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List of works by Norio Shibata

2-Diazo-1-phenyl-2-((trifluoromethyl)sulfonyl)ethan-1-one: Another Utility for Electrophilic Trifluoromethylthiolation Reactions

scientific article published on 28 January 2016

2-Fluoro-1,3-benzodithiole-1,1,3,3-tetraoxide: a reagent for nucleophilic monofluoromethylation of aldehydes

scientific article published in February 2010

A DBFOX-Ph-based combinatorial catalyst for enantioselective fluorination of aryl acetyl and 3-butenoyl thiazolidinones.

scientific article published in September 2009

A dynamic kinetic asymmetric transformation in the alpha-hydroxylation of racemic malonates and its application to biologically active molecules.

scientific article

A phthalocyanine-subphthalocyanine heterodinuclear dimer: comparison of spectroscopic properties with those of homodinuclear dimers of constituting units

scientific article published on 01 March 2014

A proximity biotinylation-based approach to identify protein-E3 ligase interactions induced by PROTACs and molecular glues

scientific article published on 10 January 2022

A small-molecule inhibitor of SOD1-Derlin-1 interaction ameliorates pathology in an ALS mouse model.

scientific article published on 10 July 2018

A sterically demanding organo-superbase avoids decomposition of a naked trifluoromethyl carbanion directly generated from fluoroform

scientific article published in March 2013

Access to benzo-fused nine-membered heterocyclic alkenes with a trifluoromethyl carbinol moiety via a double decarboxylative formal ring-expansion process under palladium catalysis.

scientific article

Activation of Saturated Fluorocarbons to Synthesize Spirobiindanes, Monofluoroalkenes, and Indane Derivatives

scientific article published on 19 June 2019

Alkynyl Cinchona Catalysts affect Enantioselective Trifluoromethylation for Efavirenz under Metal-Free Conditions

scientific article published on 14 October 2016

An IMiD-induced SALL4 degron system for selective degradation of target proteins

scientific article published on 18 September 2020

An eccentric rod-like linear connection of two heterocycles: synthesis of pyridine trans-tetrafluoro-λ6-sulfanyl triazoles.

scientific article

Anionic Triflyldiazomethane: Generation and Its Application for Synthesis of Pyrazole-3-triflones via [3 + 2] Cycloaddition Reaction

scientific article published on 10 January 2018

Assessment of Protein Binding of 5-Hydroxythalidomide Bioactivated in Humanized Mice with Human P450 3A-Chromosome or Hepatocytes by Two-Dimensional Electrophoresis/Accelerator Mass Spectrometry.

scientific article published on 27 July 2016

Asymmetric Desymmetrization via Metal-Free C-F Bond Activation: Synthesis of 3,5-Diaryl-5-fluoromethyloxazolidin-2-ones with Quaternary Carbon Centers

scientific article published on 22 June 2016

Asymmetric Electrophilic Difluoromethylthiolation of Indanone-Based β-Keto Esters Using Difluoromethanesulfonyl Hypervalent Iodonium Ylides

scientific article published on 09 January 2019

Asymmetric allylic monofluoromethylation and methylation of Morita-Baylis-Hillman carbonates with FBSM and BSM by cooperative cinchona alkaloid/FeCl2 catalysis

scientific article published on 01 September 2011

Asymmetric synthesis of agrochemically attractive trifluoromethylated dihydroazoles and related compounds under organocatalysis

scientific article

Asymmetric synthesis of both mirror images of 3'-fluorothalidomide by enantiodivergent fluorination using a single, cinchona alkaloid

scientific article published on 21 December 2010

Asymmetric synthesis of α-deuterated α-amino acids

scientific article published on 01 August 2017

Asymmetric synthesis of α-trifluoromethoxy ketones with a tetrasubstituted α-stereogenic centre via the palladium-catalyzed decarboxylative allylic alkylation of allyl enol carbonates

scientific article published on 01 May 2018

Biological evaluation of both enantiomers of fluoro-thalidomide using human myeloma cell line H929 and others.

