List of works - Marco Pallavicini

4-Oxystilbene compounds are selective ligands for neuronal nicotinic alphaBungarotoxin receptors.

scientific article published on July 1998

5-(2-Pyrrolidinyl)oxazolidinones and 2-(2-pyrrolidinyl)benzodioxanes: synthesis of all the stereoisomers and alpha4beta2 nicotinic affinity

scientific article

6-methoxy-7-benzofuranoxy and 6-methoxy-7-indolyloxy analogues of 2-[2-(2,6-Dimethoxyphenoxy)ethyl]aminomethyl-1,4-benzodioxane (WB4101):1 discovery of a potent and selective α1D-adrenoceptor antagonist.

scientific article

Affinity and activity profiling of unichiral 8-substituted 1,4-benzodioxane analogues of WB4101 reveals a potent and selective α1B-adrenoceptor antagonist.

scientific article

An investigation into the influence of counterion on the RS-propranolol and S-propranolol skin permeability.

scientific article published in March 2010

Benzodioxane-benzamides as new bacterial cell division inhibitors

scientific article published on 18 October 2014

Cardiovascular and pulmonary activity of platelet-activating factor (PAF-acether) and its derivatives.

scientific article

Characterization of in vitro metabolites of JWH-018, JWH-073 and their 4-methyl derivatives, markers of the abuse of these synthetic cannabinoids

scientific article published on 12 March 2014

Construction of human ghrelin receptor (hGHS-R1a) model using a fragmental prediction approach and validation through docking analysis

scientific article published on June 2006

Corrigendum to “Synthesis and α4β2 nicotinic affinity of unichiral 5-(2-pyrrolidinyl)oxazolidinones and 2-(2-pyrrolidinyl)benzodioxanes” [Bioorg. Med. Chem. Lett. 16 (2006) 5610–5615]

scholarly article published in Bioorganic & Medicinal Chemistry Letters

Design, synthesis and binding affinity of acetylcholine carbamoyl analogues

scientific article published on 18 September 2013

Exploring the space of histidine containing dipeptides in search of novel efficient RCS sequestering agents

scientific article published on 30 May 2013

Farnesyltransferase inhibitors: CAAX mimetics based on different biaryl scaffolds

scientific article published on 30 April 2014

From 2-aminomethyl-1,4-benzodioxane enantiomers to unichiral 2-cyano- and 2-carbonyl-substituted benzodioxanes via dichloroamine

scientific article published on 26 June 2014

Identification of 1-butyl-3-(1-(4-methyl)naphtoyl)indole detected for the first time in “herbal high” products on the Italian market

article

Modelling of full-length human alpha4beta2 nicotinic receptor by fragmental approach and analysis of its binding modes

scientific article

Modifications at C(5) of 2-(2-Pyrrolidinyl)-Substituted 1,4-Benzodioxane Elicit Potent α4β2 Nicotinic Acetylcholine Receptor Partial Agonism with High Selectivity over the α3β4 Subtype

scientific article published on 16 December 2020

New Ras CAAX mimetics: design, synthesis, antiproliferative activity, and RAS prenylation inhibition

scientific article published on 17 July 2009

Peptidomimetic inhibitors of farnesyltransferase with high in vitro activity and significant cellular potency

scientific article published on 8 September 2007

Potent anti-glioblastoma agents by hybridizing the onium-alkyloxy-stilbene based structures of an alpha7-, alpha9-nAChR antagonist and of a pro-oxidant mitocan

scientific article published on 26 November 2018

Predicting the physicochemical profile of diastereoisomeric histidine-containing dipeptides by property space analysis

scientific article published on 8 May 2012

QSAR study for a novel series of ortho disubstituted phenoxy analogues of alpha1-adrenoceptor antagonist WB4101.

scientific article published on 5 June 2006

QSAR study for a novel series of ortho monosubstituted phenoxy analogues of alpha1-adrenoceptor antagonist WB4101.

scientific article

Structure-affinity studies for a novel series of homochiral naphtho and tetrahydronaphtho analogues of alpha 1 antagonist WB-4101.

scientific article published in September 2004

Synthesis and alpha4beta2 nicotinic affinity of 2-pyrrolidinylmethoxyimines and prolinal oxime ethers

scientific article published in December 2004

Synthesis and α4β2 nicotinic affinity of unichiral 5-(2-pyrrolidinyl)oxazolidinones and 2-(2-pyrrolidinyl)benzodioxanes

scientific article published in 2006

Synthesis of homochiral 5- and 8-substituted 2-[((2-(2,6-dimethoxyphenoxy)-ethyl)amino)methyl]-1,4-benzodioxanes and electrophoretic determination of their enantiomeric excess

scientific article published on 01 February 2001

Thiazole- and imidazole-containing peptidomimetic inhibitors of protein farnesyltransferase

scientific article published on 13 July 2011

Unichiral 2-(2'-pyrrolidinyl)-1,4-benzodioxanes: the 2R,2'S diastereomer of the N-methyl-7-hydroxy analogue is a potent α4β2- and α6β2-nicotinic acetylcholine receptor partial agonist

scientific article published on 11 October 2011

WB4101-related compounds: new, subtype-selective alpha1-adrenoreceptor antagonists (or inverse agonists?).

scientific article published in November 2006

List of works by Marco Pallavicini

4-Oxystilbene compounds are selective ligands for neuronal nicotinic alphaBungarotoxin receptors.

