Search filters

Authors whose works are in public domain in at least one jurisdiction

List of works by Daniel Hoyer

(+/-)[125Iodo] cyanopindolol, a new ligand for beta-adrenoceptors: identification and quantitation of subclasses of beta-adrenoceptors in guinea pig.

scientific article published in January 1981

125ITyr10-cortistatin14 labels all five somatostatin receptors ⬇️

scientific article published on May 1, 1998

125IodoBE 2254, a New Radioligand for α1-Adrenoceptors ⬇️

scientific article published on January 1, 1982

5-HT Receptor Classification and Nomenclature: Towards a Harmonization with the Human Genome ⬇️

scientific article published on April 1, 1997

5-HT Receptor Nomenclature: Naming Names, Does It Matter? A Tribute to Maurice Rapport

scientific article published on 7 March 2017

5-HT-1 Receptors

5-HT-1A Receptor

5-HT-1B Receptor

5-HT-1D Receptor

5-HT-1E Receptor

5-HT-1F Receptor

5-HT-2 Receptors

5-HT-2A Receptor

5-HT-2B Receptor

5-HT-2C Receptor

5-HT-3 Receptor

5-HT-3A Receptor

5-HT-3B Receptor

5-HT-4 Receptor

5-HT-5 Receptors

5-HT-6 Receptor

5-HT-7 Receptor

5-HT1-like receptors mediate 5-hydroxytryptamine-induced contraction of guinea-pig isolated iliac artery ⬇️

scientific article published on February 1, 1991

5-HT1A-receptors mediate stimulation of adenylate cyclase in rat hippocampus

scientific article published in August 1986

5-HT1D receptor-mediated inhibition of forskolin-stimulated adenylate cyclase activity in calf substantia nigra

scientific article

5-Hydroxytryptamine (5-HT) receptor superfamilies

5-Hydroxytryptamine Receptors

5-Hydroxytryptamine1 recognition sites in rat brain: Heterogeneity of non-5-hydroxytryptamine1a/1c binding sites revealed by quantitative receptor autoradiography

scientific article published on 01 March 1993

5-hydroxytryptamine3 receptors in the human brain: autoradiographic visualization using [3H]ICS 205-930.

scientific article published in January 1989

A Comparative Study of Outer Membrane Proteome between Paired Colistin-Susceptible and Extremely Colistin-Resistant Klebsiella pneumoniae Strains

A comparative autoradiographic study of 5-HT1D binding sites in human and guinea-pig brain using different radioligands

scientific article published in January 1994

A proposed new nomenclature for 5-HT receptors.

scientific article

A short history of the 5-HT2C receptor: from the choroid plexus to depression, obesity and addiction treatment

scientific article published on 7 March 2017

ABP688, a novel selective and high affinity ligand for the labeling of mGlu5 receptors: identification, in vitro pharmacology, pharmacokinetic and biodistribution studies

scientific article published on 21 October 2006

AQW051, a novel, potent and selective α7 nicotinic ACh receptor partial agonist: pharmacological characterization and phase I evaluation

scientific article

Adult siRNA-induced knockdown of mGlu7 receptors reduces anxiety in the mouse

scientific article published on 17 April 2013

Agonist properties of putative small-molecule somatostatin sst2 receptor-selective antagonists

scientific article published on April 2003

Agonist/antagonist interactions with cloned human 5-HT1A receptors: variations in intrinsic activity studied in transfected HeLa cells

scientific article published on 01 March 1992

Alignment of receptor nomenclature with the human genome: classification of 5-HT1B and 5-HT1D receptor subtypes.

scientific article published on March 1996

An invitation for comprehensive single-compound reviews on the pharmacological properties of newly launched drugs

scholarly article by Martin C. Michel et al published 22 September 2013 in Naunyn-Schmiedeberg's Archives of Pharmacology

