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List of works by Scott G. Franzblau

"Studies on biodiversity of Vietnam and Laos" 1998-2005: examining the impact.

scientific article published in March 2006

(+)-Totarol from Chamaecyparis nootkatensis and activity against Mycobacterium tuberculosis

scientific article

12,34-Oxamanzamines, novel biocatalytic and natural products from manzamine producing Indo-Pacific sponges

2,6-hexadecadiynoic acid and 2,6-nonadecadiynoic acid: novel synthesized acetylenic fatty acids as potent antifungal agents

scientific article

2-methoxylated fatty acids in marine sponges: defense mechanism against mycobacteria?

scientific article published in July 2004

3,5-Dialkoxypyridine analogues of bedaquiline are potent antituberculosis agents with minimal inhibition of the hERG channel

scientific article published on 15 February 2019

5-tert-butyl-N-pyrazol-4-yl-4,5,6,7-tetrahydrobenzo[d]isoxazole-3-carboxamide derivatives as novel potent inhibitors of Mycobacterium tuberculosis pantothenate synthetase: initiating a quest for new antitubercular drugs

scientific article published on 13 March 2008

6-Cyano Analogues of Bedaquiline as Less Lipophilic and Potentially Safer Diarylquinolines for Tuberculosis

scientific article

6-Hydrogen-8-Methylquinolones Active Against Replicating and Non-replicating Mycobacterium tuberculosis

scientific article published on 10 September 2012

A Potentially New Treatment for Tuberculosis; Will a Diarylquinoline Work for Leprosy?

scientific article published on 01 March 2005

A microbiological assessment of novel nitrofuranylamides as anti-tuberculosis agents

scientific article published on 07 August 2008

A new antitubercular mulinane diterpenoid from Azorella madreporica Clos

scientific article published on July 1998

A novel combinatorial biocatalytic approach for producing antibacterial compounds effective against Mycobacterium tuberculosis (TB).

scientific article published on 8 June 2013

A novel indigoid anti-tuberculosis agent

scientific article

Active Site Loop Dynamics of a Class IIa Fructose 1,6-Bisphosphate Aldolase from Mycobacterium tuberculosis

scientific article

Activity of 7-methyljuglone in combination with antituberculous drugs against Mycobacterium tuberculosis

scientific article

Activity of Scottish plant, lichen and fungal endophyte extracts against Mycobacterium aurum and Mycobacterium tuberculosis

scientific article published in May 2010

Advanced applications of counter-current chromatography in the isolation of anti-tuberculosis constituents from Dracaena angustifolia

scientific article published on 11 January 2007

Advent of Imidazo[1,2-a]pyridine-3-carboxamides with Potent Multi- and Extended Drug Resistant Antituberculosis Activity

scientific article

Agelasine F from a Philippine Agelas sp. sponge exhibits in vitro antituberculosis activity

scientific article published in May 2000

Airborne antituberculosis activity of Eucalyptus citriodora essential oil.

scientific article published on 18 March 2014

Allylic thiocyanates as a new class of antitubercular agents

scientific article published on 21 August 2012

An NMR method towards the routine chiral determination of natural products

scientific article

An antimicrobial guanidine-bearing sesterterpene from the cultured cyanobacterium Scytonema sp. ⬇️

scientific article published on November 2009

An antimycobacterial pleuromutilin analogue effective against dormant bacilli

scientific article

An ethnobotanical survey of medicinal plants of Laos toward the discovery of bioactive compounds as potential candidates for pharmaceutical development.

scientific article published on 2 December 2011

Anti-TB polyynes from the roots of Angelica sinensis ⬇️

scientific article published on July 2008

Anti-infective discorhabdins from a deep-water alaskan sponge of the genus Latrunculia

scientific article published on March 2010

Anti-tuberculosis constituents from the stem bark of Micromelum hirsutum. ⬇️

scientific article

Antimalarial bromophycolides J-Q from the Fijian red alga Callophycus serratus ⬇️

scientific article published on April 2009

Antimycobacterial Rufomycin Analogues from Streptomyces atratus Strain MJM3502 ⬇️

scientific article published on 07 February 2020

Antimycobacterial activities of dehydrocostus lactone and its oxidation products

scientific article published on October 1998

Antimycobacterial activity of (E)-phytol and derivatives: a preliminary structure-activity study.

