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List of works by Abdelrahman S. Mayhoub

Alkoxyphenylthiazoles with broad-spectrum activity against multidrug-resistant gram-positive bacterial pathogens.

scientific article published on 25 April 2018

Amyloid-β probes: Review of structure-activity and brain-kinetics relationships

scientific article published on 28 May 2013

An investigation of phenylthiazole antiflaviviral agents ⬇️

scientific article published on May 3, 2011

An unexpected synthesis of 3,5-diaryl-1,2,4-thiadiazoles from thiobenzamides and methyl bromocyanoacetate.

scientific article

Anti-biofilm activity and synergism of novel thiazole compounds with glycopeptide antibiotics against multidrug-resistant staphylococci

scientific article published on 15 October 2014

Antibacterial Characterization of Novel Synthetic Thiazole Compounds against Methicillin-Resistant Staphylococcus pseudintermedius

scientific article

Balancing Physicochemical Properties of Phenylthiazole Compounds with Antibacterial Potency by Modifying the Lipophilic Side Chain

scientific article published on 27 November 2019

Biochemical and structural analysis of aminoglycoside acetyltransferase Eis from Anabaena variabilis

scientific article

Biphenylthiazole antibiotics with an oxadiazole linker: An approach to improve physicochemical properties and oral bioavailability

scientific article

Design and Synthesis of Imidazopyrazolopyridines as Novel Selective COX-2 Inhibitors.

scientific article published on 21 August 2015

Design, synthesis and structure-activity relationship study of novel pyrazole-based heterocycles as potential antitumor agents.

scientific article published on October 2010

Design, synthesis, and biological evaluation of thiazoles targeting flavivirus envelope proteins

scientific article

Diphenylpyrroles: Novel p53 activators

scientific article published on 3 June 2014

Discovery and characterization of potent thiazoles versus methicillin- and vancomycin-resistant Staphylococcus aureus

scientific article published on 14 January 2014

From Phenylthiazoles to Phenylpyrazoles: Broadening the Antibacterial Spectrum toward Carbapenem-Resistant Bacteria

scientific article published on 19 August 2019

Hepatitis C RNA-dependent RNA polymerase inhibitors: a review of structure-activity and resistance relationships; different scaffolds and mutations.

scientific article published on 29 March 2012

Investigating the Antibacterial Activity of Biphenylthiazoles against Methicillin- and Vancomycin-Resistant Staphylococcus aureus (MRSA and VRSA).

scientific article published on 24 April 2017

Modifying the lipophilic part of phenylthiazole antibiotics to control their drug-likeness

scientific article published on 31 October 2019

Naphthylthiazoles: Targeting Multidrug-Resistant and Intracellular Staphylococcus aureus with Biofilm Disruption Activity

scientific article published on 08 October 2018

Novel 4-heteroaryl-antipyrines as DPP-IV inhibitors

scientific article published on 29 May 2015

Optimization of the aromatase inhibitory activities of pyridylthiazole analogues of resveratrol

scientific article published on 11 February 2012

Optimization of thiazole analogues of resveratrol for induction of NAD(P)H:quinone reductase 1 (QR1) ⬇️

scientific article published on October 23, 2012

Optimizing thiadiazole analogues of resveratrol versus three chemopreventive targets

scientific article published on 25 September 2011

Oxadiazolylthiazoles as novel and selective antifungal agents

scientific article published on 10 January 2020

Phenylthiazole Antibacterial Agents Targeting Cell Wall Synthesis Exhibit Potent Activity in Vitro and in Vivo against Vancomycin-Resistant Enterococci.

scientific article published on March 2017

Phenylthiazoles with nitrogenous side chain: An approach to overcome molecular obesity

scientific article published on 10 August 2019

Phenylthiazoles with tert-Butyl side chain: Metabolically stable with anti-biofilm activity.

scientific article

Potent 1,2,4-Triazino[5,6 b]indole-3-thioether Inhibitors of the Kanamycin Resistance Enzyme Eis from Mycobacterium tuberculosis

scientific article published on 30 March 2018

Recent advances in the therapeutic applications of pyrazolines.

scientific article published on 08 March 2012

Regioselective synthesis and antitumor screening of some novel N-phenylpyrazole derivatives

scientific article published on 12 October 2007

Second-Generation Phenylthiazole Antibiotics with Enhanced Pharmacokinetic Properties

scientific article published on 17 May 2016

Single step synthesis of new fused pyrimidine derivatives and their evaluation as potent Aurora-A kinase inhibitors.

scientific article published on 20 May 2011

Synthesis and analgesic/anti-inflammatory evaluation of fused heterocyclic ring systems incorporating phenylsulfonyl moiety

scientific article

Synthesis and antibacterial evaluation of a novel series of synthetic phenylthiazole compounds against methicillin-resistant Staphylococcus aureus (MRSA).

scientific article published on 7 March 2015

Synthesis and structure-activity relationship studies of pyrazole-based heterocycles as antitumor agents.

scientific article published on July 2010

Synthesis of new N-phenylpyrazole derivatives with potent antimicrobial activity

scientific article published on 15 February 2008

The tamoxifen metabolite norendoxifen is a potent and selective inhibitor of aromatase (CYP19) and a potential lead compound for novel therapeutic agents ⬇️

scientific article published on August 4, 2011

Unexpected N-acetylation of capreomycin by mycobacterial Eis enzymes

scientific article published on 11 December 2012

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