Animal Models of Addiction and Neuropsychiatric Disorders and Their Role in Drug Discovery: Honoring the Legacy of Athina Markou

scientific article published on 22 February 2018

Antidepressants influence somatostatin levels and receptor pharmacology in brain

scientific journal article

Anxiety and increased 5-HT1A receptor response in NCAM null mutant mice

scientific article

Applications of a rat multiple tissue gene expression data set.

scientific article published in April 2004

Assessing allosteric ligand-receptor interactions

Astrocytes: Adhesion Molecules and Immunomodulation

scientific article published in January 2016

Autoradiographic analysis of somatostatin SRIF1 and SRIF2 receptors in the human brain and pituitary

scientific article published on 01 February 1997

Autoradiography of 5-HT receptors: A critical appraisal

scientific article published on 01 January 1991

Beta(2)/beta(3)-di- and alpha/beta(3)-tetrapeptide derivatives as potent agonists at somatostatin sst(4) receptors

scientific article published on 24 January 2003

Binding and functional properties of the novel somatostatin analogue KE 108 at native mouse somatostatin receptors

scientific article

Binding characteristics of (+)-, (+/-)- and (-)-[125iodo] cyanopindolol to guinea-pig left ventricle membranes

scientific article published in March 1982

Binding of 125I-cyanopindolol to beta-1-adrenoceptors in a high and low affinity state

scientific article

Biological activity of somatostatin receptors in GC rat tumour somatotrophs: evidence with sst1-sst5 receptor-selective nonpeptidyl agonists

scientific article published in April 2003

Blunted 5-HT1A receptor-mediated responses and antidepressant-like behavior in mice lacking the GABAB1a but not GABAB1b subunit isoforms.

scientific article published on 9 January 2017

Brain somatostatin: a candidate inhibitory role in seizures and epileptogenesis.

scientific article

Brain sphingosine-1-phosphate receptors: implication for FTY720 in the treatment of multiple sclerosis

scientific article published on 08 September 2007

Calcineurin inhibits desensitization of cloned rat 5-HT1C receptors

scientific article published on September 1993

Changes of AMPA receptors in MPTP monkeys with levodopa-induced dyskinesias

scientific article

Characterisation of 5-HT3 recognition sites in membranes of NG 108-15 neuroblastoma-glioma cells with [3H]ICS 205-930.

scientific article

Characterisation of human recombinant somatostatin receptors. 1. Radioligand binding studies

scientific article

Characterisation of human recombinant somatostatin receptors. 4. Modulation of phospholipase C activity.

scientific article

Characterisation of the fish sst3 receptor, a member of the SRIF1 receptor family: atypical pharmacological features.

scientific article published on March 1999

Characterization and distribution of somatostatin SS-1 and SRIF-1 binding sites in rat brain: identitity with SSTR-2 receptors

scientific article published on 01 March 1995

Characterization of IBE 2254 Binding to Alpha - Adrenergic Receptors on Intact DDT Smooth Muscle Cells: Comparison with Membrane1Binding and Correlation with Phosphoinositides Breakdown ⬇️

scientific article published on January 1, 1984

Characterization of the 5-HT1B recognition site in rat brain: binding studies with (-)[125I]iodocyanopindolol

scientific article published in November 1985

Chronic mianserin or eltoprazine treatment in rats: effects on the elevated plus-maze test and on limbic 5-HT2C receptor levels

scientific article published in September 1994

Classification and nomenclature of somatostatin receptors

scientific article

Cloning, expression, functional coupling and pharmacological characterization of the rat dopamine D 4 receptor

scientific article published on 01 May 2000

Co-expression of somatostatin SSTR-3 and SSTR-4 receptor messenger RNAs in the rat brain

scientific article published on 01 January 1995

Comparison of functional profiles at human recombinant somatostatin sst2 receptor: simultaneous determination of intracellular Ca2+ and luciferase expression in CHO-K1 cells

scientific article published on 22 March 2004

Compensatory changes in the hippocampus of somatostatin knockout mice: upregulation of somatostatin receptor 2 and its function in the control of bursting activity and synaptic transmission

scientific article published in May 2006

Competitive antagonism by recognized 5-HT2 receptor antagonists at 5-HT1C receptors in pig choroid plexus

scientific article published on August 1991

Competitive interaction of agonists and antagonists with 5-HT3 recognition sites in membranes of neuroblastoma cells labelled with [3H]ICS 205-930.

