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List of works by Kuo-Shyan Lin

(18)F-AmBF3-MJ9: a novel radiofluorinated bombesin derivative for prostate cancer imaging.

scientific article

(18)F-trifluoroborate derivatives of [des-arg(10)]kallidin for imaging bradykinin b1 receptor expression with positron emission tomography

scientific article published on 09 February 2015

2-Fluoropyridine prosthetic compounds for the 18F labeling of bombesin analogues

scientific article

225Ac-H4py4pa for Targeted Alpha Therapy

scientific article published on 09 April 2020

A Metal-Free DOTA-Conjugated 18F-Labeled Radiotracer: [18F]DOTA-AMBF3-LLP2A for Imaging VLA-4 Over-Expression in Murine Melanoma with Improved Tumor Uptake and Greatly Enhanced Renal Clearance

scientific article published on 08 April 2019

A Systematic Review of Molecular Imaging Agents Targeting Bradykinin B1 and B2 Receptors

scientific article published on 17 August 2020

A new high affinity technetium analogue of bombesin containing DTPA as a pharmacokinetic modifier

scientific article published in November 2004

A new high affinity technetium-99m-bombesin analogue with low abdominal accumulation

scientific article published in January 2005

A novel nicotinic acetylcholine receptor antagonist radioligand for PET studies

scientific article

An organotrifluoroborate for broadly applicable one-step 18F-labeling

scientific article published on 04 September 2014

Bench to Bedside: Albumin Binders for Improved Cancer Radioligand Therapies

scientific article published on 23 January 2019

Comparative evaluation of positron emission tomography radiotracers for imaging the norepinephrine transporter: (S,S) and (R,R) enantiomers of reboxetine analogs ([11C]methylreboxetine, 3-Cl-[11C]methylreboxetine and [18F]fluororeboxetine), (R)-[11C

scientific article

Comparison of biological properties of [177 Lu]Lu-ProBOMB1 and [177 Lu]Lu-NeoBOMB1 for GRPR targeting

scientific article published on 11 January 2020

Design and synthesis of a short-chain bitistatin analogue for imaging thrombi and emboli

scientific article published in September 2004

Design, Synthesis, and Initial Evaluation of High-Affinity Technetium Bombesin Analogues

scientific article published on March 1, 1998

Design, synthesis and evaluation of (18)F-labeled bradykinin B1 receptor-targeting small molecules for PET imaging.

scientific article published on 27 June 2016

Design, synthesis and structure-activity relationship of rhenium 2-arylbenzothiazoles as β-amyloid plaque binding agents

scientific article published on 24 January 2013

Dual mode fluorescent (18)F-PET tracers: efficient modular synthesis of rhodamine-[cRGD]2-[(18)F]-organotrifluoroborate, rapid, and high yielding one-step (18)F-labeling at high specific activity, and correlated in vivo PET imaging and ex vivo fluor

scientific article

Effects of Linker Modification on Tumor-to-Kidney Contrast of 68Ga-Labeled PSMA-Targeted Imaging Probes

scientific article published on 03 July 2018

Effects of adding an albumin binder chain on [177Lu]Lu-DOTATATE

scientific article published on 09 August 2018

Enhancing Treatment Efficacy of Lu-PSMA-617 with the Conjugation of an Albumin-Binding Motif: Preclinical Dosimetry and Endoradiotherapy Studies

scientific article published on 05 October 2018

Evaluation of 99mTc-sulfonamide and sulfocoumarin derivatives for imaging carbonic anhydrase IX expression

scientific article published on 13 April 2018

Evaluation of Met-Val-Lys as a Renal Brush Border Enzyme-Cleavable Linker to Reduce Kidney Uptake of 68Ga-Labeled DOTA-Conjugated Peptides and Peptidomimetics

scientific article published on 25 August 2020

Evaluation of a new norepinephrine transporter PET ligand in baboons, both in brain and peripheral organs

scientific article published on December 15, 2003

Functionally Versatile and Highly Stable Chelator for 111In and 177Lu: Proof-of-Principle Prostate-Specific Membrane Antigen Targeting

scientific article published on 05 May 2019

H2CHXhox: Rigid Cyclohexane-Reinforced Nonmacrocyclic Chelating Ligand for [nat/67/68Ga]Ga3

scientific article published on 16 March 2020

H2hox: Dual-Channel Oxine-Derived Acyclic Chelating Ligand for 68Ga Radiopharmaceuticals

scientific article published on 10 July 2018

High-Contrast CXCR4-Targeted <sup>18</sup>F-PET Imaging Using a Potent and Selective Antagonist

scientific article published on 30 November 2020

Imaging Bradykinin B1 Receptor with 68Ga-Labeled [des-Arg10]Kallidin Derivatives: Effect of the Linker on Biodistribution and Tumor Uptake

scientific article published on 02 July 2015

Improving the stability of C-labeled L-methionine with ascorbate

scientific article published on 04 October 2017

Insight into the Development of PET Radiopharmaceuticals for Oncology

scientific article published on 21 May 2020

Kit-like 18F-labeling of RGD-19F-Arytrifluroborate in high yield and at extraordinarily high specific activity with preliminary in vivo tumor imaging

scientific article published on June 27, 2013

Melanoma Imaging Using 18F-Labeled α-Melanocyte-Stimulating Hormone Derivatives with Positron Emission Tomography

scientific article published on 10 May 2018

Modeling and analysis of PET studies with norepinephrine transporter ligands: the search for a reference region.

