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List of works by Nadège Loaëc

5-Substituted 3-chlorokenpaullone derivatives are potent inhibitors of Trypanosoma brucei bloodstream forms

scientific article

9- and 11-Substituted 4-azapaullones are potent and selective inhibitors of African trypanosoma

scientific article

CDK Inhibitors Roscovitine and CR8 Trigger Mcl-1 Down-Regulation and Apoptotic Cell Death in Neuroblastoma Cells

scientific article

Discovery of pyrido[3,4-g]quinazoline derivatives as CMGC family protein kinase inhibitors: Design, synthesis, inhibitory potency and X-ray co-crystal structure

scientific article

Exploration of the imidazo[1,2-b]pyridazine scaffold as a protein kinase inhibitor

scientific article published on 22 September 2016

Identification of CLK1 Inhibitors by a Fragment-linking Based Virtual Screening

scientific article

Modulating Innate and Adaptive Immunity by (R)-Roscovitine: Potential Therapeutic Opportunity in Cystic Fibrosis

scientific article published on 18 March 2016

Novel Adociaquinone Derivatives from the Indonesian Sponge Xestospongia sp.

scientific article published on 28 April 2015

Synthesis and biological evaluation of N-arylbenzo[b]thieno[3,2-d]pyrimidin-4-amines and their pyrido and pyrazino analogues as Ser/Thr kinase inhibitors

scientific article

Synthesis and molecular modelling studies of 8-arylpyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-amines as multitarget Ser/Thr kinases inhibitors

scientific article published on 23 December 2014

Synthesis, resolution, and biological evaluation of atropisomeric (aR)- and (aS)-16-methyllamellarins N: unique effects of the axial chirality on the selectivity of protein kinases inhibition

scientific article published on 13 September 2013

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