scientific article published on February 1998

Antimycobacterial activity of substituted isosteres of pyridine- and pyrazinecarboxylic acids

scientific article published on June 1998

Antimycobacterial activity of substituted isosteres of pyridine- and pyrazinecarboxylic acids. 2.

scientific article

Antimycobacterial agents from selected Mexican medicinal plants

scientific article

Antimycobacterial compounds from Piper sanctum

scientific article published in December 2004

Antimycobacterial cycloartanes from Borrichia frutescens

scientific article published on December 1996

Antimycobacterial ergosterol-5,8-endoperoxide from Ajuga remota

scientific article

Antimycobacterial eudesmanolides from Inula helenium and Rudbeckia subtomentosa

scientific article

Antimycobacterial evaluation of germacranolides

scientific article published on September 1998

Antimycobacterial flavones from Haplopappus sonorensis

scientific article published in April 2003

Antimycobacterial terpenoids from Juniperus communis L. (Cuppressaceae).

scientific article published on 13 September 2009

Antitubercular activity and inhibitory effect on Epstein-Barr virus activation of sterols and polyisoprenepolyols from an edible mushroom, Hypsizigus marmoreus ⬇️

scientific article published on June 2005

Antitubercular activity of the semi-polar extractives of Uvaria rufa

scientific article published in October 2012

Antitubercular activity of triterpenoids from Asteraceae flowers

scientific article published in January 2005

Antitubercular activity of triterpenoids from Lippia turbinata.

scientific article

Antitubercular constituents from Premna odorata Blanco

scientific article published on 23 April 2014

Antitubercular constituents from the hexane fraction of Morinda citrifolia Linn. (Rubiaceae).

scientific article published in November 2002

Antitubercular constituents of Valeriana laxiflora

scientific article

Antitubercular sterols from Thalia multiflora Horkel ex Koernicke

scientific article published in October 2005

Antitubercular triterpenes and phytosterols from Pandanus tectorius Soland. var. laevis

scientific article published on 14 December 2007

Antituberculosis Cycloartane Triterpenoids from Radermachera boniana ⬇️

scientific article published on 06 April 2011

Antituberculotic and Antiprotozoal Activities of Primin, a Natural Benzoquinone:In vitro andin vivo Studies

scientific article published on 01 November 2006

Bioactive bromophycolides R-U from the Fijian red alga Callophycus serratus ⬇️

scientific article

Bioactive metabolites of Diaporthe sp. P133, an endophytic fungus isolated from Pandanus amaryllifolius

scientific article

Biological evaluation of plants of Laos used in the treatment of tuberculosis in Lao traditional medicine

scientific article

Byrsonima fagifolia Niedenzu Apolar Compounds with Antitubercular Activity.

scientific article published on 15 June 2011

Callophycoic acids and callophycols from the Fijian red alga Callophycus serratus ⬇️

scientific article

Carbamidocyclophanes F and G with Anti-Mycobacterium tuberculosis Activity from the Cultured Freshwater Cyanobacterium Nostoc sp ⬇️

scientific article

Carcinogenic effects of N-nitroso-3-(substituted phenylimino)-indolin-2-one derivatives

scientific article published on July 2012

Characterization of Intracellular Activity of Antitubercular Constituents the Roots of Euclea natalensis

scientific article published in January 2005

Chemical Diversity and Antimicrobial Potential of Cultivable Fungi from Deep-Sea Sediments of the Gulf of Mexico

scientific article published in 2021

Chlorinated Coumarins from the Polypore MushroomFomitopsis officinalisand Their Activity againstMycobacterium tuberculosis ⬇️

scientific article (publication date: 25 October 2013)

