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List of works by Charles M. Heard

A Time-Kill Assay Study on the Synergistic Bactericidal Activity of Pomegranate Rind Extract and Zn (II) against Methicillin-Resistant Staphylococcus aureus (MRSA), Staphylococcus epidermidis, Escherichia coli, and Pseudomonas aeruginosa

scientific article published in 2021

A novel diffusion cell model for the in vitro assessment of transcutaneous breast cancer therapeutics: effect of permeants on MCF-7 cells cultured within the receptor compartment.

scientific article published on 2 April 2010

A novel ex vivo skin model for the assessment of the potential transcutaneous anti-inflammatory effect of topically applied Harpagophytum procumbens extract

scientific article published on 19 April 2009

A therapeutic dose of primaquine can be delivered across excised human skin from simple transdermal patches

scientific article published in October 1999

Binding of doxycycline to keratin, melanin and human epidermal tissue

scientific article published in March 2002

Binding of primaquine to epidermal membranes and keratin

scientific article published in May 2003

Delivery of atovaquone and proguanil across sublingual membranes, in vitro

scientific article published on 26 May 2011

Dermal and transcutaneous delivery of the major glycoside constituents of Harpagophytum procumbens (Devil's Claw) in vitro

scientific article published on 10 April 2008

Design, synthesis and in vitro degradation of a novel co-drug for the treatment of psoriasis.

scientific article published on 17 April 2013

Differential permeation of propranolol enantiomers across human skin in vitro from formulations containing an enantioselective excipient

scientific article

Discovery of Novel 2-Aniline-1,4-naphthoquinones as Potential New Drug Treatment for Leber's Hereditary Optic Neuropathy (LHON)

scientific article published on 12 November 2020

Distribution of esterase activity in porcine ear skin, and the effects of freezing and heat separation

scientific article published on 08 May 2012

Does solute stereochemistry influence percutaneous penetration?

scientific article published on 01 January 1995

Effect of the major glycosides of Harpagophytum procumbens (Devil's Claw) on epidermal cyclooxygenase-2 (COX-2) in vitro

scientific article published on 16 April 2008

Effects of membrane type and liquid/liquid phase boundary on in vitro release of ketoprofen from gel formulations

scientific article

Enantiomeric resolution of some 2-arylpropionic acids using L-(-)-serine-impregnated silica as stationary phase by thin layer chromatography

scientific article published in August 2003

Enhanced in vitro transdermal delivery of caffeine using a temperature- and pH-sensitive nanogel, poly(NIPAM-co-AAc).

scientific article published on 30 May 2013

Enhanced topical delivery and anti-inflammatory activity of methotrexate from an activated nanogel

scientific article published on 30 June 2010

Enhanced topical delivery and ex vivo anti-inflammatory activity from a betamethasone dipropionate formulation containing fish oil.

scientific article published on 31 July 2009

Estimation of the relative antiinflammatory efficacies of six commercial preparations of Harpagophytum procumbens (Devil's Claw).

scientific article published in March 2010

Film drying and complexation effects in the simultaneous skin permeation of ketoprofen and propylene glycol from simple gel formulations.

scientific article

In Vitro Topical Delivery of Chlorhexidine to the Cornea: Enhancement Using Drug-Loaded Contact Lenses and β-Cyclodextrin Complexation, and the Importance of Simulating Tear Irrigation

scientific article published on 20 March 2020

In vitro delivery of anti-breast cancer agents directly via the mammary papilla (nipple).

scientific article published on 16 December 2009

In vitro delivery of novel, highly potent anti-varicella zoster virus nucleoside analogues to their target site in the skin.

scientific article published on June 2004

In vitro dermal and transdermal delivery of doxycycline from ethanol/migliol 840 vehicles

scientific article published in November 1999

In vitro transcutaneous delivery of ketoprofen and essential polyunsaturated fatty acids from a fish oil vehicle incorporating 1,8-cineole

scientific article published in January 2005

In vitro transdermal delivery of caffeine, theobromine, theophylline and catechin from extract of Guarana, Paullinia Cupana

scientific article published on 04 April 2006

In vitro transdermal delivery of the major catechins and caffeine from extract of Camellia sinensis

scientific article published in September 2004

In vivo response of GsdmA3Dfl/+ mice to topically applied anti-psoriatic agents: effects on epidermal thickness, as determined by optical coherence tomography and H&E staining

scientific article published in March 2011

In-vitro transcutaneous delivery of ketoprofen and polyunsaturated fatty acids from a pluronic lecithin organogel vehicle containing fish oil

scientific article published on 01 July 2006

In-vitro transcutaneous delivery of tamoxifen and gamma-linolenic acid from borage oil containing ethanol and 1,8-cineole

scientific article published in November 2004

Inter- and intralaboratory variation of in vitro diffusion cell measurements: an international multicenter study using quasi-standardized methods and materials.