scientific article published in January 1989

Contemporary Anti-Ebola Drug Discovery Approaches and Platforms

Coupling of human nicotinic acetylcholine receptors alpha 7 to calcium channels in GH3 cells.

scientific article published on 24 December 2004

Curcumin Attenuates Colistin-Induced Peripheral Neurotoxicity in Mice

scientific article published on 20 February 2020

Decahydroisoquinoline derivatives as novel non-peptidic, potent and subtype-selective somatostatin sst(3) receptor antagonists

scientific article published on 21 January 2010

Design and Synthesis of γ-Dipeptide Derivatives with Submicromolar Affinities for Human Somatostatin Receptors

scientific article published on 01 February 2003

Design, synthesis, and biological activities of potent and selective somatostatin analogues incorporating novel peptoid residues.

scientific article published in July 1998

Differential Expression of Five Somatostatin Receptor Subtypes, SSTR1-5, in the CNS and Peripheral Tissue ⬇️

scientific article published on 01 January 1994

Direct visualization of serotonin1D receptors in the human brain using a new iodinated radioligand

scientific article (publication date: March 1992)

Discovery of 1H-pyrazolo[3,4-b]pyridines as potent dual orexin receptor antagonists (DORAs).

scientific article published on 19 October 2015

Discovery of novel non-peptidic beta-alanine piperazine amide derivatives and their optimization to achiral, easily accessible, potent and selective somatostatin sst1 receptor antagonists

scientific article published on 27 January 2009

Distinct effects of IPSU and suvorexant on mouse sleep architecture

scientific article published on 10 December 2013

Distinct functional properties of native somatostatin receptor subtype 5 compared with subtype 2 in the regulation of ACTH release by corticotroph tumor cells.

scientific article published on 15 March 2005

Distribution and characterisation of somatostatin receptor mRNA and binding sites in the brain and periphery.

scientific article published on May 2000

Distribution and second messenger coupling of four somatostatin receptor subtypes expressed in brain

scientific article

Distribution of 5-HT Receptors in the Central Nervous System

Drug design at peptide receptors: somatostatin receptor ligands

scientific article

Editorial: Reporting guidelines for psychopharmacology

scientific article published on 26 February 2016

Effect of 5,7-dihydroxytryptamine lesion on mianserin-induced conditioned place aversion and on 5-hydroxytryptamine1C receptors in the rat brain

scientific article published in October 1993

Effect of somatostatin on nitric oxide production in human retinal pigment epithelium cell cultures

scientific article published in May 2004

Embryonic and postnatal mRNA distribution of five somatostatin receptor subtypes in the rat brain

scientific article published on 01 December 1995

Emerging use of non-viral RNA interference in the brain

scientific article published in April 2007

Endothelin receptors in the human coronary artery, ventricle and atrium

article

Ergoline derivatives as highly potent and selective antagonists at the somatostatin sst 1 receptor

scientific article published on 26 December 2007

Evidence for the presence of 5-HT1B receptor messenger RNA in neurons of the rat trigeminal ganglia

article

Experimental design and analysis and their reporting II: updated and simplified guidance for authors and peer reviewers

scientific article published in April 2018

Experimental design and analysis and their reporting: new guidance for publication in BJP.

scientific article published on July 2015

Extended radioligand binding profile of iloperidone: a broad spectrum dopamine/serotonin/norepinephrine receptor antagonist for the management of psychotic disorders

scientific article published in December 2001

Fish somatostatin sst3 receptor: comparison of radioligand and GTPgammaS binding, adenylate cyclase and phospholipase C activities reveals different agonist-dependent pharmacological signatures.

scientific article published on January 2005

Functional characterisation of the putative somatostatin sst2 receptor antagonist CYN 154806.