Comparative in vitro antimicrobial activity of Chinese medicinal herbs

scientific article published in March 1986

Comprehensive analysis of methods used for the evaluation of compounds against Mycobacterium tuberculosis

scientific article published on 30 August 2012

Constituents of Senecio chionophilus with potential antitubercular activity

scientific article published in September 2004

Construction and functionalization of fused pyridine ring leading to novel compounds as potential antitubercular agents

scientific article published on 05 June 2012

Counter-current chromatography based analysis of synergy in an anti-tuberculosis ethnobotanical

scientific article

Crystallization and preliminary X-ray characterization of the glpX-encoded class II fructose-1,6-bisphosphatase from Mycobacterium tuberculosis

scientific article

Current prospects of synthetic curcumin analogs and chalcone derivatives against mycobacterium tuberculosis

scientific article

Cytotoxic constituents from Lobaria scrobiculata and a comparison of two bioassays for their evaluation

scientific article

Dereplication of pentacyclic triterpenoids in plants by GC-EI/MS.

scientific article published in March 2006

Derivatives of 3-isoxazolecarboxylic acid esters: a potent and selective compound class against replicating and nonreplicating Mycobacterium tuberculosis

scientific article published on January 2012

Design and Syntheses of Anti-Tuberculosis Agents Inspired by BTZ043 Using a Scaffold Simplification Strategy

scientific article

Design, Synthesis, and Pharmacological Evaluation of Mefloquine-Based Ligands as Novel Antituberculosis Agents

scientific article published on 01 November 2007

Design, Synthesis, and SAR Studies of Mefloquine-Based Ligands as Potential Antituberculosis Agents

scientific article published on 01 June 2006

Design, synthesis and anti-tubercular evaluation of new 2-acylated and 2-alkylated amino-5-(4-(benzyloxy)phenyl)thiophene-3-carboxylic acid derivatives. Part 1.

scientific article published on 19 May 2011

Design, synthesis and investigation on the structure-activity relationships of N-substituted 2-aminothiazole derivatives as antitubercular agents

scientific article

Design, synthesis, and structure-activity relationship studies of tryptanthrins as antitubercular agents

scientific article published on 29 January 2013

Diguanidino and "reversed" diamidino 2,5-diarylfurans as antimicrobial agents

scientific article

Discovery and characterization of the tuberculosis drug lead ecumicin ⬇️

scientific article published on 19 November 2014

Discovery and development of the covalent hydrates of trifluoromethylated pyrazoles as riboflavin synthase inhibitors with antibiotic activity against Mycobacterium tuberculosis

scientific journal article

Discovery and optimization of benzotriazine di-N-oxides targeting replicating and nonreplicating Mycobacterium tuberculosis

scientific article

Discovery of New Cyclic Lipodepsipeptide Orfamide N via Partnership with Middle School Students from the Boys and Girls Club

scientific article published on 24 October 2024

Discovery of a capuramycin analog that kills nonreplicating Mycobacterium tuberculosis and its synergistic effects with translocase I inhibitors

scientific article

Discovery of selective menaquinone biosynthesis inhibitors against Mycobacterium tuberculosis

scientific article

Diterpenes from Solidago rugosa

scientific article published on January 1995

Efficacy of quinoxaline-2-carboxylate 1,4-di-N-oxide derivatives in experimental tuberculosis

scientific article published on 14 July 2008

Enhancing hit identification in Mycobacterium tuberculosis drug discovery using validated dual-event Bayesian models

scientific article

Ethnobotanical approach versus random approach in the search for new bioactive compounds: Support of a hypothesis ⬇️

scientific article published on January 1, 2012

Ethnobotany/ethnopharmacology and mass bioprospecting: issues on intellectual property and benefit-sharing.

