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List of works by Balázs Volk

(Phenylpiperazinyl-butyl)oxindoles as selective 5-HT7 receptor antagonists

scientific article

5-HT6/7 receptor antagonists facilitate dopamine release in the cochlea via a GABAergic disinhibitory mechanism.

scientific article

A novel GABA(A) alpha 5 receptor inhibitor with therapeutic potential

scientific article published on 10 July 2015

A novel tool for structure assignment of hydroxylated metabolites of (arylpiperazinylbutyl)oxindole derivatives based on relative HPLC retention times

scientific article published on 11 March 2019

Application of the systems chemistry approach on the ammonolysis of 1-ethoxycarbonyl- and 1-phenoxycarbonyl-3-(2-thienyl)oxindoles. A method to predict reactivity

scientific article published on 27 August 2012

Basicity-Tuned Reactivity: <i>diaza</i>-[1,2]-Wittig versus <i>diaza</i>-[1,3]-Wittig Rearrangements of 3,4-Dihydro-2<i>H</i>-1,2,3-benzothiadiazine 1,1-Dioxides

scientific article published on 31 December 2020

Cytochrome P450 catalyzed nitric oxide synthesis: a theoretical study

scientific article published on 01 February 2000

Development and Evaluation of Two Potential 5-HT7 Receptor PET Tracers: [18F]ENL09 and [18F]ENL10

scientific article published on 22 April 2019

Evaluation of 3-Ethyl-3-(phenylpiperazinylbutyl)oxindoles as PET Ligands for the Serotonin 5-HT₇ Receptor: Synthesis, Pharmacology, Radiolabeling, and in Vivo Brain Imaging in Pigs

scientific article published on 13 April 2015

First total synthesis of β-carboline alkaloid trigonostemine G and its derivatives

scientific article published on 29 May 2019

Interactions of non-charged tadalafil stereoisomers with cyclodextrins: capillary electrophoresis and nuclear magnetic resonance studies

scientific article published on 19 August 2014

Literature Survey and Further Studies on the 3-Alkylation of N-Unprotected 3-Monosubstituted Oxindoles. Practical Synthesis of N-Unprotected 3,3-Disubstituted Oxindoles and Subsequent Transformations on the Aromatic Ring.

scientific article published on 26 December 2016

Medicinal chemistry of 5-HT5A receptor ligands: a receptor subtype with unique therapeutical potential.

scientific article published on January 2010

Optimization of (arylpiperazinylbutyl)oxindoles exhibiting selective 5-HT₇ receptor antagonist activity.

scientific article published on 16 September 2011

Rearrangement of o-(pivaloylaminomethyl)benzaldehydes: an experimental and computational study

scientific article published on 13 July 2020

Study on the Alkylation Reactions of N(7)-Unsubstituted 1,3-Diazaoxindoles.

scientific article published on 19 May 2017

Synthesis and Biochemical Evaluation of Lid-Open D-Amino Acid Oxidase Inhibitors

scientific article published on 14 January 2019

Synthesis and in vitro evaluation of oxindole derivatives as potential radioligands for 5-HT(7) receptor imaging with PET.

scientific article published on 31 August 2012

Synthesis of 8-Fluoro-3,4-dihydroisoquinoline and Its Transformation to 1,8-Disubstituted Tetrahydroisoquinolines

scientific article published on 26 May 2018

Synthesis of Indolo[2,3-<i>c</i>]quinolin-6(7<i>H</i>)-ones and Antimalarial Isoneocryptolepine. Computational Study on the Pd-Catalyzed Intramolecular C-H Arylation

scientific article published on 30 November 2020

Synthesis of new tricyclic imidazotriazepine derivatives condensed with various heterocycles.

scientific article published on 19 July 2017

The medicinal chemistry of serotonin receptor modulators

scientific article published in January 2010

Thermal Ring Contraction Reactions of 9-Aryl-5H,7H-[1,2,5]thiadiazolo[3,4-h][2,3,4]benzothiadiazepine 6,6-Dioxides. Experimental and Computational Studies for Understanding the Course of the Transformations.

scientific article published on 17 January 2017