scientific article published in March 2005

Is there a role for topically delivered eicosapentaenoic acid in the treatment of psoriasis?

scientific article

Ketoprofen: release from, permeation across and rheology of simple gel formulations that simulate increasing dryness

scientific article

Nanogel particulates located within diffusion cell receptor phases following topical application demonstrates uptake into and migration across skin

scientific article published on 15 September 2010

Permeation of quinine across sublingual mucosa, in vitro

scientific article

Pharmaceutical applications for molecularly imprinted polymers

scientific article published on 01 February 2000

Potentiated virucidal activity of pomegranate rind extract (PRE) and punicalagin against Herpes simplex virus (HSV) when co-administered with zinc (II) ions, and antiviral activity of PRE against HSV and aciclovir-resistant HSV.

scientific article

Pre-treatment with Aloe vera juice does not enhance the in vitro permeation of ketoprofen across skin

scientific article published on 14 December 2009

Preferential pi-pi complexation between tamoxifen and borage oil/gamma linolenic acid: transcutaneous delivery and NMR spectral modulation

scientific article published in September 2005

Probing the permeation enhancement of mefenamic acid by ethanol across full-thickness skin, heat-separated epidermal membrane and heat-separated dermal membrane

scientific article published on 11 August 2007

Probing the skin permeation of eicosapentaenoic acid and ketoprofen 2. Comparative depth profiling and metabolism of eicosapentaenoic acid

scientific article published on 12 December 2006

Probing the skin permeation of fish oil/EPA and ketoprofen

scientific article published on 12 February 2007

Probing the skin permeation of fish oil/EPA and ketoprofen-3. Effects on epidermal COX-2 and LOX

scientific article published on 25 June 2007

Scope and limitations of the co-drug approach to topical drug delivery.

scientific article

Simultaneous permeation of tamoxifen and gamma linolenic acid across excised human skin. Further evidence of the permeation of solvated complexes.

scientific article

Skin penetration enhancement of mefenamic acid by ethanol and 1,8-cineole can be explained by the 'pull' effect

scientific article published on 16 May 2006

Skin permeation and ex vivo skin metabolism of O-acyl haloperidol ester prodrugs.

scientific article

Skin permeation enhancement potential of Aloe Vera and a proposed mechanism of action based upon size exclusion and pull effect

scientific article published in October 2006

Solvent content and macroviscosity effects on the in vitro transcutaneous delivery and skin distribution of ketoprofen from simple gel formulations.

scientific article published on 20 May 2005

Synthesis of haloperidol prodrugs and their hydrolysis by porcine liver esterase

scientific article

Targeted dermal delivery of highly potent anti-varicella zoster virus nucleoside analogues from saturated solutions and ethanolic oil-in-water creams

scientific article

The effects of betamethasone dipropionate and fish oil on HaCaT proliferation and apoptosis.

scientific article

The effects of topically applied polyNIPAM-based nanogels and their monomers on skin cyclooxygenase expression, ex vivo.

scientific article published on 9 January 2013

The in vitro delivery of NSAIDs across skin was in proportion to the delivery of essential fatty acids in the vehicle--evidence that solutes permeate skin associated with their solvation cages?

scientific article published in August 2003

Therapeutic and Cytotoxic Effects of the Novel Antipsoriasis Codrug, Naproxyl–Dithranol, on HaCaT Cells ⬇️

scientific article published on September 21, 2011

Thin layer chromatographic resolution of some 2-arylpropionic acid enantiomers using L-(-)-serine, L-(-)-threonine and a mixture of L-(-)-serine and L-(-)-threonine-impregnated silica gel as stationary phases.

scientific article

Topical Delivery of Retinyl Ascorbate Co-Drug

article

Topical delivery of a naproxen-dithranol co-drug: in vitro skin penetration, permeation, and staining

scientific article published on 25 September 2010

Topical delivery of retinyl ascorbate co-drug. 1. Synthesis, penetration into and permeation across human skin

scientific article

Topical delivery of retinyl ascorbate co-drug. 2. Comparative skin tissue and keratin binding studies

scientific article published in November 2004

Topical delivery of retinyl ascorbate. 3. Influence of follicle sealing and skin stretching

scientific article published on 19 November 2007

Topical delivery of retinyl ascorbate: 4. Comparative anti-oxidant activity towards DPPH.

scientific article published in May 2005

Topically applied KTTKS: a review ⬇️

scientific article published on 03 May 2011

Transdermal delivery enhancement of haloperidol from gel formulations by 1,8-cineole

scientific article published in June 2008

Triclosan: release from transdermal adhesive formulations and in vitro permeation across human epidermal membranes

scientific article published in March 2002

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