List of works - Tove Tuntland

3,4,5-Trisubstituted isoxazoles as novel PPARδ agonists. Part 2

scientific article published on 22 August 2006

A chemically induced vaccine strategy for prostate cancer.

scientific article published on 21 September 2011

A modern in vivo pharmacokinetic paradigm: combining snapshot, rapid and full PK approaches to optimize and expedite early drug discovery ⬇️

scientific article published on September 13, 2012

A monoselective sphingosine-1-phosphate receptor-1 agonist prevents allograft rejection in a stringent rat heart transplantation model

scientific article published in November 2006

Arylaminoethyl carbamates as a novel series of potent and selective cathepsin S inhibitors

scientific article published on 28 July 2006

Cell-based optimization of novel benzamides as potential antimalarial leads

scientific article published on 29 October 2009

Design, synthesis, and biological evaluations of novel oxindoles as HIV-1 non-nucleoside reverse transcriptase inhibitors. Part 2.

scientific article published on 7 February 2006

Design, synthesis, and structure–activity-relationship of phenyl imidazoles as potent Smoothened antagonists

scientific article published on 13 September 2012

Discovery and biological evaluation of benzo[a]carbazole-based small molecule agonists of the thrombopoietin (Tpo) receptor

scientific article

Discovery of BAF312 (Siponimod), a Potent and Selective S1P Receptor Modulator

scientific article

Discovery of novel 1H-imidazol-2-yl-pyrimidine-4,6-diamines as potential antimalarials

scientific article published on 2 June 2010

Efflux of zidovudine and 2',3'-dideoxyinosine out of the cerebrospinal fluid when administered alone and in combination to Macaca nemestrina

scientific article published on 01 February 1994

Gene expression signatures and small-molecule compounds link a protein kinase to Plasmodium falciparum motility

scientific article

Modulation of TNFalpha, IL-10 and IL-12p40 levels by a ceramide-1-phosphate analog, PCERA-1, in vivo and ex vivo in primary macrophages.

scientific article published on 29 January 2009

N-Acylthiadiazolines, a new class of liver X receptor agonists with selectivity for LXRbeta.

scientific article published on August 2007

No Effect of Vitamin B-6 Against Premenstrual Tension: A controlled clinical study

scientific article published on 01 January 1985

Novel bisaryl substituted thiazoles and oxazoles as highly potent and selective peroxisome proliferator-activated receptor delta agonists

scientific article published in January 2010

Snapshot PK: a rapid rodent in vivo preclinical screening approach.

scientific article

Synthesis and SAR of arylaminoethyl amides as noncovalent inhibitors of cathepsin S: P3 cyclic ethers

scientific article published on 28 July 2006

Synthesis and SAR of succinamide peptidomimetic inhibitors of cathepsin S

scientific article published on 27 February 2007

Synthesis and evaluation of arylaminoethyl amides as noncovalent inhibitors of cathepsin S. Part 3: Heterocyclic P3

scientific article published on 30 January 2006

List of works by Tove Tuntland

3,4,5-Trisubstituted isoxazoles as novel PPARδ agonists. Part 2

A chemically induced vaccine strategy for prostate cancer.

A modern in vivo pharmacokinetic paradigm: combining snapshot, rapid and full PK approaches to optimize and expedite early drug discovery ⬇️

A monoselective sphingosine-1-phosphate receptor-1 agonist prevents allograft rejection in a stringent rat heart transplantation model

Arylaminoethyl carbamates as a novel series of potent and selective cathepsin S inhibitors

Cell-based optimization of novel benzamides as potential antimalarial leads

Design, synthesis, and biological evaluations of novel oxindoles as HIV-1 non-nucleoside reverse transcriptase inhibitors. Part 2.

Design, synthesis, and structure–activity-relationship of phenyl imidazoles as potent Smoothened antagonists

Discovery and biological evaluation of benzo[a]carbazole-based small molecule agonists of the thrombopoietin (Tpo) receptor

Discovery of BAF312 (Siponimod), a Potent and Selective S1P Receptor Modulator

Discovery of novel 1H-imidazol-2-yl-pyrimidine-4,6-diamines as potential antimalarials

Efflux of zidovudine and 2',3'-dideoxyinosine out of the cerebrospinal fluid when administered alone and in combination to Macaca nemestrina

Gene expression signatures and small-molecule compounds link a protein kinase to Plasmodium falciparum motility

Modulation of TNFalpha, IL-10 and IL-12p40 levels by a ceramide-1-phosphate analog, PCERA-1, in vivo and ex vivo in primary macrophages.

N-Acylthiadiazolines, a new class of liver X receptor agonists with selectivity for LXRbeta.

No Effect of Vitamin B-6 Against Premenstrual Tension: A controlled clinical study

Novel bisaryl substituted thiazoles and oxazoles as highly potent and selective peroxisome proliferator-activated receptor delta agonists

Snapshot PK: a rapid rodent in vivo preclinical screening approach.

Synthesis and SAR of arylaminoethyl amides as noncovalent inhibitors of cathepsin S: P3 cyclic ethers

Synthesis and SAR of succinamide peptidomimetic inhibitors of cathepsin S

Synthesis and evaluation of arylaminoethyl amides as noncovalent inhibitors of cathepsin S. Part 3: Heterocyclic P3