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List of works by Saeed Emami

(E)- and (Z)-1,2,4-triazolylchromanone oxime ethers as conformationally constrained antifungals

scientific article published in August 2004

1,2,3-Triazole-based kojic acid analogs as potent tyrosinase inhibitors: Design, synthesis and biological evaluation

scientific article published on 31 October 2018

1,2-Diaryl-2-hydroxyiminoethanones as dual COX-1 and β-amyloid aggregation inhibitors: biological evaluation and in silico study

scientific article published on 11 October 2014

1-[(2-arylthiazol-4-yl)methyl]azoles as a new class of anticonvulsants: design, synthesis, in vivo screening, and in silico drug-like properties.

scientific article published on 15 September 2011

2-Amino-4-(nitroalkyl)-4H-chromene-3-carbonitriles as New Cytotoxic Agents

scientific article published on January 2013

2-Hydroxyphenacyl azoles and related azolium derivatives as antifungal agents

scientific article published on 4 November 2007

2-Substituted-5-nitroheterocycles: in vitro anti-Helicobacter pylori activity and structure-activity relationship study

scientific article published in November 2009

2H-chromene derivatives bearing thiazolidine-2,4-dione, rhodanine or hydantoin moieties as potential anticancer agents.

scientific article published on 2 November 2012

3-imidazolyl-substituted flavans as potential antifungal agents: synthesis, stereochemical properties, and antifungal activity.

scientific article published in September 2009

5,7-Dihydroxychromone-2-carboxylic acid and it's transition-metal (Mn and Zn) chelates as non-thiol radioprotective agents

scientific article published on 17 May 2007

5-Nitroimidazole-based 1,3,4-thiadiazoles: heterocyclic analogs of metronidazole as anti-Helicobacter pylori agents

scientific article published on 22 December 2010

9H-Carbazole Derivatives Containing the N-Benzyl-1,2,3-triazole Moiety as New Acetylcholinesterase Inhibitors.

scientific article

A new boronic acid fluorescent sensor based on fluorene for monosaccharides at physiological pH

scientific article published on 25 February 2015

Acetophenone benzoylhydrazones as antioxidant agents: Synthesis, in vitro evaluation and structure-activity relationship studies

scientific article published on 19 June 2018

An overview of azoles targeting sterol 14α-demethylase for antileishmanial therapy

scientific article

Anticonvulsant and antiepileptogenic effects of azolylchromanones on lithium-pilocarpine induced seizures and pentylenetetrazole-kindling model of epilepsy

scientific article published on 28 December 2007

Antinociceptive properties of new coumarin derivatives bearing substituted 3,4-dihydro-2H-benzothiazines.

scientific article

Antituberculosis agents. V. Synthesis, evaluation of in vitro antituberculosis activity and cytotoxicity of some 2-(5-nitro-2-furyl)-1,3,4-thiadiazole derivatives

scientific article published on September 2002

Asymmetrical 2,6-bis(benzylidene)cyclohexanones: Synthesis, cytotoxic activity and QSAR study

scientific article published on 28 January 2012

Azolylchromans as a novel scaffold for anticonvulsant activity

scientific article published on 24 January 2006

Benzofuran-derived benzylpyridinium bromides as potent acetylcholinesterase inhibitors.

scientific article

Chromene-based synthetic chalcones as potent antileishmanial agents: synthesis and biological activity

scientific article published on 10 March 2010

Complexes of 2-hydroxyacetophenone semicarbazones: A novel series of superoxide dismutase mimetics

scientific article published in April 2010

Conformationally constrained analogs of N-substituted piperazinylquinolones: synthesis and antibacterial activity of N-(2,3-dihydro-4-hydroxyimino-4H-1-benzopyran-3-yl)-piperazinylquinolones

scientific article published on July 2009

Coumarin-based bioactive compounds: facile synthesis and biological evaluation of coumarin-fused 1,4-thiazepines.

scientific article published on 29 August 2011

Current developments of coumarin-based anti-cancer agents in medicinal chemistry.

scientific article published on 17 August 2015

Cytotoxic Activity and DNA Binding Property of New Aminopyrimidine Derivatives

scholarly article

Cytotoxic activity evaluation and QSAR study of chromene-based chalcones.

