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List of works by Markus R. Heinrich

4-Biphenylalanine- and 3-Phenyltyrosine-Derived Hydroxamic Acids as Inhibitors of the JumonjiC-Domain-Containing Histone Demethylase KDM4A.

scientific article published on 9 August 2016

4-Substituted tert-butyl phenylazocarboxylates--synthetic equivalents for the para-phenyl radical cation

scientific article published on December 2010

A convergent approach to gamma-carbonyl vinyl boronates

scientific article published on 11 May 2005

Alanine-glyoxylate aminotransferase 2 (AGXT2) polymorphisms have considerable impact on methylarginine and β-aminoisobutyrate metabolism in healthy volunteers

scientific article

Allylation and vinylation of aryl radicals generated from diazonium salts

scientific article published on 14 November 2007

Aryl Radical Selectivity in Biphasic Systems

scientific article published on 06 January 2020

Base-Induced Radical Carboamination of Nonactivated Alkenes with Aryldiazonium Salts

scientific article published on 04 December 2015

Benzyl Phenylsemicarbazides: A Chemistry-Driven Approach Leading to G Protein-Biased Dopamine D4 Receptor Agonists with High Subtype Selectivity

scientific article published on 30 October 2019

Development of Photoactivatable Allosteric Modulators for the Chemokine Receptor CXCR3.

scientific article published on 16 February 2016

Development of flavonoid-based inverse agonists of the key signaling receptor US28 of human cytomegalovirus

scientific article published on 14 June 2013

Enhancing the catalytic activity of 4-(dialkylamino)pyridines by conformational fixation

scientific article published on 01 October 2003

Fast and efficient (18) F-labeling by [(18) f]fluorophenylazocarboxylic esters

scientific article published on 11 December 2013

Fluoro-substituted phenylazocarboxamides: Dopaminergic behavior and N-arylating properties for irreversible binding

scientific article published on 17 December 2014

Generation and intermolecular capture of cyclopropylacyl radicals

scientific article published on 01 December 2004

Generation and ring opening of aziridine N-carbonyl radicals

scientific article published on 3 November 2005

Hydrogen Peroxide Promoted Mizoroki-Heck Reactions of Phenyldiazenes with Acrylates, Acrylamides, and Styrenes

scientific article published on 14 March 2016

Hydroxy- and aminophenyl radicals from arenediazonium salts

scientific article published on 14 March 2011

Identification of novel allosteric modulators for the G-protein coupled US28 receptor of human cytomegalovirus

scientific article published on 02 July 2011

In Situ Conformational Fixation of the Amide Bond Enables General Access to Medium-Sized Lactams via Ring-Closing Metathesis

scientific article published on 11 December 2018

Intermolecular Olefin Functionalisation Involving Aryl Radicals Generated from Arenediazonium Salts

article

Intermolecular radical carboaminohydroxylation of olefins with aryl diazonium salts and TEMPO

scientific article published on 17 August 2007

Intermolecular radical carbofluorination of non-activated alkenes

scientific article published on 10 October 2014

Ligand-biased and probe-dependent modulation of chemokine receptor CXCR3 signaling by negative allosteric modulators.

scientific article published on 05 February 2015

Manganese(IV)-mediated hydroperoxyarylation of alkenes with aryl hydrazines and dioxygen from air

scientific article published on 15 April 2014

Microwave-Assisted Rapid One-Pot Synthesis of Fused and Non-Fused Indoles and 5-[18 F]Fluoroindoles from Phenylazocarboxylates

scientific article

Modern Developments in Aryl Radical Chemistry

scientific article published on January 1, 2012

Nitrogen Oxides and Nitric Acid Enable the Sustainable Hydroxylation and Nitrohydroxylation of Benzenes under Visible Light Irradiation

scientific article published on 24 November 2017

Nucleophilic substitutions and radical reactions of phenylazocarboxylates

scientific article published on 18 January 2012

Oxidative Nitration of Styrenes for the Recycling of Low-Concentrated Nitrogen Dioxide in Air.

