List of works - Thomas L. Mindt

"Click-to-chelate": design and incorporation of triazole-containing metal-chelating systems into biomolecules of diagnostic and therapeutic interest

scientific article published in January 2008

"Click-to-chelate": in vitro and in vivo comparison of a 99mTc(CO)3-labeled N(tau)-histidine folate derivative with its isostructural, clicked 1,2,3-triazole analogue

scientific article

1,2,3-Triazole Stabilized Neurotensin-Based Radiopeptidomimetics for Improved Tumor Targeting.

scientific article published on 8 September 2015

1,2,3-Triazoles as amide bond mimics: triazole scan yields protease-resistant peptidomimetics for tumor targeting

scientific article published on 5 July 2013

1,2,3-Triazoles as amide-bond surrogates in peptidomimetics.

scientific article published on January 2013

A "click chemistry" approach to the efficient synthesis of multiple imaging probes derived from a single precursor

scientific article published on 5 October 2009

A bombesin-shepherdin radioconjugate designed for combined extra- and intracellular targeting

scientific article published on 27 May 2014

A click approach to structurally diverse conjugates containing a central di-1,2,3-triazole metal chelate

scientific article

A solid phase-assisted approach for the facile synthesis of a highly water-soluble zirconium-89 chelator for radiopharmaceutical development.

scientific article

An octadentate bifunctional chelating agent for the development of stable zirconium-89 based molecular imaging probes

scientific article published on October 2014

Click-to-Chelate: development of technetium and rhenium-tricarbonyl labeled radiopharmaceuticals

scientific article published on 12 March 2013

Comparison of the octadentate bifunctional chelator DFO*-pPhe-NCS and the clinically used hexadentate bifunctional chelator DFO-pPhe-NCS for 89Zr-immuno-PET

scientific article published on 30 August 2016

Convergent Synthesis of 2H-Chromenes - a Formal [3+3] Cycloaddition by a One-pot, Three-Step Cascade.

scientific article published on December 2011

Cu(I)-catalyzed intramolecular cyclization of alkynoic acids in aqueous media: a "click side reaction".

scientific article published on 29 November 2007

Development of 68Ga- and 89Zr-Labeled Exendin-4 as Potential Radiotracers for the Imaging of Insulinomas by PET

article

Dual-targeting conjugates designed to improve the efficacy of radiolabeled peptides

scientific article published on 16 August 2012

EANM guideline for the preparation of an Investigational Medicinal Product Dossier (IMPD)

scientific article published on 01 November 2014

Effect of amino acid infusion on potassium serum levels in neuroendocrine tumour patients treated with targeted radiopeptide therapy

scientific article published on 07 May 2011

Electrocyclic Ring Closure of the Enols of Vinyl Quinones. A2H-Chromene Synthesis

scientific article published on 01 November 2001

Evaluation of a novel radiofolate in tumour-bearing mice: promising prospects for folate-based radionuclide therapy

scientific article

Expression of different neurokinin-1 receptor (NK1R) isoforms in glioblastoma multiforme: potential implications for targeted therapy

scientific article published on 19 February 2014

Fluorescent gallium and indium bis(thiosemicarbazonates) and their radiolabelled analogues: synthesis, structures and cellular confocal fluorescence imaging investigations.

scientific article published on 19 May 2011

Fluorine-18 click radiosynthesis and preclinical evaluation of a new 18F-labeled folic acid derivative

scientific article published in December 2008

Glycated 99m Tc-Tricarbonyl-Labeled Peptide Conjugates for Tumor Targeting by "Click-to-Chelate".

scientific article published on 30 November 2016

Guidance on current good radiopharmacy practice for the small-scale preparation of radiopharmaceuticals using automated modules: a European perspective

scientific article published on 01 August 2014

Heterocycle Annulation of Enolizable Vinyl Quinone Imides. Dihydroquinolines and Quinolines from Thermal 6π-Electrocyclizations and Indoles from Photochemical Cyclizations

scientific article published on 01 November 2002

Imaging of activated macrophages in experimental osteoarthritis using folate-targeted animal single-photon-emission computed tomography/computed tomography

scientific article published on 01 July 2011

Manganese in PET imaging: Opportunities and challenges

scientific article published on 01 June 2019

Metal chelating systems synthesized using the copper(I) catalyzed azide-alkyne cycloaddition.

scientific article

Methoxinine - an alternative stable amino acid substitute for oxidation-sensitive methionine in radiolabelled peptide conjugates

scientific article published on 5 January 2017

Modification of different IgG1 antibodies via glutamine and lysine using bacterial and human tissue transglutaminase

scientific article

Molecular assembly of multifunctional ⁹⁹(m)Tc radiopharmaceuticals using "clickable" amino acid derivatives.

scientific article published on December 2010

Novel chemoselective (18)F-radiolabeling of thiol-containing biomolecules under mild aqueous conditions.

scientific article published on 4 April 2016

Position paper on requirements for toxicological studies in the specific case of radiopharmaceuticals

article

Probing the Backbone Function of Tumor Targeting Peptides by an Amide-to-Triazole Substitution Strategy

scientific article published on 26 August 2015

Radiolabeled antagonistic bombesin peptidomimetics for tumor targeting.