scientific article published in July 2005

Nitroimidazole-Containing H2dedpa and H2CHXdedpa Derivatives as Potential PET Imaging Agents of Hypoxia with (68)Ga.

scientific article published on 30 April 2015

Novel 177Lu-labeled Albumin-binder-conjugated PSMA-targeting Agents with Extremely High Tumor Uptake and Enhanced Tumor-to-kidney Absorbed Dose Ratio

scientific article published on 28 August 2020

PET Imaging of Carbonic Anhydrase IX Expression of HT-29 Tumor Xenograft Mice with (68)Ga-Labeled Benzenesulfonamides.

scientific article

Positron Emission Tomography Imaging of the Gastrin-Releasing Peptide Receptor with a Novel Bombesin Analogue

scientific article published on 16 January 2019

Preliminary evaluation of 18F-labeled LLP2A-trifluoroborate conjugates as VLA-4 (α4β1 integrin) specific radiotracers for PET imaging of melanoma.

scientific article published on 12 March 2018

Radiolabeled B9958 Derivatives for Imaging Bradykinin B1 Receptor Expression with Positron Emission Tomography: Effect of the Radiolabel-Chelator Complex on Biodistribution and Tumor Uptake

scientific article published on 27 June 2016

Radiolabeled R954 Derivatives for Imaging Bradykinin B1 Receptor Expression with Positron Emission Tomography

scientific article published on 17 January 2017

Single step 18F-labeling of dimeric cycloRGD for functional PET imaging of tumors in mice

scientific article published on 3 October 2013

Synthesis and C-11 labeling of three potent norepinephrine transporter selective ligands ((R)-nisoxetine, lortalamine, and oxaprotiline) for comparative PET studies in baboons.

scientific article

Synthesis and Evaluation of [18F]FEtLos and [18F]AMBF3Los as Novel 18F-Labelled Losartan Derivatives for Molecular Imaging of Angiotensin II Type 1 Receptors

scientific article published on 18 April 2020

Synthesis and beta-amyloid binding properties of rhenium 2-phenylbenzothiazoles

scientific article published on 27 February 2009

Synthesis and evaluation of (18)F-labeled 4-nitrobenzyl derivatives for imaging tumor hypoxia with positron emission tomography: Comparison of 2-[(18)F]fluoroethyl carbonate and 2-[(18)F]fluoroethyl carbamate.

scientific article published on 19 November 2015

Synthesis and evaluation of (18)F-labeled tertiary benzenesulfonamides for imaging carbonic anhydrase IX expression in tumours with positron emission tomography.

scientific article published on 17 May 2014

Synthesis and evaluation of (18)F-trifluoroborate derivatives of triphenylphosphonium for myocardial perfusion imaging.

scientific article published on 22 February 2016

Synthesis and evaluation of 18F-labeled carbonic anhydrase IX inhibitors for imaging with positron emission tomography

scientific article published on 07 March 2013

Synthesis and evaluation of a 68Ga-labeled bradykinin B1 receptor agonist for imaging with positron emission tomography

scientific article published on 23 November 2016

Synthesis and evaluation of an 18 F-labeled trifluoroborate derivative of 2-nitroimidazole for imaging tumor hypoxia with positron emission tomography.

scientific article

Synthesis and evaluation of an F-labeled boramino acid analog of aminosuberic acid for PET imaging of the antiporter system x

scientific article published on 08 June 2018

Synthesis and positron emission tomography studies of C-11-labeled isotopomers and metabolites of GTS-21, a partial alpha7 nicotinic cholinergic agonist drug.

scientific article

Synthesis and positron emission tomography studies of carbon-11-labeled imatinib (Gleevec).

scientific article

Synthesis, enantiomeric resolution, F-18 labeling and biodistribution of reboxetine analogs: promising radioligands for imaging the norepinephrine transporter with positron emission tomography

scientific article published in May 2005

Synthesis, enantiomeric resolution, and selective C-11 methylation of a highly selective radioligand for imaging the norepinephrine transporter with positron emission tomography

scientific article published in August 2004

Toward 18 F-Labeled Theranostics: A Single Agent that Can Be Labeled with 18 F, 64 Cu, or 177 Lu

scientific article published on 04 December 2019

[68Ga]Ga/[177Lu]Lu-BL01, a Novel Theranostic Pair for Targeting C-X-C Chemokine Receptor 4

scientific article published on 04 October 2019

[nat/44Sc(pypa)]-: Thermodynamic Stability, Radiolabeling, and Biodistribution of a Prostate-Specific-Membrane-Antigen-Targeting Conjugate

scientific article published on 24 January 2020

f-[18F]fluoroethanol and 3-[18F]fluoropropanol: facile preparation, biodistribution in mice, and their application as nucleophiles in the synthesis of [18F]fluoroalkyl aryl ester and ether PET tracers

scientific article published on 14 June 2013

tBu4octapa-alkyl-NHS for metalloradiopeptide preparation

scientific article published on 27 May 2020