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List of works by Jonathan L. Katz

2-Substituted 3β-Aryltropane Cocaine Analogs Produce Atypical Effects without Inducing Inward-Facing Dopamine Transporter Conformations.

scientific article

2-isoxazol-3-phenyltropane derivatives of cocaine: molecular and atypical system effects at the dopamine transporter.

scientific article published on 11 February 2014

2D QSAR modeling and preliminary database searching for dopamine transporter inhibitors using genetic algorithm variable selection of Molconn Z descriptors

scientific article published in November 2000

3'-Chloro-3 alpha-(diphenylmethoxy)tropane but not 4'-chloro-3 alpha-(diphenylmethoxy)tropane produces a cocaine-like behavioral profile

scientific article

7-OH-DPAT antagonizes dopamine D2 receptor-inhibited adenylyl cyclase activity

scientific article published on 01 January 1994

A Role for Sigma Receptors in Stimulant Self Administration and Addiction.

scientific article

A Role for Sigma Receptors in Stimulant Self-Administration and Addiction

scientific article published on 22 January 2017

A behavioral economic analysis of the effects of rimcazole on reinforcing effects of cocaine injection and food presentation in rats

scientific article published on 09 August 2019

A comparison of responding maintained under second-order schedules of intramuscular cocaine injection or food presentation in squirrel monkeys ⬇️

scientific article published on November 1, 1979

A comparison of the effects of the D1 receptor antagonists SCH 23390 and SCH 39166 on suppression of feeding behavior by the D1 agonist SKF38393.

scientific article published in January 1994

A further assessment of a role for Toll-like receptor 4 in the reinforcing and reinstating effects of opioids

scientific article published on 01 April 2020

A role for sigma receptors in stimulant self-administration and addiction

scientific article published on 8 December 2015

Abuse liability of mitragynine assessed with a self-administration procedure in rats

scientific article published on 23 July 2018

Agonist efficacy, drug dependence, and medications development: preclinical evaluation of opioid, dopaminergic, and GABAA-ergic ligands.

scientific article

An influence of delayed reinforcement on the effectiveness of psychostimulants to enhance indices of attention under a five-choice serial reaction time procedure in male rats

scientific article published in October 2013

Assessment of cocaine-like discriminative stimulus effects of dopamine D3 receptor ligands.

scientific article

Assessment of reinforcing effects of benztropine analogs and their effects on cocaine self-administration in rats: comparisons with monoamine uptake inhibitors

scientific article published on 19 February 2009

Assessment of the influence of histaminergic actions on cocaine-like effects of 3alpha-diphenylmethoxytropane analogs

scientific article

Behavioral economics of food reinforcement and the effects of prefeeding, extinction, and eticlopride in dopamine D2 receptor mutant mice.

scientific article published on 02 February 2011

Behavioral effects of benzodiazepine antagonists in chlordiazepoxide tolerant and non-tolerant rats

scientific article published in January 1989

Behavioral effects of cocaine alone and in combination with selective dopamine antagonists in the squirrel monkey.

scientific article

Behavioral effects of dopaminergic agonists and antagonists alone and in combination in the squirrel monkey

scientific article published in January 1993

Behavioral effects of rimcazole analogues alone and in combination with cocaine

scientific article published in May 2003

Behavioral, biological, and chemical perspectives on atypical agents targeting the dopamine transporter

scientific article

Blockade of Cocaine or σ Receptor Agonist Self Administration by Subtype-Selective σ Receptor Antagonists.

scientific article published on 21 April 2016

Carbamazepine produces nonspecific effects on cocaine self-administration in rats

scientific article published in January 1992

Choice for response alternatives differing in reinforcement frequency in dopamine D2 receptor mutant and Swiss-Webster mice

scientific article published on 28 February 2014

Citalopram enhances cocaine's subjective effects in rats.

scientific article

Cocaine and food as reinforcers: effects of reinforcer magnitude and response requirement under second-order fixed-ratio and progressive-ratio schedules

scientific article

Cocaine and several sigma receptor ligands inhibit dopamine uptake in rat caudate-putamen.

scientific article

Cocaine-induced endocannabinoid release modulates behavioral and neurochemical sensitization in mice

scientific article published on 04 August 2013

Cocaine-like neurochemical effects of antihistaminic medications.

