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List of works by Jerome Waser

1,3-Difunctionalization of Aminocyclopropanes via Dielectrophilic Intermediates

scientific article published on 21 August 2019

1-Alkynyltriazenes as Functional Analogues of Ynamides

scientific article published on 16 September 2015

A Highly Chemoselective and Practical Alkynylation of Thiols

scientific article published on 18 June 2013

A Palladium-Catalyzed Aminoalkynylation Strategy towards Bicyclic Heterocycles: Synthesis of (±)-Trachelanthamidine

scientific article published on 15 April 2011

Alkynylation of Thiols with Ethynylbenziodoxolone (EBX) Reagents: α- or β- π-Addition?

scientific article published on 14 December 2015

Alkynylation of radicals: spotlight on the "Third Way" to transfer triple bonds

scientific article published on 13 August 2019

Alkynylation with Hypervalent Iodine Reagents

scientific article published on 01 January 2016

Alkynylations and Vinylations

Azidation of β-Keto Esters and Silyl Enol Ethers with a Benziodoxole Reagent

scientific article published on 17 June 2013

Benziodoxol(on)e Reagents as Tools in Organic Synthesis: The Background behind the Discovery at the Laboratory of Catalysis and Organic Synthesis

article

Benziodoxole-based hypervalent iodine reagents for atom-transfer reactions.

scientific article published on 27 August 2010

C-Terminal Bioconjugation of Peptides through Photoredox Catalyzed Decarboxylative Alkynylation

scientific article published on 08 May 2019

C2-Selective Direct Alkynylation of Indoles

scientific article published on 18 December 2012

Catalytic Enantioselective Ring-Opening Reactions of Cyclopropanes

scientific article published on 29 May 2020

Catalytic Enantiospecific [3+2] Annulation of Aminocyclopropanes with Ketones

scientific article published on 15 March 2012

Catalytic Formal Homo-Nazarov Cyclization

scientific article (publication date: 19 February 2009)

Catalytic Friedel–Crafts Reaction of Aminocyclopropanes

scientific article published on 01 July 2013

Catalytic Hydrohydrazination of a Wide Range of Alkenes with a Simple Mn Complex

scientific article published on 01 August 2004

Catalytic [3+2] Annulation of Aminocyclopropanes for the Enantiospecific Synthesis of Cyclopentylamines

scientific article published on 26 October 2011

Catalytic selective cyclizations of aminocyclopropanes: formal synthesis of aspidospermidine and total synthesis of goniomitine.

scientific article

Cobalt-Catalyzed Hydroazidation of Olefins: Convenient Access to Alkyl Azides

scientific article published on 01 June 2005

Cobalt-Catalyzed Hydrohydrazination of Dienes and Enynes:  Access to Allylic and Propargylic Hydrazides

scientific article published on 01 September 2005

Convenient synthesis of alkylhydrazides by the cobalt-catalyzed hydrohydrazination reaction of olefins and azodicarboxylates

scientific article

Copper-Catalyzed Oxy-Alkynylation of Diazo Compounds with Hypervalent Iodine Reagents

scientific article published on 12 February 2016

Copper-Catalyzed Oxyalkynylation of C-S Bonds in Thiiranes and Thiethanes with Hypervalent Iodine Reagents

scientific article published on 31 December 2019

Copper-Catalyzed Oxyvinylation of Diazo Compounds

scientific article published on 01 May 2020

Cyclic Hypervalent Iodine Reagents and Iron Catalysts: The Winning Team for Late-Stage CH Azidation

scientific article published on 30 March 2015

Cyclic Hypervalent Iodine Reagents for Atom-Transfer Reactions: Beyond Trifluoromethylation

scientific article published on 16 February 2016

Cyclic Hypervalent Iodine Reagents for Azidation: Safer Reagents and Photoredox-Catalyzed Ring Expansion

Cyclic Hypervalent Iodine Reagents: Enabling Tools for Bond Disconnection via Reactivity Umpolung

scientific article published on 28 November 2018

Cyclization and annulation reactions of nitrogen-substituted cyclopropanes and cyclobutanes

scientific article published on 27 June 2014

C‐Terminal Bioconjugation of Peptides through Photoredox Catalyzed Decarboxylative Alkynylation

