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List of works by Cenzo Congiu

A new convenient synthetic method and preliminary pharmacological characterization of triazinediones as prokineticin receptor antagonists

scientific article published on 14 May 2014

Amidrazones as precursors of biologically active compounds--synthesis of diaminopyrazoles for evaluation of anticancer activity

scientific article published on January 2006

Design, synthesis, and in vitro antitumor activity of new 1,4-diarylimidazole-2-ones and their 2-thione analogues

scientific article published on 15 December 2007

Effect of lysine at C-terminus of the Dmt-Tic opioid pharmacophore.

scientific article published on September 2006

Flavones and structurally related 4-chromenones inhibit carbonic anhydrases by a different mechanism of action compared to coumarins

scientific article published on 27 March 2012

Further studies on the effect of lysine at the C-terminus of the Dmt-Tic opioid pharmacophore.

scientific article published on 22 February 2007

In vitro antimycobacterial activity of newly synthesised S-alkylisothiosemicarbazone derivatives and synergistic interactions in combination with rifamycins against Mycobacterium avium.

scientific article published on July 2005

Inhibition of fatty acid amide hydrolase and cyclooxygenase by the N-(3-methylpyridin-2-yl)amide derivatives of flurbiprofen and naproxen

scientific article published on 8 October 2013

Inhibitory effect of positively charged triazine antagonists of prokineticin receptors on the transient receptor vanilloid type-1 (TRPV1) channel.

scientific article published on 17 July 2015

Inhibitory properties of ibuprofen and its amide analogues towards the hydrolysis and cyclooxygenation of the endocannabinoid anandamide.

scientific article published on 6 January 2012

New bis(pyridyl)methane derivatives from 4-hydroxy-2-pyridones: synthesis and antitumoral activity

scientific article published on January 2003

New potential anticancer agents based on the anthranilic acid scaffold: synthesis and evaluation of biological activity

scientific article published on December 2005

Novel 2-amino-isoflavones exhibit aryl hydrocarbon receptor agonist or antagonist activity in a species/cell-specific context

scientific article published on 7 April 2012

PPARγ controls pregnancy outcome through activation of EG-VEGF: new insights into the mechanism of placental development

scientific article

Prokineticin receptor 1 antagonist PC-10 as a biomarker for imaging inflammatory pain

scientific article published on 18 March 2011

Synthesis and antimycobacterial activity of new S-alkylisothiosemicarbazone derivatives.

scientific article published in March 2002

Synthesis and antiproliferative activity of 2,6-dibenzylamino-3,5-dicyanopyridines on human cancer cell lines.

scientific article published on 30 August 2005

Synthesis and antitumor evaluation of 6-thioxo-, 6-oxo- and 2,4-dioxopyrimidine derivatives.

scientific article

Synthesis and antitumour activity of 4-hydroxy-2-pyridone derivatives

scientific article published in May 2000

Synthesis and biological evaluation of novel acylhydrazone derivatives as potential antitumor agents

scientific article published on 22 August 2013

Synthesis and carbonic anhydrase I, II, IX and XII inhibition studies of 4-N,N-disubstituted sulfanilamides incorporating 4,4,4-trifluoro-3-oxo-but-1-enyl, phenacylthiourea and imidazol-2(3H)-one/thione moieties

scientific article published on 21 February 2014

Synthesis and carbonic anhydrase I, II, IX and XII inhibitory activity of sulfamates incorporating piperazinyl-ureido moieties

scientific article published on 21 July 2015

Synthesis and evaluation of anticancer activity of 2-arylamino-6-trifluoromethyl-3-(hydrazonocarbonyl)pyridines.

scientific article

Synthesis and evaluation of antitumoral activity of ester and amide derivatives of 2-arylamino-6-trifluoromethyl-3-pyridinecarboxylic acids.

scientific article

Synthesis and evaluation of paracetamol esters as novel fatty acid amide hydrolase inhibitors.

scientific article

Synthesis and in vitro antitumor activity of new 4,5-dihydropyrazole derivatives.

scientific article published on 9 August 2010

Synthesis and in vitro antitumoral activity of new 3,5-dicyanopyridine derivatives.

scientific article published on 19 November 2006

Synthesis and in vitro antitumoral activity of new N-phenyl-3-pyrrolecarbothioamides.

scientific article published in February 2003

Synthesis and in vitro antitumoral activity of new hydrazinopyrimidine-5-carbonitrile derivatives

scientific article published on 26 September 2005

Synthesis of new 2-arylamino-6-trifluoromethylpyridine-3-carboxylic acid derivatives and investigation of their analgesic activity

scientific article (publication date: August 2004)

Synthesis of new N-(2-(trifluoromethyl)pyridin-4-yl)anthranilic acid derivatives and their evaluation as anticancer agents.

scientific article

Synthesis of sulfonamides incorporating piperazinyl-ureido moieties and their carbonic anhydrase I, II, IX and XII inhibitory activity

scientific article published on 26 July 2015

Synthetic Flavonoids, Aminoisoflavones: Interaction and Reactivity with Metal-Free and Metal-Associated Amyloid-β Species

scientific article

TRPV1 modulators: Synthesis and in vitro evaluation of 1-heteroaryl piperidinecarboxamide and piperazinylurea derivatives

scientific article published on 06 June 2015

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