List of works - Andrey P. Antonchick

2,3-Epoxybrassinosteroids are intermediates in the biosynthesis of castasterone in seedlings of Secale cereale

scientific article published in January 2005

A Highly Enantioselective Brønsted Acid Catalyzed Reaction Cascade

scientific article published on 01 January 2008

A Metal-Free Oxidative Dehydrogenative Diels-Alder Reaction for Selective Functionalization of Alkylbenzenes

scientific article

A framework for identification of actionable cancer genome dependencies in small cell lung cancer

scientific article

A highly enantioselective Brønsted acid catalyzed cascade reaction: organocatalytic transfer hydrogenation of quinolines and their application in the synthesis of alkaloids

scientific article (publication date: 26 May 2006)

Aerobic, Metal-Free, and Catalytic Dehydrogenative Coupling of Heterocycles: En Route to Hedgehog Signaling Pathway Inhibitors

scientific article published on 16 March 2018

Asymmetric Brønsted Acid Catalysis: Catalytic Enantioselective Synthesis of Highly Biologically Active Dihydroquinazolinones

scientific article published on 01 January 2009

Asymmetric synthesis of indolines by catalytic enantioselective reduction of 3H-indoles

scientific article published on October 2010

Biology-Oriented Synthesis of 3,3-Spiro(2-tetrahydrofuranyl)oxindoles

Biology-oriented synthesis of benzopyrano[3,4- c ]pyrrolidines

scientific article published on 04 March 2015

Biosynthesis of 2,3-epoxybrassinosteroids in seedlings of Secale cereale

scientific article published in August 2003

Brønsted-Acid-Catalyzed Activation of Nitroalkanes: A Direct Enantioselective Aza-Henry Reaction

scientific article published on 08 April 2008

Cascade Multicomponent Synthesis of Indoles, Pyrazoles, and Pyridazinones by Functionalization of Alkenes

scientific article published on 06 October 2014

Catalytic Aerobic Oxidation and Tandem Enantioselective Cycloaddition in Cascade Multicomponent Synthesis

scientific article published on 11 February 2015

Catalytic Asymmetric Aminoallylation of Aldehydes: A Catalytic Enantioselective Aza-Cope Rearrangement

scientific article published on 01 January 2008

Catalytic Enantioselective Synthesis of a Pyrrolizidine-Alkaloid-Inspired Compound Collection with Antiplasmodial Activity

scientific article published on 20 February 2018

Catalytic Selective Metal-Free Cross-Coupling of Heteroaromatic N-Oxides with Organosilanes

scientific article published on 23 April 2019

Catalytic Transfer Hydrogenation Using Biomass as Hydrogen Source

scientific article published on 22 August 2018

Catalytic asymmetric exo-selective [6+3] cycloaddition of iminoesters with fulvenes.

scientific article published in September 2013

Catalytic enantioselective 1,3-dipolar cycloadditions of azomethine ylides for biology-oriented synthesis

scientific article

Catalytic enantioselective synthesis of functionalized tropanes reveals novel inhibitors of hedgehog signaling.

scientific article

Chiral Brønsted Acids in the Catalytic Asymmetric Nazarov Cyclization—The First Enantioselective Organocatalytic Electrocyclic Reaction

scientific article published on 01 January 2007

Copper(I)-Catalyzed Radical Addition of Acetophenones to Alkynes in Furan Synthesis

scientific article published on 17 August 2015

Copper-Catalyzed (2+1) Annulation of Acetophenones with Maleimides: Direct Synthesis of Cyclopropanes

scientific article published on 10 June 2015

Direct Selective Oxidative Cross-Coupling of Simple Alkanes with Heteroarenes

scientific article published on 31 January 2013

Direct enantioselective access to 4-substituted tetrahydroquinolines by catalytic asymmetric transfer hydrogenation of quinolines

scientific article published on 12 August 2011

Discovery of inhibitors of the Wnt and Hedgehog signaling pathways through the catalytic enantioselective synthesis of an iridoid-inspired compound collection

scientific article published on 2 October 2013

Dual Catalysis: A Combined Enantioselective Brønsted Acid and Metal-Catalyzed Reaction—Metal Catalysis with Chiral Counterions

scientific article published on 01 January 2007

Enantiodivergent Combination of Natural Product Scaffolds Enabled by Catalytic Enantioselective Cycloaddition

scientific article published on 19 May 2016

Enantioselective Formal C(sp3 )−H Bond Activation in the Synthesis of Bioactive Spiropyrazolone Derivatives

scientific article published on 04 December 2018

Enantioselective Synthesis of Five-Membered-Ring Atropisomers with a Chiral Rh(III) Complex

scientific article published on 13 November 2020

Enantioselective Synthesis of the Spiro-Tropanyl Oxindole Scaffold Through Bimetallic Relay Catalysis