scientific article

Design of conformationally constrained azole antifungals: efficient synthesis and antifungal activity of trans-3-imidazolylflavanones

scientific article published in April 2009

Design, synthesis and anticholinesterase activity of novel benzylidenechroman-4-ones bearing cyclic amine side chain

scientific article published on 29 April 2015

Design, synthesis and biological evaluation of flexible and rigid analogs of 4H-1,2,4-triazoles bearing 3,4,5-trimethoxyphenyl moiety as new antiproliferative agents

scientific article published on 21 September 2019

Design, synthesis and evaluation of novel multi-target-directed ligands for treatment of Alzheimer's disease based on coumarin and lipoic acid scaffolds

scientific article published on 02 May 2018

Design, synthesis and in vitro study of 5,6-diaryl-1,2,4-triazine-3-ylthioacetate derivatives as COX-2 and β-amyloid aggregation inhibitors.

scientific article published on 18 February 2015

Design, synthesis, biological evaluation and docking study of 5-oxo-4,5-dihydropyrano[3,2-c]chromene derivatives as acetylcholinesterase and butyrylcholinesterase inhibitors

scientific article published on 11 August 2013

Design, synthesis, in vivo and in silico evaluation of phenacyl triazole hydrazones as new anticonvulsant agents

scientific article published on 7 March 2018

Design, synthesis, pharmacological evaluation, and docking study of new acridone-based 1,2,4-oxadiazoles as potential anticonvulsant agents.

scientific article published in February 2016

Discovery of benzylthio analogs of fluconazole as potent antifungal agents.

scientific article published on 23 April 2018

Down-regulation of peroxin synthesis by silencing RNA (siRNA): A novel hypothesis for treatment of leishmaniasis

scientific article published in July 2016

Experimental Study on the Reduction of Loratadine Particle Size through Confined Liquid Impinging Jets

scientific article published on 20 July 2020

Facile synthesis and antiproliferative activity of 7H-benzo[7,8]chromeno[2,3-d]pyrimidin-8-amines.

scientific article published on 21 December 2016

Functionalized N(2-oxyiminoethyl) piperazinyl quinolones as new cytotoxic agents

scientific article published on January 2007

Halogenated flavanones as potential apoptosis-inducing agents: synthesis and biological activity evaluation

scientific article published on 02 November 2012

Hypothesis: The potential application of doxorubicin against cutaneous leishmaniasis

scientific article published on January 2015

Imidazo[2,1-b]thiazole derivatives as new inhibitors of 15-lipoxygenase.

scientific article

Imidazolylchromanone oxime ethers as potential anticonvulsant agents: Anticonvulsive evaluation in PTZ-kindling model of epilepsy and SAR study

scientific article published on 10 December 2010

Imidazolylchromanones containing alkyl side chain as lanosterol 14α-demethylase inhibitors: synthesis, antifungal activity and docking study.

scientific article published on 14 March 2013

Imidazolylchromanones containing non-benzylic oxime ethers: synthesis and molecular modeling study of new azole antifungals selective against Cryptococcus gattii

scientific article published on 11 February 2014

In Vitro Activities of Novel Azole Compounds ATTAF-1 and ATTAF-2 against Fluconazole-Susceptible and -Resistant Isolates of Candida Species.

scientific article published on 24 October 2016

In vitro and in vivo evaluation of kojic acid against Toxoplasma gondii in experimental models of acute toxoplasmosis

scientific article published on 20 March 2019

In vitro antileishmanial activity of novel azoles (3-imidazolylflavanones) against promastigote and amastigote stages of Leishmania major

scientific article published on 22 December 2016

Indole in the target-based design of anticancer agents: A versatile scaffold with diverse mechanisms.

scientific article published on 24 February 2018

Indole-derived chalcones as anti-dermatophyte agents: In vitro evaluation and in silico study

scientific article published on 23 December 2019

Indolinone-based acetylcholinesterase inhibitors: synthesis, biological activity and molecular modeling.

