August 2003

Structure-activity relationships of sugar-based peptidomimetics as modulators of amyloid β-peptide early oligomerization and fibrillization

scientific article published on 10 September 2014

Synthesis of 2-CF(3)-tetrahydroquinoline and quinoline derivatives from CF(3)-N-aryl-aldimine

scientific article published on 01 August 2000

Synthesis of substituted 8-aminoquinolines and phenanthrolines through a Povarov approach

scientific article published on 18 October 2010

The fluorous effect in biomolecular applications ⬇️

scientific article published on June 20, 2011

The use of 4,4,4-trifluorothreonine to stabilize extended peptide structures and mimic β-strands.

scientific article published on 21 December 2017

Trifluoromethyl nitrones: from fluoral to optically active hydroxylamines

scientific article published on 11 May 2010

α- and β-hydrazino acid-based pseudopeptides inhibit the chymotrypsin-like activity of the eukaryotic 20S proteasome.

scientific article

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