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List of works by Antonio Carrieri

1,3-Benzothiazoles as Antimicrobial Agents

2-(2-Phenylcyclopropyl)imidazolines: reversed enantioselective interaction at I(1) and I(2) imidazoline receptors

scientific article

2-Aminobenzothiazole derivatives: search for new antifungal agents

scientific article published on 9 April 2013

2-D and 3-D modeling of imidazoline receptor ligands: insights into pharmacophore

scientific article published on 01 May 1997

2D- and 3D-QSAR of tocainide and mexiletine analogues acting as Na(v)1.4 channel blockers

scientific article published on 14 October 2008

4H-1,4-benzothiazine, dihydro-1,4-benzothiazinones and 2-amino-5-fluorobenzenethiol derivatives: design, synthesis and in vitro antimicrobial screening

scientific article published on 07 December 2011

Alpha2-Adrenergic Receptors in Intestinal Epithelial Cells: Mechanisms of Signaling, Role, and Regulation

Alpha2-adrenoreceptors profile modulation and high antinociceptive activity of (S)-(-)-2-[1-(biphenyl-2-yloxy)ethyl]-4,5-dihydro-1H-imidazole.

scientific article

Alpha2-adrenoreceptors profile modulation. 4. From antagonist to agonist behavior

scientific article published on 25 June 2008

Alpidem analogues containing a GABA or glycine moiety as new anticonvulsant agents

scientific article published in March 2003

Beyond the Canonical Endocannabinoid System. A Screening of PPAR Ligands as FAAH Inhibitors

scientific article published on 24 September 2020

Binding models of reversible inhibitors to type-B monoamine oxidase

scientific article

Binding of Tracizolines to the Imidazoline Receptor: Role of Lipophilicity in Quantitative Structure-Activity Relationship Modelsa

scientific article published on 01 June 1999

Comparative molecular field analysis (CoMFA) and docking studies of non-nucleoside HIV-1 RT inhibitors (NNIs)

scientific article

Comparative molecular field analysis of some pyridazinone-containing alpha1-antagonists

scientific article published on 01 November 1999

Conformationally constrained butyrophenones with mixed dopaminergic (D(2)) and serotoninergic (5-HT(2A), 5-HT(2C)) affinities: synthesis, pharmacology, 3D-QSAR, and molecular modeling of (aminoalkyl)benzo- and -thienocycloalkanones as putative atypi

scientific article

Coumarin, chromone, and 4(3H)-pyrimidinone novel bicyclic and tricyclic derivatives as antiplatelet agents: synthesis, biological evaluation, and comparative molecular field analysis

scientific article published in January 2003

Crystallographic study of PET radio-tracers in clinical evaluation for early diagnosis of Alzheimers

scientific article published on 4 October 2014

Design, synthesis and biological evaluation of a class of bioisosteric oximes of the novel dual peroxisome proliferator-activated receptor α/γ ligand LT175.

scientific article

Dioxane and oxathiane nuclei: suitable substructures for muscarinic agonists

scientific article published on 21 October 2006

Distant collaboration in drug discovery: the LINK3D project

scientific article

Enhanced solubility and antibacterial activity of lipophilic fluoro-substituted N-benzoyl-2-aminobenzothiazoles by complexation with β-cyclodextrins

scientific article

High affinity central benzodiazepine receptor ligands. Part 2: quantitative structure-activity relationships and comparative molecular field analysis of pyrazolo[4,3-c]quinolin-3-ones.

scientific article published in February 2001

High affinity central benzodiazepine receptor ligands: synthesis and structure-activity relationship studies of a new series of pyrazolo[4,3-c]quinolin-3-ones.

scientific article published in April 1998

In vitro effectiveness of anidulafungin against Candida sp. biofilms

scientific article published on 11 September 2013

In vitro interactions between anidulafungin and nonsteroidal anti-inflammatory drugs on biofilms of Candida spp.