scientific article

Functional effects of d-Phe-c[Cys-Tyr-d-Trp-Lys-Val-Cys]-Trp-NH2 and differential changes in somatostatin receptor messenger RNAs, binding sites and somatostatin release in kainic acid-treated rats

scientific article published on 01 April 1995

Genetic deletion of somatostatin receptor 1 alters somatostatinergic transmission in the mouse retina

scientific article published in December 2003

Global down-regulation of gene expression in the brain using RNA interference, with emphasis on monoamine transporters and GPCRs: implications for target characterization in psychiatric and neurological disorders

scientific article published in January 2006

Goals and practicalities of immunoblotting and immunohistochemistry: A guide for submission to the British Journal of Pharmacology

scientific article published in February 2018

High affinity of SDZ HTF-919 related molecules for calf and human caudate 5-HT4 receptors

scientific article

Highly N-Methylated Somatostatin Analogs: Synthesis, Biological Activity and Structure-Activity Relationship Studies

Hippocampal 5-HT7 receptors signal phosphorylation of the GluA1 subunit to facilitate AMPA receptor mediated-neurotransmission in vitro and in vivo

scientific article published on 15 January 2016

Hippocampal sst(1) receptors are autoreceptors and do not affect seizures in rats

scientific article published in March 2010

Homogeneous 5-HT1D recognition sites in the human substantia nigra identified with a new iodinated radioligand

scientific article published in September 1991

Hyperdopaminergia and altered locomotor activity in GABAB1-deficient mice.

scientific article published on 5 April 2006

Hypnotics with novel modes of action

scientific article published on 17 January 2020

Identification and SAR of potent and selective non-peptide obeline somatostatin sst1 receptor antagonists

article

Identification and characterization of a type five-like somatostatin receptor in goldfish pituitary

scientific article

Identification and pharmacological characterization of somatostatin receptors in rat lung

scientific article published in July 1997

Identification of 5HT2-receptors on longitudinal muscle of the guinea pig ileum

scientific article published in January 1984

Identification of a 5-HT1 recognition site in human brain membranes different from 5-HT1A, 5-HT1B and 5-HT1C sites

scientific article

Identification of a novel series of orexin receptor antagonists with a distinct effect on sleep architecture for the treatment of insomnia

scientific article published on 18 September 2013

Identification of serotonin 5-HT3 recognition sites by radioligand binding in NG108-15 neuroblastoma-glioma cells

scientific article published on 01 November 1987

Identity of inhibitory presynaptic 5-hydroxytryptamine (5-HT) autoreceptors in the rat brain cortex with 5-HT1B binding sites

scientific article published in January 1986

Impact of the human genome project on the principles for classification and nomenclature of 5-HT receptors

scientific article

Implications of stereoselectivity in radioligand binding studies

Improving Oral Bioavailability of Peptides by Multiple N-Methylation: Somatostatin Analogues

scientific article published on 01 January 2008

Increased exploratory activity of APP23 mice in a novel environment is reversed by siRNA.

scientific article

Inhibition of 5-carboxamidotryptamine-induced relaxation of guinea-pig ileum correlates with [125I]LSD binding

scientific article published on 01 September 1986

Inhibition of cAMP Accumulation Via Recombinant Human Serotonin 5-HT 1A Receptors: Considerations on Receptor Effector Coupling across Systems ⬇️

scientific article published on April 1, 1997

Interaction of psychotropic drugs with central 5-HT3 recognition sites: fact or artifact?

scientific article published on 01 November 1989

Interaction of the alpha-adrenoceptor agonist oxymetazoline with serotonin 5-HT1A, 5-HT1B, 5-HT1C and 5-HT1D receptors

scientific article

Interfering with the brain: use of RNA interference for understanding the pathophysiology of psychiatric and neurological disorders

scientific article

Is the sumatriptan (GR 43175)-induced endothelium-dependent relaxation of pig coronary arteries mediated by 5-HT1D receptors?