scientific article

Induction of apoptosis through tubulin inhibition in human cancer cells by new chromene-based chalcones

scientific article

Isochaihulactone analogues: synthesis and anti-proliferative activity of novel dibenzylbutyrolactones.

scientific article published on 7 October 2010

Kojic acid and its manganese and zinc complexes as potential radioprotective agents

scientific article published on 04 October 2006

Kojic acid-natural product conjugates as mushroom tyrosinase inhibitors

scientific article published on 16 June 2020

Management of multi-drug resistant Helicobacter pylori infection by supplementary, complementary and alternative medicine; a review.

scientific article

Mannich bases of 7-piperazinylquinolones and kojic acid derivatives: synthesis, in vitro antibacterial activity and in silico study.

scientific article published on 11 August 2013

Modification of 7-piperazinylquinolone antibacterials to promising anticancer lead compounds: Synthesis and in vitro studies

scientific article published on 15 December 2019

Molecular Modeling and Structural Stability of Wild-Type and Mutant CYP51 from Leishmania major: In Vitro and In Silico Analysis of a Laboratory Strain.

scientific article published on 19 March 2018

Multi-structure docking analysis of BACE1 crystal structures and non-peptidic ligands

scientific article published on 28 June 2017

N-(2-(Piperazin-1-yl)phenyl)arylamide Derivatives as β-Secretase (BACE1) Inhibitors: Simple Synthesis by Ugi Four-Component Reaction and Biological Evaluation

scientific article published on 19 March 2015

N-Substituted piperazinyl quinolones as potential cytotoxic agents: structure-activity relationships study

scientific article

New 5-(nitroheteroaryl)-1,3,4-thiadiazols containing acyclic amines at C-2: synthesis and SAR study for their antileishmanial activity

scientific article published on 31 May 2012

New 7-piperazinylquinolones containing (benzo[d]imidazol-2-yl)methyl moiety as potent antibacterial agents

scientific article published on 07 June 2018

New indole-based chalconoids as tubulin-targeting antiproliferative agents.

scientific article published on 7 September 2017

New potent antifungal triazole alcohols containing N-benzylpiperazine carbodithioate moiety: Synthesis, in vitro evaluation and in silico study

scientific article published on 12 June 2019

New racemic annulated pyrazolo[1,2-b]phthalazines as tacrine-like AChE inhibitors with potential use in Alzheimer's disease

scientific article

New tacrine-derived AChE/BuChE inhibitors: Synthesis and biological evaluation of 5-amino-2-phenyl-4H-pyrano[2,3-b]quinoline-3-carboxylates.

scientific article

New tetracyclic tacrine analogs containing pyrano[2,3-c]pyrazole: efficient synthesis, biological assessment and docking simulation study

scientific article published on 18 October 2014

New thiazole-2(3H)-thiones containing 4-(3,4,5-trimethoxyphenyl) moiety as anticancer agents

scientific article published on 15 October 2019

Nitroimidazolyl-1,3,4-thiadiazole-based anti-leishmanial agents: synthesis and in vitro biological evaluation

scientific article published on 9 April 2008

Novel 3-phenylcoumarin-lipoic acid conjugates as multi-functional agents for potential treatment of Alzheimer's disease

scientific article published on 02 May 2018

Novel Tc-2-arylimidazo[2,1-b]benzothiazole derivatives as SPECT imaging agents for amyloid-β plaques

scientific article published on 29 April 2019

Novel antileishmanial chalconoids: synthesis and biological activity of 1- or 3-(6-chloro-2H-chromen-3-yl)propen-1-ones.

scientific article published on 28 December 2009

Novel coumarin-3-carboxamides bearing N-benzylpiperidine moiety as potent acetylcholinesterase inhibitors.

scientific article

Novel triazole alcohol antifungals derived from fluconazole: design, synthesis, and biological activity

scientific article published on 03 September 2014

One-pot, four-component synthesis of novel cytotoxic agents 1-(5-aryl-1,3,4-oxadiazol-2-yl)-1-(1H-pyrrol-2-yl)methanamines

scientific article published on 16 March 2014

Phthalimide-Derived N-Benzylpyridinium Halides Targeting Cholinesterases: Synthesis and Bioactivity of New Potential Anti-Alzheimer's Disease Agents.

