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List of works by Anders Skov Kristensen

2-arylureidobenzoic acids: selective noncompetitive antagonists for the homomeric kainate receptor subtype GluR5.

scientific article published on December 2003

A Heteromeric Snake Toxin and the Molecular Details of Pain Perception ⬇️

scholarly article by Kristian Strømgaard & Anders S Kristensen published 15 March 2012 in Angewandte Chemie International Edition

A high-affinity, dimeric inhibitor of PSD-95 bivalently interacts with PDZ1-2 and protects against ischemic brain damage

scientific article

Analogues of 3-Hydroxyisoxazole-Containing Glutamate Receptor Ligands Based on the 3-Hydroxypyrazole-Moiety: Design, Synthesis and Pharmacological Characterization

scientific article published on 22 May 2014

Assessment of structurally diverse philanthotoxin analogues for inhibitory activity on ionotropic glutamate receptor subtypes: discovery of nanomolar, nonselective, and use-dependent antagonists

scientific article published on October 2010

Binding of ArgTX-636 in the NMDA receptor ion channel

scientific article published on 24 May 2014

Binding site residues control inhibitor selectivity in the human norepinephrine transporter but not in the human dopamine transporter

scientific article

Bioisosteric modifications of 2-arylureidobenzoic acids: selective noncompetitive antagonists for the homomeric kainate receptor subtype GluR5.

scientific article published in December 2004

Cell-permeable and plasma-stable peptidomimetic inhibitors of the postsynaptic density-95/N-methyl-D-aspartate receptor interaction.

scientific article

Characterization of intracellular regions in the human serotonin transporter for phosphorylation sites.

scientific article

Conformational Changes in the 5-HT3A Receptor Extracellular Domain Measured by Voltage-Clamp Fluorometry

scientific article published on 03 October 2019

Correlation between anticonvulsant activity and inhibitory action on glial gamma-aminobutyric acid uptake of the highly selective mouse gamma-aminobutyric acid transporter 1 inhibitor 3-hydroxy-4-amino-4,5,6,7-tetrahydro-1,2-benzisoxazole and its N-

scientific article

Deciphering the kinetic binding mechanism of dimeric ligands using a potent plasma-stable dimeric inhibitor of postsynaptic density protein-95 as an example.

scientific article

Design and synthesis of highly potent and plasma-stable dimeric inhibitors of the PSD-95-NMDA receptor interaction

scientific article published in January 2009

Design, synthesis, and pharmacology of a highly subtype-selective GluR1/2 agonist, (RS)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)propionic acid (Cl-HIBO).

scientific article published in May 2003

Detecting protein-protein interactions in living cells: development of a bioluminescence resonance energy transfer assay to evaluate the PSD-95/NMDA receptor interaction

scientific article published on 4 June 2009

Development of potent fluorescent polyamine toxins and application in labeling of ionotropic glutamate receptors in hippocampal neurons.

scientific article published on 24 July 2013

Evaluation of PhTX-74 as subtype-selective inhibitor of GluA2-containing AMPA receptors.

scientific article

From the selective serotonin transporter inhibitor citalopram to the selective norepinephrine transporter inhibitor talopram: synthesis and structure-activity relationship studies.

scientific article

Glutamate receptors: variation in structure-function coupling

scientific article published on 6 January 2006

Inhibition of AMPA receptors by polyamine toxins is regulated by agonist efficacy and stargazin

scientific article published on 22 February 2014

Interaction of antidepressants with the serotonin and norepinephrine transporters: mutational studies of the S1 substrate binding pocket

scientific article published on 19 October 2012

Ionotropic glutamate-like receptor  2 binds D-serine and glycine

scientific article

Location of the antidepressant binding site in the serotonin transporter: importance of Ser-438 in recognition of citalopram and tricyclic antidepressants.

scientific article

Mechanism of Ca2+/calmodulin-dependent kinase II regulation of AMPA receptor gating ⬇️

scientific article published on April 24, 2011

Modeling and mutational analysis of the binding mode for the multimodal antidepressant drug vortioxetine to the human 5-HT3A receptor

scientific article published on 26 September 2018

Modulation of the dimer interface at ionotropic glutamate-like receptor delta2 by D-serine and extracellular calcium

scientific article

Molecular basis for selective serotonin reuptake inhibition by the antidepressant agent fluoxetine (Prozac).

scientific article

Molecular cloning, expression and characterization of a bovine serotonin transporter

scientific article published in July 1999

Mutational Analysis and Modeling of Negative Allosteric Modulator Binding Sites in AMPA Receptors

scientific article published on 03 October 2019

Mutational mapping and modeling of the binding site for (S)-citalopram in the human serotonin transporter.

scientific article

Mutational scanning of the human serotonin transporter reveals fast translocating serotonin transporter mutants

scientific article published in March 2004

Neuroscience: an intrusive chaperone

scientific article published in June 2005

On the neurotoxicity of glutaric, 3-hydroxyglutaric, and trans-glutaconic acids in glutaric acidemia type 1.

scientific article

Probing backbone hydrogen bonding in PDZ/ligand interactions by protein amide-to-ester mutations.

scientific article

Recent advances in the understanding of the interaction of antidepressant drugs with serotonin and norepinephrine transporters.

scientific article

Small molecules from spiders used as chemical probes.

scientific article published on 27 October 2011

Solid-phase synthesis and biological evaluation of Joro spider toxin-4 from Nephila clavata.

scientific article published on 28 December 2010

Species-scanning mutagenesis of the serotonin transporter reveals residues essential in selective, high-affinity recognition of antidepressants

scientific article published in October 2001

Structural rearrangement of the intracellular domains during AMPA receptor activation

scientific article published on 16 June 2016

Structure-activity relationship studies of N-methylated and N-hydroxylated spider polyamine toxins as inhibitors of ionotropic glutamate receptors

scientific article published on 29 May 2014

Structure-activity relationship studies of argiotoxins: selective and potent inhibitors of ionotropic glutamate receptors

scientific article

Structure-activity relationship studies of citalopram derivatives: examining substituents conferring selectivity for the allosteric site in the 5-HT transporter

scientific article published on 23 December 2015

Substrate and Inhibitor-Specific Conformational Changes in the Human Serotonin Transporter Revealed by Voltage-Clamp Fluorometry.

scientific article

Subunit-specific agonist activity at NR2A-, NR2B-, NR2C-, and NR2D-containing N-methyl-D-aspartate glutamate receptors

scientific article published on 10 July 2007

Synthesis and biological activity of argiotoxin 636 and analogues: selective antagonists for ionotropic glutamate receptors

scientific article published in January 2009

Targeting protein-protein interactions with trimeric ligands: high affinity inhibitors of the MAGUK protein family

scientific article

The glutamate receptor GluR5 agonist (S)-2-amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic acid and the 8-methyl analogue: synthesis, molecular pharmacology, and biostructural characterization

scientific article

The structure of a mixed GluR2 ligand-binding core dimer in complex with (S)-glutamate and the antagonist (S)-NS1209.

scientific article published on 31 January 2006

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