scientific article published in July 1989

JN403, in vitro characterization of a novel nicotinic acetylcholine receptor alpha7 selective agonist

scientific article published on 25 January 2007

Kinetic properties of "dual" orexin receptor antagonists at OX1R and OX2R orexin receptors

scientific article published on 3 December 2013

Lemborexant. Dual orexin receptor antagonist, Treatment of insomnia

Linear, Peptidase-Resistantβ2/β3-Di- andα/β3-Tetrapeptide Derivatives with Nanomolar Affinities to a Human Somatostatin Receptor, Preliminary Communication

article by Dieter Seebach et al published 14 November 2001 in Helvetica Chimica Acta

Localisation by autoradiography of neuronal 5-HT3 receptors in the mouse CNS

scientific article published on 01 July 1988

Localization of somatostatin (SRIF) SSTR-1, SSTR-2 and SSTR-3 receptor mRNA in rat brain by in situ hybridization.

scientific article published on February 1994

Localization of the 5-hydroxytryptamine2C receptor protein in human and rat brain using specific antisera.

scientific article

Mechanistic Insights From Global Metabolomics Studies into Synergistic Bactericidal Effect of a Polymyxin B Combination With Tamoxifen Against Cystic Fibrosis MDR

scholarly article by Maytham Hussein et al published 2018 in Computational and Structural Biotechnology Journal

Mesulergine, a selective serotonin-2 ligand in the rat cortex, does not label these receptors in porcine and human cortex: evidence for species differences in brain serotonin-2 receptors

scientific article published in November 1984

Metabolomics Study of the Synergistic Killing of Polymyxin B in Combination with Amikacin against Polymyxin-Susceptible and -Resistant Pseudomonas aeruginosa

scientific article published on 20 December 2019

Molecular Mechanisms of Neurotoxicity Induced by Polymyxins and Chemoprevention

Molecular biology of 5-HT receptors

scientific article

Molecular biology of 5-HT receptors

scholarly article

Molecular cloning and pharmacological characterization of a somatostatin receptor subtype in the gymnotiform fish Apteronotus albifrons.

scientific article

Molecular pharmacology of 5-HT1 and 5-HT2 recognition sites in rat and pig brain membranes: radioligand binding studies with [3H]5-HT, [3H]8-OH-DPAT, (-)[125I]iodocyanopindolol, [3H]mesulergine and [3H]ketanserin

scientific article published on November 1985

Molecular pharmacology of 5-HT1D recognition sites: radioligand binding studies in human, pig and calf brain membranes

scientific article

Molecular pharmacology of somatostatin receptors

scientific article published on November 1994

Molecular pharmacology of somatostatin-receptor subtypes.

scientific article published on September 1994

Molecular, pharmacological and functional diversity of 5-HT receptors

scientific article (publication date: April 2002)

NMR-Solution Structures and Affinities for the Human Somatostatin G-Protein-Coupled Receptors hsst1â 5 of CF3 Derivatives of Sandostatin® (Octreotide)

Native somatostatin sst2 and sst5 receptors functionally coupled to Gi/o-protein, but not to the serum response element in AtT-20 mouse tumour corticotrophs

scientific article published on 15 May 2003

Neurochemical and behavioral consequences of widespread gene knockdown in the adult mouse brain by using nonviral RNA interference

scholarly article

Neuropeptide Receptors – Drug Development

article

Neuropeptide receptor positive allosteric modulation in epilepsy: galanin modulation revealed

scientific article

Neuropeptides and neuropeptide receptors: drug targets, and peptide and non-peptide ligands: a tribute to Prof. Dieter Seebach

scientific article

Neuropeptidomics of mouse hypothalamus after imipramine treatment reveal somatostatin as a potential mediator of antidepressant effects

scientific article

New Open-Chain and Cyclic Tetrapeptides, Consisting ofα-,β2-, andβ3-Amino-Acid Residues, as Somatostatin Mimics - A Survey