scientific article published on 22 February 2016

Polyoxygenated cinnamoylcoumarins as conformationally constrained analogs of cytotoxic diarylpentanoids: synthesis and biological activity.

scientific article published on 8 August 2013

Promising antileishmanial activity of novel imidazole antifungal drug luliconazole against Leishmania major: In vitro and in silico studies

scientific article published on 21 May 2018

Promising antileishmanial effectiveness of doxorubicin and Doxil against Leishmania major: An in vitro assay

scientific article

Quinoline-based imidazole-fused heterocycles as new inhibitors of 15-lipoxygenase.

scientific article published on 17 July 2016

Radioprotective effects of kojic acid against mortality induced by gamma irradiation in mice.

scientific article

Recent advances of chroman-4-one derivatives: synthetic approaches and bioactivities

scientific article

Recent advances of cytotoxic chalconoids targeting tubulin polymerization: Synthesis and biological activity.

scientific article published on June 2016

Recent applications of 1,3-thiazole core structure in the identification of new lead compounds and drug discovery

scientific article published on 13 April 2015

Replacement of the methylene of dihydrochalcones with oxygen: synthesis and biological evaluation of 2-phenoxyacetophenones

scientific article published on 13 July 2012

Repurposing azole antifungals into antileishmanials: Novel 3-triazolylflavanones with promising in vitro antileishmanial activity against Leishmania major

scientific article published on 21 December 2018

Selective hydrogenation of 4-carboxybenzaldehyde over palladium catalysts supported with different structural organization

Selective leishmanicidal effect of 1,3,4-thiadiazole derivatives and possible mechanism of action against Leishmania species

scientific article published on 16 December 2008

Stereoselective synthesis and antifungal activity of (Z)-trans-3-azolyl-2-methylchromanone oxime ethers

scientific article published in November 2004

Stereoselective synthesis and in vitro antifungal evaluation of (E)- and (Z)-imidazolylchromanone oxime ethers

scientific article

Stereospecific deuteration of alpha-furanosyl azomycin nucleosides: a model reaction for tritium radiolabeling

scientific article published on 25 April 2008

Straightforward synthesis of thiazoline-incorporated chalconoids from phenacyl halides

scientific article

Structural features of new quinolones and relationship to antibacterial activity against Gram-positive bacteria

scientific article

Structure-activity relationship study of a series of N-substituted piperazinyl-fluoroquinolones as anti-Helicobacter pylori agents

scientific article

Synthesis and Evaluation of 2(3H)-Thiazole Thiones as Tyrosinase Inhibitors

article published in 2012

Synthesis and anti-Helicobacter pylori activity of 5-(nitroaryl)-1,3,4-thiadiazoles with certain sulfur containing alkyl side chain

scientific article published on 15 April 2008

Synthesis and anti-cancer activity evaluation of new dimethoxylated chalcone and flavanone analogs

scientific article published on 08 September 2014

Synthesis and anti-cholinesterase activity of new 7-hydroxycoumarin derivatives

scientific article published on 24 May 2014

Synthesis and anti-leishmanial activity of 5-(5-nitrofuran-2-yl)-1,3,4-thiadiazol-2-amines containing N-[(1-benzyl-1H-1,2,3-triazol-4-yl)methyl] moieties

scientific article published on 30 January 2012

Synthesis and antibacterial activity of N-(5-benzylthio-1,3,4-thiadiazol-2-yl) and N-(5-benzylsulfonyl-1,3,4-thiadiazol-2-yl)piperazinyl quinolone derivatives

scientific article published in October 2005

Synthesis and antibacterial activity of N-[2-(5-bromothiophen-2-yl)-2-oxoethyl] and N-[(2-5-bromothiophen-2-yl)-2-oximinoethyl] derivatives of piperazinyl quinolones.

scientific article published in October 2005

Synthesis and antibacterial activity of N-[2-[5-(methylthio)thiophen-2-yl]-2-oxoethyl] and N-[2-[5-(methylthio)thiophen-2-yl]-2-(oxyimino)ethyl]piperazinylquinolone derivatives.