scientific article

Bis(pentafluorosulfanyl)phenyl azide as an expeditious tool for click chemistry toward antitumor pharmaceuticals

scientific article published on 3 March 2014

C-F bond activation of unactivated aliphatic fluorides: synthesis of fluoromethyl-3,5-diaryl-2-oxazolidinones by desymmetrization of 2-aryl-1,3-difluoropropan-2-ols

scientific article published on 04 November 2012

Catalytic Asymmetric 1,3-Dipolar Cycloaddition of β-Fluoroalkylated α,β-Unsaturated 2-Pyridylsulfones with Nitrones for Chiral Fluoroalkylated Isoxazolidines and γ-Amino Alcohols

scientific article published on 9 January 2017

Catalytic and highly enantioselective reactions of alpha-sulfonyl carbanions with chiral bis(oxazoline)s

scientific article published in January 2008

Catalytic asymmetric synthesis of enantioenriched heterocycles bearing a C-CF3 stereogenic center.

scientific article

Catalytic enantioselective Michael addition of 1-fluorobis(phenylsulfonyl)methane to alpha,beta-unsaturated ketones catalyzed by cinchona alkaloids

scientific article published in January 2008

Catalytic enantioselective hydrophosphonylation of ketimines using cinchona alkaloids

scientific article published on 01 December 2009

Catalytic enantioselective synthesis of β-trifluoromethyl pyrrolines

scientific article published on 24 February 2012

Catalytic enantioselective trifluoromethylation of azomethine imines with trimethyl(trifluoromethyl)silane.

scientific article published in January 2009

Catalytic trifluoromethylation of aryl- and vinylboronic acids by 2-cyclopropyl-1-(trifluoromethyl)benzo[b]thiophenium triflate

scientific article published on 18 March 2015

Chiral discrimination between thalidomide enantiomers using a solid surface with two-dimensional chirality.

scientific article published in January 2004

Cinchona alkaloid catalyzed enantioselective fluorination of allyl silanes, silyl enol ethers, and oxindoles

scientific article published on January 2008

Cinchona alkaloid-catalyzed asymmetric trifluoromethylation of alkynyl ketones with trimethylsilyl trifluoromethane

scientific article published on 18 October 2010

Cinchona alkaloid-catalyzed enantioselective monofluoromethylation reaction based on fluorobis(phenylsulfonyl)methane chemistry combined with a Mannich-type reaction

scientific article published on 27 April 2007

Cinchona alkaloid/Ti(IV)-catalyzed enantioselective enamine-trifluoropyruvate condensation-cyclization reaction and its application to drug-like heterocycles

scientific article published on June 2010

Cinchona alkaloid/sulfinyl chloride combinations: enantioselective sulfinylating agents of alcohols.

scientific article published in February 2005

Cinchona alkaloids/TMAF combination-catalyzed nucleophilic enantioselective trifluoromethylation of aryl ketones.

scientific article published on 10 August 2007

Cinchona-alkaloid-catalyzed enantioselective direct aldol-type reaction of oxindoles with ethyl trifluoropyruvate

scientific article published in January 2007

Construction of Fluorinated Benzoxathiin Skeleton by Successive Perfluorophenylthiolation/Cyclization of Activated α-Methylene Ketones by Perfluorophenyl Diethylaminosulfur Difluoride

scientific article published on 13 February 2017

Copper-catalyzed enantioselective three-component synthesis of optically active propargylamines from aldehydes, amines, and aliphatic alkynes

scientific article published in February 2010

Copper-catalyzed regioselective trifluoromethylthiolation of pyrroles by trifluoromethanesulfonyl hypervalent iodonium ylide

scientific article published on 16 February 2015

Corrigendum: Regioisomer-Free C 4h β-Tetrakis(tert-butyl)metallo-phthalocyanines: Regioselective Synthesis and Spectral Investigations

scientific article published in September 2015

Cu-mediated chemoselective trifluoromethylation of benzyl bromides using shelf-stable electrophilic trifluoromethylating reagents

scientific article published on 13 June 2011

Cytotoxic effect of amide derivatives of trifluoromethionine against the enteric protozoan parasite Entamoeba histolytica

scientific article published on 12 November 2009

DBFOX-Ph/metal complexes: evaluation as catalysts for enantioselective fluorination of 3-(2-arylacetyl)-2-thiazolidinones.

