Search filters

List of works by Roland J. Pieters

A New Chemical Probe for Proteomics of Carbohydrate-Binding Proteins

scientific article published on 01 February 2005

A facile synthesis of the GalNAcbeta1-->4Gal target sequence of respiratory pathogens.

scientific article published in October 2005

A hybrid polymer to target blood group dependence of cholera toxin

scientific article published on 01 December 2019

A new chemical probe for the detection of the cancer-linked galectin-3

scientific article published on 30 October 2006

A proteinaceous fraction of wheat bran may interfere in the attachment of enterotoxigenic E. coli K88 (F4+) to porcine epithelial cells

scientific article

Activity Based High-Throughput Screening for Novel O-GlcNAc Transferase Substrates Using a Dynamic Peptide Microarray

scientific article

Adhesion inhibition of F1C-fimbriated Escherichia coli and Pseudomonas aeruginosa PAK and PAO by multivalent carbohydrate ligands.

scientific article

Bacterial Adhesion of Streptococcus suis to Host Cells and Its Inhibition by Carbohydrate Ligands.

scientific article

Cross-platform comparison of glycan microarray formats.

scientific article published on 22 March 2014

Demystifying O-GlcNAcylation: hints from peptide substrates

scientific article published on 01 November 2018

Detection of galectin-3 by novel peptidic photoprobes

scientific article published on 21 October 2006

Detection of pathogenic Streptococcus suis bacteria using magnetic glycoparticles.

scientific article published on 22 March 2010

Development of a microarray detection method for galectin cancer proteins based on ligand binding ⬇️

scientific article published on November 10, 2012

Efficient microwave-assisted synthesis of multivalent dendrimeric peptides using cycloaddition reaction (click) chemistry

scientific article published on 19 August 2005

Efficient synthesis of phenylene-ethynylene rods and their use as rigid spacers in divalent inhibitors.

scientific article published on 31 January 2013

Enhanced Inhibition of Influenza A Virus Adhesion by Di- and Trivalent Hemagglutinin Inhibitors

scientific article published on 28 June 2019

Enhanced membrane pore formation by multimeric/oligomeric antimicrobial peptides

scientific article published on 18 October 2007

Enhancing membrane disruption by targeting and multivalent presentation of antimicrobial peptides

scientific article published on 14 April 2012

Functional Characterization of Cholera Toxin Inhibitors Using Human Intestinal Organoids

scientific article published on 27 June 2016

Functional assay for shiga-like toxin via detection by antibody capture and multivalent galabiose binding.

scientific article

Functionalization of a Rigid Divalent Ligand for LecA, a Bacterial Adhesion Lectin

scientific article published on 9 March 2015

Galectin-3-Binding Glycomimetics that Strongly Reduce Bleomycin-Induced Lung Fibrosis and Modulate Intracellular Glycan Recognition

scientific article

Homodimeric galectin-7 (p53-induced gene 1) is a negative growth regulator for human neuroblastoma cells

scientific article

ITAM-derived phosphopeptide-containing dendrimers as multivalent ligands for Syk tandem SH2 domain.

scientific article published on 7 August 2009

Identification of laminin-binding motifs of Yersinia pestis plasminogen activator by phage display

scientific article published in June 2005

Identification of peptide ligands for malignancy- and growth-regulating galectins using random phage-display and designed combinatorial peptide libraries.

scientific article

Inhibition and detection of galectins.

scientific article

Inhibition of O-GlcNAc transferase (OGT) by peptidic hybrids

scientific article published on 18 April 2018

Inhibition of P-fimbriated Escherichia coli adhesion by multivalent galabiose derivatives studied by a live-bacteria application of surface plasmon resonance.

scientific article published on 10 July 2007

Inhibition of Streptococcus suis adhesion by dendritic galabiose compounds at low nanomolar concentration.

scientific article

Interference of the galactose-dependent binding of lectins by novel pentapeptide ligands

scientific article published in March 2004

Intervention with bacterial adhesion by multivalent carbohydrates.

scientific article published on November 2007

Intracellular Hydrolysis of Small-Molecule O-Linked N-Acetylglucosamine Transferase Inhibitors Differs among Cells and Is Not Required for Its Inhibition

scientific article published on 25 July 2020

Lactulose synergizes with CpG-ODN to modulate epithelial and immune cells cross talk

scientific article published on 01 January 2019

Maximising multivalency effects in protein-carbohydrate interactions

scientific article published on 15 April 2009

Measuring O-GlcNAc cleavage by OGA and cell lysates on a peptide microarray

scientific article published on 29 May 2017

Microwave-assisted, tin-mediated, regioselective 3-O-alkylation of galactosides

Multivalent carbohydrate recognition on a glycodendrimer-functionalized flow-through chip.

