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List of works by Marius Hoener

A UGT2B10 splicing polymorphism common in african populations may greatly increase drug exposure

scientific article published on 12 December 2014

A functional NR4A nuclear receptor DNA-binding domain is required for organ development in Caenorhabditis elegans

scientific article

A new perspective for schizophrenia: TAAR1 agonists reveal antipsychotic- and antidepressant-like activity, improve cognition and control body weight.

scientific article published on 29 May 2012

A partial trace amine-associated receptor 1 agonist exhibits properties consistent with a methamphetamine substitution treatment

scientific article published on 19 May 2016

A renaissance in trace amines inspired by a novel GPCR family

scientific article

Acetylcholinesterase inhibitors rapidly activate Trk neurotrophin receptors in the mouse hippocampus

scientific article published on 30 July 2011

Activation of the trace amine-associated receptor 1 prevents relapse to cocaine seeking

scientific article

Activation of trace amine-associated receptor 1 attenuates schedule-induced polydipsia in rats

scientific article published on 24 October 2018

An automated system for the analysis of G protein-coupled receptor transmembrane binding pockets: alignment, receptor-based pharmacophores, and their application

scientific article published in September 2005

Are there differences between the secretion characteristics of NGF and BDNF? Implications for the modulatory role of neurotrophins in activity-dependent neuronal plasticity

scientific article

Brain-specific overexpression of trace amine-associated receptor 1 alters monoaminergic neurotransmission and decreases sensitivity to amphetamine

scientific article

Caenorhabditis elegans MPP+ model of Parkinson's disease for high-throughput drug screenings

scientific article

Cytochrome P450 enzymes contribute to the metabolism of LSD to nor-LSD and 2-oxo-3-hydroxy-LSD: Implications for clinical LSD use

scientific article published on 11 April 2019

Darkness reduces BDNF expression in the visual cortex and induces repressive chromatin remodeling at the BDNF gene in both hippocampus and visual cortex

scientific article published on 8 July 2010

Discovery and Characterization of 2-Aminooxazolines as Highly Potent, Selective, and Orally Active TAAR1 Agonists

scientific article

Duloxetine inhibits effects of MDMA ("ecstasy") in vitro and in humans in a randomized placebo-controlled laboratory study

scientific article

Effects of sodium chloride, Triton X-100, and alkaline pH on the measurable contents and sedimentability of the nerve growth factor (NGF) antigen in adult rat hippocampal tissue extracts

scientific article published in August 1997

Effects of the new psychoactive substances diclofensine, diphenidine, and methoxphenidine on monoaminergic systems

scientific article published on 7 December 2017

Effects of the α₂-adrenergic agonist clonidine on the pharmacodynamics and pharmacokinetics of 3,4-methylenedioxymethamphetamine in healthy volunteers.

scientific article published on 27 October 2011

Electrophysiological Phenotype in Angelman Syndrome Differs Between Genotypes

scientific article published on 19 January 2019

G protein-coupled receptor transmembrane binding pockets and their applications in GPCR research and drug discovery: a survey

scientific article published in January 2011

Geldanamycin restores a defective heat shock response in vivo

scientific article

Glycosyl-phosphatidylinositol-specific phospholipase D. Interaction with and stimulation by apolipoprotein A-I

scientific article published on 01 July 1993

How Female Mice Attract Males: A Urinary Volatile Amine Activates a Trace Amine-Associated Receptor That Induces Male Sexual Interest

scholarly article by Anja Harmeier et al published 2018 in Frontiers in Pharmacology

In Vitro Characterization of Psychoactive Substances at Rat, Mouse, and Human Trace Amine-Associated Receptor 1.

scientific article published on 20 January 2016

Incretin-like effects of small molecule trace amine-associated receptor 1 agonists.

scientific article

Interaction Between the Trace Amine-Associated Receptor 1 and the Dopamine D2 Receptor Controls Cocaine's Neurochemical Actions

scientific article published on 24 October 2017

Isolation and characterization of a phosphatidylinositol-glycan-anchor-specific phospholipase D from bovine brain

scientific article published in July 1990

Metabolites of the ring-substituted stimulants MDMA, methylone and MDPV differentially affect human monoaminergic systems

scientific article published on 30 April 2019

Monoamine receptor interaction profiles of 4-aryl-substituted 2,5-dimethoxyphenethylamines (2C-BI derivatives)

scientific article published on 04 May 2019

Monoamine receptor interaction profiles of 4-thio-substituted phenethylamines (2C-T drugs).

scientific article published on 15 July 2017

Monoamine transporter and receptor interaction profiles of a new series of designer cathinones.

scientific article

Monoamine transporter and receptor interaction profiles of novel psychoactive substances: para-halogenated amphetamines and pyrovalerone cathinones

scientific article

Nerve growth factor (NGF) content in adult rat brain tissues is several-fold higher than generally reported and is largely associated with sedimentable fractions

scientific article

Opioid-induced inhibition of the human 5-HT and noradrenaline transporters in vitro: link to clinical reports of serotonin syndrome.

scientific article published on 6 December 2017

Optimisation of imidazole compounds as selective TAAR1 agonists: discovery of RO5073012

scientific article published on 23 June 2012

PRONOUNCED HYPERACTIVITY, COGNITIVE DYSFUNCTIONS AND BDNF DYSREGULATION IN DOPAMINE TRANSPORTER KNOCKOUT RATS.

scientific article published on 18 January 2018

Partial cortical devascularization results in elevations of cortical nerve growth factor and increases nerve growth factor protein within basal forebrain cholinergic neurons.