scientific article published on 19 January 2006

Synthesis and antibacterial activity of N-[5-(chlorobenzylthio)-1,3,4-thiadiazol-2-yl] piperazinyl quinolone derivatives

scientific article published on 01 February 2007

Synthesis and antibacterial activity of levofloxacin derivatives with certain bulky residues on piperazine ring

scientific article published on 14 January 2007

Synthesis and antibacterial activity of new 7-piperazinyl-quinolones containing a functionalized 2-(furan-3-yl)ethyl moiety

scientific article published on 01 January 2007

Synthesis and antibacterial activity of new N-[2-(thiophen-3-yl)ethyl] piperazinyl quinolones

scientific article published on 01 June 2007

Synthesis and antibacterial activity of new fluoroquinolones containing a substituted N-(phenethyl)piperazine moiety

scientific article published on 27 April 2006

Synthesis and antibacterial activity of nitroaryl thiadiazole-gatifloxacin hybrids.

scientific article published on 19 September 2008

Synthesis and antibacterial activity of nitroaryl thiadiazole-levofloxacin hybrids

scientific article published on 01 November 2006

Synthesis and antibacterial activity of novel levofloxacin derivatives containing a substituted thienylethyl moiety

scientific article published on 30 August 2012

Synthesis and antibacterial activity of quinolone-based compounds containing a coumarin moiety

scientific article published in January 2008

Synthesis and anticancer activity of N-substituted 2-arylquinazolinones bearing trans-stilbene scaffold

scientific article published on 26 March 2015

Synthesis and anticholinergic activity of 4-hydroxycoumarin derivatives containing substituted benzyl-1,2,3-triazole moiety.

scientific article published on 20 July 2015

Synthesis and anticholinesterase activity of coumarin-3-carboxamides bearing tryptamine moiety.

scientific article

Synthesis and antifungal activity of 1-[(2-benzyloxy)phenyl]-2-(azol-1-yl)ethanone derivatives: exploring the scaffold flexibility

scientific article published on 28 October 2011

Synthesis and antileishmanial activity of 5-(5-nitroaryl)-2-substituted-thio-1,3,4-thiadiazoles

scientific article published on 28 June 2010

Synthesis and antileishmanial activity of novel 5-(5-nitrofuran-2-y1)-1,3,4-thiadiazoles with piperazinyl-linked benzamidine substituents

scientific article published on 31 March 2011

Synthesis and antioxidant properties of substituted 3-benzylidene-7-alkoxychroman-4-ones

scientific article published on 17 October 2007

Synthesis and biological assessment of ciprofloxacin-derived 1,3,4-thiadiazoles as anticancer agents

scientific article published on 15 October 2020

Synthesis and biological evaluation of 2-phenylthiazole-4-carboxamide derivatives as anticancer agents

scientific article published on 16 September 2010

Synthesis and biological evaluation of 3-(trimethoxyphenyl)-2(3H)-thiazole thiones as combretastatin analogs.

scientific article published on 25 October 2013

Synthesis and biological evaluation of 4-amino-5-cinnamoylthiazoles as chalcone-like anticancer agents.

scientific article published on 6 January 2018

Synthesis and biological evaluation of 5-benzylidenerhodanine-3-acetic acid derivatives as AChE and 15-LOX inhibitors

scientific article published on 22 June 2015

Synthesis and biological evaluation of fluconazole analogs with triazole-modified scaffold as potent antifungal agents

scientific article published on 16 February 2015

Synthesis and biological evaluation of new N-benzylpyridinium-based benzoheterocycles as potential anti-Alzheimer's agents

scientific article published on 13 November 2018

Synthesis and biological evaluation of new coumarins bearing 2,4-diaminothiazole-5-carbonyl moiety

scientific article published on 07 June 2018

Synthesis and biological evaluation of novel imidazopyrimidin-3-amines as anticancer agents

scientific article published on 8 November 2016

Synthesis and biological evaluation of quinazolinone-based hydrazones with potential use in Alzheimer's disease

scientific article published on 25 July 2017

Synthesis and cytotoxic activity of novel poly-substituted imidazo[2,1-c][1,2,4]triazin-6-amines

scientific article

Synthesis and cytotoxic properties of novel (E)-3-benzylidene-7-methoxychroman-4-one derivatives.