scientific article

Ethnopharmacological evaluation of the informant consensus model on anti-tuberculosis claims among the Manus

scientific article

Eucapsitrione, an anti-Mycobacterium tuberculosis anthraquinone derivative from the cultured freshwater cyanobacterium Eucapsis sp ⬇️

scientific article

Evaluation of a modified antimycobacterial susceptibility test using Middlebrook 7H10 agar containing 2,3-diphenyl-5-thienyl-(2)-tetrazolium chloride

scientific article published on 06 March 2006

Evaluation of antiprotozoal and antimycobacterial activities of the resin glycosides and the other metabolites of Scrophularia cryptophila

scientific article published on 29 August 2007

Evaluation of gyrase B as a drug target in Mycobacterium tuberculosis

scientific article published on 2 November 2011

Evaluation of the flora of Puerto Rico for in vitro antiplasmodial and antimycobacterial activities

scientific article published in November 2001

Facile transformation of Biginelli pyrimidin-2(1H)-ones to pyrimidines. In vitro evaluation as inhibitors of Mycobacterium tuberculosis and modulators of cytostatic activity

scientific article published on 15 March 2011

From serendipity to rational antituberculosis drug discovery of mefloquine-isoxazole carboxylic acid esters

scientific article published in November 2009

Generation and exploration of new classes of antitubercular agents: The optimization of oxazolines, oxazoles, thiazolines, thiazoles to imidazo[1,2-a]pyridines and isomeric 5,6-fused scaffolds

scientific article published on 16 February 2012

HTS, chemical hybridization, and drug design identify a chemically unique antituberculosis agent-coupling serendipity and rational approaches to drug discovery

scientific article

Hapalindole-related alkaloids from the cultured cyanobacterium Fischerella ambigua ⬇️

scientific article published on 19 October 2010

Hytramycins V and I, anti-Mycobacterium tuberculosis hexapeptides from a Streptomyces hygroscopicus strain

scientific article published on 13 November 2013

ICAT-based comparative proteomic analysis of non-replicating persistent Mycobacterium tuberculosis

scientific article published on 20 December 2005

Identification and characterization of novel inhibitors of mPTPB, an essential virulent phosphatase from Mycobacterium tuberculosis

scientific article

Identification of Pyrazolo[1,5-]pyridine-3-carboxamide Diaryl Derivatives as Drug Resistant Antituberculosis Agents

article published in 2019

Identification of a small molecule with activity against drug-resistant and persistent tuberculosis

scientific article

Identification of novel inhibitors of nonreplicating Mycobacterium tuberculosis using a carbon starvation model

scientific article

Identification, synthesis, and pharmacological evaluation of tetrahydroindazole based ligands as novel antituberculosis agents

scientific article published in January 2010

Improved BM212 MmpL3 inhibitor analogue shows efficacy in acute murine model of tuberculosis infection

scientific article

Improved green fluorescent protein reporter gene-based microplate screening for antituberculosis compounds by utilizing an acetamidase promoter.

scientific article

In Vitro Activities of Enantiopure and Racemic 1'-Acetoxychavicol Acetate against Clinical Isolates of Mycobacterium tuberculosis

scientific article published on 18 September 2017

In vitro and in vivo activities of macrolide derivatives against Mycobacterium tuberculosis

scientific article

In vitro and in vivo activities of ruthenium(II) phosphine/diimine/picolinate complexes (SCAR) against Mycobacterium tuberculosis

scientific article

In vitro and in vivo antimycobacterial activities of ketone and amide derivatives of quinoxaline 1,4-di-N-oxide

scientific article published on 23 May 2008

In vitro susceptibility of Mycobacterium tuberculosis to extracts of Eucalyptus camaldulensis and Eucalyptus torelliana and isolated compounds

scientific article

In vivo and in vitro evaluation of highly specific thiolate carrier group copper(II) and zinc(II) complexes on Ehrlich ascites carcinoma tumor model

scientific article published on 15 September 2010

Indole alkaloids from the leaves of Philippine Alstonia scholaris

scientific article published in May 2005

Indole alkaloids from two cultured cyanobacteria, Westiellopsis sp. and Fischerella muscicola ⬇️

scientific article

Induction of pyruvate decarboxylase in Candida utilis

scientific article published on 01 January 1983

Inhibiting enoyl-ACP reductase (FabI) across pathogenic microorganisms by linear sesquiterpene lactones from Anthemis auriculata

scientific article

Inhibition of Mycobacterium tuberculosis Methionine Aminopeptidases by Bengamide Derivatives

scientific article

Inhibition of Mycobacterium tuberculosis growth by saringosterol from Lessonia nigrescens.