scientific article

Combinations of cocaine with other dopamine uptake inhibitors: assessment of additivity

scientific article

Comparative behavioral pharmacology and toxicology of cocaine and its ethanol-derived metabolite, cocaine ethyl-ester (cocaethylene).

scientific article published in January 1992

Comparative structure-activity relationships of benztropine analogues at the dopamine transporter and histamine H(1) receptors

scientific article

Comparison of interactions of D1-like agonists, SKF 81297, SKF 82958 and A-77636, with cocaine: locomotor activity and drug discrimination studies in rodents.

scientific article

Compounds of novel structure having kappa-agonist behavioral effects in rhesus monkeys

scientific article published on November 1982

Continuing implications of the early evidence against the drive-reduction hypothesis of the behavioral effects of drugs

scientific article published on 29 August 2002

Contributions to drug abuse research of Steven R. Goldberg's behavioral analysis of stimulus-stimulus contingencies

scientific article

DAT isn't all that: cocaine reward and reinforcement require Toll-like receptor 4 signaling

scientific article published on 3 February 2015

Decreases in cocaine self-administration with dual inhibition of the dopamine transporter and σ receptors

scientific article

Design and synthesis of 1-(3-(dimethylamino)propyl)-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-5-carbonitrile (citalopram) analogues as novel probes for the serotonin transporter S1 and S2 binding sites.

scientific article published on 02 December 2013

Design and synthesis of a novel photoaffinity ligand for the dopamine and serotonin transporters based on 2beta-carbomethoxy-3beta-biphenyltropane.

scientific article

Dexfenfluramine neurotoxicity in brains of non-human primates

scientific article published in December 1991

Differential antagonism of the effects of dopamine D1-receptor agonists on feeding behavior in the rat

scientific article published on January 1, 1992

Differential efficacies of dopamine D1 receptor agonists for stimulating adenylyl cyclase in squirrel monkey and rat.

scientific article published in June 1993

Differential modulation of methamphetamine-mediated behavioral sensitization by overexpression of Mu opioid receptors in nucleus accumbens and ventral tegmental area.

scientific article published on 10 November 2015

Differential relationships among dopamine transporter affinities and stimulant potencies of various uptake inhibitors.

scientific article published in October 1994

Discovery of drugs to treat cocaine dependence: behavioral and neurochemical effects of atypical dopamine transport inhibitors.

scientific article

Discriminative stimulus effects of inhaled cocaine in squirrel monkeys

scientific article published in January 1991

Discriminative stimulus effects of intravenous l-nicotine and nicotine analogs or metabolites in squirrel monkeys

scientific article published in January 1989

Discriminative stimulus effects of intravenous nicotine in squirrel monkeys

scientific article published in May 1988

Dopamine D₂-Like Receptors and Behavioral Economics of Food Reinforcement.

scientific article published on 24 July 2015

Dopamine Transporter Dynamics of -Substituted Benztropine Analogs with Atypical Behavioral Effects

scholarly article by Weimin C Hong et al published September 2018 in Journal of Pharmacology and Experimental Therapeutics

Dopamine transporter binding without cocaine-like behavioral effects: synthesis and evaluation of benztropine analogs alone and in combination with cocaine in rodents

scientific article

Dopamine transporter-dependent and -independent striatal binding of the benztropine analog JHW 007, a cocaine antagonist with low abuse liability

scientific article

Dopaminergic mediation of the discriminative stimulus effects of bupropion in rats.

scientific article published in November 1997

Drug effects on responding maintained by stimulus-reinforcer and response-reinforcer contingencies ⬇️

scientific article published on September 1, 1978

Dual DAT/sigma1 receptor ligands based on 3-(4-(3-(bis(4-fluorophenyl)amino)propyl)piperazin-1-yl)-1-phenylpropan-1-ol

scientific article

Dual probes for the dopamine transporter and sigma1 receptors: novel piperazinyl alkyl-bis(4'-fluorophenyl)amine analogues as potential cocaine-abuse therapeutic agents

