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List of works by Kenichiro Shimokawa

(-)-Ternatin inhibits adipogenesis and lipid metabolism in 3T3-L1 cells

scientific article published on 21 February 2009

Biological activity, structural features, and synthetic studies of (-)-ternatin, a potent fat-accumulation inhibitor of 3T3-L1 adipocytes

scientific article published on February 2008

Convergent synthesis and in vivo inhibitory effect on fat accumulation of (-)-ternatin, a highly N-methylated cyclic peptide

scientific article published on 08 June 2007

Derivatization of inhibitor of apoptosis protein (IAP) ligands yields improved inducers of estrogen receptor α degradation.

scientific article published on 15 March 2018

Design, synthesis, and biological evaluation of biotin-labeled (-)-ternatin, a potent fat-accumulation inhibitor against 3T3-L1 adipocytes

scientific article published on 6 November 2008

Development of protein degradation inducers of oncogenic BCR-ABL protein by conjugation of ABL kinase inhibitors and IAP ligands.

scientific article

Different Degradation Mechanisms of Inhibitor of Apoptosis Proteins (IAPs) by the Specific and Nongenetic IAP-dependent Protein Eraser (SNIPER)

scientific article published on 26 October 2018

Fragment-based drug discovery of potent and selective MKK3/6 inhibitors

scientific article published on 17 November 2015

Importance of the backbone conformation of (-)-ternatin in its fat-accumulation inhibitory activity against 3T3-L1 adipocytes

scientific article published on 7 January 2009

In Vivo Knockdown of Pathogenic Proteins via Specific and Nongenetic Inhibitor of Apoptosis Protein (IAP)-dependent Protein Erasers (SNIPERs).

scientific article

Pharmacological difference between degrader and inhibitor against oncogenic BCR-ABL kinase

scientific article published in Scientific Reports

Structure-based hybridization of the bioactive natural products rhizonin A and ternatin leading to a selective fat-accumulation inhibitor against 3T3-L1 adipocytes

scientific article published on 6 December 2008

Synthesis and inhibitory effect on fat accumulation of (-)-ternatin derivatives modified in the beta-OH-D-Leu(7) moiety

scientific article published on 22 November 2007

Targeting the Allosteric Site of Oncoprotein BCR-ABL as an Alternative Strategy for Effective Target Protein Degradation.

scientific article published on 14 September 2017

Whole structure-activity relationships of the fat-accumulation inhibitor (-)-ternatin: recognition of the importance of each amino acid residue

scientific article published on 18 September 2008

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