5-(2-Pyrrolidinyl)oxazolidinones and 2-(2-pyrrolidinyl)benzodioxanes: synthesis of all the stereoisomers and alpha4beta2 nicotinic affinity

6-methoxy-7-benzofuranoxy and 6-methoxy-7-indolyloxy analogues of 2-[2-(2,6-Dimethoxyphenoxy)ethyl]aminomethyl-1,4-benzodioxane (WB4101):1 discovery of a potent and selective α1D-adrenoceptor antagonist.

Affinity and activity profiling of unichiral 8-substituted 1,4-benzodioxane analogues of WB4101 reveals a potent and selective α1B-adrenoceptor antagonist.

An investigation into the influence of counterion on the RS-propranolol and S-propranolol skin permeability.

Benzodioxane-benzamides as new bacterial cell division inhibitors

Cardiovascular and pulmonary activity of platelet-activating factor (PAF-acether) and its derivatives.

Characterization of in vitro metabolites of JWH-018, JWH-073 and their 4-methyl derivatives, markers of the abuse of these synthetic cannabinoids

Construction of human ghrelin receptor (hGHS-R1a) model using a fragmental prediction approach and validation through docking analysis

Corrigendum to “Synthesis and α4β2 nicotinic affinity of unichiral 5-(2-pyrrolidinyl)oxazolidinones and 2-(2-pyrrolidinyl)benzodioxanes” [Bioorg. Med. Chem. Lett. 16 (2006) 5610–5615]

Design, synthesis and binding affinity of acetylcholine carbamoyl analogues

Exploring the space of histidine containing dipeptides in search of novel efficient RCS sequestering agents

Farnesyltransferase inhibitors: CAAX mimetics based on different biaryl scaffolds

From 2-aminomethyl-1,4-benzodioxane enantiomers to unichiral 2-cyano- and 2-carbonyl-substituted benzodioxanes via dichloroamine

Identification of 1-butyl-3-(1-(4-methyl)naphtoyl)indole detected for the first time in “herbal high” products on the Italian market

Modelling of full-length human alpha4beta2 nicotinic receptor by fragmental approach and analysis of its binding modes

Modifications at C(5) of 2-(2-Pyrrolidinyl)-Substituted 1,4-Benzodioxane Elicit Potent α4β2 Nicotinic Acetylcholine Receptor Partial Agonism with High Selectivity over the α3β4 Subtype

New Ras CAAX mimetics: design, synthesis, antiproliferative activity, and RAS prenylation inhibition

Peptidomimetic inhibitors of farnesyltransferase with high in vitro activity and significant cellular potency

Potent anti-glioblastoma agents by hybridizing the onium-alkyloxy-stilbene based structures of an alpha7-, alpha9-nAChR antagonist and of a pro-oxidant mitocan

Predicting the physicochemical profile of diastereoisomeric histidine-containing dipeptides by property space analysis

QSAR study for a novel series of ortho disubstituted phenoxy analogues of alpha1-adrenoceptor antagonist WB4101.

QSAR study for a novel series of ortho monosubstituted phenoxy analogues of alpha1-adrenoceptor antagonist WB4101.

Structure-affinity studies for a novel series of homochiral naphtho and tetrahydronaphtho analogues of alpha 1 antagonist WB-4101.

Synthesis and alpha4beta2 nicotinic affinity of 2-pyrrolidinylmethoxyimines and prolinal oxime ethers

Synthesis and α4β2 nicotinic affinity of unichiral 5-(2-pyrrolidinyl)oxazolidinones and 2-(2-pyrrolidinyl)benzodioxanes

Synthesis of homochiral 5- and 8-substituted 2-[((2-(2,6-dimethoxyphenoxy)-ethyl)amino)methyl]-1,4-benzodioxanes and electrophoretic determination of their enantiomeric excess

Thiazole- and imidazole-containing peptidomimetic inhibitors of protein farnesyltransferase

Unichiral 2-(2'-pyrrolidinyl)-1,4-benzodioxanes: the 2R,2'S diastereomer of the N-methyl-7-hydroxy analogue is a potent α4β2- and α6β2-nicotinic acetylcholine receptor partial agonist

WB4101-related compounds: new, subtype-selective alpha1-adrenoreceptor antagonists (or inverse agonists?).