scientific article

Effects of 4'-chloro-3 alpha-(diphenylmethoxy)-tropane on mesostriatal, mesocortical, and mesolimbic dopamine transmission: comparison with effects of cocaine

scientific article

Effects of H1-receptor antagonists on responding punished by histamine injection or electric shock presentation in squirrel monkeys

scientific article published in January 1986

Effects of N-substituted analogs of benztropine: diminished cocaine-like effects in dopamine transporter ligands

scientific article published on 30 January 2004

Effects of a selective kappa-opioid agonist, U-50,488H, on morphine dependence in rats

scientific article published in October 1989

Effects of adenosine analogs alone and in combination with caffeine in the squirrel monkey

scientific article published in February 1988

Effects of caramiphen and phencyclidine alone and in combination on behavior in the rat

scientific article published on 01 March 1994

Effects of clonidine and morphine on opioid withdrawal in rhesus monkeys

scientific article published on January 1986

Effects of clonidine and some ?-adrenergic antagonists alone and in combination on schedule-controlled behavior in pigeons and mice ⬇️

scientific article published on January 1, 1984

Effects of cocaine and its quaternary derivative cocaine methiodide on cardiovascular function in squirrel monkeys

scientific article published in March 1992

Effects of cocaine, chlordiazepoxide, and chlorpromazine on responding of squirrel monkeys under second-order schedules of IM cocaine injection or food presentation

scientific article published in January 1983

Effects of d-amphetamine and ethanol alone and in combination on schedule-controlled responding of pigeons ⬇️

scientific article published on June 28, 1979

Effects of d-amphetamine and ethanol on responding of squirrel monkeys maintained under fixed-ratio schedules of food presentation and stimulus-shock termination

scientific article published on January 1978

Effects of dopamine D1-like receptor agonists on food-maintained operant behavior in rats.

scientific article

Effects of ethylketazocine and morphine alone and in combination with naloxone on schedule-controlled behavior in pigeons

scientific article published in January 1987

Effects of muscarinic M1 receptor blockade on cocaine-induced elevations of brain dopamine levels and locomotor behavior in rats

scientific article

Effects of quinpirole and SKF 38393 alone and in combination in squirrel monkeys trained to discriminate cocaine

scientific article published in January 1992

Effects of the selective sigma receptor ligand, 1-(2-phenethyl)piperidine oxalate (AC927), on the behavioral and toxic effects of cocaine ⬇️

scientific article published on March 21, 2011

Elucidation of structural elements for selectivity across monoamine transporters: novel 2-[(diphenylmethyl)sulfinyl]acetamide (modafinil) analogues

scientific article

Enantioselective synthesis of S-(+)-2beta-carboalkoxy-3alpha-[bis(4-fluorophenyl)methoxy]tropanes as novel probes for the dopamine transporter

scientific article published in May 2002

Erratum to: behavioral economics of food reinforcement and the effects of prefeeding, extinction, and eticlopride in dopamine D₂ receptor mutant mice

scientific article published on 01 May 2015

Ethanol, pentobarbital, and chlordiazepoxide effects in squirrel monkeys responding under fixed-ratio food presentation and stimulus-shock termination schedules

scientific article published on March 1978

Evaluation of the neurotoxic potential of N,N-dimethylamphetamine: an illicit analog of methamphetamine

scientific article published on 01 June 1989

Evaluation of the neurotoxicity of N-methyl-1-(4-methoxyphenyl)-2-aminopropane (para-methoxymethamphetamine, PMMA)

scientific article (publication date: 4 September 1992)

Further delineation between typical and atypical dopamine uptake inhibitors: effects on food-maintained behavior and food consumption

scientific article published on 06 December 2016

Further studies of the reinforcing effects of benztropine analogs in rhesus monkeys

scientific article

Highly Selective Chiral N-Substituted 3α-[Bis(4‘-fluorophenyl)methoxy]tropane Analogues for the Dopamine Transporter: Synthesis and Comparative Molecular Field Analysis

scientific article published on 01 March 2000

Human cocaine-seeking behavior and its control by drug-associated stimuli in the laboratory

scientific article published in February 2005

Identification of a dopamine transporter ligand that blocks the stimulant effects of cocaine.

