List of works - Sun-Joon Min

(E)-2,2'-[3-(2-Nitro-phen-yl)prop-2-ene-1,1-di-yl]bis-(3-hy-droxy-5,5-dimethyl-cyclo-hex-2-en-1-one).

scientific article

(E)-2,2'-[3-(4-Chloro-phen-yl)prop-2-ene-1,1-di-yl]bis-(3-hy-droxy-5,5-di-methyl-cyclo-hex-2-en-1-one).

scientific article published on 27 July 2013

2,2-[(E)-3,3-Diphenyl-prop-2-ene-1,1-di-yl]bis-(3-hy-droxy-cyclo-hex-2-en-1-one).

scientific article

5-HT7 receptor modulators: Amino groups attached to biphenyl scaffold determine functional activity

scientific article published on 21 July 2016

9-[(E)-2-(4-Chloro-phen-yl)ethen-yl]-3,3,6,6-tetra-methyl-2,3,4,5,6,7,8,9-octa-hydro-1H-xanthene-1,8-dione.

scientific article published on 18 September 2013

A Potential PET Radiotracer for the 5-HT2C Receptor: Synthesis and in Vivo Evaluation of 4-(3-[18F]fluorophenethoxy)pyrimidine

scientific article published on 14 February 2017

A concise synthesis of tetrabenazine: an intramolecular aza-Prins-type cyclization via oxidative C-H activation

scientific article published on 21 November 2011

A fluorogenic substrate of beta-lactamases and its potential as a probe to detect the bacteria resistant to the third-generation oxyimino-cephalosporins.

scientific article published on 30 October 2015

A potent, selective and cell-active allosteric inhibitor of protein arginine methyltransferase 3 (PRMT3)

scientific article

An Approach to the Synthesis of Tricholomalide A: An Effective Means for Achieving Homo-Robinson Annulation.

scientific article published on May 2008

Cell-Penetrating Peptide-Patchy Deformable Polymeric Nanovehicles with Enhanced Cellular Uptake and Transdermal Delivery

scientific article published on 08 June 2018

Cell-penetrating peptide-conjugated lipid/polymer hybrid nanovesicles for endoplasmic reticulum-targeting intracellular delivery

scientific article published on 08 December 2020

Construction of 8-Azabicyclo[3.2.1]octanes via Sequential DDQ-Mediated Oxidative Mannich Reactions of N-Aryl Pyrrolidines

scientific article published on 30 January 2018

Copper(I)-Catalyzed Synthesis of 1,4-Disubstituted 1,2,3-Triazoles from Azidoformates and Aryl Terminal Alkynes

scientific article published on 05 April 2018

Creating quaternary centers with high exo stereoselectivity using activated alpha-alkynyl dienophiles

scientific article published on 27 July 2007

Crystal structure of (E)-5,5-dimethyl-2-[3-(4-nitro-phen-yl)allyl-idene]cyclo-hexane-1,3-dione

scientific article published on 13 June 2015

Crystal structure of (E)-N-[(E)-3-(4-meth-oxy-phen-yl)allyl-idene]naphthalen-1-amine.

scientific article published on 24 October 2014

Development of carbapenem-based fluorogenic probes for the clinical screening of carbapenemase-producing bacteria

scientific article published on 04 November 2019

Discovery and biological evaluation of tetrahydrothieno[2,3-c]pyridine derivatives as selective metabotropic glutamate receptor 1 antagonists for the potential treatment of neuropathic pain.

scientific article published on 30 April 2015

Discovery of Potent and Selective Allosteric Inhibitors of Protein Arginine Methyltransferase 3 (PRMT3).

scientific article

Discovery of benzimidazole derivatives as modulators of mitochondrial function: A potential treatment for Alzheimer's disease.

scientific article

Discovery of β-Arrestin Biased Ligands of 5-HT7R

article

ESET methylates UBF at K232/254 and regulates nucleolar heterochromatin plasticity and rDNA transcription.

scientific article

Efficient synthesis of mibefradil analogues: an insight into in vitro stability

scientific article

Evaluation of Chemical Interactions between Small Molecules in the Gas Phase Using Chemical Force Microscopy.