scientific article published on 20 May 2008

Decarboxylative allylation of trifluoroethyl sulfones and approach to difluoromethyl compounds

scientific article published on 10 October 2012

Defluorosilylation of fluoroarenes and fluoroalkanes

scientific article published in Nature Communications

Deoxyfluorination of acyl fluorides to trifluoromethyl compounds by FLUOLEAD<sup>®</sup>/Olah's reagent under solvent-free conditions

scientific article published on 14 December 2020

Design and synthesis of galactose-conjugated fluorinated and non-fluorinated proline oligomers: towards antifreeze molecules

scientific article published on 01 August 2018

Design, synthesis and optical properties of unsymmetrical subphthalocyanine trimer connected by phloroglucinol via axial positions

scientific article published on 01 January 2016

Design, synthesis, and spectroscopic investigation of zinc dodecakis(trifluoroethoxy)phthalocyanines conjugated with deoxyribonucleosides

scientific article published in December 2006

Desymmetrization-like catalytic enantioselective fluorination of malonates and its application to pharmaceutically attractive molecules.

scientific article published in January 2008

Diastereoselective additive trifluoromethylation/halogenation of isoxazole triflones: synthesis of all-carbon-functionalized trifluoromethyl isoxazoline triflones

scientific article published on 13 February 2014

Difluoromethanesulfonyl hypervalent iodonium ylides for electrophilic difluoromethylthiolation reactions under copper catalysis

scientific article

Difluoromethylation of Terminal Alkynes by Fluoroform

scientific article published on 16 July 2015

Difluoromethylthiolation of Phenols and Related Compounds with a HF2CSO2Na/Ph2PCl/Me3SiCl System

scientific article published on 06 February 2017

Direct nucleophilic trifluoromethylation of carbonyl compounds by potent greenhouse gas, fluoroform: Improving the reactivity of anionoid trifluoromethyl species in glymes

scientific article published in Scientific Reports

Efficient access to extended Yagupolskii-Umemoto-type reagents: triflic acid catalyzed intramolecular cyclization of ortho-ethynylaryltrifluoromethylsulfanes

scientific article published in January 2010

Efficient access to trifluoromethyl diarylpyrrolines and their N-oxides through enantioselective conjugate addition of nitromethane to β,β-disubstituted enones

scientific article published on 18 April 2013

Electrophilic Triflyl-arylation and Triflyl-pyridylation by Unsymmetrical Aryl/Pyridyl-λ3-iodonium Salts: Synthesis of Aryl and Pyridyl Triflones

scientific article

Enantiomerization of Allylic Trifluoromethyl Sulfoxides Studied by HPLC Analysis and DFT Calculations

scientific article published on 21 December 2015

Enantioselective 5-endo-dig carbocyclization of β-ketoesters with internal alkynes employing a four-component catalyst system

scientific article published on 15 March 2012

Enantioselective Benzylation and Allylation of α-Trifluoromethoxy Indanones under Phase-Transfer Catalysis

scientific article published on 30 July 2019

Enantioselective C--C bond formation to sulfonylimines through use of the 2-pyridinesulfonyl group as a novel stereocontroller

scientific article

Enantioselective Friedel-Crafts reaction of beta-trifluoromethylated acrylates with pyrroles and its application to the synthesis of trifluorinated heliotridane

scientific article published in March 2010

Enantioselective Trichloromethylation of MBH-Fluorides with Chloroform Based on Silicon-assisted C-F Activation and Carbanion Exchange Induced by a Ruppert-Prakash Reagent

scientific article published on 21 October 2015

Enantioselective aza-Morita-Baylis-Hillman reactions of acrylonitrile catalyzed by palladium(II) pincer complexes having C2-symmetric chiral bis(imidazoline) ligands

scientific article published on 17 September 2012

Enantioselective electrophilic trifluoromethylation of beta-keto esters with Umemoto reagents induced by chiral nonracemic guanidines.

scientific article published on 10 July 2009

Enantioselective fluorination mediated by N-fluoroammonium salts of cinchona alkaloids: first enantioselective synthesis of BMS-204352 (MaxiPost).

scientific article published in March 2003

Enantioselective fluorination mediated by cinchona alkaloid derivatives/Selectfluor combinations: reaction scope and structural information for N-fluorocinchona alkaloids

scientific article published on 01 July 2001

Enantioselective monofluoromethylation of aldehydes with 2-fluoro-1,3-benzodithiole-1,1,3,3-tetraoxide catalyzed by a bifunctional cinchona alkaloid-derived thiourea-titanium complex

scientific article published on 23 October 2013

Enantioselective synthesis of (R)-convolutamydine A with new N-heteroarylsulfonylprolinamides.