scientific article

Inhibitory effect of oxygenated cholestan-3β-ol derivatives on the growth of Mycobacterium tuberculosis

scientific article published on 14 September 2013

Inhibitory effect of sterols from Ruprechtia triflora and diterpenes from Calceolaria pinnifolia on the growth of Mycobacterium tuberculosis

scientific article published in July 2003

Insights into the Chemical Diversity of Selected Fungi from the Tza Itzá Cenote of the Yucatan Peninsula

scientific article published on 28 March 2022

Isolation of Tryptanthrin and Reassessment of Evidence for Its Isobaric Isostere Wrightiadione in Plants of the Wrightia Genus

article

Lahorenoic Acids A–C, ortho-Dialkyl-Substituted Aromatic Acids from the Biocontrol Strain Pseudomonas aurantiaca PB-St2

scientific article published on 12 February 2013

Library synthesis using 5,6,7,8-tetrahydro-1,6-naphthyridines as scaffolds

scientific article

Low-oxygen-recovery assay for high-throughput screening of compounds against nonreplicating Mycobacterium tuberculosis

scientific article published on 8 January 2007

Manadomanzamines A and B: a novel alkaloid ring system with potent activity against mycobacteria and HIV-1.

scientific article

Manzamine B and E and ircinal A related alkaloids from an Indonesian Acanthostrongylophora sponge and their activity against infectious, tropical parasitic, and Alzheimer's diseases ⬇️

scientific article published on 2 June 2006

Mce3R Stress-Resistance Pathway Is Vulnerable to Small-Molecule Targeting That Improves Tuberculosis Drug Activities

scientific article published on 03 May 2019

Metal complexes of carboxamidrazone analogs as antitubercular agents. 1. Synthesis, X-ray crystal-structures, spectroscopic properties and antimycobacterial activity against Mycobacterium tuberculosis H(37)Rv

scientific article published in June 2002

Microplate Alamar Blue Assay (MABA) and Low Oxygen Recovery Assay (LORA) for Mycobacterium tuberculosis

scientific article published in January 2015

Modification of the side chain of micromolide, an anti-tuberculosis natural product

scientific article published in October 2008

Mycobacterium tuberculosis and cholinesterase inhibitors from Voacanga globosa

scientific article published on 19 April 2011

Mycobacterium tuberculosis growth inhibition by constituents of Sapium haematospermum

scientific article published in April 2004

NMR and molecular mechanics study of pyrethrins I and II

scientific article

NOC chemistry for tuberculosis-further investigations on the structure-activity relationships of antitubercular isoxazole-3-carboxylic acid ester derivatives

scientific article published on October 2010

Natural product leads for drug discovery: isolation, synthesis and biological evaluation of 6-cyano-5-methoxyindolo[2,3-a]carbazole based ligands as antibacterial agents ⬇️

scientific article published on 4 September 2009

New C-3′ hydroxamate-substituted and more lipophilic cyclic hydroxamate cephalosporin derivatives as a potential new generation of selective antimicrobial agents

scientific article published on 01 November 2006

New finding of an anti-TB compound in the genus Marsypopetalum (Annonaceae) from a traditional herbal remedy of Laos

scientific article

New perspectives on natural products in TB drug research

scientific article

New phenylethanoids from Buddleja cordata subsp. cordata

scientific article published in April 2000

Novel insights into the mechanism of inhibition of MmpL3, a target of multiple pharmacophores in Mycobacterium tuberculosis

scientific article

Novel thiolactone-isatin hybrids as potential antimalarial and antitubercular agents

scientific article published on 2 March 2011

Oleanane triterpenes from Junellia tridens.