scientific article

Interactions of clonidine and naloxone on schedule-controlled behavior in opioid-naive mice

scientific article

Interactions of cocaine with dopamine D₂-like antagonists in squirrel monkeys

scientific article

Interactions of cocaine with dopamine uptake inhibitors or dopamine releasers in rats discriminating cocaine

scientific article published on 14 February 2006

Intravenous cocaine induced-activity and behavioural sensitization in norepinephrine-, but not dopamine-transporter knockout mice

scientific article published in August 2002

Intravenous cocaine-induced activity in A/J and C57BL/6J mice: behavioral sensitization and conditioned activity

scientific article

Introduction to modern cryptography (CRC, 2008) ⬇️

Investigation of the potential pharmacokinetic and pharmaco-dynamic drug interaction between AHN 1-055, a potent benztropine analog used for cocaine abuse, and cocaine after dosing in rats using intracerebral microdialysis

scientific article published in July 2006

Isothiocyanate derivatives of 9-[3-(cis-3,5-dimethyl-1-piperazinyl)propyl]carbazole (rimcazole): irreversible ligands for the dopamine transporter

scientific article

Lack of Specific Involvement of (+)-Naloxone and (+)-Naltrexone on the Reinforcing and Neurochemical Effects of Cocaine and Opioids

scientific article published on 14 June 2016

Lack of cocaine-like discriminative-stimulus effects of σ-receptor agonists in rats.

scientific article published on September 2011

Lethal effects of cocaine are reduced by the dopamine-1 receptor antagonist SCH 23390 but not by haloperidol

scientific article published in January 1989

Locomotor and discriminative-stimulus effects of cocaine in dopamine D5 receptor knockout mice

scientific journal article

Mechanisms of amphetamine action illuminated through optical monitoring of dopamine synaptic vesicles in Drosophila brain

scientific article

Methohexital and cocaine self-administration under fixed-ratio and second-order schedules

scientific article published in February 1991

Methylphenidate and impulsivity: a comparison of effects of methylphenidate enantiomers on delay discounting in rats

scientific article published on 24 August 2013

Modafinil potentiates cocaine self-administration by a dopamine-independent mechanism: possible involvement of gap junctions

scientific article published on 27 April 2020

Modification of the effects of naloxone in morphine-dependent mice

scientific article published on 01 January 1989

Modulation of opioid receptor affinity and efficacy via N-substitution of 9β-hydroxy-5-(3-hydroxyphenyl)morphan: Synthesis and computer simulation study

scientific article

Modulation of the lethal effects of cocaine by cholinomimetics

scientific article published in January 1989

Muscarinic preferential M(1) receptor antagonists enhance the discriminative-stimulus effects of cocaine in rats

scientific article

N-8-Substituted benztropinamine analogs as selective dopamine transporter ligands

scientific article

N-methylation dissociates methamphetamine's neurotoxic and behavioral pharmacologic effects

scientific article

N-substituted benztropine analogs: selective dopamine transporter ligands with a fast onset of action and minimal cocaine-like behavioral effects

scientific article

Novel N-substituted 3 alpha-[bis(4'-fluorophenyl)methoxy]tropane analogues: selective ligands for the dopamine transporter

scientific article published in December 1997

Novel azido and isothiocyanato analogues of [3-(4-phenylalkylpiperazin-1-yl)propyl]bis(4-fluorophenyl)amines as potential irreversible ligands for the dopamine transporter.

scientific article published on December 2004

Novel tropane-based irreversible ligands for the dopamine transporter

scientific article

Opioid activation of toll-like receptor 4 contributes to drug reinforcement

scientific article

Opioid receptor subtype-specific cross-tolerance to the effects of morphine on schedule-controlled behavior in mice

scientific article

Pharmacodynamic assessment of the benztropine analogues AHN-1055 and AHN-2005 using intracerebral microdialysis to evaluate brain dopamine levels and pharmacokinetic/pharmacodynamic modeling

scientific article published on 7 April 2005

Pharmacological characterization of a dopamine transporter ligand that functions as a cocaine antagonist

scientific article

Pharmacological specificity of enhanced sensitivity to naltrexone in rats

scientific article published in January 1993

Place conditioning and locomotor effects of N-substituted, 4',4''-difluorobenztropine analogs in rats

scientific article published on 2 March 2005

Potential toxic interactions of cocaine and mazindol

scientific article published in July 1989

Preclinical efficacy of N-substituted benztropine analogs as antagonists of methamphetamine self-administration in rats

scientific article

Preference for distinct functional conformations of the dopamine transporter alters the relationship between subjective effects of cocaine and stimulation of mesolimbic dopamine

scientific article

Preparation and Characterization of Tetrabenazine Enantiomers against Vesicular Monoamine Transporter 2.