scientific article published in January 2008

Enantioselective synthesis of AG-041R by using N-heteroarenesulfonyl cinchona alkaloid amides as organocatalysts

scientific article published on 26 June 2012

Enantioselective synthesis of chiral sulfinates using chiral diamines

scientific article published in February 2005

Enantioselective synthesis of epoxides having a tetrasubstituted trifluoromethylated carbon center: methylhydrazine-induced aerobic epoxidation of β,β-disubstituted enones

scientific article published on 21 January 2013

Enantioselective synthesis of imidazolines with quaternary stereocenters by organocatalytic reaction of N-(heteroarenesulfonyl)imines with isocyanoacetates

scientific article published on 01 June 2012

Enantioselective synthesis of trifluoromethyl-substituted 2-isoxazolines: asymmetric hydroxylamine/enone cascade reaction

scientific article published on 01 August 2010

Enzymatic resolution and evaluation of enantiomers of cis-5'-hydroxythalidomide

scientific article published on 28 March 2008

First enantioselective synthesis of (R)-convolutamydine B and E with N-(heteroarenesulfonyl)prolinamides

scientific article published on 01 July 2009

Fluorobis(phenylsulfonyl)methane: a fluoromethide equivalent and palladium-catalyzed enantioselective allylic monofluoromethylation

scientific article published in July 2006

Fluorothalidomide: a characterization of maternal and developmental toxicity in rabbits and mice

scientific article published on 19 April 2011

Gas/Liquid-Phase Micro-Flow Trifluoromethylation using Fluoroform: Trifluoromethylation of Aldehydes, Ketones, Chalcones, and -Sulfinylimines

scientific article published on 05 February 2019

Highly C-selective difluoromethylation of β-ketoesters by using TMSCF2Br/lithium hydroxide/N,N,N-trimethylhexadecan-1-ammonium bromide

scientific article published on 01 August 2018

Highly Diastereoselective Synthesis of Trifluoromethyl Indolines by Interceptive Benzylic Decarboxylative Cycloaddition of Nonvinyl, Trifluoromethyl Benzoxazinanones with Sulfur Ylides under Palladium Catalysis

scientific article published on 23 February 2018

Highly Enantioselective Reactions of Configurationally Labile Epimeric Diamine Complexes of LithiatedS-Benzyl Thiocarbamates

article

Highly enantioselective catalytic fluorination and chlorination reactions of carbonyl compounds capable of two-point binding.

scientific article published in July 2005

Highly enantioselective monofluoromethylation of C2-arylindoles using FBSM under chiral phase-transfer catalysis

scientific article published on 17 June 2013

Highly enantioselective reactions of alpha-sulfonyl carbanions of trifluoromethyl sulfones.

scientific article published in January 2007

Human cytochrome P450 oxidation of 5-hydroxythalidomide and pomalidomide, an amino analogue of thalidomide

scientific article published on 24 December 2013

Human liver microsomal cytochrome P450 3A enzymes involved in thalidomide 5-hydroxylation and formation of a glutathione conjugate

scientific article published on June 2010

IF5 affects the final stage of the Cl-F exchange fluorination in the synthesis of pentafluoro-λ6-sulfanyl-pyridines, pyrimidines and benzenes with electron-withdrawing substituents

scientific article published on 17 May 2017

Importance of a Fluorine Substituent for the Preparation of meta- and para-Pentafluoro-λ(6) -sulfanyl-Substituted Pyridines

scientific article published on 03 August 2016

In vivo drug interactions of the teratogen thalidomide with midazolam: heterotropic cooperativity of human cytochrome P450 in humanized TK-NOG mice.

scientific article

In vivo formation of a glutathione conjugate derived from thalidomide in humanized uPA-NOG mice

scientific article published on 7 February 2011

In vivo formation of dihydroxylated and glutathione conjugate metabolites derived from thalidomide and 5-Hydroxythalidomide in humanized TK-NOG mice.