scientific article published on 8 February 2018

General Enantioselective C-H Activation with Efficiently Tunable Cyclopentadienyl Ligands

scientific article

Highly Enantioselective Catalytic Synthesis of Neurite Growth-Promoting Secoyohimbanes

scientific article published on 01 April 2013

Highly Enantioselective Catalytic [6+3] Cycloadditions of Azomethine Ylides

scientific article published on 14 August 2012

Highly enantioselective synthesis and cellular evaluation of spirooxindoles inspired by natural products

scientific article published on 11 July 2010

Hypervalent Iodine(III) in Direct Carbon–Hydrogen Bond Functionalization

Hypervalent Iodine(III) in Direct Oxidative Amination of Arenes with Heteroaromatic Amines

scientific article published on 02 September 2015

Hypervalent Iodine-Mediated Selective Oxidative Functionalization of (Thio)chromones with Alkanes

scientific article published on 06 March 2014

Iridium(iii)-catalyzed regioselective C7-sulfonamidation of indoles.

scientific article published on 13 May 2016

Metal-Free Annulation of Arenes with 2-Aminopyridine Derivatives: The Methyl Group as a Traceless Non-Chelating Directing Group

scientific article published on 18 June 2014

Metal-Free Brønsted Acid Catalyzed Transfer Hydrogenation - New Organocatalytic Reduction of Quinolines

Metal-Free Cross-Dehydrogenative Coupling of Heterocycles with Aldehydes

scientific article published on 10 January 2013

Metal-Free C–O Bond Functionalization: Catalytic Intramolecular and Intermolecular Benzylation of Arenes

scientific article published on 14 June 2018

Metal-Free Electrocyclization at Ambient Temperature: Synthesis of 1-Arylcarbazoles

Metal-Free Oxidative C-C Bond Formation through C-H Bond Functionalization.

scientific article

Metal-Free Oxidative C-H Bond Amination at Ambient Temperature

Metal-Free Radical Azidoarylation of Alkenes: Rapid Access to Oxindoles by Cascade CN and CC Bond-Forming Reactions

scientific article published on 20 June 2013

Metal-free direct oxidative intermolecular diarylation of anilides at ambient temperature assisted by cascade selective formation of C–C and C–N bonds

scientific article published on 13 February 2012

Natural product fragment combination to performance-diverse pseudo-natural products

scientific article published on 25 March 2021

Organocatalytic Oxidative Annulation of Benzamide Derivatives with Alkynes

scientific article published on 21 May 2014

Organocatalytic enantioselective reduction of pyridines

scientific article

Organocatalytic, Oxidative, Intramolecular CH Bond Amination and Metal-free Cross-Amination of Unactivated Arenes at Ambient Temperature

scientific article published on 26 July 2011

Organocatalytic, oxidative, intermolecular amination and hydrazination of simple arenes at ambient temperature.

scientific article published on 16 October 2012

Oxidative Heterocycle Formation Using Hypervalent Iodine(III) Reagents

scientific article published on 01 January 2016

Oxidative regioselective amination of chromones exposes potent inhibitors of the hedgehog signaling pathway

scientific article

Palladium-Catalyzed Double CH Activation Directed by Sulfoxides in the Synthesis of Dibenzothiophenes

scientific article published on 19 April 2011

Phosphine-catalyzed dearomatizing [3+2] annulations of isoquinolinium methylides with allenes.

scientific article published in January 2015

Preparation of (25R)- and (25S)-26-functionalized steroids as tools for biosynthetic studies of cholic acids

scientific article published on 26 March 2005

Programmable enantioselective one-pot synthesis of molecules with eight stereocenters

Regioselective Metal-Free Cross-Coupling of Quinoline N-Oxides with Boronic Acids

scientific article published on 11 June 2015

Regioselective annulation of nitrosopyridine with alkynes: straightforward synthesis of N-oxide-imidazopyridines

scientific article published on 01 April 2015

Remarkably Low Catalyst Loading in Brønsted Acid Catalyzed Transfer Hydrogenations: Enantioselective Reduction of Benzoxazines, Benzothiazines, and Benzoxazinones

scientific article published on 01 October 2006

Rhodium(II)-Catalyzed Enantioselective Synthesis of Troponoids

scientific article published on 08 May 2015

Rhodium(III)-Catalyzed Direct Oxidative Cross Coupling at the C5 Position of Chromones with Alkenes

scientific article published on 28 November 2012

Rhodium(III)-Catalyzed Direct Regioselective Synthesis of 7-Substituted Indoles

scientific article published on 28 October 2013

Selective, Catalytic, and Metal-Free Coupling of Electron-Rich Phenols and Anilides Using Molecular Oxygen as Terminal Oxidant