Dearomatization of electron poor six-membered N-heterocycles through [3 + 2] annulation with aminocyclopropanes

scientific article published on 25 August 2017

Direct Alkynylation of Thiophenes: Cooperative Activation of TIPS-EBX with Gold and Brønsted Acids

scientific article published on 01 September 2010

Direct alkynylation of indole and pyrrole heterocycles

scientific article published in January 2009

Divergent Access to (1,1) and (1,2)-Azidolactones from Alkenes using Hypervalent Iodine Reagents

scientific article

Divergent Reactivity of Thioalkynes in Lewis Acid Catalyzed Annulations with Donor-Acceptor Cyclopropanes

scientific article published on 19 July 2016

Dynamic Kinetic Asymmetric [3 + 2] Annulation Reactions of Aminocyclopropanes

scientific article published on 21 April 2014

Electrophilic alkynylation: the dark side of acetylene chemistry

scientific article published on 18 April 2012

Enantioselective Carboetherification/Hydrogenation for the Synthesis of Amino Alcohols via a Catalytically Formed Chiral Auxiliary

scientific article published on 02 October 2020

Enantioselective Copper-Catalyzed Oxy-Alkynylation of Diazo Compounds

scientific article published on 16 June 2017

Enantioselective Synthesis of Homoallylic Azides and Nitriles via Palladium-Catalyzed Decarboxylative Allylation

scientific article published on 18 November 2015

Enantioselective synthesis of polycyclic carbocycles via an alkynylation-allylation-cyclization strategy

scientific article published on 15 October 2014

Ethynyl Benziodoxolones for the Direct Alkynylation of Heterocycles: Structural Requirement, Improved Procedure for Pyrroles, and Insights into the Mechanism

scientific article published on 21 March 2012

Ethynyl benziodoxolones: functional terminators for cell-penetrating poly(disulfide)s

Ethynyl-1,2-benziodoxol-3(1 H)-one (EBX): An Exceptional Reagent for the Ethynylation of Keto, Cyano, and Nitro Esters

scientific article published on 01 August 2010

Ethynylbenziodazolones (EBZ) as Electrophilic Alkynylation Reagents for the Highly Enantioselective Copper‐Catalyzed Oxyalkynylation of Diazo Compounds

scientific article published on 16 May 2019

Fast and highly chemoselective alkynylation of thiols with hypervalent iodine reagents enabled through a low energy barrier concerted mechanism

scientific article published on 13 November 2014

Fine-tuned organic photoredox catalysts for fragmentation-alkynylation cascades of cyclic oxime ethers

scientific article published on 21 July 2018

Formal Homo-Nazarov and Other Cyclization Reactions of Activated Cyclopropanes

scientific article published on 23 November 2011

Frontispiece: Indole- and Pyrrole-BX: Bench-Stable Hypervalent Iodine Reagents for Heterocycle Umpolung

General and Practical Formation of Thiocyanates from Thiols

scientific article published on 17 December 2014

Gold-Catalyzed Regioselective Synthesis of 2- and 3-Alkynyl Furans

scientific article published on 10 May 2013

Gold-catalyzed direct alkynylation of tryptophan in peptides using TIPS-EBX.

scientific article published on 19 April 2016

Gold-catalyzed domino cyclization-alkynylation reactions with EBX reagents: new insights into the reaction mechanism

scientific article published on 6 September 2017

Heterotetracenes: Flexible Synthesis and in Silico Assessment of the Hole-Transport Properties

scientific article published on 13 April 2017

Hydrazines and Azides via the Metal-Catalyzed Hydrohydrazination and Hydroazidation of Olefins

scientific article published on 01 September 2006

In situ tether formation from amines and alcohols enabling highly selective Tsuji-Trost allylation and olefin functionalization

scientific article

Indole Alkaloids Synthesis via a Selective Cyclization of Aminocyclopropanes ⬇️

scientific article published on January 1, 2012

Indole- and Pyrrole-BX: Bench-Stable Hypervalent Iodine Reagents for Heterocycle Umpolung

scientific article

Intramolecular palladium-catalyzed alkene carboalkynylation

Iridium- and Rhodium-Catalyzed Directed C-H Heteroarylation of Benzaldehydes with Benziodoxolone Hypervalent Iodine Reagents

scientific article published on 21 February 2018

Iron-Catalyzed [3 + 2] Annulation of Aminocyclopropanes with Aldehydes: Stereoselective Synthesis of Aminotetrahydrofurans

scientific article published on 21 December 2011

Lewis Acid Catalyzed Enantioselective Desymmetrization of Donor-Acceptor meso-Diaminocyclopropanes

scientific article published on 20 February 2018

Low-Temperature Intramolecular [4+2] Cycloaddition of Allenes with Arenes for the Synthesis of Diene Ligands

scientific article published on 20 November 2020

Low‐Temperature Intramolecular [4+2] Cycloaddition of Allenes with Arenes for the Synthesis of Diene Ligands

scientific article

Metal-Free Electrophilic Alkynylation of Sulfenate Anions with Ethynylbenziodoxolone Reagents.