scientific article

Facile diverted synthesis of pyrrolidinyl triazoles using organotrifluoroborate: discovery of potential mPTP blockers.

scientific article

Facile synthesis and biological evaluation of 3,3-diphenylpropanoyl piperazines as T-type calcium channel blockers

scientific article published on 12 November 2010

Identification of Optically Active Pyrimidine Derivatives as Selective 5-HT2C Modulators.

scientific article

Identification of highly potent and selective inhibitor, TIPTP, of the p22phox-Rubicon axis as a therapeutic agent for rheumatoid arthritis

scientific article published on 12 March 2020

Identification of the first in silico-designed TREK1 antagonists that block channel currents dose dependently.

scientific article published on 26 June 2016

In silico probing and biological evaluation of SETDB1/ESET-targeted novel compounds that reduce tri-methylated histone H3K9 (H3K9me3) level

scientific article

Indole-Substituted Benzothiazoles and Benzoxazoles as Selective and Reversible MAO-B Inhibitors for Treatment of Parkinson's Disease.

scientific article published on 23 March 2017

Inhibition of VEGF transcription through blockade of the hypoxia inducible factor-1α-p300 interaction by a small molecule.

scientific article

Intermolecular double Prins-type cyclization: a facile and efficient synthesis of 1,6-dioxecanes

scientific article published in January 2009

Intramolecular Diels-Alder reactions of optically active allenic ketones: chirality transfer in the preparation of substituted oxa-bridged octalones

scientific article published in August 2005

Modulation of SETDB1 activity by APQ ameliorates heterochromatin condensation, motor function, and neuropathology in a Huntington's disease mouse model

scientific article published on 01 December 2021

Novel Scaffold Identification of mGlu1 Receptor Negative Allosteric Modulators Using a Hierarchical Virtual Screening Approach.

scientific article published on 7 September 2015

Novel thienopyrimidinones as mGluR1 antagonists.

scientific article published on 8 August 2014

One-pot bifunctionalization of silica nanoparticles conjugated with bioorthogonal linkers: application in dual-modal imaging

scientific article published in 2022

Oxazolopyridines and thiazolopyridines as monoamine oxidase B inhibitors for the treatment of Parkinson's disease.

scientific article published on 11 June 2013

Performance of a Novel Fluorogenic Assay for Detection of Carbapenemase-Producing Enterobacteriaceae from Bacterial Colonies and Directly from Positive Blood Cultures

scientific article published on 23 December 2019

Remodeling of heterochromatin structure slows neuropathological progression and prolongs survival in an animal model of Huntington's disease.

scientific article

Single-carbon discrimination by selected peptides for individual detection of volatile organic compounds

scientific article published on 17 March 2015

Stereocontrolled synthesis of oxaspirobicycles via Prins-pinacol annulation

scientific article published on 01 September 2009

Synthesis and Biological Evaluation of Disubstituted Pyrimidines as Selective 5-HT2C Agonists

scientific article published on 05 September 2019

Synthesis and biological evaluation of 2-(arylethynyl)quinoline derivatives as mGluR5 antagonists for the treatment of neuropathic pain

scientific article published on 22 December 2012

Synthesis and biological evaluation of 2-substituted quinoline 6-carboxamides as potential mGluR1 antagonists for the treatment of neuropathic pain

scientific article published in January 2014

Synthesis and biological evaluation of aryl isoxazole derivatives as metabotropic glutamate receptor 1 antagonists: a potential treatment for neuropathic pain

scientific article published on 24 January 2015

Synthesis and biological evaluation of picolinamides and thiazole-2-carboxamides as mGluR5 (metabotropic glutamate receptor 5) antagonists.

