List of works - Gerd K. Wagner

2'-deoxy cyclic adenosine 5'-diphosphate ribose derivatives: importance of the 2'-hydroxyl motif for the antagonistic activity of 8-substituted cADPR derivatives

scientific article

5-Phenyluridine trihydrate

scientific article published on 12 January 2008

A facile two-step synthesis of 8-arylated guanosine mono- and triphosphates (8-aryl GXPs)

scientific article published on 13 November 2006

A fast synthetic route to GDP-sugars modified at the nucleobase

scientific article

A novel fluorescent probe for NAD-consuming enzymes

scientific article published on 31 October 2011

A novel fluorescent probe for retaining galactosyltransferases

scientific article published in July 2010

A survey of chemical methods for sugar-nucleotide synthesis.

scientific article published on 27 July 2009

Base-modified Donor Analogues Reveal Novel Dynamic Features of a Glycosyltransferase

scientific article

Base-modified NAD and AMP derivatives and their activity against bacterial DNA ligases.

scientific article

CD38 Structure-Based Inhibitor Design Using the N1-Cyclic Inosine 5'-Diphosphate Ribose Template

scientific article

Cellular effects and metabolic stability of N1-cyclic inosine diphosphoribose and its derivatives

scientific article

Conjugation to 4-aminoquinoline improves the anti-trypanosomal activity of Deferiprone-type iron chelators

scientific article published on 27 November 2012

Development of fluorescent aryltryptophans by Pd mediated cross-coupling of unprotected halotryptophans in water

scientific article published on 27 August 2008

Enzymatic synthesis of nucleobase-modified UDP-sugars: scope and limitations

scientific article published on 31 December 2014

Exploring the role of the 5-substituent for the intrinsic fluorescence of 5-aryl and 5-heteroaryl uracil nucleotides: a systematic study

scientific article

From imidazoles to pyrimidines: new inhibitors of cytokine release

scientific article published in June 2002

Glycosyltransferases and their Assays ⬇️

scientific article published on September 24, 2010

Identification of non-substrate-like glycosyltransferase inhibitors from library screening: pitfalls & hits

scientific article published on 29 November 2017

Identification of regioisomers in a series of N-substituted pyridin-4-yl imidazole derivatives by regiospecific synthesis, GC/MS, and 1H NMR.

scientific article published in May 2003

Imidazole inhibitors of cytokine release: probing substituents in the 2 position.

scientific article published in October 2002

Inhibition of galactosyltransferases by a novel class of donor analogues

scientific article published on 22 February 2012

New approaches to the treatment of inflammatory disorders small molecule inhibitors of p38 MAP kinase.

scientific article

Novel UDP-GalNAc Derivative Structures Provide Insight into the Donor Specificity of Human Blood Group Glycosyltransferase.

scientific article

Novel derivatives of UDP-glucose: concise synthesis and fluorescent properties

scientific article published on 18 June 2008

Novel substituted pyridinyl imidazoles as potent anticytokine agents with low activity against hepatic cytochrome P450 enzymes

scientific article

One-step synthesis of novel glycosyltransferase inhibitors

scientific article published on 01 December 2012

Ones, thiones, and N-oxides: an exercise in imidazole chemistry

scientific article published in July 2002

Optimised chemical synthesis of 5-substituted UDP-sugars and their evaluation as glycosyltransferase inhibitors

scientific article published on 23 October 2012

Profiling of <i>Haemophilus influenzae</i> strain R2866 with carbohydrate-based covalent probes

scientific article published on 23 December 2020

Rapid synthetic route toward structurally modified derivatives of cyclic adenosine 5'-diphosphate ribose

scientific article published in June 2005

Rationally designed squaryldiamides – a novel class of sugar-nucleotide mimics?

scientific article published on 07 June 2010

Small molecular anti-cytokine agents.

scientific article

Structural determinants for N1/N7 cyclization of nicotinamide hypoxanthine 5'-dinucleotide (NHD+) derivatives by ADP-ribosyl cyclase from aplysia californica: Ca2+-mobilizing activity of 8-substituted cyclic inosine 5'-diphosphoribose analogues in T

scientific article published on 01 August 2006

Studies on the anti-inflammatory activity of phytopharmaceuticals prepared from Arnica flowers

scientific article

The first C-glycosidic analogue of a novel galactosyltransferase inhibitor.

