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List of works by Jean Jacques Vanden Eynde

1,2-ethane bis-1-amino-4-benzamidine is active against several brain insult and seizure challenges through anti-NMDA mechanisms targeting the 3H-TCP binding site and antioxidant action.

scientific article published on 3 April 2010

1,4-diarylpiperazines and analogs as anti-tubercular agents: synthesis and biological evaluation.

scientific article

2015: A Transition Year for Pharmaceuticals?

scientific article published on 27 January 2016

2017: A Fruitful Year for Pharmaceuticals

scientific article published on 21 December 2017

2019: An Awesome Year for Pharmaceuticals

scientific article published on 01 January 2020

Alkanediamide-Linked Bisbenzamidines Are Promising Antiparasitic Agents.

scientific article published on 19 April 2016

Announcing the 2016 Pharmaceuticals Travel Award for Young Investigators

scientific article published on 27 June 2016

Announcing the 2017 Pharmaceuticals Travel Award for Young Post-Doctoral Researchers

scientific article published on 22 May 2017

Anti-plasmodial and anti-leishmanial activity of conformationally restricted pentamidine congeners

scientific article

Antitumor and Anti-Pneumocystis Carinii Activities of Novel Bisbenzamidines

Baricitinib: A 2018 Novel FDA-Approved Small Molecule Inhibiting Janus Kinases

scientific article published on 12 March 2019

Batch and continuous flow preparation of Hantzsch 1,4-dihydropyridines under microwave heating and simultaneous real-time monitoring by Raman spectroscopy. An exploratory study

scientific article published on 09 July 2014

Biological evaluation of bisbenzaldehydes against four Mycobacterium species

scientific article published on 18 March 2013

Bis(oxyphenylene)benzimidazoles: a novel class of anti-Plasmodium falciparum agents.

scientific article

Bisbenzamidines as antifungal agents. are both amidine functions required to observe an anti-Pneumocystis carinii activity?

scientific article published on 11 June 2010

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-3

scientific article published on 30 June 2018

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-5

scientific article published on 30 June 2019

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-6

scientific article published on 28 December 2019

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes⁻4

scientific article published on 31 December 2018

COVID-19: A Brief Overview of the Discovery Clinical Trial

scientific article published on 10 April 2020

COVID-19: An Update About the Discovery Clinical Trial

scientific article published on 14 May 2020

Correction to: Affinity capillary electrophoresis for identification of active drug candidates in myotonic dystrophy type 1

scientific article published on 01 January 2019

Design and synthesis of N¹,N⁵-bis[4-(5-alkyl-1,2,4-oxadiazol-3-yl)phenyl]glutaramides as potential antifungal prodrugs

scientific article published on 12 September 2013

Designing a high performance, stable spectroscopic biosensor for the binding of large and small molecules

scientific article published on 24 August 2017

Evaluation of bisbenzamidines as inhibitors for matriptase-2.

scientific article published on 26 May 2016

Evidences for the formation of bisbenzamidine-heme complexes in cell-free systems

scientific article published on 01 April 2004

Fragment-Based Design of Symmetrical Bis-benzimidazoles as Selective Inhibitors of the Trimethoprim-Resistant, Type II R67 Dihydrofolate Reductase ⬇️

scientific article published on March 28, 2012

Highly active anti-Pneumocystis carinii compounds in a library of novel piperazine-linked bisbenzamidines and related compounds

scientific article published in November 2004

How Efficient Is My (Medicinal) Chemistry?

scientific article

Liquid-phase synthesis of polyhydroquinoline using task-specific ionic liquid technology

scientific article published in November 2006

Novel bisbenzamidines as potential drug candidates for the treatment of Pneumocystis carinii pneumonia

scientific article published in September 2004

Novel bisbenzimidazoles with antileishmanial effectiveness

scientific article

PPARs: Interference with Warburg' Effect and Clinical Anticancer Trials.

scientific article published on 8 May 2012

Parallel solution-phase synthesis of conformationally restricted congeners of pentamidine and evaluation of their antiplasmodial activities

scientific article published on May 2004

Pentamidine analogs as inhibitors of [(3)H]MK-801 and [(3)H]ifenprodil binding to rat brain NMDA receptors.

scientific article published on 14 June 2015

Pharmaceuticals Best Paper Award 2015.

scientific article published on 5 June 2015

Pharmaceuticals: Impact Factor or CiteScore™.

scientific article published on 6 July 2017

Piperazine-linked bisbenzamidines: a novel class of antileishmanial agents.

scientific article

Potential of bisbenzimidazole-analogs toward metronidazole-resistant Trichomonas vaginalis isolates.

scientific article published on 10 March 2017

Progress Confirmed for Pharmaceuticals in 2016.

scientific article published on 26 December 2016

Some non-conventional biomolecular targets for diamidines. A short survey

scientific article published on 05 March 2014

Structure-Based Design of Dimeric Bisbenzimidazole Inhibitors to an Emergent Trimethoprim-Resistant Type II Dihydrofolate Reductase Guides the Design of Monomeric Analogues

scientific article published on 10 June 2019

Tafenoquine: A 2018 Novel FDA-Approved Prodrug for the Radical Cure of Plasmodium vivax Malaria and Prophylaxis of Malaria

scientific article published on 30 July 2019

Third International Electronic Conference on Medicinal Chemistry (ECMC-3).

scientific article published on 9 February 2018

Three optimized and validated (using accuracy profiles) LC methods for the determination of pentamidine and new analogs in rat plasma

scientific article published on 02 November 2010

Trypanocidal activity of piperazine-linked bisbenzamidines and bisbenzamidoxime, an orally active prodrug.

scientific article published on 24 October 2007

Ultra high performance liquid chromatography method for the determination of pentamidine and analog in rat biological fluids.

scientific article published on 10 February 2014

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