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List of works by Felicia A. Etzkorn

205Tl nuclear magnetic resonance study of the thallium complex of lasalocid (X-537A)

scholarly article by Richard W Briggs et al published February 1980 in Journal of Magnetic Resonance

A Reduced-Amide Inhibitor of Pin1 Binds in a Conformation Resembling a Twisted-Amide Transition State

scientific article

A capillary electrophoresis mobility shift assay for protein-DNA binding affinities free in solution.

scientific article

A phosphorylated prodrug for the inhibition of Pin1.

scientific article

A prolyl-isomerase mediates dopamine-dependent plasticity and cocaine motor sensitization

scientific article

Chemical Tools To Decipher Regulation of Phosphatases by Proline Isomerization on Eukaryotic RNA Polymerase II.

scientific article published on 2 September 2015

Cis-trans proline isomerization effects on collagen triple-helix stability are limited

scientific article published in September 2009

Conformational Analysis of n→π* Interactions in Collagen Triple Helix Models

scientific article published on 04 January 2019

Conformationally locked isostere of phosphoSer-cis-Pro inhibits Pin1 23-fold better than phosphoSer-trans-Pro isostere

scientific article

Convergent synthesis of alpha-ketoamide inhibitors of Pin1.

scientific article

Crystal structures of cyclophilin A complexed with cyclosporin A and N-methyl-4-[(E)-2-butenyl]-4,4-dimethylthreonine cyclosporin A

scientific article

Cyclic Hexapeptides and Chimeric Peptides as Mimics of Tendamistat

scientific article published in 1994

Cyclohexyl ketone inhibitors of Pin1 dock in a trans-diaxial cyclohexane conformation

scientific article

Cyclophilin Inhibition by a (Z)-Alkene cis-Proline Mimic

scientific article

DNA-binding affinities of MyoD and E47 homo- and hetero-dimers by capillary electrophoresis mobility shift assay

scientific article

Design and Enantioselective Synthesis of a Peptidomimetic of the Turn in the Helix-Turn-Helix DNA-Binding Protein Motif

scientific article

Design and synthesis of a potent histone deacetylase inhibitor

scientific article

Drinking water treatment is not associated with an observed increase in neural tube defects in mice

scientific article published on 5 February 2014

Enzyme-linked enzyme-binding assay for Pin1 WW domain ligands

scientific article

Evaluation of a PK/PBAN analog with an (E)-alkene, trans-Pro isostere identifies the Pro orientation for activity in four diverse PK/PBAN bioassays

scientific article published on 3 May 2009

Evaluation of insect CAP2b analogs with either an (E)-alkene, trans- or a (Z)-alkene, cis-Pro isostere identifies the Pro orientation for antidiuretic activity in the stink bug.

scientific article published on 2 October 2012

Hinweise zur thermodynamischen Kontrolle von relativen Hydriergeschwindigkeiten an Platin Indications to a Thermodynamic Control of the Relative Rate of Hydrogenation on Platinum

Kinetic isotope effects support the twisted amide mechanism of Pin1 peptidyl-prolyl isomerase

scientific article

Peptidyl-prolyl isomerase inhibitors

scientific article

Phosphorus-Based SAHA Analogues as Histone Deacetylase Inhibitors†

scientific article published in 2003

Pin1 as an anticancer drug target

scientific article

Pin1 flips Alzheimer's switch

scientific article

Potent activity of a PK/PBAN analog with an (E)-alkene, trans-Pro mimic identifies the Pro orientation and core conformation during interaction with HevPBANR-C receptor

scientific article published on 25 March 2009

Regulation of CK2 by phosphorylation and O-GlcNAcylation revealed by semisynthesis

scientific article published on 22 January 2012

Role of the cyclosporin-A-cyclophilin complex, FK506-FK506-binding protein complex and calcineurin in the inhibition of T-cell signal transduction

Serine-cis-proline and serine-trans-proline isosteres: stereoselective synthesis of (Z)- and (E)-alkene mimics by Still-Wittig and Ireland-Claisen rearrangements

scientific article published in March 2003

Solvent-dependent stereoselectivity in a Still-Wittig rearrangement: an experimental and ab initio study

scientific article published in June 2001

Stereochemical Control in the Still-Wittig Rearrangement Synthesis of Cyclohexyl (Z)-Alkene Inhibitors of Pin1

scientific article

Stereoselective deuterium labeling of proR beta-protons in the NMR structure determination of a helix-turn-helix turn peptide mimic.

scientific article published in June 2000

Stereospecific gating of functional motions in Pin1

scientific article

Stereospecific phosphorylation by the central mitotic kinase Cdk1-cyclin B.

scientific article

Structural and Kinetic Analysis of Prolyl-isomerization/Phosphorylation Cross-Talk in the CTD Code

scientific article

The effect of a trans-locked Gly-Pro alkene isostere on collagen triple helix stability

scientific article

The immunophilins

Theoretical and experimental investigation of the energetics of cis-trans proline isomerization in peptide models

scientific article

Toward flexibility-activity relationships by NMR spectroscopy: dynamics of Pin1 ligands

scientific article published on April 2010

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