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List of works by Roger C. Whitehead

A synthetic approach to novel carvotacetone and antheminone analogues with anti-tumour activity.

scientific article published on 26 July 2013

Arene cis-dihydrodiols: useful precursors for the preparation of analogues of the anti-tumour agent, 2-crotonyloxymethyl-(4R,5R,6R)-4,5,6-trihydroxycyclohex-2-enone (COTC)

scientific article published on 21 August 2007

Deubiquitinases regulate the activity of caspase-1 and interleukin-1β secretion via assembly of the inflammasome

scientific article published on 3 December 2012

Eeyarestatin 1 interferes with both retrograde and anterograde intracellular trafficking pathways

scientific article

Eeyarestatin I inhibits Sec61-mediated protein translocation at the endoplasmic reticulum

scientific article

Exploring electronic effects on the partitioning of actinides(iii) from lanthanides(iii) using functionalised bis-triazinyl phenanthroline ligands.

scientific article published on 4 August 2016

Hydrophilic 2,9-bis-triazolyl-1,10-phenanthroline ligands enable selective Am(iii) separation: a step further towards sustainable nuclear energy.

scientific article

Inhibition of protein translocation at the endoplasmic reticulum promotes activation of the unfolded protein response

scientific article published on March 2012

Inhibitors of NQO1: identification of compounds more potent than dicoumarol without associated off-target effects.

scientific article published on 21 October 2010

Novel inhibitors of NRH:quinone oxidoreductase 2 (NQO2): crystal structures, biochemical activity, and intracellular effects of imidazoacridin-6-ones

scientific article

Pharmacological inhibitors of NAD(P)H quinone oxidoreductase, NQO1: structure/activity relationships and functional activity in tumour cells

scientific article published on 23 June 2010

Synthetic analogues of the manzamenones and plakoridines which inhibit DNA polymerase

scientific article published on 24 March 2006

Transition metal-free, visible-light mediated synthesis of 1,10-phenanthroline derived ligand systems

scientific article published on 01 July 2017