scientific article published on 5 November 2015

Synthesis and evaluation of oxime derivatives as modulators for amyloid beta-induced mitochondrial dysfunction

scientific article published on 26 December 2012

Synthesis and relative stability of 3,5-diacyl-4,5-dihydro-1H-pyrazoles prepared by dipolar cycloaddition of enones and alpha-diazoketones

scientific article published in December 2004

Synthesis of 3'-O-fluorescently mono-modified reversible terminators and their uses in sequencing-by-synthesis

scientific article published on 25 November 2013

Synthesis of 3,4-dimethylidene oxacycles through Prins-type cyclization of allenylmethylsilanes

scientific article published on 09 June 2011

Synthesis of the Tricyclic Ring Structure of Daphnanes via Intramolecular [4 + 3] Cycloaddition/SmI2-Pinacol Coupling.

scientific article published on 21 May 2015

Total synthesis and structural revision of (+/-)-tricholomalides A and B

scientific article published on August 2009

Total synthesis of paecilomycine A

scientific article published on 01 January 2007

Tubulin inhibitor identification by bioactive conformation alignment pharmacophore-guided virtual screening.

scientific article published on 6 April 2015

List of works by Sun-Joon Min

(E)-2,2'-[3-(2-Nitro-phen-yl)prop-2-ene-1,1-di-yl]bis-(3-hy-droxy-5,5-dimethyl-cyclo-hex-2-en-1-one).

(E)-2,2'-[3-(4-Chloro-phen-yl)prop-2-ene-1,1-di-yl]bis-(3-hy-droxy-5,5-di-methyl-cyclo-hex-2-en-1-one).

2,2-[(E)-3,3-Diphenyl-prop-2-ene-1,1-di-yl]bis-(3-hy-droxy-cyclo-hex-2-en-1-one).

5-HT7 receptor modulators: Amino groups attached to biphenyl scaffold determine functional activity

9-[(E)-2-(4-Chloro-phen-yl)ethen-yl]-3,3,6,6-tetra-methyl-2,3,4,5,6,7,8,9-octa-hydro-1H-xanthene-1,8-dione.

A Potential PET Radiotracer for the 5-HT2C Receptor: Synthesis and in Vivo Evaluation of 4-(3-[18F]fluorophenethoxy)pyrimidine

A concise synthesis of tetrabenazine: an intramolecular aza-Prins-type cyclization via oxidative C-H activation

A fluorogenic substrate of beta-lactamases and its potential as a probe to detect the bacteria resistant to the third-generation oxyimino-cephalosporins.

A potent, selective and cell-active allosteric inhibitor of protein arginine methyltransferase 3 (PRMT3)

An Approach to the Synthesis of Tricholomalide A: An Effective Means for Achieving Homo-Robinson Annulation.

Cell-Penetrating Peptide-Patchy Deformable Polymeric Nanovehicles with Enhanced Cellular Uptake and Transdermal Delivery

Cell-penetrating peptide-conjugated lipid/polymer hybrid nanovesicles for endoplasmic reticulum-targeting intracellular delivery

Construction of 8-Azabicyclo[3.2.1]octanes via Sequential DDQ-Mediated Oxidative Mannich Reactions of N-Aryl Pyrrolidines

Copper(I)-Catalyzed Synthesis of 1,4-Disubstituted 1,2,3-Triazoles from Azidoformates and Aryl Terminal Alkynes

Creating quaternary centers with high exo stereoselectivity using activated alpha-alkynyl dienophiles

Crystal structure of (E)-5,5-dimethyl-2-[3-(4-nitro-phen-yl)allyl-idene]cyclo-hexane-1,3-dione

Crystal structure of (E)-N-[(E)-3-(4-meth-oxy-phen-yl)allyl-idene]naphthalen-1-amine.

Development of carbapenem-based fluorogenic probes for the clinical screening of carbapenemase-producing bacteria

Discovery and biological evaluation of tetrahydrothieno[2,3-c]pyridine derivatives as selective metabotropic glutamate receptor 1 antagonists for the potential treatment of neuropathic pain.

Discovery of Potent and Selective Allosteric Inhibitors of Protein Arginine Methyltransferase 3 (PRMT3).

Discovery of benzimidazole derivatives as modulators of mitochondrial function: A potential treatment for Alzheimer's disease.

Discovery of β-Arrestin Biased Ligands of 5-HT7R

ESET methylates UBF at K232/254 and regulates nucleolar heterochromatin plasticity and rDNA transcription.

