List of works - Fabrizio Pertusati

A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF5) and pentafluoroethyl (C2F5) substituents: Improved antiproliferative agents against prostate cancer

scientific article published on 03 July 2019

Anti-flavivirus Activity of Different Tritylated Pyrimidine and Purine Nucleoside Analogues

scientific article

Chemoselective N-deacetylation of protected nucleosides and nucleotides promoted by Schwartz's reagent.

scientific article published on 22 October 2015

Conjugating a cyanine dye to a polymer surface. In search of a monomeric dye in apolar media

scientific article published on 29 February 2008

Design and synthesis of novel bicalutamide and enzalutamide derivatives as antiproliferative agents for the treatment of prostate cancer

scientific article published on 22 April 2016

Design, synthesis and biological evaluation of phosphorodiamidate prodrugs of antiviral and anticancer nucleosides

scientific article

Diastereoselective synthesis of P-chirogenic phosphoramidate prodrugs of nucleoside analogues (ProTides) via copper catalysed reaction

scientific article published on 13 April 2015

HF-Free, Direct Synthesis of Tetrabutylammonium Trifluoroborates

Kinase-independent phosphoramidate S1P1 receptor agonist benzyl ether derivatives

scientific article published on 9 February 2017

Medicinal chemistry of nucleoside phosphonate prodrugs for antiviral therapy.

scientific article published on 14 May 2012

Nucleoside Derived Antibiotics to Fight Microbial Drug Resistance: New Utilities for an Established Class of Drugs?

scientific article published on 8 September 2016

Phosphonoamidate prodrugs of C5-substituted pyrimidine acyclic nucleosides for antiviral therapy.

scientific article published on 25 April 2017

Polyfluorinated groups in medicinal chemistry.

scientific article published on January 2015

ProTides of N-(3-(5-(2'-deoxyuridine))prop-2-ynyl)octanamide as potential anti-tubercular and anti-viral agents.

scientific article published on 15 March 2014

Rational design and synthesis of novel anti-prostate cancer agents bearing a 3,5-bis-trifluoromethylphenyl moiety

scientific article published on 2 June 2016

Rational design and synthesis of novel phenylsulfonyl-benzamides as anti-prostate cancer agents.

scientific article published on 26 May 2017

Symmetrical diamidate prodrugs of nucleotide analogues for drug delivery

scientific article published on 9 March 2015

Synthesis of an apionucleoside family and discovery of a prodrug with anti-HIV activity

scientific article published on 20 May 2014

Synthesis of phosphoramidate prodrugs: ProTide approach.

scientific article published in June 2013

Synthesis of unsymmetrical 3,3'-biquinazoline-2,2'-diones by condensation of 3-aminoquinazolinones with benzoxazinones; fortuitous discovery, and further syntheses of 4-H-3-oxo-1,9a,10-triazaanthracen-9-ones

scientific article

Synthetic Approaches for the Preparation of Phosphoramidate Prodrugs of 2'-Deoxypseudoisocytidine.

scientific article

Targeting GNE Myopathy: A Dual Prodrug Approach for the Delivery of N-Acetylmannosamine 6-Phosphate

scientific article published on 20 August 2019

λ(5)-Phosphorus-Containing α-Diazo Compounds: A Valuable Tool for Accessing Phosphorus-Functionalized Molecules.

scientific article

List of works by Fabrizio Pertusati

A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF5) and pentafluoroethyl (C2F5) substituents: Improved antiproliferative agents against prostate cancer

Anti-flavivirus Activity of Different Tritylated Pyrimidine and Purine Nucleoside Analogues

Chemoselective N-deacetylation of protected nucleosides and nucleotides promoted by Schwartz's reagent.

Conjugating a cyanine dye to a polymer surface. In search of a monomeric dye in apolar media

Design and synthesis of novel bicalutamide and enzalutamide derivatives as antiproliferative agents for the treatment of prostate cancer

Design, synthesis and biological evaluation of phosphorodiamidate prodrugs of antiviral and anticancer nucleosides

Diastereoselective synthesis of P-chirogenic phosphoramidate prodrugs of nucleoside analogues (ProTides) via copper catalysed reaction

HF-Free, Direct Synthesis of Tetrabutylammonium Trifluoroborates

Kinase-independent phosphoramidate S1P1 receptor agonist benzyl ether derivatives

Medicinal chemistry of nucleoside phosphonate prodrugs for antiviral therapy.

Nucleoside Derived Antibiotics to Fight Microbial Drug Resistance: New Utilities for an Established Class of Drugs?

Phosphonoamidate prodrugs of C5-substituted pyrimidine acyclic nucleosides for antiviral therapy.

Polyfluorinated groups in medicinal chemistry.

ProTides of N-(3-(5-(2'-deoxyuridine))prop-2-ynyl)octanamide as potential anti-tubercular and anti-viral agents.

Rational design and synthesis of novel anti-prostate cancer agents bearing a 3,5-bis-trifluoromethylphenyl moiety

Rational design and synthesis of novel phenylsulfonyl-benzamides as anti-prostate cancer agents.

Symmetrical diamidate prodrugs of nucleotide analogues for drug delivery

Synthesis of an apionucleoside family and discovery of a prodrug with anti-HIV activity

Synthesis of phosphoramidate prodrugs: ProTide approach.

Synthesis of unsymmetrical 3,3'-biquinazoline-2,2'-diones by condensation of 3-aminoquinazolinones with benzoxazinones; fortuitous discovery, and further syntheses of 4-H-3-oxo-1,9a,10-triazaanthracen-9-ones

Synthetic Approaches for the Preparation of Phosphoramidate Prodrugs of 2'-Deoxypseudoisocytidine.

Targeting GNE Myopathy: A Dual Prodrug Approach for the Delivery of N-Acetylmannosamine 6-Phosphate

λ(5)-Phosphorus-Containing α-Diazo Compounds: A Valuable Tool for Accessing Phosphorus-Functionalized Molecules.