New perspective in peptide chemistry by N-alkylation

scientific article published in January 2009

Non-specific uptake of the radioligand 125I-IHYP by intact human lymphocytes: Reversal of the uptake process

scientific article published on 01 March 1982

Novel, potent, and radio-iodinatable somatostatin receptor 1 (sst1) selective analogues

scientific article published on May 2009

Orexin OX2 Receptor Antagonists as Sleep Aids

scientific article published on 2 December 2016

Orexin Receptor Antagonists

Orexin in sleep, addiction and more: is the perfect insomnia drug at hand?

scientific article

Paroxetine combined with a 5-HT(1A) receptor antagonist reversed reward deficits observed during amphetamine withdrawal in rats

scientific article published on 25 September 2004

Pathological Conditions Associated with the Disturbance of the 5-HT System

Peptide folding induces high and selective affinity of a linear and small beta-peptide to the human somatostatin receptor 4.

scientific article

Pharmacological characterisation of 5-HT receptors positively coupled to adenylyl cyclase in the rat hippocampus

scientific article

Pharmacological characterisation of native somatostatin receptors in AtT-20 mouse tumour corticotrophs

scientific article published on May 2003

Pharmacological characterisation of the goldfish somatostatin sst5 receptor

scientific article published on February 2002

Pharmacological profile of somatostatin and cortistatin receptors

scientific article published on 23 December 2007

Polymyxins for CNS infections: Pharmacology and neurotoxicity

scientific article

Preface

Presence of somatostatin sst2 receptors in the developing rat auditory system

scientific article published in December 1996

Proceedings of Neuropeptides 2004, the XIV European Neuropeptides Club meeting.

scientific article published in December 2004

RNA interference as a therapeutic strategy for treating CNS disorders

scientific article published on 28 November 2006

Rapamycin confers neuroprotection against colistin-induced oxidative stress, mitochondria dysfunction and apoptosis through the activation of autophagy and mTOR/Akt/CREB signaling pathways

scientific article published on 19 December 2017

Reaction of Fe3(CO)12 with octreotide--chemical, electrochemical and biological investigations

scientific article published on 2 February 2010

Receptor biochemistry and methodology volume 15: Serotonin receptor subtypes

scholarly article by Daniel Hoyer published January 1991 in Trends in Pharmacological Sciences

Receptor density as a factor governing the efficacy of the dopamine D4 receptor ligands, L-745,870 and U-101958 at human recombinant D4.4 receptors expressed in CHO cells

scientific article published in October 1999

Recovery of emotional behaviour in neural cell adhesion molecule (NCAM) null mutant mice through transgenic expression of NCAM180.

scientific article published in September 2000

Region-specific transcriptional changes following the three antidepressant treatments electro convulsive therapy, sleep deprivation and fluoxetine

scientific article published on 10 October 2006

Reviewer comments on Reflections on drug research by Sir James Black

scientific article published on November 2010

SAR of the arylpiperazine moiety of obeline somatostatin sst1 receptor antagonists

scientific article published on 30 April 2007

SDZ 216-525, a selective and potent 5-HT1A receptor antagonist

scientific article published in February 1993

SMAD4 protein is decreased in the dorsolateral prefrontal and anterior cingulate cortices in schizophrenia

scientific article published on 02 March 2020

SOM230: A New Therapeutic Modality for Cushing's Disease

scientific article published on 01 January 2014

SRA880, in vitro characterization of the first non-peptide somatostatin sst(1) receptor antagonist

scientific article

SST-1 Somatostatin Receptor

SST-2 Somatostatin Receptor

SST-3 Somatostatin Receptor

SST-4 Somatostatin Receptor

SST-5 Somatostatin Receptor

Saving, changing and repairing lives

Selective effects of benzodiazepines on the acquisition of conditioned taste aversion compared to attenuation of neophobia in C57BL/6 mice.