Efficient synthesis of mibefradil analogues: an insight into in vitro stability

Evaluation of Chemical Interactions between Small Molecules in the Gas Phase Using Chemical Force Microscopy.

Facile diverted synthesis of pyrrolidinyl triazoles using organotrifluoroborate: discovery of potential mPTP blockers.

Facile synthesis and biological evaluation of 3,3-diphenylpropanoyl piperazines as T-type calcium channel blockers

Identification of Optically Active Pyrimidine Derivatives as Selective 5-HT2C Modulators.

Identification of highly potent and selective inhibitor, TIPTP, of the p22phox-Rubicon axis as a therapeutic agent for rheumatoid arthritis

Identification of the first in silico-designed TREK1 antagonists that block channel currents dose dependently.

In silico probing and biological evaluation of SETDB1/ESET-targeted novel compounds that reduce tri-methylated histone H3K9 (H3K9me3) level

Indole-Substituted Benzothiazoles and Benzoxazoles as Selective and Reversible MAO-B Inhibitors for Treatment of Parkinson's Disease.

Inhibition of VEGF transcription through blockade of the hypoxia inducible factor-1α-p300 interaction by a small molecule.

Intermolecular double Prins-type cyclization: a facile and efficient synthesis of 1,6-dioxecanes

Intramolecular Diels-Alder reactions of optically active allenic ketones: chirality transfer in the preparation of substituted oxa-bridged octalones

Modulation of SETDB1 activity by APQ ameliorates heterochromatin condensation, motor function, and neuropathology in a Huntington's disease mouse model

Novel Scaffold Identification of mGlu1 Receptor Negative Allosteric Modulators Using a Hierarchical Virtual Screening Approach.

Novel thienopyrimidinones as mGluR1 antagonists.

One-pot bifunctionalization of silica nanoparticles conjugated with bioorthogonal linkers: application in dual-modal imaging

Oxazolopyridines and thiazolopyridines as monoamine oxidase B inhibitors for the treatment of Parkinson's disease.

Performance of a Novel Fluorogenic Assay for Detection of Carbapenemase-Producing Enterobacteriaceae from Bacterial Colonies and Directly from Positive Blood Cultures

Remodeling of heterochromatin structure slows neuropathological progression and prolongs survival in an animal model of Huntington's disease.

Single-carbon discrimination by selected peptides for individual detection of volatile organic compounds

Stereocontrolled synthesis of oxaspirobicycles via Prins-pinacol annulation

Synthesis and Biological Evaluation of Disubstituted Pyrimidines as Selective 5-HT2C Agonists

Synthesis and biological evaluation of 2-(arylethynyl)quinoline derivatives as mGluR5 antagonists for the treatment of neuropathic pain

Synthesis and biological evaluation of 2-substituted quinoline 6-carboxamides as potential mGluR1 antagonists for the treatment of neuropathic pain

Synthesis and biological evaluation of aryl isoxazole derivatives as metabotropic glutamate receptor 1 antagonists: a potential treatment for neuropathic pain

Synthesis and biological evaluation of picolinamides and thiazole-2-carboxamides as mGluR5 (metabotropic glutamate receptor 5) antagonists.

Synthesis and evaluation of oxime derivatives as modulators for amyloid beta-induced mitochondrial dysfunction

Synthesis and relative stability of 3,5-diacyl-4,5-dihydro-1H-pyrazoles prepared by dipolar cycloaddition of enones and alpha-diazoketones

Synthesis of 3'-O-fluorescently mono-modified reversible terminators and their uses in sequencing-by-synthesis

Synthesis of 3,4-dimethylidene oxacycles through Prins-type cyclization of allenylmethylsilanes

Synthesis of the Tricyclic Ring Structure of Daphnanes via Intramolecular [4 + 3] Cycloaddition/SmI2-Pinacol Coupling.

Total synthesis and structural revision of (+/-)-tricholomalides A and B

Total synthesis of paecilomycine A

Tubulin inhibitor identification by bioactive conformation alignment pharmacophore-guided virtual screening.