scientific article

Phomapyrrolidones A-C, antitubercular alkaloids from the endophytic fungus Phoma sp. NRRL 46751. ⬇️

scientific article published on 30 September 2013

Phytoconstituents from Alpinia purpurata and their in vitro inhibitory activity against Mycobacterium tuberculosis

scientific article published on October 2010

Potential of lichen secondary metabolites against Plasmodium liver stage parasites with FAS-II as the potential target

scientific article published on 19 June 2013

Preparation of aminoglycoside-loaded chitosan nanoparticles using dextran sulphate as a counterion

scientific article published in June 2009

Purity-activity relationships of natural products: the case of anti-TB active ursolic acid

scientific article

Quality Control of Therapeutic Peptides by H NMR HiFSA Sequencing

scientific article published on 22 February 2019

Quantitative purity-activity relationships of natural products: the case of anti-tuberculosis active triterpenes from Oplopanax horridus

scientific article published on 28 January 2013

Quinoline alkaloids from Lunasia amara inhibit Mycobacterium tuberculosis H37Rv in vitro

scientific article published on 30 March 2007

Rapid determination of growth inhibition of Mycobacterium tuberculosis by GC–MS/MS quantitation of tuberculostearic acid

scientific article published on 28 February 2013

Rational design of 5-phenyl-3-isoxazolecarboxylic acid ethyl esters as growth inhibitors of Mycobacterium tuberculosis. a potent and selective series for further drug development

scientific article published in January 2010

Recent Advances in Methodologies for the Discovery of Antimycobacterial Drugs

Release of nitrite from the antitubercular nitroimidazole drug PA-824 and analogues upon one-electron reduction in protic, non-aqueous solvent

scientific article published on 4 November 2009

Residual Complexity Does Impact Organic Chemistry and Drug Discovery: The Case of Rufomyazine and Rufomycin. ⬇️

scientific article published on 24 May 2018

Role of antibiotic ligand in nascent peptide-dependent ribosome stalling

scientific article

Rufomycins or Ilamycins: Naming Clarifications and Definitive Structural Assignments

scientific article published in 2021

Ruthenium (II) phosphine/picolinate complexes as antimycobacterial agents

scientific article published on 6 November 2009

Ruthenium(II) phosphine/diimine/picolinate complexes: inorganic compounds as agents against tuberculosis

scientific article

Scaffold-switching: an exploration of 5,6-fused bicyclic heteroaromatics systems to afford antituberculosis activity akin to the imidazo[1,2-a]pyridine-3-carboxylates

scientific article

Searching for new cures for tuberculosis: design, synthesis, and biological evaluation of 2-methylbenzothiazoles

scientific article published in November 2009

Semisynthetic studies on the manzamine alkaloids

scientific article

Sesquiterpenes from Oplopanax horridus

scientific article

Strategies in anti-Mycobacterium tuberculosis drug discovery based on phenotypic screening

scientific article published on 11 July 2019

Structural Basis for Catalysis of a Tetrameric Class IIa Fructose 1,6-Bisphosphate Aldolase from Mycobacterium tuberculosis

scientific article

Structural requirements for the antitubercular quaternized triflupromazine pharmacophore

scientific article published on 06 July 2012

Structure and anti-TB activity of trachylobanes from the liverwort Jungermannia exsertifolia ssp. cordifolia

scientific article published in April 2010

Structure-activity relationship of new anti-tuberculosis agents derived from oxazoline and oxazole benzyl esters

scientific article

Structure-activity relationships for a series of quinoline-based compounds active against replicating and nonreplicating Mycobacterium tuberculosis.

scientific article

Structure-activity relationships for amide-, carbamate-, and urea-linked analogues of the tuberculosis drug (6S)-2-nitro-6-{[4-(trifluoromethoxy)benzyl]oxy}-6,7-dihydro-5H-imidazo[2,1-b][1,3]oxazine (PA-824).

