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List of works by Kwang-Seok Oh

3D QSAR pharmacophore model based on diverse IKKβ inhibitors

article

4-Substituted quinazoline derivatives as novel EphA2 receptor tyrosine kinase inhibitors.

scientific article published on 6 August 2014

4-arylphthalazin-1(2H)-one derivatives as potent antagonists of the melanin concentrating hormone receptor 1 (MCH-R1).

scientific article published on 10 November 2011

A Novel and Orally Active Poly(ADP-Ribose) Polymerase Inhibitor, KR-33889 [2-[Methoxycarbonyl(4-methoxyphenyl) methylsulfanyl]-1H-benzimidazole-4-carboxylic Acid Amide], Attenuates Injury in in Vitro Model of Cell Death and in Vivo Model of Cardiac I

article

A comparison of assay performance between the calcium mobilization and the dynamic mass redistribution technologies for the human urotensin receptor.

scientific article published on August 2014

A novel role of G protein-coupled receptor kinase 5 in urotensin II-stimulated cellular hypertrophy in H9c2UT cells

scientific article published on 9 September 2016

A novel urotensin II receptor antagonist, KR-36996, improved cardiac function and attenuated cardiac hypertrophy in experimental heart failure.

scientific article published on 3 February 2017

A urotensin II receptor antagonist, KR36676, decreases vascular remodeling and inflammation in experimental pulmonary hypertension

scientific article published on 6 September 2016

Antihypertensive, vasorelaxant and inotropic effects of an ethanolic extract of the roots of Saururus chinensis

scientific article published on 15 April 2008

Benzo[b]thiophene-2-carboxamide derivatives as potent urotensin-II receptor antagonists

scientific article published on 26 August 2016

DeepHIT: a deep learning framework for prediction of hERG-induced cardiotoxicity

scientific article published on 05 February 2020

Design and synthesis of novel 3-(benzo[d]oxazol-2-yl)-5-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)pyridin-2-amine derivatives as selective G-protein-coupled receptor kinase-2 and -5 inhibitors.

scientific article published on 30 October 2013

Discovery of piperidinyl aminopyrimidine derivatives as IKK-2 inhibitors.

scientific article published on 17 March 2011

Effects of KR-31378, a novel ATP-sensitive potassium channel activator, on hypertrophy of H9c2 cells and on cardiac dysfunction in rats with congestive heart failure.

scientific article published on 3 May 2006

Effects of KR-33028, a novel Na+/H+exchanger-1 inhibitor, on ischemia and reperfusion-induced myocardial infarction in rats and dogs

scientific article published on 01 June 2007

Expression and purification of the anticomplementary peptide Sh-CRIT-ed1 (formerly Sh-TOR-ed1) as a tetramultimer in Escherichia coli.

scientific article published in February 2003

Growth factors mobilize multiple pools of KCa channels in developing parasympathetic neurons: role of ADP-ribosylation factors and related proteins

scientific article

IKKbeta inhibitors identification part I: homology model assisted structure based virtual screening

scientific article

IKKβ inhibitor identification: a multi-filter driven novel scaffold

scientific article published on October 15, 2010

Inhibition of complement activation by recombinant Sh-CRIT-ed1 analogues

scientific article

Kamolonol suppresses angiotensin II-induced stress fiber formation and cellular hypertrophy through inhibition of Rho-associated kinase 2 activity.

scientific article published on 24 July 2013

Large conductance Ca2+-activated K+ (BKCa) channels are involved in the vascular relaxations elicited by piceatannol isolated from Rheum undulatum rhizome

scientific article published on 24 October 2007

Pharmacological profile of KR-33028, a highly selective inhibitor of Na+/H+ exchanger.

scientific article published on 6 March 2006

Synthesis and SAR investigations of novel 2-arylbenzimidazole derivatives as melanin-concentrating hormone receptor 1 (MCH-R1) antagonists

scientific article published on 26 February 2011

Synthesis and SAR of 5-aryl-furan-2-carboxamide derivatives as potent urotensin-II receptor antagonists

scientific article published on 29 December 2018

Synthesis and SAR study of pyrrolo[3,4-b]pyridin-7(6H)-one derivatives as melanin concentrating hormone receptor 1 (MCH-R1) antagonists

scientific article published on 24 January 2013

Synthesis and structure-activity relationship of naphtho[1,2-b]furan-2-carboxamide derivatives as melanin concentrating hormone receptor 1 antagonists

scientific article published in January 2013

The Effects of Chronic Treatment with Morus bombycis KOIDZUMI in Spontaneously Hypertensive Rats

article

The orally active urotensin receptor antagonist, KR36676, attenuates cellular and cardiac hypertrophy

scientific article published on 26 March 2015

Vasorelaxant Effect of the Rootbark Extract of Paeonia moutan on Isolated Rat Thoracic Aorta

article

Vasorelaxant effect of stilbenes from rhizome extract of rhubarb (Rheum undulatum) on the contractility of rat aorta

scientific article published on 01 February 2007