scientific article

Induction of human cytochrome P450 3A enzymes in cultured placental cells by thalidomide and relevance to bioactivation and toxicity

scientific article published in January 2017

Inherent oxygen preference in enolate monofluoromethylation and a synthetic entry to monofluoromethyl ethers

scientific article published on 23 December 2010

Lewis acid-catalyzed enantioselective hydroxylation reactions of oxindoles and beta-keto esters using DBFOX ligand.

scientific article published in December 2006

Lewis acid-catalyzed tri- and difluoromethylation reactions of aldehydes.

scientific article

Modern Approaches for Asymmetric Construction of Carbon-Fluorine Quaternary Stereogenic Centers: Synthetic Challenges and Pharmaceutical Needs.

scientific article published on 2 April 2018

N-Fluoro-3-cyclohexyl-3-methyl-2,3- dihydrobenzo[1,2-d]isothiazole 1,1-Dioxide: An Efficient Agent for Electrophilic Asymmetric Fluorination of Enolates

scientific article published on 01 July 1999

NH-type of chiral Ni(II) complexes of glycine Schiff base: design, structural evaluation, reactivity and synthetic applications

scientific article published on 01 February 2014

Novel Use of CF3SO2Cl for the Metal-Free Electrophilic Trifluoromethylthiolation

scientific article published on 28 April 2016

Novel methods for the facile construction of 3,3-disubstituted and 3, 3-spiro-2H,4H-benzo[e]1,2-thiazine-1,1-diones: synthesis of (11S,12R, 14R)-2-fluoro-14-methyl-11-(methylethyl)spiro[4H-benzo[e]- 1, 2-thiazine-3,2'-cyclohexane]-1,1-dione, an agen

scientific article published on 01 November 2000

Nucleophilic fluoroalkylation/cyclization route to fluorinated phthalides

scientific article published on 19 January 2018

Organocatalytic Enantioselective Nucleophilic Alkynylation of Allyl Fluorides Affording Chiral Skipped Ene-ynes

scientific article published on 25 April 2016

Organocatalytic asymmetric synthesis of trifluoromethyl-substituted diarylpyrrolines: enantioselective conjugate cyanation of β-aryl-β-trifluoromethyl-disubstituted enones

scientific article published on 04 April 2012

Organocatalyzed Trifluoromethylation of Ketones and Sulfonyl Fluorides by Fluoroform under a Superbase System

scientific article published on 6 August 2015

Organocatalyzed regio- and enantioselective allylic trifluoromethylation of Morita-Baylis-Hillman adducts using Ruppert-Prakash reagent

scientific article published on 24 June 2011

Partially saturated fluorinated heterocycles: diastereo- and enantioselective synthesis of β-trifluoromethyl-pyrroline carboxylates

scientific article published on 01 March 2012

Pd-Catalyzed Decarboxylative Cyclization of Trifluoromethyl Vinyl Benzoxazinanones with Sulfur Ylides: Access to Trifluoromethyl Dihydroquinolines

scientific article published on 21 February 2019

Perfluoroalkyl Analogues of Diethylaminosulfur Trifluoride: Reagents for Perfluoroalkylthiolation of Active Methylene Compounds under Mild Conditions

scientific article published on 22 November 2016

Poly[(3-hexylthiophene)-block-(3-semifluoroalkylthiophene)] for polymer solar cells

scientific article published on 6 December 2010

Reactions of allyl alcohols and boronic acids with trifluoromethanesulfonyl hypervalent iodonium ylide under copper-catalysis

scientific article published on 31 July 2015

Regioisomer-Free C 4h β-Tetrakis(tert-butyl)metallo-phthalocyanines: Regioselective Synthesis and Spectral Investigations

scientific article published on 21 November 2014

Regioselective 1,4-trifluoromethylation of α,β-unsaturated ketones via a S-(trifluoromethyl)diphenylsulfonium salts/copper system

scientific article

Regioselective synthesis of heteroaryl triflones by LDA (lithium diisopropylamide)-mediated anionic thia-Fries rearrangement

scientific article published on 27 April 2012

Regioselective synthesis of pyrazole triflones based on triflyl alkyne cycloadditions

scientific article published on 04 October 2012

Remote anionic Fries rearrangement of sulfonates: regioselective synthesis of indole triflones

scientific article published on 23 January 2013

SF5-Pyridylaryl-λ3-iodonium salts and their utility as electrophilic reagents to access SF5-pyridine derivatives in the late-stage of synthesis

scientific article

Selective O-difluoromethylation of 1,3-diones by bromodifluoromethylating reagents

scientific article published on 13 February 2013

Selective synthesis of spirobiindanes, alkenyl chlorides, and monofluoroalkenes from unactivated gem-difluoroalkanes controlled by aluminum-based Lewis acids

scientific article published on 13 December 2019

Self-disproportionation of enantiomers of thalidomide and its fluorinated analogue via gravity-driven achiral chromatography: mechanistic rationale and implications.