scientific article published on 21 June 2018

Sustainable, Oxidative, and Metal-Free Annulation

scientific article published on 31 May 2017

Synthesis of C24-functionalized hydroxysterols

scientific article

Synthesis of [26,27-2H6]brassinosteroids from 23,24-bisnorcholenic acid methyl ester

scientific article published in September 2004

Synthesis of [26-2H(3)]brassinosteroids

scientific article

Synthesis of hexadeuterated 23-dehydroxybrassinosteroids

scientific article published in December 2002

Synthesis of the B-seco limonoid core scaffold

scientific article published on 16 January 2014

Synthesis of the B-seco limonoid scaffold

scientific article published on 09 May 2011

The Pictet-Spengler reaction in nature and in organic chemistry

scientific article

The therapeutic potential of phosphatase inhibitors

scientific article published on 04 May 2009

Trienamine catalyzed asymmetric synthesis and biological investigation of a cytochalasin B-inspired compound collection

scientific article

[1+1+1] Cyclotrimerization for the Synthesis of Cyclopropanes

scientific article published on 21 March 2016

[3,3]-Claisen rearrangements in 24alpha-methyl steroid synthesis. Application to campesterol, crinosterol, and Delta25-crinosterol side chain construction

scientific article

List of works by Andrey P. Antonchick

2,3-Epoxybrassinosteroids are intermediates in the biosynthesis of castasterone in seedlings of Secale cereale

A Highly Enantioselective Brønsted Acid Catalyzed Reaction Cascade

A Metal-Free Oxidative Dehydrogenative Diels-Alder Reaction for Selective Functionalization of Alkylbenzenes

A framework for identification of actionable cancer genome dependencies in small cell lung cancer

A highly enantioselective Brønsted acid catalyzed cascade reaction: organocatalytic transfer hydrogenation of quinolines and their application in the synthesis of alkaloids

Aerobic, Metal-Free, and Catalytic Dehydrogenative Coupling of Heterocycles: En Route to Hedgehog Signaling Pathway Inhibitors

Asymmetric Brønsted Acid Catalysis: Catalytic Enantioselective Synthesis of Highly Biologically Active Dihydroquinazolinones

Asymmetric synthesis of indolines by catalytic enantioselective reduction of 3H-indoles

Biology-Oriented Synthesis of 3,3-Spiro(2-tetrahydrofuranyl)oxindoles

Biology-oriented synthesis of benzopyrano[3,4- c ]pyrrolidines

Biosynthesis of 2,3-epoxybrassinosteroids in seedlings of Secale cereale

Brønsted-Acid-Catalyzed Activation of Nitroalkanes: A Direct Enantioselective Aza-Henry Reaction

Cascade Multicomponent Synthesis of Indoles, Pyrazoles, and Pyridazinones by Functionalization of Alkenes

Catalytic Aerobic Oxidation and Tandem Enantioselective Cycloaddition in Cascade Multicomponent Synthesis

Catalytic Asymmetric Aminoallylation of Aldehydes: A Catalytic Enantioselective Aza-Cope Rearrangement

Catalytic Enantioselective Synthesis of a Pyrrolizidine-Alkaloid-Inspired Compound Collection with Antiplasmodial Activity

Catalytic Selective Metal-Free Cross-Coupling of Heteroaromatic N-Oxides with Organosilanes

Catalytic Transfer Hydrogenation Using Biomass as Hydrogen Source

Catalytic asymmetric exo-selective [6+3] cycloaddition of iminoesters with fulvenes.

Catalytic enantioselective 1,3-dipolar cycloadditions of azomethine ylides for biology-oriented synthesis

Catalytic enantioselective synthesis of functionalized tropanes reveals novel inhibitors of hedgehog signaling.

Chiral Brønsted Acids in the Catalytic Asymmetric Nazarov Cyclization—The First Enantioselective Organocatalytic Electrocyclic Reaction

Copper(I)-Catalyzed Radical Addition of Acetophenones to Alkynes in Furan Synthesis

Copper-Catalyzed (2+1) Annulation of Acetophenones with Maleimides: Direct Synthesis of Cyclopropanes

Direct Selective Oxidative Cross-Coupling of Simple Alkanes with Heteroarenes

Direct enantioselective access to 4-substituted tetrahydroquinolines by catalytic asymmetric transfer hydrogenation of quinolines

Discovery of inhibitors of the Wnt and Hedgehog signaling pathways through the catalytic enantioselective synthesis of an iridoid-inspired compound collection

Dual Catalysis: A Combined Enantioselective Brønsted Acid and Metal-Catalyzed Reaction—Metal Catalysis with Chiral Counterions

Enantiodivergent Combination of Natural Product Scaffolds Enabled by Catalytic Enantioselective Cycloaddition

Enantioselective Formal C(sp3 )−H Bond Activation in the Synthesis of Bioactive Spiropyrazolone Derivatives

Enantioselective Synthesis of Five-Membered-Ring Atropisomers with a Chiral Rh(III) Complex