scientific article

Preparation and evaluation of tetrabenazine enantiomers and all eight stereoisomers of dihydrotetrabenazine as VMAT2 inhibitors

scientific article published on 23 February 2011

Proerectile effects of dopamine D2-like agonists are mediated by the D3 receptor in rats and mice.

scientific article published on 09 January 2009

R-modafinil (armodafinil): a unique dopamine uptake inhibitor and potential medication for psychostimulant abuse

scientific article

Rapid and sustained antidepressant properties of an NMDA antagonist/monoamine reuptake inhibitor identified via transporter-based virtual screening.

scientific article

Rate-dependent effects of d-and l-amphetamine on schedule-controlled responding in pigeons and squirrel monkeys

scientific article published in March 1982

Receptor binding, antagonist, and withdrawal precipitating properties of opiate antagonists

scientific article

Reinforcing effects of enantiomers of N,N-dimethylamphetamine in squirrel monkeys

scientific article published in January 1992

Reinforcing effects of sigma-receptor agonists in rats trained to self-administer cocaine

scientific article

Relations between heterogeneity of dopamine transporter binding and function and the behavioral pharmacology of cocaine

scientific article published on July 1997

Relations between stimulation of mesolimbic dopamine and place conditioning in rats produced by cocaine or drugs that are tolerant to dopamine transporter conformational change

scientific article published on 24 April 2013

Relationship between conformational changes in the dopamine transporter and cocaine-like subjective effects of uptake inhibitors

scientific article

Relationship between in vivo occupancy at the dopamine transporter and behavioral effects of cocaine, GBR 12909 [1-{2-[bis-(4-fluorophenyl)methoxy]ethyl}-4-(3-phenylpropyl)piperazine], and benztropine analogs

scientific article published on 13 July 2005

Response requirement and increases in accuracy produced by stimulant drugs in a 5-choice serial reaction-time task in rats.

scientific article

Selective effects of the D1 dopamine receptor agonist, SKF 38393, on behavior maintained by cocaine injection in squirrel monkeys

scientific article published in January 1992

Selective sigma ligands block stimulant effects of cocaine

scientific article published in August 1991

Self-administration of cocaine induces dopamine-independent self-administration of sigma agonists.

scientific article published on 28 November 2012

Sigma receptor agonists: receptor binding and effects on mesolimbic dopamine neurotransmission assessed by microdialysis.

scientific article

Stereoselective behavioral effects of N6-phenylisopropyl-adenosine and antagonism by caffeine

scientific article published in January 1985

Stimulants as specific inducers of dopamine-independent σ agonist self-administration in rats

scientific article

Structure-Activity Relationships at the Monoamine Transporters for a Novel Series of Modafinil (2-[(diphenylmethyl)sulfinyl]acetamide) Analogues

scientific article

Structure-activity relationship comparison of (S)-2beta-substituted 3alpha-(bis[4-fluorophenyl]methoxy)tropanes and (R)-2beta-substituted 3beta-(3,4-dichlorophenyl)tropanes at the dopamine transporter

scientific article

Structure-activity relationship studies on a novel series of (S)-2beta-substituted 3alpha-[bis(4-fluoro- or 4-chlorophenyl)methoxy]tropane analogues for in vivo investigation

scientific article

Structure-activity relationships at monoamine transporters for a series of N-substituted 3alpha-(bis[4-fluorophenyl]methoxy)tropanes: comparative molecular field analysis, synthesis, and pharmacological evaluation

scientific article

Structure-activity relationships at the monoamine transporters and sigma receptors for a novel series of 9-[3-(cis-3, 5-dimethyl-1-piperazinyl)propyl]carbazole (rimcazole) analogues

scientific article

Structure-activity relationships for a novel series of citalopram (1-(3-(dimethylamino)propyl)-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-5-carbonitrile) analogues at monoamine transporters

scientific article

Synthesis and biological evaluation of 2-substituted 3beta-tolyltropane derivatives at dopamine, serotonin, and norepinephrine transporters

scientific article

Synthesis and biological evaluation of meperidine analogues at monoamine transporters

scientific article (publication date: 10 March 2005)