scientific article published on 12 April 2013

Synthesis and evaluation of 4-substituted coumarins as novel acetylcholinesterase inhibitors

scientific article published on 18 March 2013

Synthesis and free radical scavenging activity of coumarin derivatives containing a 2-methylbenzothiazoline motif

scientific article published on 25 August 2011

Synthesis and hypoxia selective radiosensitization potential of beta-2-FAZA and beta-3-FAZL: fluorinated azomycin beta-nucleosides

scientific article published in March 2009

Synthesis and in vitro anti-Helicobacter pylori activity of N-[5-(5-nitro-2-heteroaryl)-1,3,4-thiadiazol-2-yl]thiomorpholines and related compounds

scientific article

Synthesis and in vitro anti-Toxoplasma gondii activity of a new series of aryloxyacetophenone thiosemicarbazones

scientific article published on 20 August 2019

Synthesis and in vitro anti-leishmanial activity of 1-[5-(5-nitrofuran-2-yl)-1,3,4-thiadiazol-2-yl]- and 1-[5-(5-nitrothiophen-2-yl)-1,3,4-thiadiazol-2-yl]-4-aroylpiperazines

scientific article published on 20 February 2008

Synthesis and in vitro cytotoxic activity of novel chalcone-like agents

scientific article

Synthesis and in vitro leishmanicidal activity of 2-(1-methyl-5-nitro-1H-imidazol-2-yl)-5-substituted-1,3,4-thiadiazole derivatives

scientific article published on 10 August 2005

Synthesis and in-vitro antibacterial activity of 5-substituted 1-methyl-4-nitro-1H-imidazoles.

scientific article published in August 2008

Synthesis and in-vitro cytotoxicity of poly-functionalized 4-(2-arylthiazol-4-yl)-4H-chromenes.

scientific article published on July 2010

Synthesis and structure-activity relationship study of benzofuran-based chalconoids bearing benzylpyridinium moiety as potent acetylcholinesterase inhibitors.

scientific article

Synthesis and structure-activity relationship study of tacrine-based pyrano[2,3-c]pyrazoles targeting AChE/BuChE and 15-LOX.

scientific article published on 21 July 2016

Synthesis of 4‐Hydroxycoumarin‐Based Triazoles/Oxadiazoles as Novel Anticancer Agents

scientific article published in 2022

Synthesis, biological evaluation and docking study of 3-aroyl-1-(4-sulfamoylphenyl)thiourea derivatives as 15-lipoxygenase inhibitors

scientific article published on 24 May 2014

Synthesis, computational study and cytotoxicity of 4-hydroxycoumarin-derived imines/enamines

scientific article published on 22 April 2020

Synthesis, in vitro antifungal activity and in silico study of 3-(1,2,4-triazol-1-yl)flavanones.

scientific article

Synthesis, in vitro antifungal evaluation and in silico study of 3-azolyl-4-chromanone phenylhydrazones.

scientific article published on 4 October 2012

Synthesis, in vitro cytotoxicity and apoptosis inducing study of 2-aryl-3-nitro-2H-chromene derivatives as potent anti-breast cancer agents

scientific article published on 6 September 2014

The effects of plant cover on population of pear psylla (Cacopsylla pyricola) and its predators

scientific article published in 2017

The importance of triazole scaffold in the development of anticonvulsant agents

scientific article published on 11 January 2016

Tropolone alkaloids from Colchicum kurdicum (Bornm.) Stef. (Colchicaceae) as the potent novel antileishmanial compounds; purification, structure elucidation, antileishmanial activities and molecular docking studies

scientific article published on 27 April 2020

Ultrastructural Investigation of Leishmania major Promastigotes Treated with A New Potent Antileishmanial Azole Using Scanning Electron and Atomic Force Microscopes

scientific article published on 01 January 2018

Utility of aptamers for antileishmanial drug targets: A potential hypothesis

scientific article published on January 2017

β-Ionone and its analogs as promising anticancer agents

scientific article published on 20 July 2016

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