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List of works by Akihiro Sugawara

5-O-Mycaminosyltylonolide antibacterial derivatives: design, synthesis and bioactivity

scientific article published on 31 May 2017

An inducible cell-cell fusion system with integrated ability to measure the efficiency and specificity of HIV-1 entry inhibitors

scientific article

Argifin; efficient solid phase total synthesis and evaluation of analogues of acyclic peptide

scientific article

Associating HIV-1 envelope glycoprotein structures with states on the virus observed by smFRET

scientific article published on 10 April 2019

Asymmetric Total Synthesis of Indole Alkaloids Containing an Indoline Spiroaminal Framework

scientific article published on 6 July 2015

Asymmetric total synthesis of neoxaline

scientific article published on 19 August 2013

Azithromycin, a 15-membered macrolide antibiotic, inhibits influenza A(H1N1)pdm09 virus infection by interfering with virus internalization process

scientific article published on 12 July 2019

Borrelidin analogues with antimalarial activity: design, synthesis and biological evaluation against Plasmodium falciparum parasites

scientific article published on 26 February 2013

Cinatrins D and E, and virgaricin B, three novel compounds produced by a fungus, Virgaria boninensis FKI-4958. ⬇️

scientific article

Computational analysis of the binding affinities of the natural-product cyclopentapeptides argifin and argadin to chitinase B from Serratia marcescens

scientific article published on 8 February 2008

Computer-aided rational molecular design of argifin-derivatives with increased inhibitory activity against chitinase B from Serratia marcescens.

scientific article published on 9 April 2009

Creation of Customized Bioactivity within a 14-Membered Macrolide Scaffold: Design, Synthesis, and Biological Evaluation Using a Family-18 Chitinase

scientific article

Crystal Structures of HIV-1 gp120 Envelope Glycoprotein in Complex with NBD Analogues That Target the CD4-Binding Site

scientific article

Design and synthesis via click chemistry of 8,9-anhydroerythromycin A 6,9-hemiketal analogues with anti-MRSA and -VRE activity

scientific article

Design, synthesis and biological evaluation of small molecule inhibitors of CD4-gp120 binding based on virtual screening

scientific article

Human acidic mammalian chitinase as a novel target for anti-asthma drug design using in silico screening

scientific article published in April 2013

Jietacins, azoxy antibiotics with potent nematocidal activity: Design, synthesis, and biological evaluation against parasitic nematodes

scientific article published on 28 December 2017

Jietacins, azoxy natural products, as novel NF-κB inhibitors: Discovery, synthesis, biological activity, and mode of action

scientific article published on 29 May 2019

Leucomycin A3, a 16-membered macrolide antibiotic, inhibits influenza A virus infection and disease progression.

scientific article published on 5 February 2014

Macrolides Promote CCL2-Mediated Macrophage Recruitment and Clearance of Nasopharyngeal Pneumococcal Colonization in Mice

scientific article published on 12 March 2015

Macrolides sensitize EGFR-TKI-induced non-apoptotic cell death via blocking autophagy flux in pancreatic cancer cell lines.

scientific article published on 9 November 2015

Macrolides with promotive activity of monocyte to macrophage differentiation

scientific article published in January 2005

Molecular modeling of human acidic mammalian chitinase in complex with the natural-product cyclopentapeptide chitinase inhibitor argifin

scientific article published on 25 July 2009

NMR spectroscopy and computational analysis of interaction between Serratia marcescens chitinase B and a dipeptide derived from natural-product cyclopentapeptide chitinase inhibitor argifin ⬇️

scientific article published on August 15, 2010

Non-antibiotic 12-membered macrolides: design, synthesis and biological evaluation in a cigarette-smoking model

scientific article published on 30 September 2015

Novel 12-membered non-antibiotic macrolides from erythromycin A; EM900 series as novel leads for anti-inflammatory and/or immunomodulatory agents

scientific article published on 07 April 2011

Novel 12-membered non-antibiotic macrolides, EM900 series with anti-inflammatory and/or immunomodulatory activity; synthesis, structure-activity relationships and in vivo study

scientific article

Solid-phase total synthesis of the chitinase inhibitor Argadin using a supported acetal resin.

scientific article published on 3 July 2009

Three-Dimensional Solution Structure of Bottromycin A2: A Potent Antibiotic Active against Methicillin-Resistant Staphylococcus aureus and Vancomycin-Resistant Enterococci ⬇️

scientific article published on January 1, 2012

Three-dimensional solution structure of EM703 with potent promoting activity of monocyte-to-macrophage differentiation

scientific article published on 09 February 2006

Total syntheses of the AChE inhibitors (-)-arisugacins F and G

scientific article published on 01 August 2003

Toward the total synthesis of luminamicin; an anaerobic antibiotic: construction of highly functionalized cis-decalin containing a bridged ether moiety

scientific article published on 5 July 2017

Two New Terpenes Isolated from Dictyostelium Cellular Slime Molds

scientific article published on 23 June 2020

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