scientific article

Shelf-stable electrophilic trifluoromethylating reagents: A brief historical perspective.

scientific article published on 16 June 2010

Silver-induced self-immolative Cl-F exchange fluorination of arylsulfur chlorotetrafluorides: synthesis of arylsulfur pentafluorides

scientific article published on 17 October 2017

Simulation of Human Plasma Concentrations of Thalidomide and Primary 5-Hydroxylated Metabolites Explored with Pharmacokinetic Data in Humanized TK-NOG Mice.

scientific article

Stereodivergent trifluoromethylation of N-sulfinylimines by fluoroform with either organic-superbase or organometallic-base.

scientific article published on 10 April 2018

Stereoselective Synthesis of β-Lactam-triflones under Catalyst-Free Conditions

scientific article published on 09 November 2015

Stereoselective synthesis of vinyl triflones and heteroaryl triflones through anionic O→C(vinyl) and N→C(vinyl) trifluoromethanesulfonyl migration reactions.

scientific article published on 15 October 2013

Sterically Demanding Unsymmetrical Diaryl-λ(3)-iodanes for Electrophilic Pentafluorophenylation and an Approach to α-Pentafluorophenyl Carbonyl Compounds with an All-Carbon Stereocenter

scientific article published on 17 September 2014

Stille cross-coupling of secondary and tertiary α-(trifluoromethyl)-benzyl chlorides with allylstannanes

scientific article published on 01 June 2018

Structural bases of IMiD selectivity that emerges by 5-hydroxythalidomide

scientific article published on 14 September 2020

Structural basis of thalidomide enantiomer binding to cereblon

scientific article

Structure of isopenicillin N synthase complexed with substrate and the mechanism of penicillin formation

scientific article

Studies of Halogen Bonding Induced by Pentafluorosulfanyl Aryl Iodides: A Potential Group of Halogen Bond Donors in a Rational Drug Design

scientific article published on 07 October 2019

Successive C-C bond cleavage, fluorination, trifluoromethylthio- and pentafluorophenylthiolation under metal-free conditions to provide compounds with dual fluoro-functionalization.

scientific article

Super-Sensitive Protonation Behavior of Trifluoroethoxy-Substituted Phthalocyanines and Their Application to Solvent Discrimination

scientific article published on 10 September 2018

Synthesis and configurational stability of (S)- and (R)-deuteriothalidomides

scientific article published in January 2010

Synthesis and optical properties of subphthalocyanine homo- and heterodimers axially connected via a hydroquinone linker

scientific article published on 20 July 2015

Synthesis and properties of trifluoroethoxy-coated binuclear phthalocyanine.

scientific article published on 28 March 2008

Synthesis of Aryl Triflones through the Trifluoromethanesulfonylation of Benzynes.

scientific article published on 27 February 2018

Synthesis of Both Enantiomers of Nine-Membered CF3 -Substituted Heterocycles Using a Single Chiral Ligand: Palladium-Catalyzed Decarboxylative Ring Expansion with Kinetic Resolution

scientific article published on 31 January 2020

Synthesis of Chiral Nonracemic α-Difluoromethylthio Compounds with Tetrasubstituted Stereogenic Centers via a Palladium-Catalyzed Decarboxylative Asymmetric Allylic Alkylation

scientific article published on 08 November 2018

Synthesis of Chiral gem-Difluoromethylene Compounds by Enantioselective Ethoxycarbonyldifluoromethylation of MBH Fluorides via Silicon-Assisted C-F Bond Activation

scientific article published on 04 November 2020

Synthesis of Diaryliodonium Salts Having Pentafluorosulfanylarenes and Their Application to Electrophilic Pentafluorosulfanylarylation of C-, O-, N-, and S-Nucleophiles

scientific article published on 29 May 2015

Synthesis of Phthalocyanines with a Pentafluorosulfanyl Substituent at Peripheral Positions

scientific article published on 24 July 2015

Synthesis of Sulfur Perfluorophenyl Compounds Using a Pentafluorobenzenesulfonyl Hypervalent Iodonium Ylide.