scientific article published on April 1998

Pharmacological characterization of designer cathinones in vitro ⬇️

scientific article published on January 1, 2013

Pharmacological characterization of the aminorex analogs 4-MAR, 4,4'-DMAR, and 3,4-DMAR

scientific article published on 15 February 2019

Pharmacological profile of mephedrone analogs and related new psychoactive substances.

scientific article published on 26 July 2017

Pharmacological profile of methylphenidate-based designer drugs.

scientific article published on 17 August 2017

Pharmacological profile of novel psychoactive benzofurans

scientific article

Pharmacological profiles of aminoindanes, piperazines, and pipradrol derivatives.

scientific article published on 28 January 2014

Pharmacological profiles of compounds in preworkout supplements ("boosters")

scientific article published on 29 June 2019

Pharmacology of human trace amine-associated receptors: Therapeutic opportunities and challenges.

scientific article

Phosphatidylinositol-glycan-specific phospholipase D is an amphiphilic glycoprotein that in serum is associated with high-density lipoproteins

scientific article

Receptor Interaction Profiles of 4-Alkoxy-Substituted 2,5-Dimethoxyphenethylamines and Related Amphetamines

scientific article published on 28 November 2019

Receptor interaction profiles of novel N-2-methoxybenzyl (NBOMe) derivatives of 2,5-dimethoxy-substituted phenethylamines (2C drugs).

scientific article

Receptor interaction profiles of novel psychoactive tryptamines compared with classic hallucinogens.

scientific article published on 20 May 2016

Reversible sedimentation and masking of nerve growth factor (NGF) antigen by high molecular weight fractions from rat brain

scientific article published in October 1997

Role of trace amine-associated receptor 1 in nicotine's behavioral and neurochemical effects.

scientific article published on 5 February 2018

Role played by sodium in activity-dependent secretion of neurotrophins - revisited.

scientific article published in September 2000

Secreted retrovirus-like GAG-domain-containing protein PEG10 is regulated by UBE3A and is involved in Angelman syndrome pathophysiology

scientific article published on 17 August 2021

Selective activation of the trace amine-associated receptor 1 decreases cocaine's reinforcing efficacy and prevents cocaine-induced changes in brain reward thresholds.

scientific article published on 3 June 2015

Selective antagonists of mouse trace amine-associated receptor 1 (mTAAR1): discovery of EPPTB (RO5212773).

scientific article

Similar patterns of mitochondrial vulnerability and rescue induced by genetic modification of alpha-synuclein, parkin, and DJ-1 in Caenorhabditis elegans

scientific article

Stereochemistry of phase-1 metabolites of mephedrone determines their effectiveness as releasers at the serotonin transporter

scientific article published on 02 January 2019

TAAR1 Modulates Cortical Glutamate NMDA Receptor Function

scientific article

TAAR1 activation modulates monoaminergic neurotransmission, preventing hyperdopaminergic and hypoglutamatergic activity

scientific article

TAAR1 levels and sub-cellular distribution are cell line but not breast cancer subtype specific

scientific article published on 21 May 2019

TAAR1-dependent effects of apomorphine in mice.

scientific article published on 13 June 2014

Taar1-mediated modulation of presynaptic dopaminergic neurotransmission: role of D2 dopamine autoreceptors.

scientific article published on 22 February 2014

The Caenorhabditis elegans NR4A nuclear receptor is required for spermatheca morphogenesis

scientific article

The Trace Amine-Associated Receptor 1 Agonist RO5256390 Blocks Compulsive, Binge-like Eating in Rats

scientific article published on 6 October 2016

The antidepressant-like effects of glutamatergic drugs ketamine and AMPA receptor potentiator LY 451646 are preserved in bdnf⁺/⁻ heterozygous null mice

scientific article

The impact of Bdnf gene deficiency to the memory impairment and brain pathology of APPswe/PS1dE9 mouse model of Alzheimer's disease

scientific article published on 03 July 2013

The norepinephrine transporter inhibitor reboxetine reduces stimulant effects of MDMA ("ecstasy") in humans

scientific article (publication date: August 2011)

The psychostimulant (±)-cis-4,4'-dimethylaminorex (4,4'-DMAR) interacts with human plasmalemmal and vesicular monoamine transporters

scientific article published on 23 June 2018

The selective antagonist EPPTB reveals TAAR1-mediated regulatory mechanisms in dopaminergic neurons of the mesolimbic system

scientific article

The trace amine-associated receptor 1 modulates methamphetamine's neurochemical and behavioral effects.

scientific article

Trace Amine-Associated Receptor 1 Agonists as Narcolepsy Therapeutics

scientific article published on 18 October 2016

Trace Amine-Associated Receptor 1 Regulates Wakefulness and EEG Spectral Composition.

scientific article

Trace Amines and Their Receptors

scientific article published on 01 July 2018

Trace amine associated receptor 1 signaling in activated lymphocytes

scientific article published in December 2012

Trace amine-associated receptor 1 activation silences GSK3β signaling of TAAR1 and D2R heteromers

scientific article

Trace amine-associated receptor 1 agonism promotes wakefulness without impairment of cognition in Cynomolgus macaques

scientific article published on 06 April 2019

Trace amine-associated receptor 1 modulates dopaminergic activity

scientific article

Trace amine-associated receptor 1 partial agonism reveals novel paradigm for neuropsychiatric therapeutics.

scientific article

Trace amine-associated receptors form structurally and functionally distinct subfamilies of novel G protein-coupled receptors

scientific article

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