scientific article published on 11 December 2013

Radiolabelling of the octadentate chelators DFO* and oxoDFO* with zirconium-89 and gallium-68

scientific article published on 13 July 2020

Structure-Activity Relationship Studies of Amino Acid Substitutions in Radiolabeled Neurotensin Conjugates

scientific article published on 23 November 2015

Synthesis and Preclinical Evaluation of Radiolabeled [103Ru]BOLD-100

scientific article published on 15 November 2023

TESOTf-induced rearrangement of quinols. Efficient construction of the fully functionalized carbon skeleton of the griseusins by a divergent-reconvergent approach

scientific article published on April 2006

Toward the Optimization of Bombesin-Based Radiotracers for Tumor Targeting.

scientific article published on 07 April 2016

“Click to Chelate”: Synthesis and Installation of Metal Chelates into Biomolecules in a Single Step

scientific article published on 01 November 2006

List of works by Thomas L. Mindt

"Click-to-chelate": design and incorporation of triazole-containing metal-chelating systems into biomolecules of diagnostic and therapeutic interest

"Click-to-chelate": in vitro and in vivo comparison of a 99mTc(CO)3-labeled N(tau)-histidine folate derivative with its isostructural, clicked 1,2,3-triazole analogue

1,2,3-Triazole Stabilized Neurotensin-Based Radiopeptidomimetics for Improved Tumor Targeting.

1,2,3-Triazoles as amide bond mimics: triazole scan yields protease-resistant peptidomimetics for tumor targeting

1,2,3-Triazoles as amide-bond surrogates in peptidomimetics.

A "click chemistry" approach to the efficient synthesis of multiple imaging probes derived from a single precursor

A bombesin-shepherdin radioconjugate designed for combined extra- and intracellular targeting

A click approach to structurally diverse conjugates containing a central di-1,2,3-triazole metal chelate

A solid phase-assisted approach for the facile synthesis of a highly water-soluble zirconium-89 chelator for radiopharmaceutical development.

An octadentate bifunctional chelating agent for the development of stable zirconium-89 based molecular imaging probes

Click-to-Chelate: development of technetium and rhenium-tricarbonyl labeled radiopharmaceuticals

Comparison of the octadentate bifunctional chelator DFO*-pPhe-NCS and the clinically used hexadentate bifunctional chelator DFO-pPhe-NCS for 89Zr-immuno-PET

Convergent Synthesis of 2H-Chromenes - a Formal [3+3] Cycloaddition by a One-pot, Three-Step Cascade.

Cu(I)-catalyzed intramolecular cyclization of alkynoic acids in aqueous media: a "click side reaction".

Development of 68Ga- and 89Zr-Labeled Exendin-4 as Potential Radiotracers for the Imaging of Insulinomas by PET

Dual-targeting conjugates designed to improve the efficacy of radiolabeled peptides

EANM guideline for the preparation of an Investigational Medicinal Product Dossier (IMPD)

Effect of amino acid infusion on potassium serum levels in neuroendocrine tumour patients treated with targeted radiopeptide therapy

Electrocyclic Ring Closure of the Enols of Vinyl Quinones. A2H-Chromene Synthesis

Evaluation of a novel radiofolate in tumour-bearing mice: promising prospects for folate-based radionuclide therapy

Expression of different neurokinin-1 receptor (NK1R) isoforms in glioblastoma multiforme: potential implications for targeted therapy

Fluorescent gallium and indium bis(thiosemicarbazonates) and their radiolabelled analogues: synthesis, structures and cellular confocal fluorescence imaging investigations.

Fluorine-18 click radiosynthesis and preclinical evaluation of a new 18F-labeled folic acid derivative

Glycated 99m Tc-Tricarbonyl-Labeled Peptide Conjugates for Tumor Targeting by "Click-to-Chelate".

Guidance on current good radiopharmacy practice for the small-scale preparation of radiopharmaceuticals using automated modules: a European perspective

Heterocycle Annulation of Enolizable Vinyl Quinone Imides. Dihydroquinolines and Quinolines from Thermal 6π-Electrocyclizations and Indoles from Photochemical Cyclizations

Imaging of activated macrophages in experimental osteoarthritis using folate-targeted animal single-photon-emission computed tomography/computed tomography

Manganese in PET imaging: Opportunities and challenges

Metal chelating systems synthesized using the copper(I) catalyzed azide-alkyne cycloaddition.

Methoxinine - an alternative stable amino acid substitute for oxidation-sensitive methionine in radiolabelled peptide conjugates

Modification of different IgG1 antibodies via glutamine and lysine using bacterial and human tissue transglutaminase

Molecular assembly of multifunctional ⁹⁹(m)Tc radiopharmaceuticals using "clickable" amino acid derivatives.

Novel chemoselective (18)F-radiolabeling of thiol-containing biomolecules under mild aqueous conditions.

Position paper on requirements for toxicological studies in the specific case of radiopharmaceuticals

Probing the Backbone Function of Tumor Targeting Peptides by an Amide-to-Triazole Substitution Strategy

Radiolabeled antagonistic bombesin peptidomimetics for tumor targeting.

Radiolabelling of the octadentate chelators DFO* and oxoDFO* with zirconium-89 and gallium-68

Structure-Activity Relationship Studies of Amino Acid Substitutions in Radiolabeled Neurotensin Conjugates

Synthesis and Preclinical Evaluation of Radiolabeled [103Ru]BOLD-100

TESOTf-induced rearrangement of quinols. Efficient construction of the fully functionalized carbon skeleton of the griseusins by a divergent-reconvergent approach

Toward the Optimization of Bombesin-Based Radiotracers for Tumor Targeting.

“Click to Chelate”: Synthesis and Installation of Metal Chelates into Biomolecules in a Single Step