scientific article published on 22 July 2009

Separating Probability and Reversal Learning in a Novel Probabilistic Reversal Learning Task for Mice

scientific article published on 01 January 2019

Serotonin increases the production of inositol phosphates and mobilises calcium via the 5-HT2 receptor in A7r5 smooth muscle cells

scientific article published in June 1986

Serotonin receptors in the human brain. I. Characterization and autoradiographic localization of 5-HT1A recognition sites. Apparent absence of 5-HT1B recognition sites

scientific article published in June 1986

Serotonin receptors in the human brain. II. Characterization and autoradiographic localization of 5-HT1C and 5-HT2 recognition sites

scientific article published in June 1986

Serotoninergic System

Sex differences in mouse models of fear inhibition: Fear extinction, safety learning, and fear–safety discrimination

scientific article published on 15 April 2019

Sex: A change in our guidelines to authors to ensure that this is no longer an ignored experimental variable

scientific article published on 23 August 2019

Similar distribution of [125I]sarafotoxin-6b and [125I]endothelin-1, -2, -3 binding sites in the human kidney

scientific article published on 01 February 1990

Somatostatin

Somatostatin

Somatostatin Receptor Gene Family - Subtype Selectivity for Ligand Binding

article

Somatostatin Receptors

Somatostatin receptor 1 selective analogues: 2. N(alpha)-Methylated scan

scientific article published in January 2005

Somatostatin receptor subtypes 2 and 4 affect seizure susceptibility and hippocampal excitatory neurotransmission in mice

scientific article published in September 2002

Somatostatin receptors differentially affect spontaneous epileptiform activity in mouse hippocampal slices

scientific article published in November 2004

Somatostatin receptors in the Rhesus monkey brain: localization and pharmacological characterization

scientific article published on 01 May 1996

Somatostatin receptors in the developing rat brain

scientific article published in February 1996

Somatostatin receptors in wildtype and somatostatin deficient mice and their involvement in nitric oxide physiology in the retina

scientific article

Somatostatin sst2 receptor knock-out mice: localisation of sst1-5 receptor mRNA and binding in mouse brain by semi-quantitative RT-PCR, in situ hybridisation histochemistry and receptor autoradiography.

scientific article

Somatostatin, Alzheimer's disease and cognition: an old story coming of age?

scientific article published on 10 July 2009

Somatostatin-28 modulates prepulse inhibition of the acoustic startle response, reward processes and spontaneous locomotor activity in rats

scientific article

Sputum Active Polymyxin Lipopeptides: Activity against Cystic Fibrosis Pseudomonas aeruginosa Isolates and Their Interactions with Sputum Biomolecules

scientific article published on 22 March 2018

Status of somatostatin receptor messenger RNAs and binding sites in rat brain during kindling epileptogenesis

scientific article published in December 1996

Structural and compositional determinants of cortistatin activity

article

Study of the calcium dynamics of the human alpha4beta2, alpha3beta4 and alpha1beta1gammadelta nicotinic acetylcholine receptors

scientific article published on 27 June 2002

Subtypes of alpha 1-adrenoceptors in hippocampus of pigs, guinea-pigs, calves and humans: regional differences

scientific article published in January 1990

Suvorexant for the treatment of insomnia

scientific article

Synthesis and Biological Evaluation of a Cyclo-β-tetrapeptide as a Somatostatin Analogue

scientific article

Synthesis and structure-activity relationships of teixobactin

scientific article published on 02 December 2019

T-2 toxin neurotoxicity: role of oxidative stress and mitochondrial dysfunction

scientific article published on 30 September 2019

THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: G protein‐coupled receptors ⬇️

journal article from 'British Journal of Pharmacology' published in 2021

The 5-hydroxytryptamine 5-HT1D receptor subtype is negatively coupled to adenylate cyclase in calf substantia nigra

scientific article published on 01 June 1988

The BJP expects authors to share data

scientific article published on 01 December 2019

The Cyclo-β-Tetrapeptide (β-HPhe-β-HThr-β-HLys-β-HTrp): Synthesis, NMR Structure in Methanol Solution, and Affinity for Human Somatostatin Receptors