Enantioselective Synthesis of the Spiro-Tropanyl Oxindole Scaffold Through Bimetallic Relay Catalysis

General Enantioselective C-H Activation with Efficiently Tunable Cyclopentadienyl Ligands

Highly Enantioselective Catalytic Synthesis of Neurite Growth-Promoting Secoyohimbanes

Highly Enantioselective Catalytic [6+3] Cycloadditions of Azomethine Ylides

Highly enantioselective synthesis and cellular evaluation of spirooxindoles inspired by natural products

Hypervalent Iodine(III) in Direct Carbon–Hydrogen Bond Functionalization

Hypervalent Iodine(III) in Direct Oxidative Amination of Arenes with Heteroaromatic Amines

Hypervalent Iodine-Mediated Selective Oxidative Functionalization of (Thio)chromones with Alkanes

Iridium(iii)-catalyzed regioselective C7-sulfonamidation of indoles.

Metal-Free Annulation of Arenes with 2-Aminopyridine Derivatives: The Methyl Group as a Traceless Non-Chelating Directing Group

Metal-Free Brønsted Acid Catalyzed Transfer Hydrogenation - New Organocatalytic Reduction of Quinolines

Metal-Free Cross-Dehydrogenative Coupling of Heterocycles with Aldehydes

Metal-Free C–O Bond Functionalization: Catalytic Intramolecular and Intermolecular Benzylation of Arenes

Metal-Free Electrocyclization at Ambient Temperature: Synthesis of 1-Arylcarbazoles

Metal-Free Oxidative C-C Bond Formation through C-H Bond Functionalization.

Metal-Free Oxidative C-H Bond Amination at Ambient Temperature

Metal-Free Radical Azidoarylation of Alkenes: Rapid Access to Oxindoles by Cascade CN and CC Bond-Forming Reactions

Metal-free direct oxidative intermolecular diarylation of anilides at ambient temperature assisted by cascade selective formation of C–C and C–N bonds

Natural product fragment combination to performance-diverse pseudo-natural products

Organocatalytic Oxidative Annulation of Benzamide Derivatives with Alkynes

Organocatalytic enantioselective reduction of pyridines

Organocatalytic, Oxidative, Intramolecular CH Bond Amination and Metal-free Cross-Amination of Unactivated Arenes at Ambient Temperature

Organocatalytic, oxidative, intermolecular amination and hydrazination of simple arenes at ambient temperature.

Oxidative Heterocycle Formation Using Hypervalent Iodine(III) Reagents

Oxidative regioselective amination of chromones exposes potent inhibitors of the hedgehog signaling pathway

Palladium-Catalyzed Double CH Activation Directed by Sulfoxides in the Synthesis of Dibenzothiophenes

Phosphine-catalyzed dearomatizing [3+2] annulations of isoquinolinium methylides with allenes.

Preparation of (25R)- and (25S)-26-functionalized steroids as tools for biosynthetic studies of cholic acids

Programmable enantioselective one-pot synthesis of molecules with eight stereocenters

Regioselective Metal-Free Cross-Coupling of Quinoline N-Oxides with Boronic Acids

Regioselective annulation of nitrosopyridine with alkynes: straightforward synthesis of N-oxide-imidazopyridines

Remarkably Low Catalyst Loading in Brønsted Acid Catalyzed Transfer Hydrogenations: Enantioselective Reduction of Benzoxazines, Benzothiazines, and Benzoxazinones

Rhodium(II)-Catalyzed Enantioselective Synthesis of Troponoids

Rhodium(III)-Catalyzed Direct Oxidative Cross Coupling at the C5 Position of Chromones with Alkenes

Rhodium(III)-Catalyzed Direct Regioselective Synthesis of 7-Substituted Indoles

Selective, Catalytic, and Metal-Free Coupling of Electron-Rich Phenols and Anilides Using Molecular Oxygen as Terminal Oxidant

Sustainable, Oxidative, and Metal-Free Annulation

Synthesis of C24-functionalized hydroxysterols

Synthesis of [26,27-2H6]brassinosteroids from 23,24-bisnorcholenic acid methyl ester

Synthesis of [26-2H(3)]brassinosteroids

Synthesis of hexadeuterated 23-dehydroxybrassinosteroids

Synthesis of the B-seco limonoid core scaffold

Synthesis of the B-seco limonoid scaffold

The Pictet-Spengler reaction in nature and in organic chemistry

The therapeutic potential of phosphatase inhibitors

Trienamine catalyzed asymmetric synthesis and biological investigation of a cytochalasin B-inspired compound collection

[1+1+1] Cyclotrimerization for the Synthesis of Cyclopropanes

[3,3]-Claisen rearrangements in 24alpha-methyl steroid synthesis. Application to campesterol, crinosterol, and Delta25-crinosterol side chain construction