scientific article published on 29 December 2011

Structure-activity relationships for analogs of the tuberculosis drug bedaquiline with the naphthalene unit replaced by bicyclic heterocycles

scientific article published on 20 February 2018

Structure-activity relationships for unit C pyridyl analogues of the tuberculosis drug bedaquiline

scientific article published on 15 February 2019

Structure-activity relationships of compounds targeting mycobacterium tuberculosis 1-deoxy-D-xylulose 5-phosphate synthase

scientific article

Structure-activity relationships of macrolides against Mycobacterium tuberculosis

scientific article published on August 2008

Structure-based design of novel benzoxazinorifamycins with potent binding affinity to wild-type and rifampin-resistant mutant Mycobacterium tuberculosis RNA polymerases

scientific article published on 5 April 2012

Succinylphosphonate esters are competitive inhibitors of MenD that show active-site discrimination between homologous alpha-ketoglutarate-decarboxylating enzymes

scientific article published in March 2010

Syntheses and Antituberculosis Activity of 1,3-Benzothiazinone Sulfoxide and Sulfone Derived from BTZ043.

scientific article

Syntheses and biological studies of novel spiropiperazinyl oxazolidinone antibacterial agents using a spirocyclic diene derived acylnitroso Diels-Alder reaction

scientific article

Syntheses and evaluation of benzodiazaborine compounds against M. tuberculosis H37Rv in vitro

scientific article published on April 1998

Syntheses and evaluation of substituted aromatic hydroxamates and hydroxamic acids that target Mycobacterium tuberculosis

scientific article published on 20 May 2015

Syntheses and studies of quinolone-cephalosporins as potential anti-tuberculosis agents

scientific article published on 30 August 2006

Syntheses of mycobactin analogs as potent and selective inhibitors of Mycobacterium tuberculosis

scientific article

Synthesis and Activity of Carbazole Derivatives Against Mycobacterium tuberculosis

scientific article published on 01 August 2006

Synthesis and Evaluation as Antitubercular Agents of 5-Arylethenyl and 5-(Hetero)aryl-3-Isoxazolecarboxylate

Synthesis and Structure−Activity Relationships of Aza- and Diazabiphenyl Analogues of the Antitubercular Drug (6S)-2-Nitro-6-{[4-(trifluoromethoxy)benzyl]oxy}-6,7-dihydro-5H-imidazo[2,1-b][1,3]oxazine (PA-824)

article

Synthesis and antimycobacterial activities of non-purine analogs of 6-aryl-9-benzylpurines: Imidazopyridines, pyrrolopyridines, benzimidazoles, and indoles

scientific article published on 20 April 2011

Synthesis and antitubercular activity of quaternized promazine and promethazine derivatives

scientific article published on 02 December 2006

Synthesis and antituberculosis activity of novel mefloquine-isoxazole carboxylic esters as prodrugs

scientific article published on 26 November 2009

Synthesis and characterization of pyruvate–isoniazid analogs and their copper complexes as potential ICL inhibitors

scientific article published on 16 March 2012

Synthesis and evaluation of analogues of the tuberculosis drug bedaquiline containing heterocyclic B-ring units.

scientific article published on 20 October 2017

Synthesis and evaluation of anti-tubercular and antibacterial activities of new 4-(2,6-dichlorobenzyloxy)phenyl thiazole, oxazole and imidazole derivatives. Part 2.

scientific article published on 12 January 2012

Synthesis and evaluation of nitrofuranylamides as novel antituberculosis agents

scientific article

Synthesis and evaluation of rifabutin analogs against Mycobacterium avium and H(37)Rv, MDR and NRP Mycobacterium tuberculosis.

scientific article

Synthesis and in vitro biological evaluation of ring B abeo-sterols as novel inhibitors of Mycobacterium tuberculosis

scientific article published on 11 September 2008

Synthesis and structure-activity relationships for extended side chain analogues of the antitubercular drug (6S)-2-nitro-6-{[4-(trifluoromethoxy)benzyl]oxy}-6,7-dihydro-5H-imidazo[2,1-b][1,3]oxazine (PA-824).