The NK1 receptor antagonist NKP608 lacks anxiolytic-like activity in Swiss-Webster mice exposed to the elevated plus-maze

scientific article published on September 2004

The Serotonin 5-HT4 Receptor. 2. Structure-Activity Studies of the Indole Carbazimidamide Class of Agonists ⬇️

scientific article published on June 23, 1995

The agonist activities of the putative antipsychotic agents, L‐745,870 and U‐101958 in HEK293 cells expressing the human dopamine D4.4 receptor ⬇️

scientific article published on July 1, 1998

The binding of serotonergic ligands to the porcine choroid plexus: characterization of a new type of serotonin recognition site

scientific article published on November 1984

The dual orexin receptor antagonist almorexant induces sleep and decreases orexin-induced locomotion by blocking orexin 2 receptors

scientific article

The enantiomer of octreotate binds to all five somatostatin receptors with almost equal micromolar affinity--a comparison with SANDOSTATIN.

scientific article published in July 2008

The impact of backbone N-methylation on the structure-activity relationship of Leu10 -teixobactin

scientific article published on 06 August 2019

The mTOR kinase inhibitor Everolimus decreases S6 kinase phosphorylation but fails to reduce mutant huntingtin levels in brain and is not neuroprotective in the R6/2 mouse model of Huntington's disease

scientific article

The potentially beneficial central nervous system activity profile of ivacaftor and its metabolites.

scientific article published in January 2018

The role of alpha2-adrenoceptor antagonism in the anti-cataleptic properties of the atypical neuroleptic agent, clozapine, in the rat

scientific article

The rostral anterior cingulate cortex modulates the efficiency of amygdala-dependent fear learning

scientific article

The selective nicotinic acetylcholine receptor alpha7 agonist JN403 is active in animal models of cognition, sensory gating, epilepsy and pain

scientific article

The serotonin 5-HT1D receptor: a progress review

scientific article published on June 1990

The serotonin 5-HT4 receptor. 1. Design of a new class of agonists and receptor map of the agonist recognition site.

scientific article published in June 1995

The somatostatin receptor (sst1) modulates the release of somatostatin in the nucleus accumbens of the rat

scientific article published on 01 September 2004

The somatostatin sst1 receptor: an autoreceptor for somatostatin in brain and retina?

scientific article

The structure and signalling properties of 5-HT receptors: an endless diversity?

scientific article published on 01 January 1998

The β-adrenergic receptor in human lymphocytes: Subclassification by the use of a new radio-ligand, (±)−125iodocyanopindolol

scientific article published on 01 November 1981

Updating the guidelines for data transparency in the British Journal of Pharmacology - data sharing and the use of scatter plots instead of bar charts

scientific article published on September 2017

Visualization of a novel serotonin recognition site (5-HT1D) in the human brain by autoradiography

scientific article published on 01 May 1988

Withdrawal from chronic amphetamine induces depressive-like behavioral effects in rodents

scientific article published on July 2003

[125I]BE 2254, a new high affinity radioligand for α1-adrenoceptors

scientific article published on 01 July 1981

[125I]SCH 23982, a ‘selective’ D-1 receptor antagonist, labels with high affinity 5-HT1C sites in pig choroid plexus

scientific article published on 01 May 1988

[125I][Tyr3]octreotide labels human somatostatin sst2 and sst5 receptors

scientific article published on May 1998

[3H]ketanserin labels 5-HT2 receptors and alpha 1-adrenoceptors in human and pig brain membranes

scientific article

alpha 1-Adrenoceptors in the mammalian brain: similar pharmacology but different distribution in rodents and primates

scientific article published in September 1987

mGluR7 facilitates extinction of aversive memories and controls amygdala plasticity

scientific article published on 21 August 2007

siRNA-mediated knockdown of the serotonin transporter in the adult mouse brain

scientific article published in August 2005

siRNA-mediated knockdown of the serotonin transporter in the adult mouse brain

scholarly article by D R Thakker et al published 26 July 2005 in Molecular Psychiatry

Paulina is supported by:

About Paulina

Help