scientific article

Oxidative and reductive carbodiazenylation of nonactivated olefins

scientific article published on 01 January 2007

Oxidative radical arylation of anilines with arylhydrazines and dioxygen from air

scientific article published on 21 February 2014

Radical Arylation of Anilines and Pyrroles via Aryldiazotates

scientific article published on 25 April 2017

Radical Carbofluorination of Alkenes with Arylhydrazines and Selectfluor: Additives, Mechanistic Pathways, and Polar Effects

scientific article published on 25 January 2019

Radical arylation of phenols, phenyl ethers, and furans

scientific article published in February 2010

Radical arylation of tyrosine and its application in the synthesis of a highly selective neurotensin receptor 2 ligand

scientific article

Radical carbonitrosation and recycling of the waste gas nitrogen monoxide

scientific article

Radiosynthesis and validation of ¹⁸F-FP-CMT, a phenyltropane with superior properties for imaging the dopamine transporter in living brain.

scientific article

Reductive carbodiazenylation of nonactivated olefins via aryl diazonium salts

scientific article published on 01 July 2006

Regioselective Radical Arylation of 3-Hydroxypyridines

scientific article published on 22 June 2016

Regioselective radical arylation of anilines with arylhydrazines

scientific article published on 15 November 2012

Regiospecific Introduction of Halogens on the 2-Aminobiphenyl Subunit Leading to Highly Potent and Selective M3 Muscarinic Acetylcholine Receptor Antagonists and Weak Inverse Agonists

scientific article published on 09 April 2020

Strongly Directing Substituents in the Radical Arylation of Substituted Benzenes

scientific article published on 10 October 2016

Sustainable Synthesis of Balsalazide and Sulfasalazine Based on Diazotization with Low Concentrations of Nitrogen Dioxide in Air.

scientific article published on 5 January 2017

Switching and Conformational Fixation of Amides Through Proximate Positive Charges

scientific article published on 01 July 2015

Synthesis and application of the first radioligand targeting the allosteric binding pocket of chemokine receptor CXCR3

scientific article published on 11 June 2012

Synthesis and biological evaluation of biphenyl amides that modulate the US28 receptor

scientific article published on 21 November 2013

Synthesis and evaluation of fluoro substituted pyridinylcarboxamides and their phenylazo analogues for potential dopamine D3 receptor PET imaging.

scientific article published in December 2014

Synthesis of (S)-(+)-cericlamine through lipase-catalyzed aminolysis of azo acetates

scientific article published on 22 March 2012

Synthesis of Spirocyclohexadienones through Radical Cascade Reactions Featuring 3-Fold Carbon-Carbon Bond Formation.

scientific article

Synthesis of amino- and hydroxybiphenyls by radical chain reaction of arenediazonium salts

scientific article published on 01 January 2008

Synthesis, biological evaluation and radiolabelling by 18F-fluoroarylation of a dopamine D3-selective ligand as prospective imaging probe for PET.

scientific article published on 26 October 2010

The Gomberg-Bachmann reaction for the arylation of anilines with aryl diazotates

scientific article published on 06 August 2012

The trapping of phenyldiazenes in cycloaddition reactions

scientific article published on 25 August 2014

Thermally Induced Carbohydroxylation of Styrenes with Aryldiazonium Salts

scientific article published on 8 June 2016

Twofold carbon-carbon bond formation by intra- and intermolecular radical reactions of aryl diazonium salts

scientific article published on 13 May 2013

Visible-Light-Induced, Catalyst-Free Radical Arylations of Arenes and Heteroarenes with Aryldiazonium Salts

scientific article

Zinc-Mediated Allylation and Benzylation of Phenylazocarboxylic Esters

scientific article published on 06 October 2015

[18F]Fluorophenylazocarboxylates: Design and Synthesis of Potential Radioligands for Dopamine D3 and μ-Opioid Receptor

scientific article published on 6 December 2017