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List of works by Venkatesan Jayaprakash

2-[(4,6-Di-amino-pyrimidin-2-yl)sulfan-yl]-N-(2-methyl-phen-yl)acetamide

scientific article published on 5 July 2014

5' Adenosine Monophosphate-Activated Protein Kinase Modulators as Anticancer Agents

scientific article published on 11 February 2016

A novel N-hydroxy-N'-aminoguanidine derivative inhibits ribonucleotide reductase activity: Effects in human HL-60 promyelocytic leukemia cells and synergism with arabinofuranosylcytosine (Ara-C).

scientific article published on 16 September 2010

A novel druggable interprotomer pocket in the capsid of rhino- and enteroviruses

scientific article published on 11 June 2019

A perspective on targeting non-structural proteins to combat neglected tropical diseases: Dengue, West Nile and Chikungunya viruses.

scientific article

Anticonvulsant activity of Benkara malabarica (Linn.) root extract: In vitro and in vivo investigation.

scientific article published on 28 January 2010

Antidiabetic activity of Pterospermum acerifolium flowers and glucose uptake potential of bioactive fraction in L6 muscle cell lines with its HPLC fingerprint.

scientific article

Biphenyl urea derivatives as selective CYP1B1 inhibitors

scientific article published on September 2016

Chemical scaffolds with structural similarities to siderophores of nonribosomal peptide–polyketide origin as novel antimicrobials against Mycobacterium tuberculosis and Yersinia pestis ⬇️

scientific article published on August 26, 2011

Cink4T, a quinazolinone-based dual inhibitor of Cdk4 and tubulin polymerization, identified via ligand-based virtual screening, for efficient anticancer therapy

scientific article published on 10 January 2019

Crystal structures and Hirshfeld surface analyses of 2-[(4,6-di-amino-pyrimidin-2-yl)sulfan-yl]-N-(pyridin-2-yl)acetamide and 2-[(4,6-di-amino-pyrimidin-2-yl)sulfan-yl]-N-(pyrazin-2-yl)acetamide.

scientific article

Crystal structures of 2-[(4,6-di-amino-pyrimidin-2-yl)sulfan-yl]-N-(3-nitro-phen-yl)acetamide monohydrate and N-(2-chloro-phen-yl)-2-[(4,6-di-amino-pyrimidin-2-yl)sulfan-yl]acetamide

scientific article published on 22 July 2016

Curcumin-based pyrazoline analogues as selective inhibitors of human monoamine oxidase A

scientific article published on 08 June 2018

Design, synthesis, optimization and antiviral activity of a class of hybrid dengue virus E protein inhibitors

scientific article published on 2 March 2015

Development of CoMFA and CoMSIA models of cytotoxicity data of anti-HIV-1-phenylamino-1H-imidazole derivatives

scientific article

Development of selective and reversible pyrazoline based MAO-A inhibitors: Synthesis, biological evaluation and docking studies.

scientific article published on 25 January 2010

Evaluation of in silico, in vitro α-amylase inhibition potential and antidiabetic activity of Pterospermum acerifolium bark

scientific article published on 30 September 2013

Exploration of chlorinated thienyl chalcones: A new class of monoamine oxidase-B inhibitors

scientific article published in June 2016

Exploring the Anticancer Effects of Brominated Plastoquinone Analogs with Promising Cytotoxic Activity in MCF-7 Breast Cancer Cells via Cell Cycle Arrest and Oxidative Stress Induction

scientific article published on 23 June 2022

Histone deacetylase inhibitors: a review on class-I specific inhibition

scientific article published on January 2015

Hydroxamates of para-aminobenzoic acid as selective inhibitors of HDAC8.

scientific article published on 3 September 2014

Inhibitors of human histone deacetylase: synthesis and enzyme assay of hydroxamates with piperazine linker

scientific article published in March 2010

Monoamine Oxidase Inhibitory Activity of Ferulic Acid Amides: Curcumin-Based Design and Synthesis

scientific article published on 23 November 2015

Monoamine Oxidase Inhibitory Activity of Novel Pyrazoline Analogues: Curcumin Based Design and Synthesis.

scientific article published in December 2015

Monoamine oxidase inhibitory activity of 2-aryl-4H-chromen-4-ones.

scientific article

Monoamine oxidase inhibitory activity of 3,5-biaryl-4,5-dihydro-1H-pyrazole-1-carboxylate derivatives.

scientific article

Novel Benzylidene Thiazolidinedione Derivatives as Partial PPARγ Agonists and their Antidiabetic Effects on Type 2 Diabetes

scientific article

Phytoestrogens and their synthetic analogues as substrate mimic inhibitors of CYP1B1

scientific article published on 17 November 2018

Potent and Selective Monoamine Oxidase-B Inhibitory Activity: Fluoro- vs. Trifluoromethyl-4-hydroxylated Chalcone Derivatives

scientific article published on 04 August 2016

Progress and prospects on DENV protease inhibitors.

scientific article published on 8 April 2016

Pyrazoline based MAO inhibitors: synthesis, biological evaluation and SAR studies.

scientific article published on 25 May 2011

Pyrazoline-based mycobactin analogues as MAO-inhibitors

scientific article

Reaching beyond HIV/HCV: nelfinavir as a potential starting point for broad-spectrum protease inhibitors against dengue and chikungunya virus

article

Small molecules with structural similarities to siderophores as novel antimicrobials against Mycobacterium tuberculosis and Yersinia pestis

scientific article

Structure based virtual screening of GSK-3beta: importance of protein flexibility and induced fit

scientific article published on 14 August 2009

Synthesis and molecular modelling studies of novel sulphonamide derivatives as dengue virus 2 protease inhibitors.

scientific article published on 29 July 2015

Synthesis and ribonucleotide reductase inhibitory activity of thiosemicarbazones

scientific article

Synthesis, Biochemistry, and Computational Studies of Brominated Thienyl Chalcones: A New Class of Reversible MAO-B Inhibitors.

scientific article published on 9 May 2016

Synthesis, antimicrobial and anticancer activity of new thiosemicarbazone derivatives

scientific article published on 25 November 2010

The Mycobactin Biosynthesis Pathway: A Prospective Therapeutic Target in the Battle against Tuberculosis

scientific article published on 29 December 2020

Thiazolidinediones and PPAR orchestra as antidiabetic agents: From past to present.

scientific article published on 10 December 2016

Thiazolidone derivatives as inhibitors of chikungunya virus

scientific article published on 16 October 2014

Thiosemicarbazone derivatives, thiazolyl hydrazones, effectively inhibit leukemic tumor cell growth: Down-regulation of ribonucleotide reductase activity and synergism with arabinofuranosylcytosine

scientific article published on 14 July 2017

Towards development of selective and reversible pyrazoline based MAO-inhibitors: Synthesis, biological evaluation and docking studies

scientific article published on 12 November 2009

Validation and method development of Tadalafil in bulk and tablet dosage form by RP-HPLC

scientific article published on 29 April 2014

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