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List of works by Jean-christophe Cintrat

(S)-N-Methyldihydroquinazolinones are the Active Enantiomers of Retro-2 Derived Compounds against Toxins

scientific article

An isosparteine derivative for stereochemical assignment of stereogenic (chiral) methyl groups using tritium NMR: theory and experiment.

scientific article

Antiviral effects of Retro-2cycl and Retro-2.1 against Enterovirus 71 in vitro and in vivo

scientific article published on 5 July 2017

Carbon-centered radicals can transfer hydrogen atoms between amino acid side chains

scientific article published on 06 February 2012

Chemical inhibitors of monogalactosyldiacylglycerol synthases in Arabidopsis thaliana.

scientific article

Control of peptide nanotube diameter by chemical modifications of an aromatic residue involved in a single close contact

scientific article

Directing peptide crystallization through curvature control of nanotubes

scientific article published on 11 June 2014

Discovery of compounds blocking the proliferation of Toxoplasma gondii and Plasmodium falciparum in a chemical space based on piperidinyl-benzimidazolone analogs

scientific article

Elimination and exchange of trifluoroacetate counter-ion from cationic peptides: a critical evaluation of different approaches

scientific article published in March 2008

Experimental observation of double-walled peptide nanotubes and monodispersity modeling of the number of walls.

scientific article published on 12 February 2013

Footprinting of protein interactions by tritium labeling

scientific article published on 01 May 2010

Functional dissection of the retrograde Shiga toxin trafficking inhibitor Retro-2

scientific article published on 17 February 2020

Highly chemoselective hydrogenolysis of iodoarenes

scientific article published in February 2002

Intracellular pathogens convert macrophages from death traps into hospitable homes.

scientific article published on 20 January 2016

Localization and quantification of carbon-centered radicals on any amino acid of a protein

scientific article published on 19 June 2007

Measurement of Long-Range Interatomic Distances by Solid-State Tritium-NMR Spectroscopy

scientific article published on 17 February 2010

N-methyldihydroquinazolinone derivatives of Retro-2 with enhanced efficacy against Shiga toxin

scientific article published on 05 April 2013

Palladium-Catalyzed Chemoselective and Biocompatible Functionalization of Cysteine-Containing Molecules at Room Temperature.

scientific article

Parthenolide inhibits tubulin carboxypeptidase activity

scientific article published on 01 April 2007

Photochemical Strain-Release-Driven Cyclobutylation of C(sp3 )-Centered Radicals

scientific article published on 06 November 2019

Regioselective Halogenation of 1,4-Benzodiazepinones via CH Activation

scientific article published on 16 July 2015

Regulation of endo-lysosomal pathway and autophagic flux by broad-spectrum antipathogen inhibitor ABMA

scientific article published on 04 January 2020

Retrograde Trafficking Inhibitor of Shiga Toxins Reduces Morbidity and Mortality of Mice Infected with Enterohemorrhagic Escherichia coli

scientific article

Revisiting Old Ionophore Lasalocid as a Novel Inhibitor of Multiple Toxins

scientific article published on 01 January 2020

Scalable synthesis of cryptophane-1.1.1 and its functionalization

scientific article published in March 2010

Squalenoylation favorably modifies the in vivo pharmacokinetics and biodistribution of gemcitabine in mice.

scientific article published on 12 May 2008

Stille cross-coupling reaction of an alpha-stannyl enamide

scientific article published on 01 November 2001

Structural Role of Counterions Adsorbed on Self-Assembled Peptide Nanotubes

scientific article published on 22 December 2011

Syntaxin 5-dependent retrograde transport to the trans-Golgi network is required for adeno-associated virus transduction

scientific article

Synthesis of orthogonally protected azahistidine: application to the synthesis of a GHK analogue

scientific article published on 15 February 2009

Synthesis, Chiral Separation, Absolute Configuration Assignment, and Biological Activity of Enantiomers of Retro-1 as Potent Inhibitors of Shiga Toxin.

scientific article published on June 2015

The peptide methionine sulfoxide reductases, MsrA and MsrB (hCBS-1), are downregulated during replicative senescence of human WI-38 fibroblasts

scientific publication

The small molecule Retro-1 enhances the pharmacological actions of antisense and splice switching oligonucleotides.

scientific article published on 8 February 2013