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List of works by Oleksandr O. Grygorenko

(Chlorosulfonyl)benzenesulfonyl fluorides - versatile building blocks for combinatorial chemistry. Design, synthesis and evaluation of a covalent inhibitor library

article

1-Alkyl-5-((di)alkylamino) tetrazoles: building blocks for peptide surrogates

scientific article published on 30 December 2011

3-((Hetera)cyclobutyl)azetidines, "Stretched" Analogues of Piperidine, Piperazine, and Morpholine: Advanced Building Blocks for Drug Discovery

scientific article published on 08 January 2019

3-Benzyl-3-azabicyclo[3.1.1]heptan-6-one: a promising building block for medicinal chemistry.

scientific article published on October 2010

3-haloquinolines by Friedländer reaction of α-haloketones

scientific article published on 15 June 2011

4-Fluoro-2,4-methanoproline

scientific article published in December 2009

A conformationally restricted GABA analogue based on octahydro-1H-cyclopenta[b]pyridine scaffold

scientific article published on 04 October 2018

An Old Story in the Parallel Synthesis World: An Approach to Hydantoin Libraries

scientific article

An entry into hexahydro-2H-thieno[2,3-c]pyrrole 1,1-dioxide derivatives.

scientific article

Approach to the library of 3-hydroxy-1,5-dihydro-2H-pyrrol-2-ones through a three-component condensation.

scientific article

Approach to the library of fused pyridine-4-carboxylic acids by Combes-type reaction of acyl pyruvates and electron-rich amino heterocycles.

scientific article

Beyond the Five and Six: Evaluation of Seven-Membered Cyclic Anhydrides in the Castagnoli-Cushman Reaction

scientific article published on 21 December 2016

Bicyclic Conformationally Restricted Diamines

scientific article published on 28 June 2011

Building the Housane: Diastereoselective Synthesis and Characterization of Bicyclo[2.1.0]pentane Carboxylic Acids

scientific article published on 06 January 2020

Conformational behaviour of peptides containing a 2-pyrrolidinemethanesulfonic acid (2PyMS) residue.

scientific article

Conformationally restricted nonchiral pipecolic acid analogues

scientific article published on 01 August 2009

Cyclobutane-derived diamines: synthesis and molecular structure

scientific article published on September 2010

Far Away from Flatland. Synthesis and Molecular Structure of Dihetera[3.3.n]propellanes and Trihetera[3.3.n]propellanes: Advanced Analogues of Morpholine/Piperazine

scientific article published on 26 September 2019

Focused enumeration and assessing the structural diversity of scaffold libraries: conformationally restricted bicyclic secondary diamines.

scientific article

Impact of Fluoroalkyl Substituents on the Physicochemical Properties of Saturated Heterocyclic Amines

scientific article published in 2022

Last of the gem-Difluorocycloalkanes: Synthesis and Characterization of 2,2-Difluorocyclobutyl-Substituted Building Blocks

scientific article published on 24 April 2019

One-Pot Parallel Synthesis of 5-(Dialkylamino)tetrazoles

scientific article published on 29 August 2019

Photochemical Synthesis of 3-Azabicyclo[3.2.0]heptanes: Advanced Building Blocks for Drug Discovery.

scientific article published on 16 August 2017

Photochemical [2 + 2] Cycloaddition of Alkenyl Boronic Derivatives: An Entry into 3-Azabicyclo[3.2.0]heptane Scaffold

scientific article published on 13 April 2020

Regioselective Synthesis of Functionalized 3- or 5-Fluoroalkyl Isoxazoles and Pyrazoles from Fluoroalkyl Ynones and Binucleophiles

scientific article published on 08 November 2019

Regioselective synthesis of isoxazole and 1,2,4-oxadiazole-derived phosphonates via [3 + 2] cycloaddition

scientific article published on 01 December 2018

SAR by Space: Enriching Hit Sets from the Chemical Space

scientific article published on 26 August 2019

Scalable Synthesis of Biologically Relevant Spirocyclic Pyrrolidines

scientific article published on 24 April 2019

Straightforward hit identification approach in fragment-based discovery of bromodomain-containing protein 4 (BRD4) inhibitors

scientific article published on 09 May 2018

Sulfonimidamides and Imidosulfuric Diamides: Compounds from an Underexplored Part of Biologically Relevant Chemical Space

scientific article published on 01 April 2019

Synthesis and Structural Analysis of Angular Monoprotected Diamines Based on Spiro[3.3]heptane Scaffold

scientific article published on 25 March 2015

Synthesis of 2-azaspiro[3.3]heptane-derived amino acids: ornitine and GABA analogues

scientific article published on 27 January 2010

Synthesis of 3‐Borylated Pyrrolidines by 1,3‐Dipolar Cycloaddition of Alkenyl Boronates and Azomethine Ylide

scientific article published in 2022

Synthesis of 5-(Fluoroalkyl)isoxazole Building Blocks by Regioselective Reactions of Functionalized Halogenoximes

scientific article published on 30 October 2019

The Symbiotic Relationship Between Drug Discovery and Organic Chemistry

scientific article published on 30 October 2019

The Synthesis and Acid-base Properties of α-(Fluoromethyl)- and α-(Difluoromethyl)-substituted Cyclobutane Building Blocks

The Ukrainian Factor in Early-Stage Drug Discovery in the Context of Russian Invasion: The Case of Enamine Ltd

scientific article published in 2022

The catalytic asymmetric α-benzylation of aldehydes.

scientific article

Toward lead-oriented synthesis: one-pot version of Castagnoli condensation with nonactivated alicyclic anhydrides

scientific article published on 06 February 2014

[2+2]-Photocycloaddition of N-Benzylmaleimide to Alkenes As an Approach to Functional 3-Azabicyclo[3.2.0]heptanes

scientific article published on 12 March 2018

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