scientific article published on 27 March 2015

Synthesis and structure-activity relationships of antitubercular 2-nitroimidazooxazines bearing heterocyclic side chains

scientific article published in January 2010

Synthesis and structure-activity relationships of novel substituted 8-amino, 8-thio, and 1,8-pyrazole congeners of antitubercular rifamycin S and rifampin

scientific article

Synthesis and structure-activity relationships of varied ether linker analogues of the antitubercular drug (6S)-2-nitro-6-{[4-(trifluoromethoxy)benzyl]oxy}-6,7-dihydro-5h-imidazo[2,1-b][1,3]oxazine (PA-824).

scientific article published on September 2011

Synthesis and structure-activity studies of biphenyl analogues of the tuberculosis drug (6S)-2-nitro-6-{[4-(trifluoromethoxy)benzyl]oxy}-6,7-dihydro-5H-imidazo[2,1-b][1,3]oxazine (PA-824).

scientific article published in January 2010

Synthesis of 3-(3-aryl-pyrrolidin-1-yl)-5-aryl-1,2,4-triazines that have antibacterial activity and also inhibit inorganic pyrophosphatase

scientific article

Synthesis of non-purine analogs of 6-aryl-9-benzylpurines, and their antimycobacterial activities. Compounds modified in the imidazole ring

scientific article published on 13 August 2010

Synthesis, antimalarial and antitubercular activity of acetylenic chalcones

scientific article published on 23 December 2009

Synthesis, biological evaluation, and structure-activity relationships for 5-[(E)-2-arylethenyl]-3-isoxazolecarboxylic acid alkyl ester derivatives as valuable antitubercular chemotypes.

scientific article

Synthesis, reduction potentials, and antitubercular activity of ring A/B analogues of the bioreductive drug (6S)-2-nitro-6-{[4-(trifluoromethoxy)benzyl]oxy}-6,7-dihydro-5H-imidazo[2,1-b][1,3]oxazine (PA-824).

scientific article

Targeting mycobacterium protein tyrosine phosphatase B for antituberculosis agents

scientific article

Tetrahydroxanthene-1,3(2H)-dione derivatives from Uvaria valderramensis.

scientific article

The Mce3R Regulon Is Required for 6-Azasteroid Potentiation of Anti-TB Drug Activity

The Oxidation-sensing Regulator (MosR) Is a New Redox-dependent Transcription Factor in Mycobacterium tuberculosis

scientific article

The cyclic peptide ecumicin targeting ClpC1 is active against Mycobacterium tuberculosis in vivo

scientific article

The design, synthesis, in silico ADME profiling, antiplasmodial and antimycobacterial evaluation of new arylamino quinoline derivatives

scientific article published on 7 September 2012

Thiosemicarbazones, semicarbazones, dithiocarbazates and hydrazide/hydrazones: anti-Mycobacterium tuberculosis activity and cytotoxicity

scientific article

Trichormamides C and D, antiproliferative cyclic lipopeptides from the cultured freshwater cyanobacterium cf. Oscillatoria sp. UIC 10045. ⬇️

scientific article published on May 2015

Trypanoside, anti-tuberculosis, leishmanicidal, and cytotoxic activities of tetrahydrobenzothienopyrimidines

scientific article

UTILIZTION OF THE SUZUKI COUPLING TO ENHANCE THE ANTITUBERCULOSIS ACTIVITY OF ARYL OXAZOLES.

scientific article

Unbiased evaluation of bioactive secondary metabolites in complex matrices

scientific article

Unusual antimalarial meroditerpenes from tropical red macroalgae

scientific article

Utilization of microbial iron assimilation processes for the development of new antibiotics and inspiration for the design of new anticancer agents

scientific article published on 07 January 2009

Vaccination with Bacille-Calmette Guérin promotes mycobacterial control in guinea pig macrophages infected in vivo

scientific article published in September 2008

glpX Gene of Mycobacterium tuberculosis: Heterologous Expression, Purification, and Enzymatic Characterization of the Encoded Fructose 1,6-bisphosphatase II

article

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