scientific article

Metal-Free Oxidative Cross Coupling of Indoles with Electron-Rich (Hetero)arenes

scientific article published on 03 May 2018

One-Pot Three-Component Synthesis of Vicinal Diamines via In Situ Aminal Formation and Carboamination

scientific article published on 16 September 2016

One-Pot Three-Component Synthesis of Vicinal Diamines via In Situ Aminal Formation and Carboamination

One-pot gold-catalyzed synthesis of 3-silylethynyl indoles from unprotected o-alkynylanilines ⬇️

scientific article published on 4 May 2011

One-pot, three-component arylalkynyl sulfone synthesis

scientific article published on 29 January 2015

Palladium-Catalyzed Carbo-Oxygenation of Propargylic Amines using in Situ Tether Formation

scientific article published on 29 January 2019

Palladium-Catalyzed Carboamination of Allylic Alcohols Using a Trifluoroacetaldehyde-Derived Tether.

scientific article published on 13 June 2017

Palladium-Catalyzed Carboxy-Alkynylation of Propargylic Amines Using Carbonate Salts as Carbon Dioxide Source

Palladium-Catalyzed Vicinal Amino Alcohols Synthesis from Allyl Amines by In Situ Tether Formation and Carboetherification

scientific article published on 26 February 2015

Para-Selective Gold-Catalyzed Direct Alkynylation of Anilines

scientific article published on 19 January 2012

Pd(0)-Catalyzed Alkene Oxy- and Aminoalkynylation with Aliphatic Bromoacetylenes

scientific article published on 19 March 2013

Pd(0)-Catalyzed Oxy- and Aminoalkynylation of Olefins for the Synthesis of Tetrahydrofurans and Pyrrolidines

scientific article published on 09 November 2011

Pd-catalyzed intramolecular oxyalkynylation of alkenes with hypervalent iodine

scientific article published in January 2010

Photocatalysis with organic dyes: facile access to reactive intermediates for synthesis

scientific article published on 29 May 2020

Photocatalytic redox reactions for in-source peptide fragmentation

scientific article

Platinum-catalyzed domino reaction with benziodoxole reagents for accessing benzene-alkynylated indoles.

scientific article published on 10 March 2015

Proteome-Wide Profiling of Targets of Cysteine reactive Small Molecules by Using Ethynyl Benziodoxolone Reagents.

scientific article

Revisiting the Urech Synthesis of Hydantoins: Direct Access to Enantiopure 1,5-Substituted Hydantoins Using Cyanobenziodoxolone

scientific article published on 07 January 2019

Rhodium-catalyzed C-H functionalization of heteroarenes using indoleBX hypervalent iodine reagents.

scientific article

Room temperature alkynylation of H-phosphi(na)tes and secondary phosphine oxides with ethynylbenziodoxolone (EBX) reagents

scientific article published in November 2014

Room temperature decarboxylative cyanation of carboxylic acids using photoredox catalysis and cyanobenziodoxolones: a divergent mechanism compared to alkynylation

scientific article published on 22 December 2016

Room-Temperature Decarboxylative Alkynylation of Carboxylic Acids Using Photoredox Catalysis and EBX Reagents

scientific article published on 24 July 2015

Stereoselective synthesis of alkyl-, aryl-, vinyl- and alkynyl-substituted -enamides and enol ethers

Synthesis of (carbo)nucleoside analogues by [3+2] annulation of aminocyclopropanes.

scientific article

Synthesis of Thiochromans via [3+3] Annulation of Aminocyclopropanes with Thiophenols

scientific article published on 10 November 2020

Synthesis of aminocyclobutanes by iron-catalyzed [2+2] cycloaddition

scientific article

Synthesis of bicyclo[3.1.0]hexanes by (3 + 2) annulation of cyclopropenes with aminocyclopropanes

scientific article published on 08 October 2019

Taming Hypervalent Bonds and Strained Rings for Catalysis and Synthesis

scientific article published on 01 January 2014

Tandem Photoredox and Copper-Catalyzed Decarboxylative C(sp3)-N Coupling of Anilines and Imines Using an Organic Photocatalyst

scientific article published on 29 June 2020

Total synthesis and biological evaluation of jerantinine E.

scientific article published on 14 October 2013

Total synthesis of (-)-pseudolaric acid B

scientific article

Total synthesis of (-)-pseudolaric acid B

scientific article published in 2008

Triazene-Activated Donor-Acceptor Cyclopropanes: Ring-Opening and (3 + 2) Annulation Reactions

scientific article published on 26 May 2020

Zinc-gold cooperative catalysis for the direct alkynylation of benzofurans.

scientific article published on 29 August 2013

[4 + 2]-Annulations of Aminocyclobutanes

scientific article published on 04 February 2015

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