Synthesis and dopamine transporter affinity of the four stereoisomers of (+/-)-2-(methoxycarbonyl)-7-methyl-3-phenyl-7-azabicyclo[2.2.1]heptane

scientific article published in June 1998

Synthesis and ligand binding of eta(6)-(2beta-carbomethoxy-3beta-phenyltropane) transition metal complexes

scientific article published in March 1996

Synthesis and monoamine transporter binding of 2-(diarylmethoxymethyl)-3 beta-aryltropane derivatives

scientific article

Synthesis, dopamine transporter affinity, dopamine uptake inhibition, and locomotor stimulant activity of 2-substituted 3 beta-phenyltropane derivatives

scientific article

Synthesis, structure, dopamine transporter affinity, and dopamine uptake inhibition of 6-alkyl-3-benzyl-2-[(methoxycarbonyl)methyl]tropane derivatives

scientific article published in December 1997

Systemic and intracerebroventricular effects of opioid peptides in withdrawn morphine-dependent rhesus monkeys

scientific article published in January 1983

The Intriguing Effects of Substituents in the N-Phenethyl Moiety of Norhydromorphone: A Bifunctional Opioid from a Set of "Tail Wags Dog" Experiments

scientific article published on 06 June 2020

The cocaine-like behavioral effects of meperidine are mediated by activity at the dopamine transporter.

scientific article

The effect of 6-substituted-4',4"-difluorobenztropines on monoamine transporters and the muscarinic M1 receptor

scientific article

The effect of N-methylation on fenfluramine's neurotoxic and pharmacologic actions

scientific article published in July 1997

The effects of repeated administration of MDMA on the expression of sexual behavior in the male rat.

scientific article published in July 1991

The experimental imperative

scientific article published on 28 August 2002

The opiate quasiwithdrawal syndrome in rhesus monkeys: Comparison of naloxone-precipitated withdrawal to effects of cholinergic agents

scientific article published on 01 January 1984

The partial opioid agonist, buprenorphine, protects against lethal effects of cocaine

scientific article published on March 1991

The role of D2-like dopamine receptors in the locomotor stimulant effects of cocaine in mice

scientific article published in April 2001

The sigma-1 receptor modulates methamphetamine dysregulation of dopamine neurotransmission.

scientific article published on 20 December 2017

The stereotypy-inducing effects of N-substituted benztropine analogs alone and in combination with cocaine do not account for their blockade of cocaine self-administration

scientific article published on 14 September 2012

The unique psychostimulant profile of (±)-modafinil: investigation of behavioral and neurochemical effects in mice

scientific article published on 22 August 2016

The validity of the reinstatement model of craving and relapse to drug use.

scientific article

Tolerance to effects of morphine without cross tolerance to effects of clonidine on schedule-controlled behavior of pigeons

scientific article published in January 1986

Transcriptional responses to reinforcing effects of cocaine in the rat hippocampus and cortex

scientific article

Two types of bias in psychophysical detection and recognition procedures: nonparametric indices and effects of drugs

scientific article published in January 1989

Vigilance demand and the effects of stimulant drugs in a five-choice reaction-time procedure in mice

scientific article published on 01 December 2018

Yawning and locomotor behavior induced by dopamine receptor agonists in mice and rats.

scientific article

[3-cis-3,5-Dimethyl-(1-piperazinyl)alkyl]-bis-(4'-fluorophenyl)amine analogues as novel probes for the dopamine transporter

scientific article published in December 2001

c-Fos facilitates the acquisition and extinction of cocaine-induced persistent changes.

scientific article published in December 2006

σ Receptor Effects of N-Substituted Benztropine Analogs: Implications for Antagonism of Cocaine Self-Administration

scientific article

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