List of works by Guillaume Médard

A new chemical probe for quantitative proteomic profiling of fibroblast growth factor receptor and its inhibitors

scientific article published on 31 October 2013

Characterization of a chemical affinity probe targeting Akt kinases

scientific article published on 3 July 2013

Chemical Proteomics Reveals Ferrochelatase as a Common Off-target of Kinase Inhibitors

scientific article published on 10 February 2016

Chemical Proteomics Uncovers EPHA2 as a Mechanism of Acquired Resistance to Small Molecule EGFR Kinase Inhibition

scientific article published on 26 May 2015

Chemical Proteomics and Structural Biology Define EPHA2 Inhibition by Clinical Kinase Drugs

scientific article published on 21 October 2016

Chemoproteomic Selectivity Profiling of PIKK and PI3K Kinase Inhibitors

scientific article published on 03 April 2019

Chemoproteomics-Aided Medicinal Chemistry for the Discovery of EPHA2 Inhibitors

scientific article

Comprehensive and reproducible phosphopeptide enrichment using iron immobilized metal ion affinity chromatography (Fe-IMAC) columns

scientific article

DMSO enhances electrospray response, boosting sensitivity of proteomic experiments

scientific article published on 25 August 2013

Decrypting drug actions and protein modifications by dose- and time-resolved proteomics

scientific article published on 16 March 2023

Dynamic Proteome Alteration and Functional Modulation of Human Saliva Induced by Dietary Chemosensory Stimuli

scientific article published on 29 May 2018

Effect of Astringent Stimuli on Salivary Protein Interactions Elucidated by Complementary Proteomics Approaches.

scientific article

Evaluation of Kinase Activity Profiling Using Chemical Proteomics

scientific article published on 17 September 2015

K+ Efflux-Independent NLRP3 Inflammasome Activation by Small Molecules Targeting Mitochondria

scientific article

Label-free quantitative proteome analysis of the surface-bound salivary pellicle

scientific article published on 6 January 2017

Mitigation of Acetylcholine Esterase Activity in the 1,7-Diazacarbazole Series of Inhibitors of Checkpoint Kinase 1

scientific article

N-Heterocyclic carbenes on close-packed coinage metal surfaces: bis-carbene metal adatom bonding scheme of monolayer films on Au, Ag and Cu.

scientific article published on 28 September 2017

NVP-BHG712: Effects of Regioisomers on the Affinity and Selectivity toward the EPHrin Family

scientific article published on 20 July 2018

New affinity probe targeting VEGF receptors for kinase inhibitor selectivity profiling by chemical proteomics.

scientific article published on 22 April 2014

Optimized chemical proteomics assay for kinase inhibitor profiling.

scientific article

ProteomeTools: Systematic Characterization of 21 Post-translational Protein Modifications by Liquid Chromatography Tandem Mass Spectrometry (LC-MS/MS) Using Synthetic Peptides

Salivary Proteome Patterns Affecting Human Salt Taste Sensitivity.

scientific article published on 5 October 2017

Snapshots of Dynamic Adaptation: Two-Dimensional Molecular Architectonics with Linear Bis-Hydroxamic Acid Modules

scientific article published on 27 November 2019

Studying epigenetic complexes and their inhibitors with the proteomics toolbox

scientific article

Surface anchors target golden bullets

scientific article published on 01 January 2019

Systematic Identification of MCU Modulators by Orthogonal Interspecies Chemical Screening

scientific article published in August 2017

Target and identify: triazene linker helps identify azidation sites of labelled proteins via click and cleave strategy

scientific article

Targeted Diazotransfer Reagents Enable Selective Modification of Proteins with Azides

scientific article published on 29 March 2017

The Inflammasome Drives GSDMD-Independent Secondary Pyroptosis and IL-1 Release in the Absence of Caspase-1 Protease Activity

scientific article

The target landscape of clinical kinase drugs

scientific article

Xanthohumol C, a minor bioactive hop compound: Production, purification strategies and antimicrobial test

scientific article published on 18 July 2018

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