scientific article published on 26 January 2011

Trypanosoma brucei: chemical evidence that cathepsin L is essential for survival and a relevant drug target

scientific article

Two-Step Synthesis of Novel, Bioactive Derivatives of the Ubiquitous Cofactor Nicotinamide Adenine Dinucleotide (NAD)

scientific article published on 29 April 2011

Uncharged nucleoside inhibitors of β-1,4-galactosyltransferase with activity in cells

scientific article published on 16 February 2016

List of works by Gerd K. Wagner

2'-deoxy cyclic adenosine 5'-diphosphate ribose derivatives: importance of the 2'-hydroxyl motif for the antagonistic activity of 8-substituted cADPR derivatives

5-Phenyluridine trihydrate

A facile two-step synthesis of 8-arylated guanosine mono- and triphosphates (8-aryl GXPs)

A fast synthetic route to GDP-sugars modified at the nucleobase

A novel fluorescent probe for NAD-consuming enzymes

A novel fluorescent probe for retaining galactosyltransferases

A survey of chemical methods for sugar-nucleotide synthesis.

Base-modified Donor Analogues Reveal Novel Dynamic Features of a Glycosyltransferase

Base-modified NAD and AMP derivatives and their activity against bacterial DNA ligases.

CD38 Structure-Based Inhibitor Design Using the N1-Cyclic Inosine 5'-Diphosphate Ribose Template

Cellular effects and metabolic stability of N1-cyclic inosine diphosphoribose and its derivatives

Conjugation to 4-aminoquinoline improves the anti-trypanosomal activity of Deferiprone-type iron chelators

Development of fluorescent aryltryptophans by Pd mediated cross-coupling of unprotected halotryptophans in water

Enzymatic synthesis of nucleobase-modified UDP-sugars: scope and limitations

Exploring the role of the 5-substituent for the intrinsic fluorescence of 5-aryl and 5-heteroaryl uracil nucleotides: a systematic study

From imidazoles to pyrimidines: new inhibitors of cytokine release

Glycosyltransferases and their Assays ⬇️

Identification of non-substrate-like glycosyltransferase inhibitors from library screening: pitfalls & hits

Identification of regioisomers in a series of N-substituted pyridin-4-yl imidazole derivatives by regiospecific synthesis, GC/MS, and 1H NMR.

Imidazole inhibitors of cytokine release: probing substituents in the 2 position.

Inhibition of galactosyltransferases by a novel class of donor analogues

New approaches to the treatment of inflammatory disorders small molecule inhibitors of p38 MAP kinase.

Novel UDP-GalNAc Derivative Structures Provide Insight into the Donor Specificity of Human Blood Group Glycosyltransferase.

Novel derivatives of UDP-glucose: concise synthesis and fluorescent properties

Novel substituted pyridinyl imidazoles as potent anticytokine agents with low activity against hepatic cytochrome P450 enzymes

One-step synthesis of novel glycosyltransferase inhibitors

Ones, thiones, and N-oxides: an exercise in imidazole chemistry

Optimised chemical synthesis of 5-substituted UDP-sugars and their evaluation as glycosyltransferase inhibitors

Profiling of <i>Haemophilus influenzae</i> strain R2866 with carbohydrate-based covalent probes

Rapid synthetic route toward structurally modified derivatives of cyclic adenosine 5'-diphosphate ribose

Rationally designed squaryldiamides – a novel class of sugar-nucleotide mimics?

Small molecular anti-cytokine agents.

Structural determinants for N1/N7 cyclization of nicotinamide hypoxanthine 5'-dinucleotide (NHD+) derivatives by ADP-ribosyl cyclase from aplysia californica: Ca2+-mobilizing activity of 8-substituted cyclic inosine 5'-diphosphoribose analogues in T

Studies on the anti-inflammatory activity of phytopharmaceuticals prepared from Arnica flowers

The first C-glycosidic analogue of a novel galactosyltransferase inhibitor.

Trypanosoma brucei: chemical evidence that cathepsin L is essential for survival and a relevant drug target

Two-Step Synthesis of Novel, Bioactive Derivatives of the Ubiquitous Cofactor Nicotinamide Adenine Dinucleotide (NAD)

Uncharged nucleoside inhibitors of β-1,4-galactosyltransferase with activity in cells