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List of works by Vincent Leroux

A new strategy for treating hypertension by blocking the activity of the brain renin-angiotensin system with aminopeptidase A inhibitors

scientific article published on August 2014

Analysis of c-Met kinase domain complexes: a new specific catalytic site receptor model for defining binding modes of ATP-competitive ligands

scientific article published on December 2009

By interacting with the C-terminal Phe of apelin, Phe255 and Trp259 in helix VI of the apelin receptor are critical for internalization.

scientific article published on 30 July 2010

Coenzyme Q Biosynthesis: Evidence for a Substrate Access Channel in the FAD-Dependent Monooxygenase Coq6

scientific article

Comparison of three preprocessing filters efficiency in virtual screening: identification of new putative LXRbeta regulators as a test case

scientific article published in May 2010

Exploring c-Met kinase flexibility by sampling and clustering its conformational space.

scientific article published on 24 January 2012

Identification and pharmacological properties of E339-3D6, the first nonpeptidic apelin receptor agonist

scientific article

Identification of New Antifungal Compounds Targeting Thioredoxin Reductase of Paracoccidioides Genus

scientific article

Identification of new aminoacid amides containing the imidazo[2,1-b]benzothiazol-2-ylphenyl moiety as inhibitors of tumorigenesis by oncogenic Met signaling

scientific article published on November 4, 2011

Multiple-step virtual screening using VSM-G: overview and validation of fast geometrical matching enrichment

scientific article published on 03 January 2008

New structural insights into the apelin receptor: identification of key residues for apelin binding

scientific article published on 30 October 2014

Recent Trends and Applications in 3D Virtual Screening

scientific article published on November 1, 2012

SHEF: a vHTS geometrical filter using coefficients of spherical harmonic molecular surfaces

scientific article

Structure-based virtual screening of hypothetical inhibitors of the enzyme longiborneol synthase-a potential target to reduce Fusarium head blight disease.

scientific article