scientific article published in July 2008

Multivalent glycoconjugates as anti-pathogenic agents ⬇️

scientific article

N-Guanidino Derivatives of 1,5-Dideoxy-1,5-imino-d-xylitol are Potent, Selective, and Stable Inhibitors of β-Glucocerebrosidase

scientific article published on 22 March 2017

Nanomolar affinity, iminosugar-based chemical probes for specific labeling of lysosomal glucocerebrosidase

scientific article published on 31 October 2009

New properties of wheat bran: anti-biofilm activity and interference with bacteria quorum-sensing systems

scientific article published on 04 April 2014

Optimizing divalent inhibitors of Pseudomonas aeruginosa lectin LecA by using a rigid spacer.

scientific article

Orthoester functionalized N-guanidino derivatives of 1,5-dideoxy-1,5-imino-d-xylitol as pH-responsive inhibitors of β-glucocerebrosidase

scientific article published on 10 October 2017

Peptide microarray analysis of the cross-talk between O-GlcNAcylation and tyrosine phosphorylation

scientific article published on 5 June 2017

PhoX - an IMAC-enrichable Crosslinking Reagent

PhoX: An IMAC-Enrichable Cross-Linking Reagent

scientific article published on 19 August 2019

Potent divalent inhibitors with rigid glucose click spacers for Pseudomonas aeruginosa lectin LecA

scientific article published on 19 March 2012

Potential scorpionate antibiotics: targeted hydrolysis of lipid II containing model membranes by vancomycin-TACzyme conjugates and modulation of their antibacterial activity by Zn-ions.

scientific article

Probing the Inhibitor versus Chaperone Properties of sp2-Iminosugars towards Human β-Glucocerebrosidase: A Picomolar Chaperone for Gaucher Disease

scientific article published on 17 April 2018

Rapid screening of lectins for multivalency effects with a glycodendrimer microarray

scientific article published on September 2010

Rationally Designed Chemically Modified Glycodendrimer Inhibits Streptococcus suis Adhesin SadP at Picomolar Concentrations.

scientific article published on 2 November 2017

Rigidified multivalent lactose molecules and their interactions with mammalian galectins: a route to selective inhibitors.

scientific article

Site-specific conjugation of single domain antibodies to liposomes enhances photosensitizer uptake and photodynamic therapy efficacy.

scientific article published on 08 March 2016

Strong Inhibition of Cholera Toxin B Subunit by Affordable, Polymer-Based Multivalent Inhibitors

scientific article published on 24 January 2019

Strong Inhibition of Cholera Toxin by Multivalent GM1 Derivatives

scientific article published on 01 September 2007

Strong inhibition of cholera toxin binding by galactose dendrimers.

scientific article published on 24 September 2007

Structural Insight into Multivalent Galactoside Binding to Pseudomonas aeruginosa Lectin LecA

scientific article

Study of cross talk between phosphatases and OGA on a ZO-3-derived peptide

scientific article published on 06 February 2019

Synthesis and biological activity of polygalloyl-dendrimers as stable tannic acid mimics

scientific article published in June 2002

Synthesis and cholera toxin binding properties of multivalent GM1 mimics

scientific article published on 30 June 2004

Synthesis and evaluation of TAC-based inhibitors of papain as mimics of cystatin B

scientific article published on 01 November 2007

Synthesis and evaluation of new thiodigalactoside-based chemical probes to label galectin-3.

scientific article

Synthesis and evaluation of novel macrocyclic antifungal peptides

scientific article published on 22 August 2011

Synthesis of multivalent Streptococcus suis adhesion inhibitors by enzymatic cleavage of polygalacturonic acid and 'click' conjugation.

scientific article published on 29 February 2008

Tannic acid mimicking dendrimers as small intestine submucosa stabilizing nanomordants.

scientific article published on 18 August 2005

Tetra- versus Pentavalent Inhibitors of Cholera Toxin ⬇️

scientific article published on 21 March 2015

The influence of ligand valency on aggregation mechanisms for inhibiting bacterial toxins

scientific article published in January 2009

The vancomycin-nisin(1-12) hybrid restores activity against vancomycin resistant Enterococci

scientific article

Thiodigalactoside-Bovine Serum Albumin Conjugates as High-Potency Inhibitors of Galectin-3: An Outstanding Example of Multivalent Presentation of Small Molecule Inhibitors.

scientific article

Thiourea-based spacers in potent divalent inhibitors of Pseudomonas aeruginosa virulence lectin LecA.

scientific article published on 15 September 2015

Tuning the preference of thiodigalactoside- and lactosamine-based ligands to galectin-3 over galectin-1

scientific article published on 23 January 2013

Uptake and transport of superparamagnetic iron oxide nanoparticles through human brain capillary endothelial cells

scientific article published on 26 August 2013

Use of tetravalent galabiose for inhibition of streptococcus suis serotype 2 infection in a mouse model

scientific article published on 08 April 2013

Paulina is supported by:

About Paulina

Help