scientific article published on 22 January 2016

Investigation of platelet aggregation inhibitory activity by phenyl amides and esters of piperidinecarboxylic acids

scientific article (publication date: 3 April 2003)

Involvement of I2-imidazoline binding sites in positive and negative morphine analgesia modulatory effects

scientific article published on 26 September 2006

Ligand binding to I2 imidazoline receptor: the role of lipophilicity in quantitative structure-activity relationship models.

scientific article

Lipophilicity of teicoplanin antibiotics as assessed by reversed phase high-performance liquid chromatography: quantitative structure-property and structure-activity relationships

scientific article published in December 1994

Might the observed α(2A)-adrenoreceptor agonism or antagonism of allyphenyline analogues be ascribed to different molecular conformations?

scientific article published on 31 January 2012

Modeling the structural basis of human CCR5 chemokine receptor function: from homology model building and molecular dynamics validation to agonist and antagonist docking

scientific article published on 01 May 2006

Molecular determinants for nuclear receptors selectivity: chemometric analysis, dockings and site-directed mutagenesis of dual peroxisome proliferator-activated receptors α/γ agonists.

scientific article published on 24 February 2013

N-aryl-2,6-dimethylbenzamides, a new generation of tocainide analogues as blockers of skeletal muscle voltage-gated sodium channels

scientific article

Natural and synthetic geiparvarins are strong and selective MAO-B inhibitors. Synthesis and SAR studies

scientific article (publication date: 16 December 2002)

Neuronal nicotinic receptor agonists: a multi-approach development of the pharmacophore

scientific article published in September 2001

New serotonin 5-HT(2A), 5-HT(2B), and 5-HT(2C) receptor antagonists: synthesis, pharmacology, 3D-QSAR, and molecular modeling of (aminoalkyl)benzo and heterocycloalkanones

scientific article published in January 2002

Novel imidazoline compounds as partial or full agonists of D2-like dopamine receptors inspired by I2-imidazoline binding sites ligand 2-BFI.

scientific article published on 6 August 2010

Recent trends and future prospects in computational GPCR drug discovery: from virtual screening to polypharmacology.

scientific article published on January 2013

Repositioning of Endonuclear Receptors Binders as Potential Antibacterial and Antifungal Agents. Eptyloxìm: A Potential and Novel Gyrase B and Cytochrome Cyp51 Inhibitor.

scientific article published on 12 May 2016

Structure-Activity Relationship Studies on Tetrahydroisoquinoline Derivatives: [4'-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-ylmethyl)biphenyl-4-ol] (MC70) Conjugated through Flexible Alkyl Chains with Furazan Moieties Gives Rise to Potent and Sel

scientific article

Structure-activity relationships in 1,4-benzodioxan-related compounds. 10. Novel α1-adrenoreceptor antagonists related to openphendioxan: synthesis, biological evaluation, and α1d computational study

scientific article published on 6 August 2010

Structure-activity relationships in 1,4-benzodioxan-related compounds. 7. Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes

scientific article

Synthesis and biological evaluation of pyridazino[4,3-b]indoles and indeno[1,2-c]pyridazines as new ligands of central and peripheral benzodiazepine receptors

scientific article

Synthesis, in vitro evaluation, and molecular modeling investigation of benzenesulfonimide peroxisome proliferator-activated receptors α antagonists

scientific article published on 27 February 2016

The Versatile 2-Substituted Imidazoline Nucleus as a Structural Motif of Ligands Directed to the Serotonin 5-HT1A Receptor

scientific article published on 30 September 2016

Theoretical evidence of a salt bridge disruption as the initiating process for the alpha1d-adrenergic receptor activation: a molecular dynamics and docking study

scientific article

alpha 2-adrenoreceptors profile modulation. 2. Biphenyline analogues as tools for selective activation of the alpha 2C-subtype

scientific article published in December 2004

miRNAs for the Detection of MultiDrug Resistance: Overview and Perspectives

scientific article published on 30 April 2014

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