List of works - Yuri Bukhtiyarov

Biphenyl/diphenyl ether renin inhibitors: filling the S1 pocket of renin via the S3 pocket

scientific article

Cloning, characterization and site-directed mutagenesis of canine renin

scientific article

Design and optimization of renin inhibitors: Orally bioavailable alkyl amines

scientific article

Discovery and optimization of adamantyl carbamate inhibitors of 11β-HSD1.

scientific article published on 7 September 2010

Discovery of VTP-27999, an Alkyl Amine Renin Inhibitor with Potential for Clinical Utility

scientific article

Discovery of a Novel, Orally Efficacious Liver X Receptor (LXR) β Agonist

scientific article

Identification of 23S rRNA nucleotides neighboring the P-loop in the Escherichia coli 50S subunit.

scientific article

Identification of Inhibitors of Bacterial Transcription/Translation Machinery Utilizing a Miniaturized 1536-Well Format Screen ⬇️

scientific article published on August 1, 2001

Identification of spirooxindole and dibenzoxazepine motifs as potent mineralocorticoid receptor antagonists

scientific article

Photolabile derivatives of oligonucleotides as probes of ribosomal structure

scientific article published on 01 January 2000

Photoreactive analogues of prenyl diphosphates as inhibitors and probes of human protein farnesyltransferase and geranylgeranyltransferase type I

scientific article published on 01 August 1995

Purification and characterization of recombinant human renin for X-ray crystallization studies

scientific article

Regulation of sphingomyelin phosphodiesterase acid-like 3A gene (SMPDL3A) by liver X receptors.

scientific article

Solubilization and characterization of dehydrodolichyl diphosphate synthase from the yeast Saccharomyces carlsbergensis

scientific article published on 01 June 1993

Spirocyclic ureas: orally bioavailable 11 beta-HSD1 inhibitors identified by computer-aided drug design

scientific article published on 4 January 2010

Structure-based design and synthesis of 1,3-oxazinan-2-one inhibitors of 11β-hydroxysteroid dehydrogenase type 1.

scientific article published on 4 August 2011

Three-dimensional placement of the conserved 530 loop of 16 S rRNA and of its neighboring components in the 30 S subunit

scientific article published on 01 February 1999

List of works by Yuri Bukhtiyarov

Biphenyl/diphenyl ether renin inhibitors: filling the S1 pocket of renin via the S3 pocket

Cloning, characterization and site-directed mutagenesis of canine renin

Design and optimization of renin inhibitors: Orally bioavailable alkyl amines

Discovery and optimization of adamantyl carbamate inhibitors of 11β-HSD1.

Discovery of VTP-27999, an Alkyl Amine Renin Inhibitor with Potential for Clinical Utility

Discovery of a Novel, Orally Efficacious Liver X Receptor (LXR) β Agonist

Identification of 23S rRNA nucleotides neighboring the P-loop in the Escherichia coli 50S subunit.

Identification of Inhibitors of Bacterial Transcription/Translation Machinery Utilizing a Miniaturized 1536-Well Format Screen ⬇️

Identification of spirooxindole and dibenzoxazepine motifs as potent mineralocorticoid receptor antagonists

Photolabile derivatives of oligonucleotides as probes of ribosomal structure

Photoreactive analogues of prenyl diphosphates as inhibitors and probes of human protein farnesyltransferase and geranylgeranyltransferase type I

Purification and characterization of recombinant human renin for X-ray crystallization studies

Regulation of sphingomyelin phosphodiesterase acid-like 3A gene (SMPDL3A) by liver X receptors.

Solubilization and characterization of dehydrodolichyl diphosphate synthase from the yeast Saccharomyces carlsbergensis

Spirocyclic ureas: orally bioavailable 11 beta-HSD1 inhibitors identified by computer-aided drug design

Structure-based design and synthesis of 1,3-oxazinan-2-one inhibitors of 11β-hydroxysteroid dehydrogenase type 1.

Three-dimensional placement of the conserved 530 loop of 16 S rRNA and of its neighboring components in the 30 S subunit