List of works - Laurence Goossens

1-[4-(Methylsulfonyl)phenyl]-5-phenyl-1H-pyrazole derivatives

scientific article published on 11 August 2004

A new synthesis of pyrrolo[3,2-b]quinolines by a tandem electrocyclization–oxidation process

Antiproliferative effects of isopentenylated coumarins isolated from Phellolophium madagascariense Baker

scientific article published on August 2006

Antispasmodic and antioxidant activities of fractions and bioactive constituent davidigenin isolated from Mascarenhasia arborescens.

scientific article published on 16 May 2010

COX-2/5-LOX dual acting anti-inflammatory drugs in cancer chemotherapy.

scientific article published on January 2007

Chemotaxonomic interest of iridoids isolated from a Malagasy species: Perichlaena richardii

scientific article published in 2011

Chiral separation of new sulfonamide derivatives and evaluation of their enantioselective affinity for human carbonic anhydrase II by microscale thermophoresis and surface plasmon resonance

scientific article published on 9 January 2017

DNA Methylation Targeting: The DNMT/HMT Crosstalk Challenge

scientific article published on 05 January 2017

Discovery of orally bioavailable NK1 receptor antagonists

scientific article published in February 2003

Impact of aryloxy-linked quinazolines: a novel series of selective VEGFR-2 receptor tyrosine kinase inhibitors

scientific article published on 3 February 2011

Inhibition of tumor cell growth and angiogenesis by 7-aminoalkoxy-4-aryloxy-quinazoline ureas, a novel series of multi-tyrosine kinase inhibitors.

scientific article

New NSAIDs-NO hybrid molecules with antiproliferative properties on human prostatic cancer cell lines.

scientific article

Quinazoline derivatives as anticancer drugs: a patent review (2011 - present).

scientific article published on 24 April 2015

Quinazoline-urea, new protein kinase inhibitors in treatment of prostate cancer.

scientific article published on April 2010

Synthesis and activity of a new methoxytetrahydropyran derivative as dual cyclooxygenase-2/5-lipoxygenase inhibitor

scientific article published in March 2002

Synthesis and biological evaluation of a new family of anti-benzylanilinosulfonamides as CA IX inhibitors

scientific article

Synthesis and biological evaluation of di-aryl urea derivatives as c-Kit inhibitors.

scientific article

Synthesis and structure-activity relationships of (aryloxy)quinazoline ureas as novel, potent, and selective vascular endothelial growth factor receptor-2 inhibitors.

scientific article published on 25 January 2012

List of works by Laurence Goossens

1-[4-(Methylsulfonyl)phenyl]-5-phenyl-1H-pyrazole derivatives

A new synthesis of pyrrolo[3,2-b]quinolines by a tandem electrocyclization–oxidation process

Antiproliferative effects of isopentenylated coumarins isolated from Phellolophium madagascariense Baker

Antispasmodic and antioxidant activities of fractions and bioactive constituent davidigenin isolated from Mascarenhasia arborescens.

COX-2/5-LOX dual acting anti-inflammatory drugs in cancer chemotherapy.

Chemotaxonomic interest of iridoids isolated from a Malagasy species: Perichlaena richardii

Chiral separation of new sulfonamide derivatives and evaluation of their enantioselective affinity for human carbonic anhydrase II by microscale thermophoresis and surface plasmon resonance

DNA Methylation Targeting: The DNMT/HMT Crosstalk Challenge

Discovery of orally bioavailable NK1 receptor antagonists

Impact of aryloxy-linked quinazolines: a novel series of selective VEGFR-2 receptor tyrosine kinase inhibitors

Inhibition of tumor cell growth and angiogenesis by 7-aminoalkoxy-4-aryloxy-quinazoline ureas, a novel series of multi-tyrosine kinase inhibitors.

New NSAIDs-NO hybrid molecules with antiproliferative properties on human prostatic cancer cell lines.

Quinazoline derivatives as anticancer drugs: a patent review (2011 - present).

Quinazoline-urea, new protein kinase inhibitors in treatment of prostate cancer.

Synthesis and activity of a new methoxytetrahydropyran derivative as dual cyclooxygenase-2/5-lipoxygenase inhibitor

Synthesis and biological evaluation of a new family of anti-benzylanilinosulfonamides as CA IX inhibitors

Synthesis and biological evaluation of di-aryl urea derivatives as c-Kit inhibitors.

Synthesis and structure-activity relationships of (aryloxy)quinazoline ureas as novel, potent, and selective vascular endothelial growth factor receptor-2 inhibitors.

[4-(6,7-Disubstituted quinazolin-4-ylamino)phenyl] carbamic acid esters: a novel series of dual EGFR/VEGFR-2 tyrosine kinase inhibitors