scientific article published on 12 September 2017

Synthesis of chiral (tetrazolyl)methyl-containing acrylates via silicon-induced organocatalytic kinetic resolution of Morita-Baylis-Hillman fluorides

scientific article published on 5 January 2017

Synthesis of covalently linked binuclear clamshell phthalocyanine by double-click reaction

scientific article published on 23 October 2008

Synthesis of fluorinated allenes via palladium-catalyzed monofluoromethylation using FBSM.

scientific article published on 2 November 2009

Synthesis of fluoro-functionalized diaryl-λ3-iodonium salts and their cytotoxicity against human lymphoma U937 cells

scientific article published on 7 February 2018

Synthesis of indole and biindolyl triflones: trifluoromethanesulfonylation of indoles with Tf2O/TTBP (2,4,6-tri-tert-butylpyridine) system.

scientific article

Synthesis of trifluoroethoxy-coated binuclear phthalocyanines with click spacers and investigation of their clamshell behaviour.

scientific article

Synthesis, configurational stability and stereochemical biological evaluations of (S)- and (R)-5-hydroxythalidomides.

scientific article published on 3 March 2009

Synthetic methods for compounds having CF3-S units on carbon by trifluoromethylation, trifluoromethylthiolation, triflylation, and related reactions

scientific article

Thalidomide and its metabolite 5-hydroxythalidomide induce teratogenicity via the cereblon neosubstrate PLZF

scientific article published on 20 January 2021

Thalidomide increases human hepatic cytochrome P450 3A enzymes by direct activation of the pregnane X receptor

scientific article published on 5 February 2014

Thalidomide protects against ischemic neuronal damage induced by focal cerebral ischemia in mice

scientific article published in January 2009

The CF3-DAST-induced deacylative trifluoromethylthiolation of cyclic 1,3-diketones/lactams/lactones and its extension to deacylative pentafluorophenylthiolation

scientific article published on 01 August 2018

The Dihydroxy Metabolite of the Teratogen Thalidomide Causes Oxidative DNA Damage.

scientific article published on 26 July 2017

Transition-metal-free oxidative trifluoromethylation of unsymmetrical biaryls with trifluoromethanesulfinate

scientific article published on 10 May 2013

Trifluoroethoxy-Coated Phthalocyanine Catalyzes Perfluoroalkylation of Alkenes under Visible-Light Irradiation

scientific article published on 07 July 2017

Trifluoroethoxy-Coated Subphthalocyanine affects Trifluoromethylation of Alkenes and Alkynes even under Low-Energy Red-Light Irradiation

scientific article published on 21 February 2017

Trifluoroethoxy-Coated Subphthalocyanines Attract Small Arenes in Their π-Concave Cavity

scientific article published on 28 December 2017

Trifluoroethoxy-Coated Subphthalocyanines Attract Small Arenes in Their π-Concave Cavity

scientific article published on 15 January 2018

Trifluoroethoxy-coating improves the axial ligand substitution of subphthalocyanine

scientific article published in July 2010

Trifluoromethanesulfonyl hypervalent iodonium ylide for copper-catalyzed trifluoromethylthiolation of enamines, indoles, and β-keto esters

scientific article published on 11 June 2013

Trifluoromethyl sulfoxides from allylic alcohols and electrophilic SCF3 donor by [2,3]-sigmatropic rearrangement

scientific article published in April 2015

Trifluoromethylation of aromatic isoxazoles: regio- and diastereoselective route to 5-trifluoromethyl-2-isoxazolines

scientific article published on 01 August 2011

Trifluoromethylthiolation of allylsilanes and silyl enol ethers with trifluoromethanesulfonyl hypervalent iodonium ylide under copper catalysis

scientific article published on 17 February 2015

Understanding the Thalidomide Chirality in Biological Processes by the Self-disproportionation of Enantiomers

scientific article published in Scientific Reports